Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
11x35 3.32738405
21x39 5.03137407
31x43 3.352407
41x50 5.36375409
51x60 3.804638246
62x42 5.15188408
72x46 3.712254149
82x50 5.59315149
9E1x50 7.6773518
10E1x52 5.8479506
113x34 3.5955506
123x37 3.73225408
133x42 3.69387408
143x50 8.34812409
153x51 5.849874178
16I2x51 3.27338407
17I2x57 4.76667697
184x50 5.18937409
194x52 0.9005405
204x61 3.9165417
21E2 15.69441513
22E2x52 7.35062415
235x39 3.45587417
245x47 4.39365198
255x58 6.81213409
266x48 5.60392608
276x51 4.68563417
286x55 4.68587417
29E3 6.45578913
307x38 4.7427515
317x42 4.3729517
327x49 5.389124149
337x53 4.5711509
348x50 4.82338408
35b.1x1 1.6235404
36b.1x2 1.42337401
37b.1x4 1.54833608
38b.1x11 1.64025408
39b.b1x6 7.73363479
40b.l1x3 8.21467679
41b.b2x1 8.6122528
42b.b2x5 7.2221507
43b.b3x3 3.91112408
44b.l3x2 5.7101579
45b.b4x2 5.01662408
46b.b4x3 4.294134157
47b.b4x5 4.17154227
48b.b4x6 8.79507779
49b.b5x2 6.39675407
50b.b5x3 6.72333679
51b.b5x5 5.002754225
52b.b5x7 5.85488407
53b.l5x1 4.1265158
54b.l5x5 6.29381829
55b.b6x5 4.82825406
56b.b7x1 5.2665504
57b.b8x3 3.88788406
58b.b8x4 5.098336156
59b.l8x9 2.687384233
60b.b9x3 4.53587406
61b.l9x3 7.30617649
62b.l9x6 6.08992648
63b.b10x5 4.28517609
64b.b11x4 5.0958549
65b.l11x2 7.7473549
66b.b12x5 4.1305466
67b.b12x6 7.82529748
68b.b13x7 8.1678567
69b.l13x3 6.97367669
70b.l13x6 5.42562449
71b.b14x3 4.97262465
72b.b15x1 8.4945469
73b.b15x2 6.72488456
74b.l15x1 4.68237447
75b.l15x2 4.9263569
76b.b16x4 10.8142466
77b.b16x5 4.65662405
78b.b16x6 7.75664768
79b.b16x7 8.155754129
80b.l16x3 5.879884123
81b.b17x4 5.31954125
82b.b17x6 5.34388407
83b.b17x7 8.22087458
84b.l17x3 8.67617659
85b.l17x6 7.06549
86b.b18x3 5.31887458
87b.b18x5 5.3385405
88b.l18x1 5.84236786
89b.l18x2 5.8475487
90b.l18x3 5.83725485
91b.b19x2 7.8158556
92b.b19x4 6.32263458
93b.l19x1 7.001449
94b.l19x2 5.331559
95b.b20x2 5.345456
96b.b20x4 8.8255658
97b.b20x6 7.9675556
98b.b20x7 3.89237409
99b.l20x2 6.775409
100b.b21x1 5.22407757
101b.b21x2 2.35375406
102b.b21x7 5.22086705
103b.l21x5 3.6754104
104b.b22x5 5.49113487
105b.l22x5 7.05325209
106b.b23x6 6.26056107
107b.l23x1 8.78588426
108b.b24x4 8.187384106
109b.l24x3 4.74225405
110b.b25x3 7.556374105
111b.l25x3 8.22995119
112b.b27x3 5.19975408
113b.l27x1 12.6834629
114b.l27x2 8.117884119
115b.b28x3 4.1494577
116b.b28x4 7.245874116
117b.b28x6 8.5085119
118g.h2x11 7.77587486
119g.ctx3 5.91888409
120g.ctx16 4.3968578
121G.HN.11 1.5287502
122G.S1.05 5.65013409
123G.H1.04 4.87508637
124G.S2.04 6.426407
125G.S2.06 3.51933608
126G.S2.08 2.900124185
127G.S3.03 4.492797187
128G.S3.07 3.2486509
129G.S3.08 4.13625429
130G.H2.04 4.5734529
131G.H2.06 5.61757749
132G.H2.07 5.98842629
133G.H2.08 3.699428
134G.h2s4.01 5.41617629
135G.S4.03 3.62112407
136G.S4.04 6.19588429
137G.s4h3.01 5.200124167
138G.s4h3.03 5.48075437
139G.s4h3.04 5.7675638
140G.s4h3.05 8.97425439
141G.H3.01 7.76562439
142G.H3.06 5.40887407
143G.H3.09 5.71242609
144G.H3.12 4.0066527
145G.H3.15 3.87043728
146G.H3.17 6.099425
147G.H3.18 5.959429
148G.S5.05 3.98919839
149G.S5.07 4.1001539
150G.s5hg.01 3.7695439
151G.HG.07 5.9841539
152G.HG.15 5.66963436
153G.hgh4.02 4.98337408
154G.hgh4.05 6.7088536
155G.H4.10 5.8283537
156G.H4.12 3.99525165
157G.H4.15 4.69025409
158G.S6.02 6.852176138
159G.S6.04 7.50425439
160G.S6.05 7.5784165
161G.s6h5.01 5.24425639
162G.s6h5.02 2.9245507
163G.s6h5.05 4.0039539
164G.H5.03 5.40658638
165G.H5.08 3.7984188
166G.H5.20 3.4265408
167G.H5.23 6.44892694
168G.H5.26 2.3952508
169Lig 9.839162510
170NT 6.17483610
171I3 2.070119130
172G.s4h3.08 4.72188400
173G.h1ha.04 2.336400
174H.HA.13 1.2065400
175H.HA.16 2.0142500
176H.HE.02 1.841400
177H.hahb.06 2.469400
178H.HB.10 2.14175400
179H.hchd.01 1.989500
180H.HD.07 3.049400
181H.HE.09 0.7365400
182H.hehf.04 2.1192500
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
13x36 Lig 25.25498.913NoYes170
23x36 6x48 25.4425.202NoYes078
36x48 7x45 31.0919.075YesNo089
47x45 7x49 31.73676.973NoYes099
53x43 7x49 35.72395.1495NoYes1499
63x43 7x53 46.26744.221NoYes099
73x50 7x53 49.09336.488YesYes099
83x50 G.H5.23 56.336710.1365YesYes094
92x37 2x40 13.62547.149NoNo079
102x40 I1x50 11.71714.1655NoNo098
113x53 G.H5.23 69.41674.9065NoYes984
123x53 G.H5.19 72.97394.872NoNo088
13G.H5.15 G.H5.19 73.14932.9745NoNo088
14G.H5.15 I2x51 73.46323.1775NoYes087
15G.H5.08 I2x51 74.19723.515YesYes087
16G.H5.08 G.S3.03 74.37043.2145YesYes1887
17G.S1.04 G.S3.03 76.56785.2365NoYes067
18G.S1.04 G.S4.03 76.73463.109NoYes067
19G.H5.07 G.S4.03 95.99753.498NoYes087
20G.H5.07 G.S5.05 96.14063.144NoYes089
21G.H1.04 G.S5.05 48.91595.36YesYes379
22G.H1.04 G.S5.07 49.00553.6855YesYes379
23G.S5.07 G.s5hg.01 1004.826YesYes399
24G.S4.07 G.s5hg.01 93.3542.9725NoYes089
25G.S4.07 G.s4h3.03 93.32543.8485NoYes087
26G.H3.05 G.s4h3.03 93.1784.1685NoYes087
27G.H3.05 G.S4.06 93.08823.394NoNo087
28G.H4.15 G.S4.06 93.05946.2895YesNo097
29G.H3.09 G.H4.15 97.70835.1445YesYes099
30G.H3.09 G.S4.04 98.341511.361YesYes099
31G.S5.05 G.s6h5.01 49.64483.76YesYes399
32G.S5.07 G.s6h5.01 50.7915.3375YesYes399
331x60 I1x50 11.23952.7105YesNo068
34G.H3.08 G.S4.04 24.68033.898NoYes299
35G.H2.04 G.H3.08 24.64723.0945YesNo299
36G.H2.04 G.H2.07 49.09427.8YesYes299
37G.H2.02 G.H2.07 56.2024.941NoYes089
38G.H2.02 b.l9x6 55.92485.6615NoYes088
39G.H2.06 b.l9x6 38.27134.0585YesYes498
40G.H2.06 b.l19x1 36.8393.455YesYes499
41b.l17x5 b.l19x1 36.62533.3105NoYes069
42b.l17x5 b.l19x2 36.33354.931NoYes069
43b.l17x3 b.l19x2 25.35863.843YesYes599
44b.b19x4 b.l17x3 15.2888.282YesYes589
45b.b17x7 b.b20x6 21.159310.6645YesYes586
46b.b17x7 b.b21x1 18.46434.4195YesYes587
47G.H3.12 G.S4.04 69.54364.7745YesYes279
48G.H2.04 G.H3.12 24.59513.2565YesYes297
49b.b20x4 b.b20x6 15.94153.69YesYes586
50b.b20x2 b.l19x2 10.08894.842YesYes569
51G.H3.12 G.H3.15 44.97373.87YesYes278
52G.H3.15 G.H3.17 44.57823.085YesYes285
53G.H2.09 G.H3.17 44.27327.1955NoYes285
54G.H2.09 b.l27x1 44.00675.9265NoYes289
55b.l25x6 b.l27x1 51.258223.04NoYes289
56b.l23x1 b.l25x6 50.986722.0945YesNo268
57b.l21x7 b.l23x1 50.78324.278NoYes056
58b.l21x7 b.l23x2 50.54456.69NoNo058
59b.b23x6 b.l23x2 49.87583.1045YesNo078
60b.b23x6 b.b24x6 48.10176.2225YesNo1078
61b.b21x7 b.b24x6 48.236110.37YesNo058
62b.b21x5 b.b21x7 43.37616.465NoYes045
63b.b21x5 b.h2x1 42.72827.916NoNo045
64b.h2x1 b.h2x5 43.03693.759NoNo055
65b.h2x5 b.l24x2 42.37114.202NoNo056
66b.l22x5 b.l24x2 42.10336.62YesNo096
67b.l22x5 g.ctx6 40.0693.217YesNo096
68g.ctx3 g.ctx6 39.65666.4485YesNo096
69g.ctx3 g.ctx4 34.70963.4615YesNo097
70b.l26x5 g.ctx4 34.2743.6905NoNo057
71b.l26x3 b.l26x5 26.85548.733NoNo075
72b.l26x1 b.l26x3 26.53386.217NoNo2177
73b.b2x5 b.l26x1 26.402110.9175YesNo077
74b.b2x5 b.b3x2 25.798512.243YesNo075
75b.b3x2 b.b4x6 25.64485.1825NoYes059
76b.b4x6 b.l1x3 23.86393.226YesYes799
77b.l1x3 b.l3x2 23.7913.402YesYes799
78b.b4x2 b.l3x2 22.98956.501YesYes089
79b.b4x2 b.b5x8 22.00412.8445YesNo085
80b.b5x7 b.b5x8 21.83913.39YesNo075
81b.b4x3 b.b5x7 16.84334.923YesYes077
82b.b3x3 b.b4x3 16.27453.6505YesYes087
83b.b3x3 b.b6x5 15.47513.784YesYes086
84b.b2x4 b.b6x5 14.94713.8695NoYes066
85b.b10x4 b.b2x4 14.769715.12NoNo066
86b.l11x1 b.l9x6 16.8056.4455NoYes498
87b.b11x6 b.l11x1 16.52713.0625NoNo499
88b.b11x6 b.l9x3 12.780115.6935NoYes499
89b.b10x2 b.b10x4 14.59314.458NoNo066
90b.b10x2 b.b14x3 14.41634.7575NoYes065
91b.b14x3 b.b15x1 11.8365.4805YesYes659
92G.S1.06 G.S4.03 23.94322.9685NoYes087
93G.S1.06 G.S3.07 23.71922.9845NoYes089
94G.H1.01 G.S3.07 21.73324.078NoYes099
95G.H1.01 G.hfs2.02 21.31213.254NoNo090
96G.hfs2.02 H.hdhe.04 20.86481.732NoNo000
97H.HE.02 H.hdhe.04 12.21681.28YesNo000
982x46 3x43 10.33794.0835YesNo1499
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
2x563x324.8430NoNo7821
2x567x425.41450NoYes7721
2x577x424.7240NoYes7721
2x63E1x505.321NoYes5812
2x63Lig5.58651NoYes5010
E1x49E24.00250NoYes4321
3x22E28.3371NoYes4321
3x294x6515.8781NoNo5612
3x29Lig4.8961NoYes5010
3x32Lig4.4191NoYes8010
3x334x574.8781NoNo6812
3x33Lig4.3741NoYes6010
3x366x485.2021NoYes7812
3x36Lig8.9131NoYes7010
4x61E2x524.24451YesYes7511
4x615x393.6541YesYes7712
4x61Lig4.48251YesYes7010
4x64E29.31351NoYes4321
4x65E2x528.470NoYes6521
E2E255.2521YesYes3311
E2E2x515.85751YesNo3411
E2Lig27.9091YesYes3010
E2x51Lig3.9821NoYes4010
E2E2x528.5941YesYes3511
E2x52Lig8.0941YesYes5010
5x36E212.520NoYes5321
5x39E24.4751YesYes7321
5x35E26.7361NoYes4321
5x395x434.3531YesNo7721
6x517x373.1211YesNo7612
6x51Lig7.7031YesYes7010
6x547x345.7170NoNo5421
6x55Lig8.7811YesYes7010
6x57E36.16250NoYes5321
6x58Lig9.0191NoYes4010
6x61E33.411NoYes4321
E3Lig12.02251YesYes3010
E3E38.47551YesYes3311
7x347x384.0391NoYes4511
7x34Lig8.97951NoYes4010
7x387x424.35751YesYes5711
7x38Lig6.811YesYes5010
7x42Lig4.3391YesYes7010
1x397x423.02950YesYes7721
2x64Lig3.52551NoYes5010
3x334x613.2851NoYes6711
5x43Lig8.4791NoYes7010
6x516x553.71151YesYes7711
2x60Lig7.34250NoYes7010
2x67E23.73351NoYes4321
6x517x384.2071YesYes7511
5x436x553.92451NoYes7711
2x597x384.30NoYes6521
2x64E14.5421NoNo5011
7x31Lig15.2420NoYes3010
NTNT5.9051YesYes0011
E2NT15.7721YesYes3011
LigNT4.9291YesYes0001
E1Lig7.3511NoYes0010
4x645x354.4071NoNo4422
6x60E33.1181NoYes5321
E2E314.0261YesYes3311
6x62E23.6360NoYes1321
7x24NT2.9120NoYes0021
7x28Lig2.780NoYes0010
5x406x552.32650NoYes6721
6x587x302.1521NoNo4012
7x26E31.6981NoYes0321
7x32NT1.6260NoYes3021
2x5513x321.60650NoNo5821
6x63E30.7140NoYes0321

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
84.00Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
84.00Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
80.00Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
79.17Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
75.00Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
73.91Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
72.00Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
66.67Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
65.22Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
64.29Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
64.29Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
64.29Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
64.00Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
64.00Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
64.00Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
62.96Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
62.96Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
61.54Consensusangiotensin_onOrthosteric Ligandat1_on
61.54Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
60.71Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
60.71Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
60.71Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
59.26Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
59.26Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
59.26Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
59.26Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
59.26Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
59.26Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
58.62Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
58.33Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
57.69Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
57.69Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
57.69Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
57.69Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
57.69Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
57.69Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
57.14Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
57.14Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
57.14Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
57.14Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
57.14Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
56.67Single6IGLIRL16206IGL-ETB-IRL1620
56.67Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
56.00Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
56.00Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
56.00Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
56.00Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
56.00Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
56.00Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
55.56Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
55.56Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
55.56Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
55.56Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
55.56Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
55.56Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
55.17Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
55.17Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
55.17Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
55.17Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
54.84Single5GLHEndothelin-15GLH-ETB-Endothelin-1
54.84Single6IGKEndothelin-36IGK-ETB-Endothelin-3
54.84Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
54.84Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
54.84Consensusbombesin_onOrthosteric Ligandbb2_on
54.84Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
54.84Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
54.84Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
54.84Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
54.84Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
54.17Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
54.17Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
54.17Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
54.17Consensusorexin_onOrthosteric Ligandox2_on
53.85Single7F8XNN90567F8X-CCKA-NN9056
53.85Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
53.85Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
53.85Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
53.85Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
53.85Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
53.85Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
53.85Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
53.85Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
53.57Single6JODAngiotensin II6JOD-AT2-Angiotensin II
53.57Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
53.57Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
53.57Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
53.57Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
53.33Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
53.33Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
53.33Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
53.33Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
53.33Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
52.17Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
52.00Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
52.00Consensuscck_onOrthosteric Ligandccka_on cckb_on
52.00Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
52.00Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
51.85Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
51.85Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
51.85Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
51.85Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
51.85Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
51.85Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
51.85Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
51.85Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
51.85Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
51.72Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
51.72Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
51.72Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
51.72Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
51.72Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
51.72Single8ZRTET-18ZRT-ETB-ET-1
51.72Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
51.61Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
51.61Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
51.61Consensusbradykinin_onOrthosteric Ligandbk2_on
51.61Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
51.61Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
51.52Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
51.52Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
50.00Single4UG2CGS216804UG2-A2A-CGS21680
50.00Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
50.00Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
50.00Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
50.00Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
50.00Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
50.00Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
50.00Single7XN9L-054,5227XN9-SST2-L-054,522
50.00Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
50.00Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
50.00Single8E0GBU728E0G-μ-BU72
50.00Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
50.00Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
50.00Single8QJ2pN1628QJ2-MC4-pN162-Gs
50.00Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
50.00Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
50.00Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
50.00Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
50.00Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
50.00Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
50.00Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
50.00Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
50.00Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
50.00Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
50.00Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
50.00Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
50.00Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
50.00Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
50.00Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
48.48Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
48.48Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
48.48Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
48.28Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
48.28Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
48.28Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
48.28Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
48.28Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
48.28Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
48.28Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
48.15Single4IARErgotamine4IAR-5-HT1B-Ergotamine
48.15Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
48.15Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
48.15Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
48.15Single8WDTphotoNECA8WDT-A2A-photoNECA
48.15Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
48.15Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
48.15Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
48.15Consensuslpl_onOrthosteric Ligands1p_on lpa_on
48.15Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
48.15Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
48.15Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
48.15Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
48.15Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
48.15Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
48.15Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
48.00Single4RWADIPP-NH24RWA-δ-DIPP-NH2
48.00Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
48.00Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
48.00Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
48.00Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
48.00Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
48.00Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
48.00Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
48.00Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
48.00Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
48.00Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
48.00Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
48.00Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
48.00Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
48.00Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
47.83Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
47.83Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
47.83Single8K5DGSK2560738K5D-HCA2-GSK256073
47.83Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
47.83Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
47.83Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
47.83Consensushca_on_gpOrthosteric Ligandhca2_on_gp
47.22Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
47.22Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
46.88Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
46.88Single8IY6Endothelin-18IY6-ETB-Endothelin-1
46.88Consensusendothelin_onOrthosteric Ligandetb_on eta_on
46.88Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
46.67Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
46.67Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
46.67Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
46.67Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
46.67Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
46.67Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
46.67Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
46.67Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
46.67Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
46.67Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
46.43Single3QAKUK-4320973QAK-A2A-UK-432097
46.43Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
46.43Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
46.43Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
46.43Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
46.43Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
46.43Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
46.43Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
46.43Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
46.15Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
46.15Single7EZCUKA7EZC-A2A-UKA
46.15Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
46.15Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
46.15Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
46.15Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
46.15Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
46.15Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
46.15Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
46.15Consensuschemerin_onOrthosteric Ligandcml1_on
46.15Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
46.15Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
46.15Consensusprostanoid_offOrthosteric Ligandep_off dp_off
45.83Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
45.83Single5C1MBU725C1M-μ-BU72
45.83Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
45.83Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
45.83Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
45.83Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
45.83Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
45.83Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
45.83Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
45.45Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
45.16Single4XT3Fractalkine4XT3-US28-Fractalkine
45.16Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
45.16Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
44.83Single5WF5UK-4320975WF5-A2A-UK-432097
44.83Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
44.83Single6PT2KGCHM076PT2-δ-KGCHM07
44.83Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
44.83Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
44.83Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
44.83Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
44.83Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
44.83Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
44.83Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
44.83Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
44.44Single5WF6UK-4320975WF6-A2A-UK-432097
44.44Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
44.44Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
44.44Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
44.44Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
44.44Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
44.44Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
44.44Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
44.44Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
44.44Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
44.44Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
44.44Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
44.12Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
44.12Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
44.12Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
44.00Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
44.00Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
44.00Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
44.00Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
44.00Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
44.00Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
44.00Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
44.00Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
44.00Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
44.00Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
44.00Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
44.00Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
44.00Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
44.00Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
44.00Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
44.00Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
44.00Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
44.00Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
44.00Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
44.00Consensusrelaxin_onOrthosteric Ligandrxfp4_on
44.00Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
43.75Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
43.75Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
43.75Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
43.75Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
43.75Single9KDFRES-701-39KDF-ETB-RES-701-3
43.48Single4ZJCSB-6740424ZJC-OX1-SB-674042
43.48Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
43.48Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
43.48Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
43.48Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
43.48Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
43.48Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
43.48Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
43.48Consensushca_onOrthosteric Ligandhca2_on
43.33Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
43.33Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
43.33Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
43.33Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
43.33Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
43.33Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
43.33Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
43.33Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
43.33Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
42.86Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
42.86Single4XT1Fractalkine4XT1-US28-Fractalkine
42.86Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
42.86Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
42.86Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
42.86Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
42.86Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
42.86Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
42.86Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
42.86Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
42.86Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
42.86Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
42.86Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
42.86Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
42.86Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
42.86Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
42.86Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
42.42Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
42.42Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
42.42Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
42.31Single4XEENeurotensin4XEE-NTS1-Neurotensin
42.31Single4XESNeurotensin4XES-NTS1-Neurotensin
42.31Single6MXTSalmeterol6MXT-β2-Salmeterol
42.31Single6OS2TRV0266OS2-AT1-TRV026
42.31Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
42.31Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
42.31Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
42.31Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
42.31Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
42.31Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
42.31Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
42.31Single7YITNalfurafine7YIT-κ-Nalfurafine
42.31Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
42.31Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
42.31Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
42.31Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
42.31Single8JJLOlodaterol8JJL-β2-Olodaterol
42.31Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
42.31Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
42.31Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
42.31Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
42.31Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
42.31Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
42.31Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
42.31Consensusalpha1_offOrthosteric Ligandalpha1a_off
42.31Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
42.31Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
42.31Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
42.31Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
42.31Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
42.31Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
42.31Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
42.31Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
42.31Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
42.31Consensuslpa_offOrthosteric Ligandlpa1_off
42.31Consensuslpl_offOrthosteric Ligands1p_off lpa_off
42.31Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
42.31Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
42.31Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
42.31Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
42.31Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
41.94Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
41.94Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
41.94Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
41.94Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
41.94Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
41.94Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
41.94Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
41.67Single6TOTLemborexant6TOT-OX1-Lemborexant
41.67Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
41.67Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
41.67Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
41.67Single7UL4Alvimopan7UL4-μ-Alvimopan
41.67Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
41.67Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
41.67Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
41.67Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
41.67Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
41.67Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
41.67Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
41.67Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
41.67Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
41.67Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
41.67Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
41.67Consensusa3_onOrthosteric Liganda3a_on
41.67Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
41.67Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
41.67Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
41.67Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
41.67Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
41.67Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
41.67Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
41.67Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
41.67Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
41.67Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
41.38Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
41.38Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
41.38Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
41.38Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
41.38Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
41.38Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
41.38Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
41.38Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
41.38Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
41.38Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
41.18Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
40.74Single4BUONeurotensin4BUO-NTS1-Neurotensin
40.74Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
40.74Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
40.74Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
40.74Single6IBLArformoterol6IBL-β1-Arformoterol
40.74Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
40.74Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
40.74Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
40.74Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
40.74Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
40.74Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
40.74Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
40.74Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
40.74Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
40.74Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
40.74Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
40.74Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
40.74Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
40.74Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
40.74Consensusendothelin_offOrthosteric Ligandetb_off
40.74Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
40.74Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
40.74Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
40.74Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
40.74Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
40.74Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
40.74Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
40.62Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
40.62Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
40.62Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
40.62Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
40.48Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
40.00Single3OE0CVX153OE0-CXCR4-CVX15
40.00Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
40.00Single5N2SPSB365N2S-A1-PSB36
40.00Single5WQCEMPA5WQC-OX2-EMPA
40.00Single6D26Fevipiprant6D26-DP2-Fevipiprant
40.00Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
40.00Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
40.00Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
40.00Single6TP6Filorexant6TP6-OX1-Filorexant
40.00Single7C61Ergotamine7C61-5-HT1B-Ergotamine
40.00Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
40.00Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
40.00Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
40.00Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
40.00Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
40.00Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
40.00Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
40.00Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
40.00Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
40.00Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
40.00Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
40.00Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
40.00Single8S4DCMF-0198S4D-Apelin-CMF-019
40.00Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
40.00Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
40.00Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
40.00Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
40.00Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
40.00Single9EHSLUF76029EHS-A3A-LUF7602
40.00Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
40.00Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
40.00Consensusa3_on_gpOrthosteric Liganda3a_on_gp
40.00Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
40.00Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
40.00Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
40.00Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
40.00Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
40.00Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
40.00Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
40.00Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
40.00Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
40.00Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
40.00Consensusdp_offOrthosteric Liganddp2_off
40.00Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
40.00Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
40.00Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
40.00Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
39.39Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
39.29Single3NY9ICI118-5513NY9-β2-ICI118-551
39.29Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
39.29Single5ZTYAM102575ZTY-CB2-AM10257
39.29Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
39.29Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
39.29Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
39.29Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
39.29Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
39.29Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
39.29Single8XQJJN2418XQJ-Apelin-JN241
39.29Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
39.29Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
39.29Single9IPYJR14a9IPY-C3aB-JR14a
39.29Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
39.29Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
39.29Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
39.29Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
39.29Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
39.29Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
39.13Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
39.13Single5WS3EMPA5WS3-OX2-EMPA
39.13Single6TODEMPA6TOD-OX1-EMPA-Na
39.13Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
39.13Single7XRRLemborexant7XRR-OX2-Lemborexant
39.13Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
39.13Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
39.13Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
39.13Single8GNGIstradefylline8GNG-A2A-Istradefylline
39.13Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
39.13Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
39.13Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
39.13Consensusorexin_offOrthosteric Ligandox2_off ox1_off
39.13Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
39.13Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
38.71Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
38.71Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
38.71Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
38.71Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
38.71Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
38.71Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
38.71Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
38.71Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
38.71Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
38.71Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
38.71Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
38.71Consensusvasop-oxy_onOrthosteric Ligandv2_on
38.71Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
38.46Single2YDVNECA2YDV-A2A-NECA
38.46Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
38.46Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
38.46Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
38.46Single4UHRCGS216804UHR-A2A-CGS21680
38.46Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
38.46Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
38.46Single5G53NECA5G53-A2A-NECA-Gs
38.46Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
38.46Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
38.46Single6H7JIsoprenaline6H7J-β1-Isoprenaline
38.46Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
38.46Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
38.46Single6OS1TRV0266OS1-AT1-TRV026
38.46Single6TQ7SB-3348676TQ7-OX1-SB-334867
38.46Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
38.46Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
38.46Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
38.46Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
38.46Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
38.46Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
38.46Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
38.46Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
38.46Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
38.46Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
38.46Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
38.46Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
38.46Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
38.46Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
38.46Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
38.46Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
38.46Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
38.46Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
38.46Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
38.46Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
38.46Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
38.46Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
38.46Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
38.46Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
38.46Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
38.46Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
38.46Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
38.46Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
38.46Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
38.46Consensusa2_onOrthosteric Liganda2b_on
38.46Consensusa2_on_gpOrthosteric Liganda2b_on_gp
38.46Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
38.46Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
38.46Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
38.46Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
38.46Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
38.46Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
38.46Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
38.46Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
38.46Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
38.46Consensusneurotensin_onOrthosteric Ligandnts1_on
38.46Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
38.46Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
38.46Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
37.93Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
37.93Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
37.93Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
37.93Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
37.93Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
37.93Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
37.93Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
37.93Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
37.93Single8WKYPG-9348WKY-MC4-PG-934
37.93Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
37.93Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
37.93Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
37.93Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
37.93Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
37.93Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
37.93Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
37.84Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
37.50Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
37.50Single6PS0S-Carazolol6PS0-β2-S-Carazolol
37.50Single6PS4ICI118-5516PS4-β2-ICI118-551
37.50Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
37.50Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
37.50Single6TPGEMPA6TPG-OX2-EMPA
37.50Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
37.50Single6V9SGTPL114036V9S-OX1-GTPL11403
37.50Single7F61PF-036547467F61-H3-PF-03654746
37.50Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
37.50Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
37.50Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
37.50Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
37.50Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
37.50Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
37.50Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
37.50Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
37.50Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
37.50Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
37.50Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
37.50Single8IHKAcifran8IHK-HCA3-Acifran
37.50Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
37.50Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
37.50Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
37.50Single8K5CAcipimox8K5C-HCA2-Acipimox
37.50Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
37.50Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
37.50Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
37.50Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
37.50Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
37.50Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
37.50Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
37.50Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
37.50Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
37.50Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
37.50Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
37.50Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
37.50Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
37.50Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
37.14Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
37.14Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
37.04Single4AMIBucindolol4AMI-β1-Bucindolol
37.04Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
37.04Single4LDEBI1671074LDE-β2-BI167107
37.04Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
37.04Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
37.04Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
37.04Single6YVRNTS8-136YVR-NTS1-NTS8-13
37.04Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
37.04Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
37.04Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
37.04Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
37.04Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
37.04Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
37.04Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
37.04Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
37.04Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
37.04Single8JJ8Formoterol8JJ8-β2-Formoterol
37.04Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
37.04Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
37.04Single8XYIVUF106618XYI-CXCR3-VUF10661
37.04Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
37.04Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
37.04Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
37.04Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
37.04Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
37.04Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
37.04Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
37.04Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
37.04Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
37.04Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
37.04Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
37.04Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
37.04Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
36.67Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
36.67Single7SK5CXCL127SK5-ACKR3-CXCL12
36.67Single7XNACYN1548067XNA-SST2-CYN154806
36.67Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
36.67Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
36.67Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
36.67Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
36.36Single7SK3CXCL127SK3-ACKR3-CXCL12
36.36Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
36.36Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
36.00Single2Y04Salbutamol2Y04-β1-Salbutamol
36.00Single3NY8ICI118-5513NY8-β2-ICI118-551
36.00Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
36.00Single4EJ4Naltrindole4EJ4-δ-Naltrindole
36.00Single4GBRS-Carazolol4GBR-β2-S-Carazolol
36.00Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
36.00Single4QKX35V4QKX-β2-35V
36.00Single4YAYZD-71554YAY-AT1-ZD-7155
36.00Single6D27CAY104716D27-DP2-CAY10471
36.00Single6PS1Timolol6PS1-β2-Timolol
36.00Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
36.00Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
36.00Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
36.00Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
36.00Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
36.00Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
36.00Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
36.00Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
36.00Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
36.00Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
36.00Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
36.00Single7V3ZCP559407V3Z-CB1-CP55940
36.00Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
36.00Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
36.00Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
36.00Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
36.00Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
36.00Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
36.00Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
36.00Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
36.00Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
36.00Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.00Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.00Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.00Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.00Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.00Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.00Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.00Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.00Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.00Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.00Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
36.00Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
36.00Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
36.00Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
36.00Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
36.00Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
36.00Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
36.00Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
36.00Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
36.00Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
36.00Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
36.00Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.00Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.00Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.00Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.00Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
36.00Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
36.00Single9CHXS-Carazolol9CHX-β2-S-Carazolol
36.00Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
36.00Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
36.00Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
36.00Consensuscck_offOrthosteric Ligandccka_off
36.00Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
36.00Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
36.00Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
36.00Consensusdopamine_offOrthosteric Ligandd2_off d3_off
36.00Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
36.00Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
35.71Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
35.71Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
35.71Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
35.71Single5X93K-87945X93-ETB-K-8794
35.71Single6H7LDobutamine6H7L-β1-Dobutamine
35.71Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
35.71Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
35.71Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
35.71Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
35.71Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
35.71Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
35.71Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
35.71Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
35.71Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
35.71Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
35.71Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
35.71Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
35.71Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
35.71Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
35.71Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
35.71Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
35.71Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
35.71Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
35.71Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
35.71Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
35.71Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
35.48Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
35.48Single6W25SHU91196W25-MC4-SHU9119-Ca
35.48Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
35.48Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
35.48Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
35.48Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
35.48Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
35.48Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
35.29Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
35.29Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
34.78Single3OE9IT1t3OE9-CXCR4-IT1t
34.78Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
34.78Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
34.78Single8K5BNiacin8K5B-HCA2-Niacin
34.78Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
34.78Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
34.62Single2RH1S-Carazolol2RH1-β2-S-Carazolol
34.62Single2Y03Isoprenaline2Y03-β1-Isoprenaline
34.62Single2YCWS-Carazolol2YCW-β1-S-Carazolol
34.62Single5D6LS-Carazolol5D6L-β2-S-Carazolol
34.62Single5JQHS-Carazolol5JQH-β2-S-Carazolol
34.62Single5N2RPSB-365N2R-A2A-PSB-36-Na
34.62Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
34.62Single5WIUNemonapride5WIU-D4-Nemonapride
34.62Single5WIVNemonapride5WIV-D4-Nemonapride-Na
34.62Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
34.62Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
34.62Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
34.62Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
34.62Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
34.62Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
34.62Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
34.62Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
34.62Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
34.62Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
34.62Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
34.62Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
34.62Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
34.62Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
34.62Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
34.62Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
34.62Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
34.62Single8GNEKW-63568GNE-A2A-KW-6356-Na
34.62Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
34.62Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
34.62Single8JXSPF-61428JXS-D1-PF-6142
34.62Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
34.62Single8TF5Oleic acid8TF5-GPR6-Oleic acid
34.62Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
34.62Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
34.62Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
34.62Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
34.62Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
34.62Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
34.62Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
34.62Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
34.62Single9HAPTolvaptan9HAP-V2-Tolvaptan
34.62Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
34.62Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
34.62Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
34.62Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
34.62Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
34.62Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
34.62Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
34.62Consensusamine_offonOrthosteric Ligandamine_off amine_on
34.62Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
34.62Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
34.62Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
34.62Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
34.62Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
34.62Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
34.62Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
34.62Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
34.62Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
34.62Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
34.62Consensustrace-amine_onOrthosteric Ligandta1_on
34.48Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
34.48Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
34.48Single6PT3DPI-2876PT3-δ-DPI-287
34.48Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
34.48Single7SK9CCX6627SK9-ACKR3-CCX662
34.48Single8X5YAstemizole8X5Y-H1-Astemizole
34.48Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
34.48Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
34.48Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
34.48Consensuskisspeptin_onOrthosteric Ligandkiss1_on
34.38Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
34.38Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
34.29Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
34.29Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
33.33Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
33.33Single3P0GBI1671073P0G-β2-BI167107
33.33Single4BV0Neurotensin4BV0-NTS1-Neurotensin
33.33Single4DJHJDTic4DJH-κ-JDTic
33.33Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
33.33Single4S0VSuvorexant4S0V-OX2-Suvorexant
33.33Single5D5AS-Carazolol5D5A-β2-S-Carazolol
33.33Single5D5BS-Carazolol5D5B-β2-S-Carazolol
33.33Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
33.33Single5XR8AM8415XR8-CB1-AM841
33.33Single5XRAAM115425XRA-CB1-AM11542
33.33Single6AKXA4R6AKX-CCR5-A4R
33.33Single6B73MP11046B73-κ-MP1104
33.33Single6J21Aprepitant6J21-NK1-Aprepitant
33.33Single6TPJSuvorexant6TPJ-OX2-Suvorexant
33.33Single6WGTLSD6WGT-5-HT2A-LSD
33.33Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
33.33Single7B6WCyclazosin7B6W-α1b-Cyclazosin
33.33Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
33.33Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
33.33Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
33.33Single7F8ULintitript7F8U-CCKA-Lintitript
33.33Single7F8YDevazepide7F8Y-CCKA-Devazepide
33.33Single7FEECP559407FEE-CB1-CP55940-ZCZ011
33.33Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
33.33Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
33.33Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
33.33Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
33.33Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
33.33Single7TUYGSK682753A7TUY-GPR183-GSK682753A
33.33Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
33.33Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
33.33Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
33.33Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
33.33Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
33.33Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
33.33Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
33.33Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
33.33Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
33.33Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
33.33Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
33.33Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
33.33Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
33.33Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
33.33Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
33.33Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
33.33Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
33.33Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
33.33Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
33.33Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
33.33Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
33.33Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
33.33Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
33.33Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
33.33Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
33.33Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
33.33Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
33.33Single8IWESpermidine8IWE-TA9-Spermidine
33.33Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
33.33Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
33.33Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
33.33Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
33.33Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
33.33Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
33.33Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
33.33Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
33.33Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
33.33Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
33.33Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
33.33Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
33.33Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
33.33Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
33.33Single8XVLZibotentan8XVL-ETA-Zibotentan
33.33Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
33.33Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
33.33Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
33.33Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
33.33Single8ZWFJR14a8ZWF-C3aB-JR14a
33.33Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
33.33Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
33.33Single9BJKNaloxone9BJK-μ-Naloxone-NAM
33.33Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
33.33Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
33.33Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
33.33Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
33.33Single9M4TSilodosin9M4T-Alpha1A-Silodosin
33.33Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
33.33Consensusalpha2_offOrthosteric Ligandalpha2c_off
33.33Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
33.33Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
33.33Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
33.33Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
33.33Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
33.33Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
33.33Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
33.33Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
33.33Consensuslpa_onOrthosteric Ligandlpa1_on
33.33Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
33.33Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
33.33Consensuspac_onOrthosteric Ligandpac1_on
33.33Consensuspth_onOrthosteric Ligandpth1_on pth2_on
33.33Consensussomatostatin_offOrthosteric Ligandsst2_off
33.33Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
33.33Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
33.33Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
33.33Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
32.35Single6FJ3PTH6FJ3-PTH1-PTH
32.35Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
32.35Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
32.26Single6HLOAprepitant6HLO-NK1-Aprepitant
32.26Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
32.26Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
32.26Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
32.26Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
32.26Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
32.26Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
32.26Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
32.26Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
32.14Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
32.14Single3D4STimolol3D4S-β2-Timolol
32.14Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
32.14Single6A93Risperidone6A93-5-HT2A-Risperidone
32.14Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
32.14Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
32.14Single6KQICP559406KQI-CB1-CP55940-Org27569
32.14Single6ZG4HTL00099366ZG4-M1-HTL0009936
32.14Single7DFPSpiperone7DFP-D2-Spiperone
32.14Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
32.14Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
32.14Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
32.14Single7K15MKD0467K15-BLT1-MKD046-Na
32.14Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
32.14Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
32.14Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
32.14Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
32.14Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
32.14Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
32.14Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
32.14Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
32.14Single8JWY2-1188JWY-A2A-2-118
32.14Single8JWZAB9288JWZ-A2A-AB928-Na
32.14Single8XQJJN2418XQJ-Apelin-JN241
32.14Single9DGIZ85267113509DGI-CB1-Z8526711350
32.14Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
32.14Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
32.14Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
32.14Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
32.14Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
32.14Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
32.14Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
32.14Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
32.14Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
32.14Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
32.00Single2YDOAdenosine2YDO-A2A-Adenosine
32.00Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
32.00Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
32.00Single4MBSMaraviroc4MBS-CCR5-Maraviroc
32.00Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
32.00Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
32.00Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
32.00Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
32.00Single6IQLL7458706IQL-D4-L745870
32.00Single6KUXRS-799486KUX-α2a-RS-79948
32.00Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
32.00Single6MH8ZM-2413856MH8-A2A-ZM-241385
32.00Single6PS5S-Propranolol6PS5-β2-S-Propranolol
32.00Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
32.00Single6TP3Nemorexant6TP3-OX1-Nemorexant
32.00Single6TPNHTL66416TPN-OX2-HTL6641
32.00Single7AROLUF58337ARO-A2A-LUF5833-Na
32.00Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
32.00Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
32.00Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
32.00Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
32.00Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
32.00Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
32.00Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
32.00Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
32.00Single7UL3Famotidine7UL3-H2-Famotidine
32.00Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
32.00Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
32.00Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
32.00Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
32.00Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
32.00Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
32.00Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
32.00Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
32.00Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
32.00Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
32.00Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
32.00Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
32.00Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
32.00Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
32.00Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
32.00Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
32.00Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
32.00Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
32.00Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
32.00Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
32.00Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
32.00Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
32.00Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
32.00Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
32.00Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
32.00Single8ZPMAMD0708ZPM-CXCR4-AMD070
32.00Single9AS5Mescaline9AS5-5-HT2A-Mescaline
32.00Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
32.00Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
32.00Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
32.00Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
32.00Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
32.00Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
32.00Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
32.00Consensusalpha1_onOrthosteric Ligandalpha1a_on
32.00Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
32.00Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
32.00Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
32.00Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
32.00Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
32.00Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
32.00Consensusgrh_offOrthosteric Ligandgnrh1_off
32.00Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
31.71Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
31.43Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
31.43Consensusglp_onOrthosteric Ligandglp1_on glp2_on
31.43Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
31.25Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
31.25Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
31.25Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
31.25Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
31.25Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
31.03Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
31.03Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
31.03Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
31.03Single7UM4AS26747237UM4-5-HT5A-AS2674723
31.03Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
31.03Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
31.03Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
31.03Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
31.03Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
31.03Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
31.03Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
31.03Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
31.03Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
31.03Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.03Single8ZPLHF511168ZPL-CXCR4-HF51116
31.03Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
31.03Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
30.77Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
30.77Single2Y02Carmoterol2Y02-β1-Carmoterol
30.77Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
30.77Single3EMLZM-2413853EML-A2A-ZM-241385
30.77Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
30.77Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
30.77Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
30.77Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
30.77Single5DHGC-355DHG-NOP-C-35
30.77Single5DHHSB-6121115DHH-NOP-SB-612111
30.77Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
30.77Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
30.77Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
30.77Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
30.77Single5UIGCmpd-15UIG-A2A-Cmpd-1
30.77Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
30.77Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
30.77Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
30.77Single6H7MSalbutamol6H7M-β1-Salbutamol
30.77Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
30.77Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
30.77Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
30.77Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
30.77Single6S0LZM-2413856S0L-A2A-ZM-241385
30.77Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
30.77Single7BU7BI1671077BU7-β1-BI167107
30.77Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
30.77Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
30.77Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
30.77Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
30.77Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
30.77Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
30.77Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
30.77Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
30.77Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
30.77Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
30.77Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
30.77Single8CU6LJ-45178CU6-A2A-LJ-4517
30.77Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
30.77Single8JJOAlprenolol8JJO-β2-Alprenolol
30.77Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
30.77Single8JXRLSD8JXR-D1-LSD
30.77Single8T1WCVN4248T1W-GPR6-CVN424
30.77Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
30.77Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
30.77Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
30.77Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
30.77Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
30.77Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
30.77Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
30.77Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
30.77Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
30.77Single9H37A1IR09H37-A2A-A1IR0-Na
30.77Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
30.77Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
30.77Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
30.77Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
30.77Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
30.77Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
30.77Consensus5ht5_onOrthosteric Ligand5ht5a_on
30.77Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
30.77Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
30.77Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
30.77Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
30.77Consensusblt_onOrthosteric Ligandblt1_on
30.77Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
30.77Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
30.77Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
30.77Consensusleukotriene_onOrthosteric Ligandblt_on
30.77Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
30.56Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
30.56Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
30.56Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
30.56Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
30.56Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
30.56Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
30.43Single3OE6IT1t3OE6-CXCR4-IT1t
30.43Single6ME5Agomelatine6ME5-MT1-Agomelatine
30.43Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
30.43Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
30.43Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
30.43Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
30.43Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
30.43Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
30.30Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
30.30Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
30.30Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
30.30Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
30.30Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
30.23Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
30.00Single6KNMJN241-96KNM-Apelin-JN241-9
30.00Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
30.00Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
30.00Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
30.00Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
30.00Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
29.63Single2Y00Dobutamine2Y00-β1-Dobutamine
29.63Single5IUAQ274563485IUA-A2A-Q27456348-Na
29.63Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
29.63Single5TVNLSD5TVN-5-HT2B-LSD
29.63Single6E67BI1671076E67-β2-BI167107-Gs(CT)
29.63Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
29.63Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
29.63Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
29.63Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
29.63Single6PS6Timolol6PS6-β2-Timolol
29.63Single6S0QZM-2413856S0Q-A2A-ZM-241385
29.63Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
29.63Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
29.63Single7C4SS1P7C4S-S1P3-S1P
29.63Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
29.63Single7W41PD1762527W41-BB2-PD176252
29.63Single7WC6LSD7WC6-5-HT2A-LSD
29.63Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
29.63Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
29.63Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
29.63Single8QOTNanobody-E8QOT-μ-Nanobody-E
29.63Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
29.63Single8ZMFA1L108ZMF-5-HT2C-A1L10
29.63Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
29.63Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
29.63Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.63Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
29.63Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
29.63Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
29.63Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
29.63Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
29.63Consensusadenosine_offOrthosteric Liganda1_off a2_off
29.63Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
29.63Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
29.63Consensusbombesin_offOrthosteric Ligandbb2_off
29.63Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
29.63Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
29.63Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
29.63Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
29.63Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
29.41Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
29.41Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
29.17Single3PBLEticlopride3PBL-D3-Eticlopride
29.17Single6HLLCP999946HLL-NK1-CP99994
29.17Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
29.17Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
29.17Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
29.17Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
29.17Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
29.17Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
29.17Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
29.17Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
29.17Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
29.17Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
29.17Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
29.17Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
29.17Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
29.17Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
29.17Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
29.17Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
29.17Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
29.17Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
29.17Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
29.17Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
29.17Consensusgq_nucleotideOrthosteric Ligandgq_p2y
29.17Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
29.03Single7QA8Peptide7QA8-STE2-Peptide
29.03Single7QA8Peptide7QA8-STE2-Peptide
29.03Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
29.03Single8XWNCXCL88XWN-CXCR2-CXCL8
29.03Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
28.95Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
28.95Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
28.57Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
28.57Single6J20Aprepitant6J20-NK1-Aprepitant
28.57Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
28.57Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
28.57Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
28.57Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
28.57Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
28.57Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
28.57Single7PX4PSB-21137PX4-A2A-PSB-2113
28.57Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
28.57Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
28.57Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
28.57Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
28.57Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
28.57Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
28.57Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
28.57Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
28.57Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
28.57Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
28.57Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
28.57Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
28.57Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
28.57Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
28.57Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
28.57Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
28.57Consensustachykinin_offOrthosteric Ligandnk1_off
28.57Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
28.21Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
28.21Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
28.12Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
28.12Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
28.00Single3ODUIT1t3ODU-CXCR4-IT1t
28.00Single3PWHZM-2413853PWH-A2A-ZM-241385
28.00Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
28.00Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
28.00Single4BWBNeurotensin4BWB-NTS1-Neurotensin
28.00Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
28.00Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
28.00Single6AKYMaraviroc6AKY-CCR5-Maraviroc
28.00Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
28.00Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
28.00Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
28.00Single6ME2Ramelteon6ME2-MT1-Ramelteon
28.00Single6ME9Ramelteon6ME9-MT2-Ramelteon
28.00Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
28.00Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
28.00Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
28.00Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
28.00Single7BR3Elagolix7BR3-GnRH1-Elagolix
28.00Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
28.00Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
28.00Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
28.00Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
28.00Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
28.00Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
28.00Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
28.00Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
28.00Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
28.00Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
28.00Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
28.00Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.00Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.00Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
28.00Single8Y0HVUF114188Y0H-CXCR3-VUF11418
28.00Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
28.00Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
28.00Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
28.00Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
28.00Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
28.00Consensusangiotensin_offOrthosteric Ligandat1_off
28.00Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
28.00Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
28.00Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
27.78Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
27.78Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
27.78Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
27.78Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
27.78Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
27.78Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
27.59Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
27.59Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
27.59Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
27.59Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
27.59Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
27.59Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
27.59Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
27.59Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
27.50Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
27.50Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
27.50Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.50Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
27.27Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
27.27Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.27Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
27.27Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
27.03Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
27.03Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
27.03Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
27.03Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
27.03Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
26.92Single3REYXAC3REY-A2A-XAC
26.92Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
26.92Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
26.92Single5IU7Q274563465IU7-A2A-Q27456346-Na
26.92Single5IUBQ274563445IUB-A2A-Q27456344-Na
26.92Single5JTBZM-2413855JTB-A2A-ZM-241385
26.92Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
26.92Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
26.92Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
26.92Single5UVIZM-2413855UVI-A2A-ZM-241385
26.92Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
26.92Single6VI4JDTic6VI4-κ-JDTic
26.92Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
26.92Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
26.92Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
26.92Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
26.92Single6ZG9GSK10347026ZG9-M1-GSK1034702
26.92Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
26.92Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
26.92Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
26.92Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
26.92Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
26.92Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
26.92Single7T32ZM-2413857T32-A2A-ZM-241385
26.92Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
26.92Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
26.92Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
26.92Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
26.92Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
26.92Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
26.92Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
26.92Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
26.92Single8RLNLUF58348RLN-A2A-LUF5834
26.92Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
26.92Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.92Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
26.92Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
26.92Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
26.92Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
26.92Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
26.92Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
26.92Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
26.92Single8ZPNAMD31008ZPN-CXCR4-AMD3100
26.92Single9AS3LSD9AS3-5-HT2A-LSD
26.92Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
26.92Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
26.92Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
26.92Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
26.92Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
26.92Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
26.92Consensusa2_offOrthosteric Liganda2a_off
26.92Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
26.92Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
26.92Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
26.83Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
26.67Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
26.67Single6K1QIRL25006K1Q-ETB-IRL2500
26.67Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
26.67Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
26.67Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
26.67Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.67Single8XVUCXCL28XVU-CXCR2-CXCL2
26.67Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
26.67Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
26.67Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
26.67Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
26.47Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
26.47Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
26.47Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
26.47Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
26.32Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
26.09Single6TQ9SB-4081246TQ9-OX1-SB-408124
26.09Single8A2OTheophylline8A2O-A2A-Theophylline-Na
26.09Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.09Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
26.09Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
26.09Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
25.93Single2Y01Dobutamine2Y01-β1-Dobutamine
25.93Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
25.93Single5IU8Q274563475IU8-A2A-Q27456347-Na
25.93Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
25.93Single5T04Neurotensin5T04-NTS1-Neurotensin
25.93Single5TGZAM65385TGZ-CB1-AM6538
25.93Single5UENDU1725UEN-A1-DU172
25.93Single6DRXLisuride6DRX-5-HT2B-Lisuride
25.93Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
25.93Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
25.93Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
25.93Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
25.93Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
25.93Single7PYRPSB-21157PYR-A2A-PSB-2115
25.93Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
25.93Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
25.93Single7WC7Lisuride7WC7-5-HT2A-Lisuride
25.93Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
25.93Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
25.93Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
25.93Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
25.93Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
25.93Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
25.93Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
25.93Single8X64Desloratadine8X64-H1-Desloratadine
25.93Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
25.93Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
25.93Single9IYAONO-97105319IYA-GPR55-ONO-9710531
25.93Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
25.93Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
25.93Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
25.93Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
25.93Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
25.93Consensusalpha2_onOrthosteric Ligandalpha2b_on
25.93Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
25.93Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
25.93Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
25.81Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
25.81Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
25.71Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
25.71Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
25.71Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
25.71Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
25.71Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
25.71Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
25.64Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
25.64Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
25.64Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
25.64Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
25.58Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
25.00Single4XNWMRS25004XNW-P2Y1-MRS2500
25.00Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
25.00Single5XPRBosentan5XPR-ETB-Bosentan
25.00Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
25.00Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
25.00Single6HLPNetupitant6HLP-NK1-Netupitant
25.00Single6LUQHaloperidol6LUQ-D2-Haloperidol
25.00Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
25.00Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
25.00Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
25.00Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
25.00Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
25.00Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
25.00Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
25.00Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
25.00Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
25.00Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
25.00Single7SINNPS-21437SIN-CaS-NPS-2143
25.00Single7SINNPS-21437SIN-CaS-NPS-2143
25.00Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
25.00Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8IEBA1LYA8IEB-GPR156-A1LYA
25.00Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
25.00Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
25.00Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
25.00Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
25.00Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
25.00Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
25.00Single8KIGSHU91198KIG-MC3-SHU9119-Ca
25.00Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
25.00Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
25.00Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
25.00Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
25.00Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
25.00Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
25.00Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
25.00Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
25.00Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
25.00Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
25.00Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
25.00Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
25.00Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
25.00Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
25.00Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
25.00Single9LRCHistamine9LRC-H4-Histamine
25.00Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
25.00Consensus5ht2_onOrthosteric Ligand5ht2b_on
25.00Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
25.00Consensusblt_offOrthosteric Ligandblt1_off
25.00Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
25.00Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
25.00Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
25.00Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
25.00Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
25.00Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
25.00Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
25.00Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
25.00Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
24.39Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
24.32Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
24.32Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
24.32Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
24.32Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
24.32Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
24.32Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
24.24Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
24.24Single8IEBA1LYA8IEB-GPR156-A1LYA
24.24Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
24.14Single4U15Tiotropium4U15-M3-Tiotropium
24.14Single5TZRMK86665TZR-FFA1-MK8666
24.14Single5V54Methiothepin5V54-5-HT1B-Methiothepin
24.14Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
24.14Single6E59L-7607356E59-NK1-L-760735
24.14Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
24.14Single6OL9Tiotropium6OL9-M5-Tiotropium
24.14Single7F1TMIP-1a7F1T-CCR5-MIP-1a
24.14Single7R0CAVP7R0C-V2-AVP-Arrestin2
24.14Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
24.14Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
24.14Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
24.14Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
24.14Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
24.14Consensus5ht1_offOrthosteric Ligand5ht1b_off
24.14Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
24.14Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
24.14Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
24.14Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
24.00Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
24.00Single6TP4ACT-4622066TP4-OX1-ACT-462206
24.00Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
24.00Single7SRQLSD7SRQ-5-HT2B-LSD
24.00Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
24.00Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
24.00Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
24.00Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
24.00Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
24.00Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
24.00Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
24.00Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
24.00Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
24.00Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
24.00Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
24.00Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
24.00Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
24.00Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
24.00Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
24.00Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
23.81Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
23.68Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
23.68Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
23.68Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
23.68Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
23.68Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
23.53Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
23.53Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
23.53Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
23.40Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
23.33Single4N4WSANT-14N4W-SMO-SANT-1
23.33Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
23.33Single5CXVTiotropium5CXV-M1-Tiotropium
23.33Single6CM4Risperidone6CM4-D2-Risperidone
23.33Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
23.33Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
23.33Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
23.33Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.33Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
23.33Single8XWACXCL18XWA-CXCR2-CXCL1
23.33Single8XWMCXCL68XWM-CXCR2-CXCL6
23.33Single8XWSCXCL58XWS-CXCR2-CXCL5
23.33Single9BJKNAM9BJK-μ-Naloxone-NAM
23.33Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
23.33Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
23.08Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
23.08Single5ZKQABT-4915ZKQ-PAF-ABT-491
23.08Single6DS0Ly2660976DS0-5-HT2B-Ly266097
23.08Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
23.08Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
23.08Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
23.08Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
23.08Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
23.08Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.08Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
23.08Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
23.08Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
23.08Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
23.08Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
23.08Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
23.08Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
23.08Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
23.08Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
23.08Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
23.08Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
23.08Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.08Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
23.08Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
23.08Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
23.08Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
23.08Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
23.08Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
23.08Single9H2XA1IR19H2X-A2A-A1IR1-Na
23.08Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
23.08Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
23.08Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.08Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
23.08Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
23.08Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
23.08Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
23.08Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
23.08Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
23.08Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
23.08Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
23.08Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
23.08Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
23.08Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
23.08Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
23.08Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
22.86Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
22.86Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
22.86Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
22.58Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
22.58Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
22.58Single8XVJMacitentan8XVJ-ETA-Macitentan
22.58Single8XWFCXCL38XWF-CXCR2-CXCL3
22.58Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
22.58Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
22.22Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
22.22Single6A94Zotepine6A94-5-HT2A-Zotepine
22.22Single6AQFZM-2413856AQF-A2A-ZM-241385
22.22Single6TPKRetosiban6TPK-OT-Retosiban
22.22Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
22.22Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
22.22Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
22.22Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.22Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
22.22Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
22.22Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
22.22Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
22.22Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
22.22Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
22.22Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
22.22Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
22.22Single9ARXSerotonin9ARX-5-HT2A-Serotonin
22.22Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
22.22Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
22.22Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
22.22Consensuscalcitonin_onOrthosteric Ligandctlike_on
22.22Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
22.22Consensusvasop-oxy_offOrthosteric Ligandot_off
21.95Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
21.95Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
21.88Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.88Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
21.88Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
21.88Single9JF4PD1683689JF4-BB1-PD168368
21.88Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
21.88Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
21.74Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
21.74Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
21.74Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
21.74Single8PWNTheophylline8PWN-A2A-Theophylline
21.74Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
21.62Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
21.62Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
21.62Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
21.62Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
21.62Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
21.62Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
21.62Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
21.62Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
21.43Single4QIMANTA XV4QIM-SMO-ANTA XV
21.43Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
21.43Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
21.43Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
21.43Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
21.43Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
21.43Single6GPSMK08126GPS-CCR2-MK0812
21.43Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
21.43Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
21.43Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
21.43Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
21.43Single7YXAONO-54306087YXA-S1P5-ONO-5430608
21.43Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.43Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
21.43Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
21.43Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
21.43Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
21.43Single8X63Mepyramine8X63-H1-Mepyramine
21.43Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
21.43Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
21.43Single9AS1DMT9AS1-5-HT2A-DMT
21.43Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
21.43Single9JEAAtropine9JEA-M1-Atropine
21.43Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
21.43Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
21.43Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
21.43Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
21.43Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
21.43Consensushistamine_offOrthosteric Ligandh1_off
21.43Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
21.43Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
21.43Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
21.21Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
21.21Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
21.21Single8IEIA1LYA8IEI-GPR156-A1LYA
21.21Single8IEIA1LYA8IEI-GPR156-A1LYA
21.21Single8IEPA1LYA8IEP-GPR156-A1LYA
21.21Single8IEPA1LYA8IEP-GPR156-A1LYA
21.21Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
21.21Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
21.21Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
21.05Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
21.05Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
21.05Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
21.05Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
21.05Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
21.05Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
20.93Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
20.83Single3OE8IT1t3OE8-CXCR4-IT1t
20.83Single3RFMCaffeine3RFM-A2A-Caffeine
20.83Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
20.83Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
20.83Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
20.83Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
20.83Single9CHUNoradrenaline9CHU-β2-Noradrenaline
20.83Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
20.83Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
20.83Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
20.83Consensusp2y_offOrthosteric Ligandp2y1_off
20.83Consensussensory_onOrthosteric Ligandopsins_on
20.69Single4NTJAZD12834NTJ-P2Y12-AZD1283
20.69Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
20.69Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
20.69Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
20.69Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
20.69Single6GPXMK08126GPX-CCR2-MK0812
20.69Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
20.69Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
20.69Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
20.69Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.69Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.69Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
20.69Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
20.69Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
20.69Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
20.69Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
20.69Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
20.69Consensusep_offOrthosteric Ligandep4_off
20.69Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
20.69Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
20.69Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
20.69Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.69Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.59Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
20.51Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
20.51Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
20.51Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
20.51Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
20.51Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
20.51Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
20.45Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
20.00Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
20.00Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
20.00Single3UZAGTPL92363UZA-A2A-GTPL9236
20.00Single5V56TC1145V56-SMO-TC114
20.00Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
20.00Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
20.00Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
20.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
20.00Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
20.00Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
20.00Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
20.00Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
20.00Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
20.00Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
20.00Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
20.00Single7WC5Psilocin7WC5-5-HT2A-Psilocin
20.00Single8EA0Iperoxo8EA0-M3-Iperoxo
20.00Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
20.00Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
20.00Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
20.00Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
20.00Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
20.00Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
20.00Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
20.00Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
20.00Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
20.00Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
20.00Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
20.00Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
20.00Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
20.00Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
20.00Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
20.00Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
20.00Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
20.00Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
20.00Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
20.00Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
20.00Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
19.51Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
19.44Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
19.44Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
19.44Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
19.44Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
19.44Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
19.44Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
19.44Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
19.35Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
19.35Single4PY02MeSATP4PY0-P2Y12-2MeSATP
19.35Single5X33BIIL2605X33-BLT1-BIIL260
19.35Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
19.35Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
19.35Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
19.35Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
19.35Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
19.35Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
19.35Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.35Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single4O9RCyclopamine4O9R-SMO-Cyclopamine
19.23Single5L7IVismodegib5L7I-SMO-Vismodegib
19.23Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
19.23Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
19.23Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
19.23Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
19.23Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
19.23Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
19.23Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
19.23Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
19.23Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single9B9Y7DY9B9Y-CB1-7DY
19.23Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
19.23Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
18.92Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
18.75Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
18.75Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
18.75Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
18.75Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
18.60Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
18.60Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
18.52Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
18.52Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
18.52Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
18.52Single4QINSAG1.54QIN-SMO-SAG1.5
18.52Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
18.52Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
18.52Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
18.52Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
18.52Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
18.52Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
18.52Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
18.52Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.52Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
18.52Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
18.52Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.52Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
18.52Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
18.52Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
18.52Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
18.52Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
18.52Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
18.52Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
18.42Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
18.18Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
18.18Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
18.18Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
18.18Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
17.95Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
17.95Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
17.95Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
17.86Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
17.86Single3RZECidoxepin3RZE-H1-Cidoxepin
17.86Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
17.86Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
17.86Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
17.86Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
17.86Single6ZINSR486926ZIN-NTS1-SR48692
17.86Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
17.86Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
17.86Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
17.86Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
17.86Single8K2WAMG4878K2W-CXCR3-AMG487
17.86Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
17.86Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.86Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
17.86Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
17.86Single9BA0A1AKN9BA0-CB1-A1AKN
17.86Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
17.86Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
17.86Consensusopsins_offOrthosteric Ligandrhodopsin_off
17.86Consensussensory_offOrthosteric Ligandopsins_off
17.65Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.65Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
17.65Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
17.50Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
17.50Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
17.39Single5MZPCaffeine5MZP-A2A-Caffeine-Na
17.39Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
17.39Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
17.24Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
17.24Single4DAJTiotropium4DAJ-M3-Tiotropium
17.24Single4MQSIperoxo4MQS-M2-Iperoxo
17.24Single4U14Tiotropium4U14-M3-Tiotropium
17.24Single5DSGTiotropium5DSG-M4-Tiotropium
17.24Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
17.24Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
17.24Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.24Single7F83PF-051904577F83-Ghrelin-PF-05190457
17.24Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
17.24Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
17.24Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
17.24Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
17.24Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
17.24Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
17.14Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
16.67Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
16.67Single4JKVTaladegib4JKV-SMO-Taladegib
16.67Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
16.67Single5CGCHTL142425CGC-mGlu5-HTL14242
16.67Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
16.67Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
16.67Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
16.67Single6Z4SSR486926Z4S-NTS1-SR48692
16.67Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
16.67Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
16.67Single7WC4Serotonin7WC4-5-HT2A-Serotonin
16.67Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
16.67Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
16.67Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
16.67Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
16.67Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
16.67Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
16.67Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
16.67Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
16.67Single9B9ZA1AKO9B9Z-CB1-A1AKO
16.13Single5V57TC1145V57-SMO-TC114
16.13Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
16.13Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
16.13Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
16.13Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
16.13Single9AS9RS130-1809AS9-5-HT2A-RS130-180
16.13Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.13Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
16.00Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
16.00Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
16.00Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
15.91Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
15.79Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
15.79Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
15.62Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
15.62Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
15.62Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
15.62Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.62Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
15.62Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
15.62Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
15.62Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
15.38Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
15.38Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
15.38Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
15.38Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
15.38Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
15.38Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
15.38Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
15.38Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
15.38Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
15.38Consensusgi_sensoryOrthosteric Ligandgi_opsins
15.38Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
15.38Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
15.15Single5CGDHTL142425CGD-mGlu5-HTL14242
15.15Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
15.15Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
15.15Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.15Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
15.15Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
15.15Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
15.15Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
14.81Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
14.81Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
14.81Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
14.81Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
14.81Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
14.81Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
14.81Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
14.81Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
14.81Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
14.81Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.81Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.81Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
14.81Single9AS7Psilocin9AS7-5-HT2A-Psilocin
14.81Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
14.81Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
14.71Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
14.71Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
14.63Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
14.29Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
14.29Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
14.29Single5U09Taranabant5U09-CB1-Taranabant
14.29Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
14.29Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
14.29Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
14.29Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
14.29Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
14.29Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
14.29Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
14.29Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
14.29Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
14.29Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
14.29Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
14.29Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
13.79Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
13.79Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
13.79Single7VODCariprazine7VOD-5-HT2A-Cariprazine
13.79Single7VV6C48/807VV6-MRGPRX2-C48/80
13.33Single6IIVDaltroban6IIV-TXA2-Daltroban
13.33Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
13.33Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
13.33Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
13.33Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
13.33Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
13.16Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
12.90Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
12.90Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
12.90Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
12.90Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
12.90Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
12.90Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
12.90Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
12.90Single9HC04YI9HC0-mGlu5-4YI
12.90Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
12.90Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
12.50Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
12.50Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
12.50Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
12.50Single7P2L4YI7P2L-mGlu5-4YI
12.50Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
12.50Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
12.12Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
12.12Single6IIURamatroban6IIU-TXA2-Ramatroban
12.12Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
12.00Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
11.76Single9JH5C16:0 Ceramide9JH5-CysLT2-C16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
11.54Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
11.54Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
11.54Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
11.11Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
11.11Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
11.11Single8JPSCCL78JPS-ACKR1-CCL7
11.11Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
10.71Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
10.71Single6LI0C176LI0-GPR52-C17
10.71Single7UL2SR486927UL2-NTS1-SR48692-Na
10.71Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
10.71Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
10.71Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
10.71Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
10.71Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
10.71Consensusneurotensin_offOrthosteric Ligandnts1_off
10.71Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
10.34Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
10.34Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
10.34Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
10.00Single6FFIMMPEP6FFI-mGlu5-MMPEP
10.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
10.00Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
10.00Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Single6FFHFenobam6FFH-mGlu5-Fenobam
9.38Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
9.38Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
9.38Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
9.38Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
9.09Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
9.09Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
8.57Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
8.33Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
8.33Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
8.11Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
7.69Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
7.69Single8HS2Fab0468HS2-GPR20-Fab046
7.69Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
7.41Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
7.14Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
7.14Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
6.90Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.90Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
6.90Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
6.06Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
6.06Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
5.88Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
4.35Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
4.35Single6D35Cholesterol6D35-SMO-Cholesterol
4.35Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.35Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.35Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
4.35Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
4.35Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042
4.35Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
4.35Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
4.35Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-BHFF
4.35Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
4.35Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626
4.35Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.35Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.35Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.35Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.35Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
4.35Single7DTTCa7DTT-CaS-Ca-Ca
4.35Single7DTTCa7DTT-CaS-Ca-Ca
4.35Single7DTUTryptophan7DTU-CaS-Tryptophan
4.35Single7DTUTryptophan7DTU-CaS-Tryptophan
4.35Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.35Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.35Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.35Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.35Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.35Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.35Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.35Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.35Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.35Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.35Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.35Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.35Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
4.35Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.35Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.35Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.35Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.35Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.35Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.35Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
4.35Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
4.35Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.35Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.35Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.35Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.35Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.35Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.35Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.35Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.35Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.35Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.35Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.35Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.35Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.35Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.35Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.35Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.35Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.35Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.35Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.35Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.35Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.35Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.35Single7T9NM22 Fab7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
4.35Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.35Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.35Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.35Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.35Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.35Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.35Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
4.35Single7XW7K1-707XW7-TSH-K1-70
4.35Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.35Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.35Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.35Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.35Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.35Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.35Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.35Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.35Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.35Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.35Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.35Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.35Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
4.35Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.35Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.35Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.35Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.35Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
4.35Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
4.35Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.35Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.35Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
4.35Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
4.35Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
4.35Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
4.35Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.35Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.35Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
4.35Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.35Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.35Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.35Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.35Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.35Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.35Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.35Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.35Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.35Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.35Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.35Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.35Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.35Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.35Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.35Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.35Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
4.35Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
4.35Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
4.35Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
4.35Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
4.35Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
4.35Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.35Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.35Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.35Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.35Single8WVXNorrin8WVX-LGR4-Norrin
4.35Single8WVYNorrin8WVY-LGR4-Norrin
4.35Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.35Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.35Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.35Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.35Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.35Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.35Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.35Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.35Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.35Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.35Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.35Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.35Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.35Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.35Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
4.35Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.35Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.35Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.35Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.35Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.35Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.35Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.35Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.35Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.35Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.35Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.35Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.35Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.35Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.35Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.35Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.35Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.35Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.35Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.35Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.35Single9KHHNorrin9KHH-LGR4-Norrin
4.35Single9S37NB219S37-LGR4-NB21
4.35Single9UTBSucralose9UTB-TAS1R2; TAS1R3-Sucralose
4.17Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.17Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.17Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.17Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.17Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.17Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.17Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.17Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.17Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.17Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.17Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.17Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.17Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.17Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.17Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
4.17Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
4.00Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
4.00Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
4.00Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
3.85Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
3.85Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
3.85Single7UTZTR14027UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
3.85Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
3.85Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
3.85Single8JGBConorfamide-Tx28JGB-MRGPRX1-Conorfamide-Tx2-Gi1/β1/γ2
3.70Single5L7DCholesterol5L7D-SMO-Cholesterol
3.70Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
3.70Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
3.57Single7Y14Beta-Alanine7Y14-MRGPRD-β-Alanine
3.57Single9IVMLSN33188399IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
3.45Single7Y12Beta-Alanine7Y12-MRGPRD-β-Alanine-Gi1/β1/γ2
3.45Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
3.33Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
3.33Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
3.33Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
3.33Single8YKDDehydroepiandrosterone8YKD-ADGRG2-Dehydroepiandrosterone-chim(NtGi1-Gs)/β1/γ2
3.23Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
3.23Single8G94CD698G94-S1P1-CD69-Gi1/β1/γ2
3.12Single8IYXYL-3658IYX-GPR34-YL-365
3.03Single8Y73MPAM-158Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
2.56Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.56Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.44Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.44Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.38Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.22Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
gq_cck 8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
gq_kisspeptin 8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
gq_bradykinin 7F6H-BK2-Bradykinin-Gq/β1/γ2
7F6I-BK2-Kallidin-Gq/β1/γ2
gq_bombesin 7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
gq_angiotensin 7F6G-AT1-SAR1-AngII-Gq/β1/γ2
Net Summary
Imin 2.943
Number of Linked Nodes 1057
Number of Links 1236
Number of Hubs 182
Number of Links mediated by Hubs 731
Number of Communities 24
Number of Nodes involved in Communities 218
Number of Links involved in Communities 322
Path Summary
Number Of Nodes in MetaPath 99
Number Of Links MetaPath 98
Number of Shortest Paths 1425171
Length Of Smallest Path 3
Average Path Length 36.5196
Length of Longest Path 89
Minimum Path Strength 0.324
Average Path Strength 5.32871
Maximum Path Strength 24.227
Minimum Path Correlation 0.7
Average Path Correlation 0.963101
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 1.14943
Average % Of Corr. Nodes 31.1051
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 54.1615
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
gq_class-agq_peptide
gq_amine
gq_nucleotide



You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

Download gq_peptide.zip



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