Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1Lig 15.57082410
2G.HN.36 6.6375424
3G.hns1.01 7.9045124
4G.S3.03 4.71668
5G.S3.04 8.964137
6G.S3.06 8.0645137
7G.H2.01 9.175439
8G.H2.05 5.815438
9G.H2.06 7.54539
10G.H2.07 7.794149
11G.H3.09 5.247147109
12G.H3.13 8.27506
13G.H3.17 9.88435
14G.H3.18 5.99409
15G.S5.03 4.7154159
16G.hgh4.05 7.11406
17G.hgh4.08 9.385406
18G.H4.04 2.785404
19G.H4.10 7.8875407
20G.H4.14 7.135405
21G.H4.15 6.1875408
22G.h4s6.02 5.5407
23G.S6.01 4.5054105
24G.S6.02 8.0485158
25G.S6.05 5.63405
26G.H5.05 4.775465
27G.H5.08 6.196568
28G.H5.20 3.84408
29b.1x14 4.044547
30b.1x18 6.476546
31b.h2x1 4.755405
32b.lhb1x3 3.8175492
33b.lhb1x6 3.625693
34b.b1x6 9.6075429
35b.l1x3 8.52167629
36b.l1x6 12.445439
37b.b2x1 6.6125438
38b.b2x3 4.994526
39b.b2x5 7.66527
40b.l2x5 8.108525
41b.b3x2 5.8675425
42b.b3x3 4.485198
43b.l3x2 7.0125129
44b.b4x2 4.366508
45b.b4x3 3.9454197
46b.b4x5 4.6175407
47b.b4x6 8.8275829
48b.b4x7 8.66428
49b.l4x2 7.51424
50b.l4x3 6.705426
51b.b5x2 8.0175427
52b.b5x3 6.78629
53b.l5x1 4.2925408
54b.l5x5 9.208509
55b.b6x1 4.915439
56b.b6x5 4.34506
57b.l7x2 4.08439
58b.l7x5 4.525406
59b.b8x3 3.3475406
60b.b8x4 5.522506
61b.l9x3 8.316589
62b.l9x6 5.13667638
63b.b10x2 4.04406
64b.b10x5 4.19167609
65b.b11x4 5.4425489
66b.b11x5 3.64406
67b.b11x6 8.12489
68b.l11x2 7.68589
69b.b12x6 8.05167688
70b.b13x7 7.628577
71b.l13x3 7.52167679
72b.l13x6 7.3075439
73b.l13x7 4.685479
74b.b15x1 7.096579
75b.b15x3 4.446579
76b.l15x1 4.644537
77b.l15x2 7.455479
78b.b16x4 8.765406
79b.b16x6 8.28678
80b.b17x5 6.698547
81b.b17x7 7.8325448
82b.l17x3 8.64167649
83b.l17x6 6.9675439
84b.b18x3 4.325448
85b.l18x1 8.126116
86b.l18x3 9.01754115
87b.b19x2 6.69167646
88b.l19x2 9.1975409
89b.b20x2 8.4325446
90b.b20x4 12.552548
91b.b20x6 6.88143746
92b.b21x5 4.0425404
93b.b21x6 7.17441
94b.b21x7 5.03167605
95b.l21x5 3.92434
96b.l21x7 4.61435
97b.l22x5 6.628599
98b.b23x6 6.22286737
99b.l23x1 8.19436
100b.b24x3 4.07555
101b.b24x4 7.0775436
102b.b24x5 3.798505
103b.l24x3 3.1875405
104b.b25x7 5.91457
105b.l25x3 8.126559
106b.l25x6 11.844538
107b.l25x7 4.67457
108b.b26x3 3.955656
109b.b27x1 3.81456
110b.b27x3 6.5075458
111b.l27x1 11.1917639
112b.b28x3 4.944527
113b.b28x4 6.09456
114b.b28x6 6.555659
115g.h1x6 2.276549
116g.l1x4 5.374548
117g.ctx3 6.438509
118g.ctx6 3.44496
119g.ctx15 6.825429
120g.ctx16 6.74125828
121NT 244.647615
1221x35 6.73516
1231x36 6.2275416
1241x40 3.6825416
1251x50 4.075409
1262x39 7.0175409
1272x46 6.695409
1282x47 5.03508
1292x50 9.97408
1302x60 7.725407
131E1 11.1862814
1323x30 3.3725406
1333x32 6.162516
1343x36 5.032516
1353x40 6.455418
1363x42 6.53167609
1373x44 4.53508
1383x46 9.375409
1393x49 9.86568
140I2 10.24381366
1414x50 5.844209
1424x64 10.42407
143E2 12.3283615
1445x57 10.1125408
1455x58 3.53254219
1465x68 4.234569
1476x44 6.314219
1486x46 5.18254217
1496x47 6.304518
1506x48 7.022518
1517x33 7.0975416
1527x38 12.4225417
1537x41 5.545417
1547x42 9.252509
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1G.h2s4.01 b.l5x5 86.677313.03NoYes099
2G.H2.07 G.h2s4.01 87.12973.01YesNo099
3G.H2.07 G.S3.08 99.6058.58YesNo099
4G.S3.07 G.S3.08 99.69331.46NoNo099
5G.S1.06 G.S3.07 99.78154.07NoNo089
6G.S1.06 G.S3.05 49.9358.48NoNo088
7G.S1.04 G.S3.05 49.99742.83NoNo078
8G.S1.04 G.S3.03 1003.65NoYes078
9G.S1.02 G.S3.03 33.27363.39NoYes668
10G.S1.02 I2 33.24093.39NoYes666
113x49 I2 91.692316.91YesYes686
122x42 3x49 84.07264.69NoYes098
132x42 3x42 47.56215.69NoYes099
142x46 3x42 33.16447.97YesYes099
152x46 2x50 54.99377.31YesYes098
162x50 3x39 25.981221.75YesNo088
172x53 3x39 38.435512.26NoNo088
182x53 3x36 33.24495.61NoYes086
193x36 Lig 28.05328.08YesYes160
20G.S1.06 G.S4.03 49.9352.85NoNo087
21G.S1.04 G.S4.03 49.99742.85NoNo077
22G.S3.01 G.S3.03 33.27365.24NoYes658
23G.S3.01 I2 33.240911.8NoYes656
24G.H5.08 G.S3.03 33.47984.29YesYes688
25G.H5.08 I2 33.316310.72YesYes686
262x42 3x46 36.38713.98NoYes099
272x46 3x46 33.19916.63YesYes099
283x42 4x50 13.70937.5YesYes099
292x49 4x50 13.08383.71NoYes2089
302x49 3x39 12.9375.96NoNo088
312x50 7x45 28.41228.2YesNo089
326x48 7x45 25.894310.54YesNo189
336x48 7x41 24.26217.46YesYes187
347x41 Lig 18.9444.56YesYes170
35b.l3x1 b.l5x5 52.04636.57NoYes099
36b.l1x6 b.l3x1 26.043810.85YesNo099
37b.l1x6 b.l27x1 25.692820.89YesYes399
38b.b2x1 b.l3x1 25.91996.76YesNo089
39b.b2x1 b.l27x1 26.33755.79YesYes389
40b.l5x5 b.l7x2 26.43045.69YesYes099
41b.l7x2 b.l9x6 26.06443.52YesYes398
42G.H2.04 G.H2.07 17.32249NoYes1499
43G.H2.04 G.H3.08 17.1954.86NoNo098
44G.H3.08 G.S4.04 17.07217.31NoNo089
45G.H3.09 G.S4.04 12.60594.29YesNo099
46G.H3.06 G.H4.14 10.23523.98NoYes065
47b.l25x6 b.l27x1 44.346422.99YesYes389
48b.l23x1 b.l25x6 17.402610.72YesYes368
49b.l11x1 b.l9x6 24.89938.69NoYes098
50b.b11x6 b.l11x1 24.77723.71YesNo099
51b.b11x6 b.l9x3 23.778616.74YesYes899
52b.b11x4 b.l9x3 22.57395.48YesYes899
53b.b10x3 b.b11x4 21.32173.38NoYes089
54b.b10x3 b.b6x2 18.85993.38NoNo088
55b.b10x2 b.b6x2 18.74473.38YesNo068
56b.l21x7 b.l23x1 16.91523.11YesYes356
57b.b23x6 b.l21x7 15.43994.03YesYes375
58b.b23x6 b.b24x6 12.04189.65YesNo078
59b.b21x7 b.b24x6 11.5910.61YesNo058
60b.b22x1 b.l25x6 25.842410.35NoYes088
61b.b22x1 b.b22x2 10.56163.2NoNo088
62b.b22x2 b.b26x3 10.31586.01NoYes086
63b.b23x1 b.b24x5 13.8894.47NoYes055
64b.b22x1 b.l25x7 15.03443.17NoYes087
652x46 2x47 11.51984.87YesYes098
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
5x41Lig4.160NoYes5010
5x42Lig6.431NoYes6010
6x53Lig8.931NoYes5010
5x48Lig5.070NoYes4010
7x37Lig6.351NoYes8010
5x44Lig21.391NoYes6010
7x38Lig12.061YesYes7010
7x41Lig4.561YesYes7010
2x61Lig7.21NoYes7010
3x36Lig8.081YesYes6010
3x32Lig4.781YesYes6010
E2Lig7.481YesYes5010
1x36Lig7.311YesYes6010
E1Lig8.081YesYes4010
E2x52Lig3.381NoYes6010
1x28Lig2.821NoYes3010
1x32Lig3.160NoYes5010
1x33Lig4.361NoYes3010
LigNT116.681YesYes0501
1x29Lig9.641NoYes1010
NTNT661.161YesYes5511
1x25NT4.360NoYes1521
1x24NT10.551NoYes2521
1x28NT13.971NoYes3511
1x291x332.981NoNo1311
1x357x344.071YesNo6622
1x357x38181YesYes6721
1x361x407.541YesYes6612
1x362x614.871YesNo6711
1x362x625.191YesNo6312
1x402x623.041YesNo6322
2x532x572.920NoNo8722
2x533x365.610NoYes8621
2x563x324.150NoYes6621
2x573x329.580NoYes7621
2x603x328.360YesYes7621
E1E122.381YesYes4411
E1E2x508.711YesNo4912
3x26E16.991NoYes8421
E1E213.621YesYes4511
3x24E13.560NoYes4421
3x25E13.771NoYes9421
3x25E2x507.281NoNo9922
3x323x363.941YesYes6611
3x363x403.591YesYes6812
3x365x443.941YesNo6611
3x406x484.131YesYes8822
3x407x413.591YesYes8721
4x68E219.371NoYes6521
4x685x389.991NoNo6522
E2E214.351YesYes5511
E2x50E2x523.271NoNo9621
5x38E24.81NoYes5521
5x395x428.710NoNo4621
6x487x417.461YesYes8721
6x537x313.271NoNo5412
6x537x3310.611NoYes5612
7x317x335.611NoYes4622
7x337x3710.781YesNo6821
7x347x3810.081NoYes6721
7x387x429.551YesYes7912
7x417x426.571YesYes7912
1x26Lig2.770NoYes2010
E3Lig1.190NoYes4010

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
95.45Consensuscalcitonin_onOrthosteric Ligandctlike_on
75.86Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
68.00Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
61.54Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
61.29Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
60.71Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
60.00Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
59.26Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
58.62Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
57.69Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
57.14Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
57.14Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
55.17Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
55.17Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
54.84Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
53.33Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
53.33Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
53.33Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
51.72Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
51.72Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
51.61Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
51.52Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
50.00Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
50.00Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
50.00Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
50.00Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
48.39Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
48.39Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
48.28Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
48.15Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
47.22Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
46.88Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
46.67Single6FJ3PTH6FJ3-PTH1-PTH
46.67Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
46.15Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
45.95Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
45.16Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
45.16Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
45.16Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
44.83Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
44.83Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
44.83Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
44.74Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
43.33Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
42.86Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
42.42Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
41.94Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
41.38Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
41.38Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
41.18Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
41.18Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
40.62Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
40.00Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
40.00Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
40.00Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
40.00Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
40.00Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
40.00Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
40.00Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
40.00Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
39.47Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
39.39Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
39.39Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
39.39Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
39.39Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
39.39Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
39.39Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
39.39Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
39.39Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
39.29Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
38.89Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
38.71Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
38.71Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
38.71Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
38.71Consensuspac_onOrthosteric Ligandpac1_on
38.71Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
38.24Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
37.93Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
37.84Consensuspth_onOrthosteric Ligandpth1_on pth2_on
37.50Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
37.50Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
37.50Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
37.50Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
37.50Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
37.50Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
37.50Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
37.14Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
37.04Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
36.67Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
36.36Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
36.36Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
36.36Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
36.36Consensusglp_onOrthosteric Ligandglp1_on glp2_on
36.36Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
36.11Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
36.11Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
36.11Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
35.29Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
35.29Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
35.29Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
35.29Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
35.29Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
35.29Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
35.29Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
35.29Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
35.29Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
35.29Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
35.14Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
35.14Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
35.14Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
34.48Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
34.48Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
34.38Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
34.38Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
34.29Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
34.29Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
34.21Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
33.33Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
33.33Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
33.33Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
33.33Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
33.33Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
33.33Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
33.33Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
33.33Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
33.33Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
33.33Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
33.33Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
32.43Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
32.43Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
32.43Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
32.43Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
32.35Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
32.35Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
32.35Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
32.35Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
32.26Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
32.14Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
31.58Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
31.58Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
31.25Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
31.25Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
30.30Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
30.30Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
29.73Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
29.41Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
29.41Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
29.27Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
28.95Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
28.57Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
28.57Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
28.57Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
28.57Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
28.21Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
28.12Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
27.78Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
27.59Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
27.03Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
27.03Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
25.81Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
25.71Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
25.64Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
25.00Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
25.00Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
25.00Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
24.14Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
24.00Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
23.81Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
23.53Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.53Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
23.33Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
23.08Single2YDOAdenosine2YDO-A2A-Adenosine
23.08Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
22.86Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
22.86Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
22.58Single4UG2CGS216804UG2-A2A-CGS21680
22.58Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
22.58Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
22.22Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
22.22Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
22.22Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
22.22Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
22.22Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
22.22Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
22.22Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
22.22Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
22.22Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
22.22Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
22.22Consensushca_on_gpOrthosteric Ligandhca2_on_gp
22.22Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
21.88Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
21.62Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
21.62Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
21.62Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
21.62Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
21.62Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
21.62Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
21.43Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
21.43Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
21.43Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
21.43Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
21.43Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
21.43Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
21.43Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
21.43Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
21.43Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
21.21Single3QAKUK-4320973QAK-A2A-UK-432097
21.21Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
21.21Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
21.21Single7XNACYN1548067XNA-SST2-CYN154806
21.21Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
21.21Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
21.21Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
21.21Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
21.21Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
21.21Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
21.05Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
20.83Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
20.69Single2YDVNECA2YDV-A2A-NECA
20.69Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
20.69Single4UHRCGS216804UHR-A2A-CGS21680
20.69Single5G53NECA5G53-A2A-NECA-Gs
20.69Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
20.69Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
20.69Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
20.69Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
20.69Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
20.69Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
20.59Single5WF5UK-4320975WF5-A2A-UK-432097
20.59Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
20.59Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
20.59Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
20.59Consensusangiotensin_onOrthosteric Ligandat1_on
20.59Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
20.59Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
20.59Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
20.59Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
20.59Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
20.59Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
20.51Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
20.00Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
20.00Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
20.00Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
20.00Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
20.00Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
20.00Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
20.00Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
20.00Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
20.00Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
20.00Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
20.00Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
20.00Single8K5BNiacin8K5B-HCA2-Niacin
20.00Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
20.00Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
20.00Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
20.00Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
20.00Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
20.00Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
20.00Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
20.00Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
20.00Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
20.00Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
20.00Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
20.00Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
20.00Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
20.00Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
20.00Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
20.00Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
20.00Consensusvasop-oxy_onOrthosteric Ligandv2_on
20.00Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
19.44Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
19.44Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
19.44Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
19.44Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
19.44Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
19.44Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
19.44Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
19.44Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
19.44Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
19.44Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
19.44Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
19.44Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
19.35Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
19.35Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
19.35Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
19.35Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
19.35Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
19.35Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
19.35Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
19.35Consensuscck_onOrthosteric Ligandccka_on cckb_on
19.35Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
19.35Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
19.23Single5U09Taranabant5U09-CB1-Taranabant
19.23Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
19.23Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
19.23Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
19.23Single8IWESpermidine8IWE-TA9-Spermidine
19.23Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
19.23Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
19.23Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
18.92Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
18.92Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
18.92Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
18.92Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
18.92Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
18.75Single3NY9ICI118-5513NY9-β2-ICI118-551
18.75Single5WF6UK-4320975WF6-A2A-UK-432097
18.75Single5ZTYAM102575ZTY-CB2-AM10257
18.75Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
18.75Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
18.75Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
18.75Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
18.75Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
18.75Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
18.75Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
18.75Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
18.75Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
18.75Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
18.52Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
18.52Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
18.52Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
18.52Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
18.52Single8K5CAcipimox8K5C-HCA2-Acipimox
18.52Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
18.52Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
18.52Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
18.52Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
18.52Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
18.52Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
18.52Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
18.52Consensushca_onOrthosteric Ligandhca2_on
18.42Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
18.42Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
18.42Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
18.42Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
18.42Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
18.42Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
18.18Single4XT1Fractalkine4XT1-US28-Fractalkine
18.18Single7QA8Peptide7QA8-STE2-Peptide
18.18Single7QA8Peptide7QA8-STE2-Peptide
18.18Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
18.18Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
18.18Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
18.18Single8WDTphotoNECA8WDT-A2A-photoNECA
18.18Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
18.18Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
18.18Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
18.18Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
18.18Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
18.18Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
18.18Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
18.18Consensussomatostatin_offOrthosteric Ligandsst2_off
18.18Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.95Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
17.95Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
17.95Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
17.95Consensusbradykinin_onOrthosteric Ligandbk2_on
17.95Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
17.95Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
17.86Single4DAJTiotropium4DAJ-M3-Tiotropium
17.86Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
17.86Single5TGZAM65385TGZ-CB1-AM6538
17.86Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
17.86Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
17.86Single8K5DGSK2560738K5D-HCA2-GSK256073
17.86Single8T1WCVN4248T1W-GPR6-CVN424
17.86Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
17.86Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
17.86Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
17.86Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
17.86Single9AS1DMT9AS1-5-HT2A-DMT
17.86Single9CHXS-Carazolol9CHX-β2-S-Carazolol
17.86Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
17.86Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
17.86Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
17.86Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
17.65Single6HLOAprepitant6HLO-NK1-Aprepitant
17.65Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
17.65Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
17.65Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
17.65Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
17.65Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
17.65Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
17.50Single5GLHEndothelin-15GLH-ETB-Endothelin-1
17.50Single6IGKEndothelin-36IGK-ETB-Endothelin-3
17.50Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
17.50Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
17.50Consensusbombesin_onOrthosteric Ligandbb2_on
17.50Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
17.50Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
17.50Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
17.50Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
17.50Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
17.24Single5JQHS-Carazolol5JQH-β2-S-Carazolol
17.24Single5N2RPSB-365N2R-A2A-PSB-36-Na
17.24Single5N2SPSB365N2S-A1-PSB36
17.24Single5TVNLSD5TVN-5-HT2B-LSD
17.24Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
17.24Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
17.24Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
17.24Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
17.24Single6PS6Timolol6PS6-β2-Timolol
17.24Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
17.24Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
17.24Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
17.24Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
17.24Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
17.24Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
17.24Single8TF5Oleic acid8TF5-GPR6-Oleic acid
17.24Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
17.24Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
17.24Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
17.24Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
17.24Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
17.24Single9B9ZA1AKO9B9Z-CB1-A1AKO
17.24Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
17.24Consensusadenosine_offOrthosteric Liganda1_off a2_off
17.24Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
17.24Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
17.24Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
17.24Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
17.24Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
17.24Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
17.24Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.24Consensustrace-amine_onOrthosteric Ligandta1_on
17.14Single3OE0CVX153OE0-CXCR4-CVX15
17.14Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
17.14Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
17.14Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.14Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
17.14Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.14Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.14Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
17.14Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
17.14Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
17.14Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
17.14Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
16.67Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
16.67Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
16.67Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
16.67Single5XR8AM8415XR8-CB1-AM841
16.67Single5XRAAM115425XRA-CB1-AM11542
16.67Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
16.67Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
16.67Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
16.67Single6WGTLSD6WGT-5-HT2A-LSD
16.67Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
16.67Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
16.67Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
16.67Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
16.67Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
16.67Single7PX4PSB-21137PX4-A2A-PSB-2113
16.67Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
16.67Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
16.67Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
16.67Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
16.67Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
16.67Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
16.67Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
16.67Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
16.67Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
16.67Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
16.67Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
16.67Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
16.67Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
16.67Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
16.67Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
16.67Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
16.67Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
16.67Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
16.67Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
16.67Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
16.67Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
16.67Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
16.67Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
16.67Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
16.67Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
16.67Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
16.67Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
16.67Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
16.67Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
16.67Consensusrelaxin_onOrthosteric Ligandrxfp4_on
16.67Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
16.67Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
16.28Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
16.22Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
16.22Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
16.22Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
16.22Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
16.22Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
16.22Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
16.22Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
16.22Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
16.22Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
16.22Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
16.22Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
16.22Single8ZRTET-18ZRT-ETB-ET-1
16.22Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
16.22Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
16.22Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
16.13Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
16.13Single4XEENeurotensin4XEE-NTS1-Neurotensin
16.13Single4XESNeurotensin4XES-NTS1-Neurotensin
16.13Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
16.13Single5CXVTiotropium5CXV-M1-Tiotropium
16.13Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
16.13Single6OS2TRV0266OS2-AT1-TRV026
16.13Single6YVRNTS8-136YVR-NTS1-NTS8-13
16.13Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
16.13Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
16.13Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
16.13Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
16.13Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
16.13Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
16.13Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
16.13Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
16.13Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
16.13Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
16.13Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
16.13Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
16.13Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
16.13Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
16.13Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
16.13Single9DGIZ85267113509DGI-CB1-Z8526711350
16.13Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
16.13Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
16.13Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
16.13Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
16.13Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
16.13Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
16.13Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
16.13Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
16.13Consensuslpa_offOrthosteric Ligandlpa1_off
16.13Consensuslpl_offOrthosteric Ligands1p_off lpa_off
16.13Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
16.13Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
16.13Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
16.13Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
16.13Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
16.00Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.00Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.00Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
16.00Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
16.00Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
16.00Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
16.00Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
16.00Single9LRCHistamine9LRC-H4-Histamine
16.00Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
16.00Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
16.00Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
15.79Single4XT3Fractalkine4XT3-US28-Fractalkine
15.79Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
15.79Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
15.79Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
15.79Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
15.79Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
15.79Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
15.62Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
15.62Single4BUONeurotensin4BUO-NTS1-Neurotensin
15.62Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
15.62Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
15.62Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
15.62Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
15.62Single7EZCUKA7EZC-A2A-UKA
15.62Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
15.62Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
15.62Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
15.62Single7UM4AS26747237UM4-5-HT5A-AS2674723
15.62Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
15.62Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
15.62Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
15.62Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
15.62Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
15.62Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
15.62Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
15.62Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
15.62Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
15.62Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
15.62Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
15.62Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single8XVUCXCL28XVU-CXCR2-CXCL2
15.62Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
15.62Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
15.62Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
15.62Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
15.62Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
15.62Consensuschemerin_onOrthosteric Ligandcml1_on
15.62Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
15.62Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
15.62Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
15.62Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
15.56Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
15.56Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
15.38Single3OE9IT1t3OE9-CXCR4-IT1t
15.38Single4O9RCyclopamine4O9R-SMO-Cyclopamine
15.38Single6LI0C176LI0-GPR52-C17
15.38Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
15.38Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
15.38Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
15.38Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
15.38Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
15.38Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
15.38Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
15.38Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
15.38Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
15.38Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
15.38Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
15.38Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
15.38Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
15.38Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
15.38Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
15.38Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
15.38Single9B9Y7DY9B9Y-CB1-7DY
15.38Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
15.38Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
15.38Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
15.15Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
15.15Single7SK9CCX6627SK9-ACKR3-CCX662
15.15Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
15.15Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
15.15Single7XN9L-054,5227XN9-SST2-L-054,522
15.15Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
15.15Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
15.15Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
15.15Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
15.15Single8QJ2pN1628QJ2-MC4-pN162-Gs
15.15Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
15.15Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
15.15Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
15.15Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
15.15Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
15.00Single6IGLIRL16206IGL-ETB-IRL1620
15.00Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
15.00Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
15.00Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
15.00Consensusendothelin_onOrthosteric Ligandetb_on eta_on
15.00Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
14.81Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
14.81Single3ODUIT1t3ODU-CXCR4-IT1t
14.81Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
14.81Single4BWBNeurotensin4BWB-NTS1-Neurotensin
14.81Single4QINSAG1.54QIN-SMO-SAG1.5
14.81Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
14.81Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
14.81Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
14.81Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
14.81Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
14.81Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
14.81Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
14.81Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
14.81Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
14.81Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
14.81Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
14.81Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
14.81Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
14.81Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
14.81Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
14.81Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
14.81Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
14.81Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
14.81Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
14.81Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
14.81Single8GNGIstradefylline8GNG-A2A-Istradefylline
14.81Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
14.81Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
14.81Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
14.81Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
14.81Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
14.81Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
14.81Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
14.81Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
14.81Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
14.81Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
14.81Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
14.81Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
14.81Single8Y0HVUF114188Y0H-CXCR3-VUF11418
14.81Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
14.81Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
14.81Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
14.81Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
14.81Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
14.81Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
14.81Consensusalpha2_offOrthosteric Ligandalpha2c_off
14.81Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
14.81Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
14.81Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
14.81Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
14.81Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
14.71Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
14.71Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
14.71Single7F8XNN90567F8X-CCKA-NN9056
14.71Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
14.71Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
14.71Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
14.71Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
14.71Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.71Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
14.71Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
14.71Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.71Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
14.71Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
14.71Consensuslpl_onOrthosteric Ligands1p_on lpa_on
14.71Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
14.71Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
14.29Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
14.29Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
14.29Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
14.29Single5IU7Q274563465IU7-A2A-Q27456346-Na
14.29Single5IUBQ274563445IUB-A2A-Q27456344-Na
14.29Single5JTBZM-2413855JTB-A2A-ZM-241385
14.29Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
14.29Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
14.29Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
14.29Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
14.29Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
14.29Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
14.29Single6PS0S-Carazolol6PS0-β2-S-Carazolol
14.29Single6PS4ICI118-5516PS4-β2-ICI118-551
14.29Single6PS5S-Propranolol6PS5-β2-S-Propranolol
14.29Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
14.29Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
14.29Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
14.29Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
14.29Single7AROLUF58337ARO-A2A-LUF5833-Na
14.29Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
14.29Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
14.29Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
14.29Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
14.29Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
14.29Single7F61PF-036547467F61-H3-PF-03654746
14.29Single7SK5CXCL127SK5-ACKR3-CXCL12
14.29Single7T32ZM-2413857T32-A2A-ZM-241385
14.29Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
14.29Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
14.29Single7UL3Famotidine7UL3-H2-Famotidine
14.29Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
14.29Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
14.29Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
14.29Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
14.29Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
14.29Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
14.29Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
14.29Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
14.29Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
14.29Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
14.29Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
14.29Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
14.29Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
14.29Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
14.29Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
14.29Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
14.29Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
14.29Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8IHKAcifran8IHK-HCA3-Acifran
14.29Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
14.29Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
14.29Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
14.29Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
14.29Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
14.29Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
14.29Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
14.29Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
14.29Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
14.29Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
14.29Single9AS5Mescaline9AS5-5-HT2A-Mescaline
14.29Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9BA0A1AKN9BA0-CB1-A1AKN
14.29Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
14.29Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
14.29Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
14.29Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
14.29Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
14.29Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
14.29Consensusa2_offOrthosteric Liganda2a_off
14.29Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
14.29Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
14.29Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
14.29Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
14.29Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
14.29Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
14.29Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
14.29Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
14.29Consensusgrh_offOrthosteric Ligandgnrh1_off
14.29Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
14.29Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
14.29Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
14.29Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
14.29Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
13.95Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
13.89Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
13.89Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
13.89Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
13.89Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
13.89Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
13.89Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
13.89Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
13.89Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
13.89Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
13.79Single2Y04Salbutamol2Y04-β1-Salbutamol
13.79Single3EMLZM-2413853EML-A2A-ZM-241385
13.79Single3NY8ICI118-5513NY8-β2-ICI118-551
13.79Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
13.79Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
13.79Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
13.79Single4GBRS-Carazolol4GBR-β2-S-Carazolol
13.79Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
13.79Single4MQSIperoxo4MQS-M2-Iperoxo
13.79Single4QKX35V4QKX-β2-35V
13.79Single4U14Tiotropium4U14-M3-Tiotropium
13.79Single5DSGTiotropium5DSG-M4-Tiotropium
13.79Single5IU8Q274563475IU8-A2A-Q27456347-Na
13.79Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
13.79Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
13.79Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
13.79Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
13.79Single5T04Neurotensin5T04-NTS1-Neurotensin
13.79Single5UENDU1725UEN-A1-DU172
13.79Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
13.79Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
13.79Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
13.79Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
13.79Single6D27CAY104716D27-DP2-CAY10471
13.79Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
13.79Single6H7MSalbutamol6H7M-β1-Salbutamol
13.79Single6IIVDaltroban6IIV-TXA2-Daltroban
13.79Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
13.79Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
13.79Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
13.79Single6PS1Timolol6PS1-β2-Timolol
13.79Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
13.79Single6S0LZM-2413856S0L-A2A-ZM-241385
13.79Single6TOTLemborexant6TOT-OX1-Lemborexant
13.79Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
13.79Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
13.79Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
13.79Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
13.79Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
13.79Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
13.79Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
13.79Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
13.79Single7PYRPSB-21157PYR-A2A-PSB-2115
13.79Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
13.79Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
13.79Single7UL4Alvimopan7UL4-μ-Alvimopan
13.79Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
13.79Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
13.79Single7V3ZCP559407V3Z-CB1-CP55940
13.79Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
13.79Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
13.79Single7WC7Lisuride7WC7-5-HT2A-Lisuride
13.79Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
13.79Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
13.79Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
13.79Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
13.79Single7YXAONO-54306087YXA-S1P5-ONO-5430608
13.79Single8CU6LJ-45178CU6-A2A-LJ-4517
13.79Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
13.79Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
13.79Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
13.79Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
13.79Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
13.79Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
13.79Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
13.79Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
13.79Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
13.79Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
13.79Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
13.79Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
13.79Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
13.79Single8JJOAlprenolol8JJO-β2-Alprenolol
13.79Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
13.79Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
13.79Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
13.79Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
13.79Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
13.79Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
13.79Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
13.79Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
13.79Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
13.79Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
13.79Single9JEAAtropine9JEA-M1-Atropine
13.79Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
13.79Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
13.79Consensus5ht5_onOrthosteric Ligand5ht5a_on
13.79Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
13.79Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
13.79Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
13.79Consensusa3_onOrthosteric Liganda3a_on
13.79Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
13.79Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
13.79Consensusdopamine_offOrthosteric Ligandd2_off d3_off
13.79Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
13.79Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
13.79Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
13.79Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
13.79Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
13.79Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
13.79Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
13.79Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
13.79Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
13.79Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
13.73Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
13.51Single6JODAngiotensin II6JOD-AT2-Angiotensin II
13.51Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
13.51Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
13.51Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
13.51Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
13.51Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
13.51Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
13.51Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
13.51Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
13.51Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
13.51Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
13.33Single2RH1S-Carazolol2RH1-β2-S-Carazolol
13.33Single2Y03Isoprenaline2Y03-β1-Isoprenaline
13.33Single2YCWS-Carazolol2YCW-β1-S-Carazolol
13.33Single4JKVTaladegib4JKV-SMO-Taladegib
13.33Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
13.33Single5C1MBU725C1M-μ-BU72
13.33Single5CGCHTL142425CGC-mGlu5-HTL14242
13.33Single5D6LS-Carazolol5D6L-β2-S-Carazolol
13.33Single5IUAQ274563485IUA-A2A-Q27456348-Na
13.33Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
13.33Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
13.33Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
13.33Single6D26Fevipiprant6D26-DP2-Fevipiprant
13.33Single6E67BI1671076E67-β2-BI167107-Gs(CT)
13.33Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
13.33Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
13.33Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
13.33Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
13.33Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
13.33Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
13.33Single6S0QZM-2413856S0Q-A2A-ZM-241385
13.33Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
13.33Single6TP6Filorexant6TP6-OX1-Filorexant
13.33Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
13.33Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
13.33Single7C4SS1P7C4S-S1P3-S1P
13.33Single7C61Ergotamine7C61-5-HT1B-Ergotamine
13.33Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
13.33Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
13.33Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
13.33Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
13.33Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
13.33Single7SINNPS-21437SIN-CaS-NPS-2143
13.33Single7SINNPS-21437SIN-CaS-NPS-2143
13.33Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
13.33Single7W41PD1762527W41-BB2-PD176252
13.33Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
13.33Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
13.33Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
13.33Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
13.33Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
13.33Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
13.33Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
13.33Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
13.33Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
13.33Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
13.33Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.33Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.33Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.33Single8GNEKW-63568GNE-A2A-KW-6356-Na
13.33Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
13.33Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
13.33Single8QOTNanobody-E8QOT-μ-Nanobody-E
13.33Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
13.33Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
13.33Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.33Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.33Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
13.33Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
13.33Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
13.33Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
13.33Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
13.33Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
13.33Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
13.33Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
13.33Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
13.33Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
13.33Single9EHSLUF76029EHS-A3A-LUF7602
13.33Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
13.33Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
13.33Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
13.33Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
13.33Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
13.33Consensusa3_on_gpOrthosteric Liganda3a_on_gp
13.33Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
13.33Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
13.33Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
13.33Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
13.33Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
13.33Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
13.33Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
13.33Consensusamine_offonOrthosteric Ligandamine_off amine_on
13.33Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
13.33Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
13.33Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
13.33Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
13.33Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
13.33Consensusbombesin_offOrthosteric Ligandbb2_off
13.33Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
13.33Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
13.33Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
13.33Consensusdp_offOrthosteric Liganddp2_off
13.33Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
13.33Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
13.33Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
13.33Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
13.33Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
13.33Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
13.33Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
13.16Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
13.16Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
13.16Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.16Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
13.16Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
13.16Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
12.90Single3P0GBI1671073P0G-β2-BI167107
12.90Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
12.90Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
12.90Single4BV0Neurotensin4BV0-NTS1-Neurotensin
12.90Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
12.90Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
12.90Single4U15Tiotropium4U15-M3-Tiotropium
12.90Single5D5AS-Carazolol5D5A-β2-S-Carazolol
12.90Single5D5BS-Carazolol5D5B-β2-S-Carazolol
12.90Single5V54Methiothepin5V54-5-HT1B-Methiothepin
12.90Single5V56TC1145V56-SMO-TC114
12.90Single5V57TC1145V57-SMO-TC114
12.90Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
12.90Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
12.90Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
12.90Single6H7JIsoprenaline6H7J-β1-Isoprenaline
12.90Single6J21Aprepitant6J21-NK1-Aprepitant
12.90Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
12.90Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
12.90Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
12.90Single6OL9Tiotropium6OL9-M5-Tiotropium
12.90Single7B6WCyclazosin7B6W-α1b-Cyclazosin
12.90Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
12.90Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
12.90Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
12.90Single7F1TMIP-1a7F1T-CCR5-MIP-1a
12.90Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
12.90Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
12.90Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
12.90Single7P2L4YI7P2L-mGlu5-4YI
12.90Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
12.90Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
12.90Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
12.90Single7TUYGSK682753A7TUY-GPR183-GSK682753A
12.90Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
12.90Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
12.90Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
12.90Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
12.90Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.90Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
12.90Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
12.90Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
12.90Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
12.90Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
12.90Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
12.90Single8E0GBU728E0G-μ-BU72
12.90Single8EA0Iperoxo8EA0-M3-Iperoxo
12.90Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
12.90Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
12.90Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
12.90Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
12.90Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
12.90Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
12.90Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
12.90Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
12.90Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
12.90Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
12.90Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
12.90Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
12.90Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
12.90Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
12.90Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
12.90Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
12.90Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
12.90Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
12.90Single9AS9RS130-1809AS9-5-HT2A-RS130-180
12.90Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
12.90Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
12.90Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
12.90Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
12.90Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
12.90Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
12.90Consensus5ht1_offOrthosteric Ligand5ht1b_off
12.90Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
12.90Consensusa2_onOrthosteric Liganda2b_on
12.90Consensusa2_on_gpOrthosteric Liganda2b_on_gp
12.90Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
12.90Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
12.90Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
12.90Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
12.90Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
12.90Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
12.90Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
12.90Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
12.90Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
12.90Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
12.90Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
12.90Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
12.90Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
12.90Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
12.90Consensuslpa_onOrthosteric Ligandlpa1_on
12.90Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
12.90Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
12.90Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
12.90Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Consensusneurotensin_onOrthosteric Ligandnts1_on
12.90Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
12.90Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
12.90Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
12.90Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
12.82Single7SK3CXCL127SK3-ACKR3-CXCL12
12.82Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
12.82Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
12.82Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
12.50Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
12.50Single3D4STimolol3D4S-β2-Timolol
12.50Single4AMIBucindolol4AMI-β1-Bucindolol
12.50Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
12.50Single4LDEBI1671074LDE-β2-BI167107
12.50Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
12.50Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
12.50Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
12.50Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
12.50Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
12.50Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
12.50Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
12.50Single6IIURamatroban6IIU-TXA2-Ramatroban
12.50Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
12.50Single6MXTSalmeterol6MXT-β2-Salmeterol
12.50Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
12.50Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
12.50Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
12.50Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
12.50Single7K15MKD0467K15-BLT1-MKD046-Na
12.50Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
12.50Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
12.50Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
12.50Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
12.50Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
12.50Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
12.50Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
12.50Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
12.50Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
12.50Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
12.50Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
12.50Single8HS2Fab0468HS2-GPR20-Fab046
12.50Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
12.50Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
12.50Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
12.50Single8JJ8Formoterol8JJ8-β2-Formoterol
12.50Single8JJLOlodaterol8JJL-β2-Olodaterol
12.50Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
12.50Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
12.50Single8JWY2-1188JWY-A2A-2-118
12.50Single8PWNTheophylline8PWN-A2A-Theophylline
12.50Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
12.50Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
12.50Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
12.50Single8XWMCXCL68XWM-CXCR2-CXCL6
12.50Single8XYIVUF106618XYI-CXCR3-VUF10661
12.50Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
12.50Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
12.50Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
12.50Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
12.50Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
12.50Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
12.50Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
12.50Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
12.50Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
12.50Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
12.50Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
12.50Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
12.50Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
12.50Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
12.50Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
12.50Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
12.50Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
12.50Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
12.50Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
12.50Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
12.50Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
12.50Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
12.50Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
12.50Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
12.50Consensusorexin_onOrthosteric Ligandox2_on
12.50Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
12.20Single8IY6Endothelin-18IY6-ETB-Endothelin-1
12.12Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
12.12Single5CGDHTL142425CGD-mGlu5-HTL14242
12.12Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
12.12Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
12.12Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
12.12Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
12.12Single6H7LDobutamine6H7L-β1-Dobutamine
12.12Single6IBLArformoterol6IBL-β1-Arformoterol
12.12Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
12.12Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
12.12Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
12.12Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
12.12Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
12.12Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
12.12Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
12.12Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
12.12Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
12.12Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.12Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
12.12Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
12.12Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
12.12Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
12.12Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
12.12Single8XWFCXCL38XWF-CXCR2-CXCL3
12.12Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
12.12Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
12.12Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
12.12Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.12Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
12.12Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
12.12Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
12.12Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
12.12Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
12.12Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.12Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.12Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
12.12Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
12.12Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
12.12Consensusprostanoid_offOrthosteric Ligandep_off dp_off
12.00Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
12.00Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
12.00Single8A2OTheophylline8A2O-A2A-Theophylline-Na
12.00Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.00Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
12.00Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
12.00Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
12.00Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
12.00Single9CHUNoradrenaline9CHU-β2-Noradrenaline
12.00Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
11.90Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
11.90Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
11.90Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
11.76Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
11.76Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
11.76Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
11.76Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
11.76Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
11.76Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
11.76Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
11.76Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
11.76Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
11.76Single8XQJJN2418XQJ-Apelin-JN241
11.76Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
11.76Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
11.76Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
11.76Single9JF4PD1683689JF4-BB1-PD168368
11.76Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
11.76Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
11.76Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
11.76Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
11.76Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
11.63Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
11.63Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
11.54Single3OE6IT1t3OE6-CXCR4-IT1t
11.54Single4XNWMRS25004XNW-P2Y1-MRS2500
11.54Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
11.54Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
11.54Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
11.54Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
11.54Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
11.54Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
11.54Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
11.54Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
11.54Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
11.54Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
11.54Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
11.54Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
11.54Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
11.54Consensus5ht2_onOrthosteric Ligand5ht2b_on
11.54Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
11.43Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
11.43Single4IARErgotamine4IAR-5-HT1B-Ergotamine
11.43Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
11.43Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
11.43Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
11.43Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
11.43Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
11.43Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
11.43Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
11.43Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
11.43Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
11.43Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
11.43Single8IEBA1LYA8IEB-GPR156-A1LYA
11.43Single8IEIA1LYA8IEI-GPR156-A1LYA
11.43Single8IEIA1LYA8IEI-GPR156-A1LYA
11.43Single8IEPA1LYA8IEP-GPR156-A1LYA
11.43Single8IEPA1LYA8IEP-GPR156-A1LYA
11.43Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
11.43Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
11.43Single8XWNCXCL88XWN-CXCR2-CXCL8
11.43Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
11.43Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
11.43Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
11.43Single9M4TSilodosin9M4T-Alpha1A-Silodosin
11.43Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
11.43Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
11.43Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
11.11Single5L7IVismodegib5L7I-SMO-Vismodegib
11.11Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
11.11Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
11.11Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
11.11Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
11.11Single7SRQLSD7SRQ-5-HT2B-LSD
11.11Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
11.11Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
11.11Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
11.11Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
11.11Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
11.11Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
11.11Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
11.11Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
11.11Single8IEBA1LYA8IEB-GPR156-A1LYA
11.11Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
11.11Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
11.11Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
11.11Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
11.11Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
11.11Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
11.11Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
11.11Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
11.11Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
11.11Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
11.11Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
11.11Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
11.11Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single9AS7Psilocin9AS7-5-HT2A-Psilocin
11.11Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
11.11Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.11Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
11.11Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
11.11Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
11.11Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
11.11Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
11.11Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
11.11Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
11.11Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
11.11Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
11.11Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
11.11Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
11.11Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
10.81Single6PT2KGCHM076PT2-δ-KGCHM07
10.81Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
10.81Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
10.81Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
10.81Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
10.81Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
10.81Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
10.81Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
10.81Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
10.81Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
10.81Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
10.81Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
10.71Single3PWHZM-2413853PWH-A2A-ZM-241385
10.71Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
10.71Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
10.71Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
10.71Single4S0VSuvorexant4S0V-OX2-Suvorexant
10.71Single5ZKQABT-4915ZKQ-PAF-ABT-491
10.71Single6AKXA4R6AKX-CCR5-A4R
10.71Single6AKYMaraviroc6AKY-CCR5-Maraviroc
10.71Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
10.71Single6ME2Ramelteon6ME2-MT1-Ramelteon
10.71Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
10.71Single6TODEMPA6TOD-OX1-EMPA-Na
10.71Single6TPJSuvorexant6TPJ-OX2-Suvorexant
10.71Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
10.71Single7BR3Elagolix7BR3-GnRH1-Elagolix
10.71Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
10.71Single7F8ULintitript7F8U-CCKA-Lintitript
10.71Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
10.71Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
10.71Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
10.71Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
10.71Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
10.71Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
10.71Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
10.71Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
10.71Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
10.71Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
10.71Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
10.71Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
10.71Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
10.71Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
10.71Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
10.71Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
10.71Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
10.71Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
10.71Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
10.71Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
10.71Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
10.71Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
10.71Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
10.71Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
10.71Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
10.71Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
10.71Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
10.71Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
10.71Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
10.71Single9H2XA1IR19H2X-A2A-A1IR1-Na
10.71Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
10.71Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
10.71Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
10.71Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
10.71Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
10.71Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
10.71Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
10.71Consensusangiotensin_offOrthosteric Ligandat1_off
10.71Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
10.71Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
10.71Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
10.71Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
10.71Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
10.71Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
10.71Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
10.71Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
10.71Consensusorexin_offOrthosteric Ligandox2_off ox1_off
10.71Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
10.71Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
10.71Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
10.71Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
10.71Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
10.71Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
10.53Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
10.53Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
10.53Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
10.53Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
10.53Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
10.53Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
10.34Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
10.34Single4MBSMaraviroc4MBS-CCR5-Maraviroc
10.34Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
10.34Single4ZJCSB-6740424ZJC-OX1-SB-674042
10.34Single5UVIZM-2413855UVI-A2A-ZM-241385
10.34Single6A94Zotepine6A94-5-HT2A-Zotepine
10.34Single6AQFZM-2413856AQF-A2A-ZM-241385
10.34Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
10.34Single6KUXRS-799486KUX-α2a-RS-79948
10.34Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
10.34Single6MH8ZM-2413856MH8-A2A-ZM-241385
10.34Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
10.34Single6TP3Nemorexant6TP3-OX1-Nemorexant
10.34Single6TPGEMPA6TPG-OX2-EMPA
10.34Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
10.34Single6V9SGTPL114036V9S-OX1-GTPL11403
10.34Single6VI4JDTic6VI4-κ-JDTic
10.34Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
10.34Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
10.34Single6ZG9GSK10347026ZG9-M1-GSK1034702
10.34Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
10.34Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
10.34Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
10.34Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
10.34Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
10.34Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
10.34Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
10.34Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
10.34Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.34Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
10.34Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
10.34Single7VV6C48/807VV6-MRGPRX2-C48/80
10.34Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
10.34Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
10.34Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.34Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
10.34Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single8JD6VU03647708JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
10.34Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
10.34Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
10.34Single8RLNLUF58348RLN-A2A-LUF5834
10.34Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
10.34Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
10.34Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
10.34Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
10.34Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
10.34Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
10.34Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
10.34Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
10.34Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
10.34Single9ARXSerotonin9ARX-5-HT2A-Serotonin
10.34Single9AS3LSD9AS3-5-HT2A-LSD
10.34Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
10.34Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
10.34Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
10.34Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
10.34Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
10.34Consensusalpha1_onOrthosteric Ligandalpha1a_on
10.34Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
10.34Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
10.34Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
10.34Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
10.34Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
10.34Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
10.26Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
10.26Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
10.00Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
10.00Single2Y01Dobutamine2Y01-β1-Dobutamine
10.00Single2Y02Carmoterol2Y02-β1-Carmoterol
10.00Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
10.00Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
10.00Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
10.00Single4EJ4Naltrindole4EJ4-δ-Naltrindole
10.00Single4QIMANTA XV4QIM-SMO-ANTA XV
10.00Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
10.00Single4YAYZD-71554YAY-AT1-ZD-7155
10.00Single5DHHSB-6121115DHH-NOP-SB-612111
10.00Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
10.00Single6DRXLisuride6DRX-5-HT2B-Lisuride
10.00Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
10.00Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
10.00Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
10.00Single7BU7BI1671077BU7-β1-BI167107
10.00Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
10.00Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
10.00Single7F83PF-051904577F83-Ghrelin-PF-05190457
10.00Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
10.00Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
10.00Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
10.00Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
10.00Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
10.00Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
10.00Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
10.00Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
10.00Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
10.00Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
10.00Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
10.00Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
10.00Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
10.00Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
10.00Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
10.00Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
10.00Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
10.00Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
10.00Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
10.00Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
10.00Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
10.00Single8JXRLSD8JXR-D1-LSD
10.00Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
10.00Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
10.00Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
10.00Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
10.00Single8X63Mepyramine8X63-H1-Mepyramine
10.00Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
10.00Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
10.00Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
10.00Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
10.00Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
10.00Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
10.00Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
10.00Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
10.00Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
10.00Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
10.00Single9H37A1IR09H37-A2A-A1IR0-Na
10.00Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
10.00Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
10.00Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
10.00Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
10.00Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
10.00Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
10.00Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
10.00Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
10.00Consensusalpha2_onOrthosteric Ligandalpha2b_on
10.00Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
10.00Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
10.00Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
10.00Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
10.00Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
10.00Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
10.00Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
10.00Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
10.00Consensushistamine_offOrthosteric Ligandh1_off
9.76Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
9.76Single9KDFRES-701-39KDF-ETB-RES-701-3
9.68Single2Y00Dobutamine2Y00-β1-Dobutamine
9.68Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
9.68Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
9.68Single5WIUNemonapride5WIU-D4-Nemonapride
9.68Single5WIVNemonapride5WIV-D4-Nemonapride-Na
9.68Single5WQCEMPA5WQC-OX2-EMPA
9.68Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
9.68Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
9.68Single6LUQHaloperidol6LUQ-D2-Haloperidol
9.68Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
9.68Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
9.68Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
9.68Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
9.68Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
9.68Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
9.68Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
9.68Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
9.68Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
9.68Single7WC6LSD7WC6-5-HT2A-LSD
9.68Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
9.68Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.68Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
9.68Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
9.68Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
9.68Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
9.68Single8JXSPF-61428JXS-D1-PF-6142
9.68Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
9.68Single8S4DCMF-0198S4D-Apelin-CMF-019
9.68Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
9.68Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
9.68Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
9.68Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
9.68Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
9.68Single8ZMFA1L108ZMF-5-HT2C-A1L10
9.68Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
9.68Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
9.68Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
9.68Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
9.68Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
9.68Single9HC04YI9HC0-mGlu5-4YI
9.68Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
9.68Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
9.68Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
9.68Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
9.68Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
9.68Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
9.68Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
9.68Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
9.68Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
9.68Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
9.68Consensusblt_offOrthosteric Ligandblt1_off
9.68Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
9.68Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
9.68Consensusep_offOrthosteric Ligandep4_off
9.68Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
9.68Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
9.68Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
9.68Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
9.68Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
9.52Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
9.38Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
9.38Single4DJHJDTic4DJH-κ-JDTic
9.38Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
9.38Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
9.38Single6J20Aprepitant6J20-NK1-Aprepitant
9.38Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
9.38Single6OS1TRV0266OS1-AT1-TRV026
9.38Single6TQ7SB-3348676TQ7-OX1-SB-334867
9.38Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
9.38Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
9.38Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
9.38Single7FEECP559407FEE-CB1-CP55940-ZCZ011
9.38Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
9.38Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
9.38Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
9.38Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.38Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
9.38Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
9.38Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.38Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
9.38Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
9.38Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
9.38Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
9.38Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
9.38Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
9.38Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
9.38Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
9.38Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
9.38Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
9.38Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
9.38Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
9.38Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
9.38Single8ZWFJR14a8ZWF-C3aB-JR14a
9.38Single9BJKNaloxone9BJK-μ-Naloxone-NAM
9.38Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
9.38Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
9.38Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
9.09Single4N4WSANT-14N4W-SMO-SANT-1
9.09Single4RWADIPP-NH24RWA-δ-DIPP-NH2
9.09Single6A93Risperidone6A93-5-HT2A-Risperidone
9.09Single6CM4Risperidone6CM4-D2-Risperidone
9.09Single6KQICP559406KQI-CB1-CP55940-Org27569
9.09Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
9.09Single6ZG4HTL00099366ZG4-M1-HTL0009936
9.09Single7DFPSpiperone7DFP-D2-Spiperone
9.09Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
9.09Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
9.09Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
9.09Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.09Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
9.09Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
9.09Single7YITNalfurafine7YIT-κ-Nalfurafine
9.09Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
9.09Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
9.09Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
9.09Single8JWZAB9288JWZ-A2A-AB928-Na
9.09Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
9.09Single8XQJJN2418XQJ-Apelin-JN241
9.09Single8XWACXCL18XWA-CXCR2-CXCL1
9.09Single8XWSCXCL58XWS-CXCR2-CXCL5
9.09Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
9.09Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
9.09Consensusalpha1_offOrthosteric Ligandalpha1a_off
9.09Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
9.09Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
9.09Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
9.09Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
9.09Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
9.09Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
9.09Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
9.09Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.82Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
8.82Single5X93K-87945X93-ETB-K-8794
8.82Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
8.82Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
8.82Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
8.82Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.82Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.82Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
8.82Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
8.82Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
8.82Single8XVJMacitentan8XVJ-ETA-Macitentan
8.82Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
8.82Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
8.82Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
8.82Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
8.82Consensusendothelin_offOrthosteric Ligandetb_off
8.82Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
8.82Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
8.82Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
8.57Single6KNMJN241-96KNM-Apelin-JN241-9
8.57Single6PT3DPI-2876PT3-δ-DPI-287
8.57Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
8.57Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
8.57Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
8.57Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
8.57Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
8.57Single8X5YAstemizole8X5Y-H1-Astemizole
8.57Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
8.57Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
8.57Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
8.57Single9IPYJR14a9IPY-C3aB-JR14a
8.57Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
8.57Consensuskisspeptin_onOrthosteric Ligandkiss1_on
8.57Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single5MZPCaffeine5MZP-A2A-Caffeine-Na
8.33Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
8.33Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
8.33Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
8.33Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
8.33Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
8.33Single8KIGSHU91198KIG-MC3-SHU9119-Ca
8.33Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
8.33Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
8.33Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
8.33Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
8.33Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
8.33Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
8.33Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
8.33Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
8.33Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
8.33Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
8.33Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
8.11Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
8.11Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
8.11Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
8.11Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
8.11Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
8.11Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
8.11Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
8.11Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
8.00Single6VCBLSN31604406VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
8.00Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
8.00Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
8.00Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
7.89Single6W25SHU91196W25-MC4-SHU9119-Ca
7.89Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
7.89Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
7.89Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
7.69Single3OE8IT1t3OE8-CXCR4-IT1t
7.69Single3RFMCaffeine3RFM-A2A-Caffeine
7.69Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
7.69Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
7.69Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
7.69Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single9IVMLSN33188399IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
7.69Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
7.69Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
7.69Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
7.69Consensusp2y_offOrthosteric Ligandp2y1_off
7.69Consensussensory_onOrthosteric Ligandopsins_on
7.50Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
7.41Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
7.41Single3UZAGTPL92363UZA-A2A-GTPL9236
7.41Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
7.41Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
7.41Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
7.41Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
7.41Single6ME5Agomelatine6ME5-MT1-Agomelatine
7.41Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
7.41Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
7.41Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
7.41Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
7.41Single8JPSCCL78JPS-ACKR1-CCL7
7.41Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
7.41Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
7.41Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
7.41Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
7.41Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
7.41Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
7.41Consensusgi_sensoryOrthosteric Ligandgi_opsins
7.41Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
7.41Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
7.41Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
7.41Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
7.41Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
7.41Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
7.14Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
7.14Single3PBLEticlopride3PBL-D3-Eticlopride
7.14Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
7.14Single6HLLCP999946HLL-NK1-CP99994
7.14Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
7.14Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
7.14Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
7.14Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
7.14Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
7.14Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
7.14Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
7.14Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
7.14Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
7.14Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
7.14Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
7.14Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
7.14Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
7.14Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
7.14Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.14Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.14Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
7.14Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
7.14Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
7.14Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
7.14Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
7.14Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
7.14Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
7.14Consensusgq_nucleotideOrthosteric Ligandgq_p2y
7.14Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
7.14Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
6.90Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
6.90Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
6.90Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
6.90Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
6.90Single5WS3EMPA5WS3-OX2-EMPA
6.90Single6B73MP11046B73-κ-MP1104
6.90Single6DS0Ly2660976DS0-5-HT2B-Ly266097
6.90Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
6.90Single6ME9Ramelteon6ME9-MT2-Ramelteon
6.90Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
6.90Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
6.90Single7F8YDevazepide7F8Y-CCKA-Devazepide
6.90Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
6.90Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
6.90Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
6.90Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
6.90Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
6.90Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
6.90Single7XRRLemborexant7XRR-OX2-Lemborexant
6.90Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
6.90Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
6.90Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
6.90Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
6.90Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
6.90Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
6.90Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
6.90Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
6.90Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
6.67Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
6.67Single3REYXAC3REY-A2A-XAC
6.67Single3RZECidoxepin3RZE-H1-Cidoxepin
6.67Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
6.67Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
6.67Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
6.67Single6FFIMMPEP6FFI-mGlu5-MMPEP
6.67Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
6.67Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
6.67Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
6.67Single6TPKRetosiban6TPK-OT-Retosiban
6.67Single6TPNHTL66416TPN-OX2-HTL6641
6.67Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
6.67Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
6.67Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
6.67Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
6.67Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
6.67Single7VODCariprazine7VOD-5-HT2A-Cariprazine
6.67Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
6.67Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
6.67Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
6.67Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
6.67Single8ZPMAMD0708ZPM-CXCR4-AMD070
6.67Single8ZPNAMD31008ZPN-CXCR4-AMD3100
6.67Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
6.67Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
6.67Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
6.67Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
6.67Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
6.67Consensusopsins_offOrthosteric Ligandrhodopsin_off
6.67Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
6.67Consensussensory_offOrthosteric Ligandopsins_off
6.67Consensusvasop-oxy_offOrthosteric Ligandot_off
6.45Single5DHGC-355DHG-NOP-C-35
6.45Single5UIGCmpd-15UIG-A2A-Cmpd-1
6.45Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
6.45Single6FFHFenobam6FFH-mGlu5-Fenobam
6.45Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
6.45Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
6.45Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
6.45Single6GPSMK08126GPS-CCR2-MK0812
6.45Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
6.45Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
6.45Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
6.45Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
6.45Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
6.45Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
6.45Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
6.45Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
6.45Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
6.45Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
6.45Single8X64Desloratadine8X64-H1-Desloratadine
6.45Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
6.45Single9IYAONO-97105319IYA-GPR55-ONO-9710531
6.45Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
6.45Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
6.45Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
6.45Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
6.45Consensusblt_onOrthosteric Ligandblt1_on
6.45Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
6.45Consensuscck_offOrthosteric Ligandccka_off
6.45Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
6.45Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
6.45Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
6.45Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
6.45Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
6.45Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
6.45Consensusleukotriene_onOrthosteric Ligandblt_on
6.45Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
6.45Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
6.25Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
6.25Single5XPRBosentan5XPR-ETB-Bosentan
6.25Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
6.25Single6GPXMK08126GPX-CCR2-MK0812
6.25Single6HLPNetupitant6HLP-NK1-Netupitant
6.25Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
6.25Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
6.25Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
6.25Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
6.25Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
6.25Single9HAPTolvaptan9HAP-V2-Tolvaptan
6.25Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
6.25Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
6.06Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
6.06Single6E59L-7607356E59-NK1-L-760735
6.06Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
6.06Single7R0CAVP7R0C-V2-AVP-Arrestin2
6.06Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
6.06Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
6.06Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
6.06Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
6.06Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
6.06Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
6.06Single8XVLZibotentan8XVL-ETA-Zibotentan
6.06Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
6.06Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
6.06Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
6.06Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
6.06Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
6.06Consensustachykinin_offOrthosteric Ligandnk1_off
5.88Single5X33BIIL2605X33-BLT1-BIIL260
5.88Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
5.88Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
5.88Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.88Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
5.88Single9BJKNAM9BJK-μ-Naloxone-NAM
5.88Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
5.71Single6K1QIRL25006K1Q-ETB-IRL2500
5.71Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
5.71Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
5.71Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.71Single8ZPLHF511168ZPL-CXCR4-HF51116
5.71Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
5.56Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
5.56Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.56Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
5.56Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
5.56Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
5.56Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
5.56Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
5.41Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.41Single8WKYPG-9348WKY-MC4-PG-934
5.41Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
5.26Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
5.26Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
5.13Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
5.13Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
5.13Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
5.00Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
4.65Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
4.55Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
4.55Single6D35Cholesterol6D35-SMO-Cholesterol
4.55Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.55Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.55Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
4.55Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
4.55Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042
4.55Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
4.55Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
4.55Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-BHFF
4.55Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
4.55Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626
4.55Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
4.55Single7DTTCa7DTT-CaS-Ca-Ca
4.55Single7DTTCa7DTT-CaS-Ca-Ca
4.55Single7DTUTryptophan7DTU-CaS-Tryptophan
4.55Single7DTUTryptophan7DTU-CaS-Tryptophan
4.55Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.55Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.55Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.55Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.55Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
4.55Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.55Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.55Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.55Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.55Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.55Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.55Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
4.55Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
4.55Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.55Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.55Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.55Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.55Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.55Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.55Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.55Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.55Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.55Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7T9NM22 Fab7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
4.55Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.55Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.55Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.55Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.55Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.55Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.55Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
4.55Single7XW7K1-707XW7-TSH-K1-70
4.55Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.55Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.55Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.55Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.55Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.55Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.55Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.55Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.55Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.55Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.55Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.55Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.55Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
4.55Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.55Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.55Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.55Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.55Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
4.55Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
4.55Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.55Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.55Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
4.55Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
4.55Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
4.55Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
4.55Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
4.55Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.55Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.55Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
4.55Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.55Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.55Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.55Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.55Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.55Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.55Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.55Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.55Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.55Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.55Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.55Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.55Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.55Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.55Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.55Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.55Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
4.55Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
4.55Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
4.55Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
4.55Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
4.55Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
4.55Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.55Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.55Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.55Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.55Single8WVXNorrin8WVX-LGR4-Norrin
4.55Single8WVYNorrin8WVY-LGR4-Norrin
4.55Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.55Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.55Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.55Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.55Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.55Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.55Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
4.55Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.55Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.55Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.55Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.55Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.55Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.55Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.55Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.55Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single9KHHNorrin9KHH-LGR4-Norrin
4.55Single9S37NB219S37-LGR4-NB21
4.55Single9UTBSucralose9UTB-TAS1R2; TAS1R3-Sucralose
4.35Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.35Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.35Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.35Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.35Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.35Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.35Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
4.35Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
4.17Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
4.17Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
4.17Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
4.17Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
4.00Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
4.00Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
4.00Single7UTZTR14027UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
4.00Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
4.00Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
3.85Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
3.85Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
3.85Single5L7DCholesterol5L7D-SMO-Cholesterol
3.85Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
3.85Single7WC4Serotonin7WC4-5-HT2A-Serotonin
3.85Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
3.70Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
3.70Single6TQ9SB-4081246TQ9-OX1-SB-408124
3.70Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
3.57Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
3.57Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
3.57Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
3.57Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
3.57Single7WC5Psilocin7WC5-5-HT2A-Psilocin
3.45Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
3.45Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
3.45Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
3.45Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
3.45Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
3.45Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
3.45Single6TP4ACT-4622066TP4-OX1-ACT-462206
3.45Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.45Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
3.45Single7UL2SR486927UL2-NTS1-SR48692-Na
3.45Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
3.45Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
3.45Single8YKDDehydroepiandrosterone8YKD-ADGRG2-Dehydroepiandrosterone-chim(NtGi1-Gs)/β1/γ2
3.45Consensusneurotensin_offOrthosteric Ligandnts1_off
3.45Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
3.33Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
3.33Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
3.33Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
3.33Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
3.33Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
3.33Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
3.33Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.33Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
3.33Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
3.33Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
3.33Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
3.33Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
3.33Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.33Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
3.33Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
3.23Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
3.23Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
3.23Single6IQLL7458706IQL-D4-L745870
3.23Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
3.23Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
3.23Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
3.23Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
3.23Single8K2WAMG4878K2W-CXCR3-AMG487
3.23Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
3.23Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.23Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
3.23Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
3.23Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
3.12Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
3.12Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
3.12Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.12Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
3.03Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
3.03Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
3.03Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.03Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
2.94Single5TZRMK86665TZR-FFA1-MK8666
2.94Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
2.94Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
2.94Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
2.94Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
2.94Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
2.94Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
2.94Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
2.86Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
2.86Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
2.86Single4PY02MeSATP4PY0-P2Y12-2MeSATP
2.86Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
2.86Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
2.86Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
2.78Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
2.78Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
2.78Single9JH5C16:0 Ceramide9JH5-CysLT2-C16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
2.70Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
2.63Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
2.63Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
2.63Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
2.63Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.63Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.63Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
2.56Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
2.50Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.50Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.44Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.38Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
2.38Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
2.27Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
ctlike_on_gp 6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
Net Summary
Imin 2.82
Number of Linked Nodes 767
Number of Links 947
Number of Hubs 154
Number of Links mediated by Hubs 587
Number of Communities 21
Number of Nodes involved in Communities 218
Number of Links involved in Communities 321
Path Summary
Number Of Nodes in MetaPath 66
Number Of Links MetaPath 65
Number of Shortest Paths 3779805
Length Of Smallest Path 3
Average Path Length 29.3444
Length of Longest Path 49
Minimum Path Strength 1.215
Average Path Strength 7.04549
Maximum Path Strength 63.615
Minimum Path Correlation 0.7
Average Path Correlation 0.990886
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 3.33333
Average % Of Corr. Nodes 41.5248
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 50.4485
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
class-b1_on_gpglucagon_on_gp
vip-pacap_on_gp
pth_on_gp
crf_on_gp
calcitonin_on_gp



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Download calcitonin_on_gp.zip



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