Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.33 1.06806604
2G.S1.06 4.5115468
3G.H1.01 4.70458469
4G.S2.04 3.00325407
5G.S2.08 3.5052536
6G.S3.03 4.56852738
7G.S3.04 7.43375417
8G.H2.07 4.49667719
9G.h2s4.01 7.88508409
10G.S4.02 4.2925418
11G.S4.03 3.6965467
12G.S4.04 4.83767409
13G.s4h3.04 4.174608
14G.H3.09 5.39807519
15G.H3.13 6.1712516
16G.H3.14 2.96853508
17G.H3.17 5.658515
18G.H3.18 5.07917419
19G.S5.05 5.24289669
20G.hgh4.05 7.35487506
21G.hgh4.20 2.31008403
22G.hgh4.21 3.64133404
23G.H4.03 2.54408404
24G.H4.08 5.666475103
25G.H4.10 8.16292407
26G.H4.12 5.8334104
27G.H4.15 7.41633408
28G.S6.02 7.4305408
29G.S6.05 7.07845105
30G.s6h5.01 5.42117469
31G.s6h5.05 3.15544669
32G.H5.03 5.74127569
33G.H5.08 5.98417438
34G.H5.17 4.663505
35G.H5.22 2.08633404
36G.H5.23 5.38383484
37G.H5.24 2.37242406
38b.1x4 1.66125403
39b.1x15 2.12492404
40b.lh12x2 5.0475408
41b.h2x1 4.48675405
42b.lhb1x3 2.62542402
43b.lhb1x6 4.035254143
44b.l1x3 10.2075409
45b.l1x6 10.4238419
46b.b2x1 5.98017418
47b.b2x5 6.11939677
48b.l3x2 6.08292409
49b.b4x6 9.66193579
50b.b5x2 4.99308407
51b.b5x3 6.152679
52b.b5x5 5.53858405
53b.b5x7 4.69625407
54b.l5x1 3.825834158
55b.l5x5 8.24544619
56b.b6x1 3.52042409
57b.b6x5 3.817506
58b.b7x1 6.38092404
59b.l7x4 2.88567409
60b.b8x3 3.35075406
61b.b8x4 5.26945156
62b.b9x4 6.69142409
63b.l9x3 6.46883619
64b.l9x6 5.36783618
65b.b10x5 4.26486709
66b.b11x4 5.12517419
67b.l11x2 6.89027519
68b.b12x6 8.54389618
69b.b12x7 5.29825459
70b.b13x7 7.5382557
71b.l13x3 7.36894659
72b.b14x3 4.72083455
73b.b15x1 6.9684559
74b.l15x2 5.02558409
75b.b16x4 10.7192456
76b.b16x6 8.26817658
77b.b17x5 7.11042447
78b.b17x7 8.012448
79b.l17x3 8.559649
80b.l17x6 6.82642409
81b.b18x3 5.66517448
82b.b18x5 5.6475405
83b.l18x1 6.12897116
84b.b19x2 6.55755646
85b.b19x4 5.97025448
86b.l19x2 6.55587549
87b.b20x4 9.92993548
88b.b20x6 6.94693546
89b.b20x7 4.12633409
90b.l20x2 5.75333409
91b.b21x1 6.568547
92b.b21x5 4.90417404
93b.b21x7 5.2875605
94b.l21x2 5.59325404
95b.l21x9 5.056406
96b.b22x5 6.103174117
97b.l22x5 6.563475149
98b.b23x6 7.088726127
99b.l23x1 5.41487516
100b.b24x4 7.375334126
101b.b24x6 6.196584128
102b.l25x3 8.77953599
103b.l25x6 11.0723518
104b.b26x3 3.86817406
105b.l27x1 11.7163619
106b.l27x2 7.98842499
107b.b28x4 6.83433596
108b.b28x6 8.68833599
109g.h1x5 1.45942406
110g.l1x4 2.83333508
111g.h2x7 2.72025405
112g.h2x11 8.377924116
113g.ctx3 5.76987509
114g.ctx6 3.25925406
115g.ctx16 5.29489608
1161x50 3.71075409
1171x60 3.80533509
118I1x50 2.5378508
1192x39 5.81408489
1202x43 4.93913589
121E1 4.27356623
1223x24 1.35975408
1233x33 4.24119729
1243x34 4.06673509
1253x37 4.33842409
1263x42 8.894726189
1273x49 4.64292489
1283x53 4.9975489
129I2 5.683181738
1304x42 3.98683438
1314x50 6.298674189
1324x53 3.69093509
133E2 9.409781727
134E2x51 6.86713529
135E2x52 5.69613528
1365x40 3.82692429
1375x58 3.7875199
138I3 3.31945208
1396x48 11.0845529
140E3 5.72067428
1417x35 4.63525409
1427x37 8.42908429
1437x50 6.07525179
1447x52 3.71233409
1458x54 3.71033409
146G.s4h3.14 0.303667400
147G.H3.01 3.89045130
148NT 7.055172420
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1b.b4x4 b.l1x3 52.31210.341NoYes089
2b.b3x6 b.l1x3 10013.2967NoYes099
3b.b3x6 b.l3x2 99.92817.805NoYes099
4b.l1x4 b.l3x2 99.27638.50467NoYes069
5G.HN.51 b.l1x4 99.05716.126NoNo046
6G.HN.51 I2 98.98113.06533NoYes348
7b.b26x2 b.b2x3 90.85245.076NoNo076
8b.b26x1 b.b26x2 90.7953.21067NoNo097
9b.b26x1 b.l27x1 90.73785.02333NoYes099
10b.l3x1 b.l5x5 11.38899.018NoYes199
11b.b2x1 b.l27x1 74.87575.72267YesYes189
12G.S1.02 I2 24.39726.496NoYes368
13G.S1.02 G.S3.03 24.15155.564NoYes368
14G.S3.01 I2 24.262511.6503NoYes358
15G.S3.01 G.S3.03 24.14093.83333NoYes358
16G.H5.08 I2 25.16076.64567YesYes388
17G.H5.08 G.S3.03 24.17093.32333YesYes388
18G.S1.04 G.S3.03 52.74363.929NoYes078
19G.S1.04 G.S4.03 52.34663.33NoYes077
20b.l25x6 b.l27x1 15.032624.5563YesYes189
21G.H3.15 G.H3.17 10.20573.22533NoYes185
22G.S2.06 G.S3.03 19.00218.46767NoYes098
23b.b2x1 b.b6x1 69.16753.113YesYes089
24b.b6x1 b.l9x6 68.8914.50933YesYes098
25G.H2.07 b.l9x6 12.35113.34433YesYes198
26G.S4.03 G.S5.05 48.09363.96367YesYes679
27G.S5.05 G.s6h5.01 10.87995.104YesYes699
28G.S5.07 G.s5hg.01 12.76714.19767NoNo099
29G.H1.08 G.S2.06 12.37285.30667NoNo099
30G.H1.04 G.H1.08 12.01743.71667NoNo079
31G.H2.06 b.l17x6 33.78496.96067NoYes099
32G.H2.06 b.b14x1 33.90045.72NoNo098
33b.b14x1 b.l9x6 34.01444.39033NoYes088
34b.l15x1 b.l17x6 34.49049.54333NoYes079
35b.l13x6 b.l15x1 34.60453.31967NoNo097
36b.l13x6 b.l9x6 34.00949.46567NoYes198
37G.S4.04 G.S5.04 11.14163.571YesNo099
38G.H5.10 G.S6.02 30.291712.602NoYes078
39G.H5.10 G.S5.03 15.53929.09367NoNo079
40G.S5.03 G.S5.05 16.35034.39533NoYes099
41G.H5.10 G.S6.04 15.56698.278NoNo079
42G.S5.05 G.S6.04 16.34765.39333YesNo099
43G.S6.02 G.h4s6.20 14.33266.082YesNo084
44G.H5.17 G.h4s6.20 12.70069.42933YesNo054
45G.H5.13 G.H5.17 12.70046.364NoYes085
46G.H5.13 G.S6.02 13.51617.416NoYes088
475x68 G.H5.17 13.24693.96967NoYes085
486x48 7x45 16.15497.33833YesNo099
493x43 7x45 19.70583.98933NoNo099
502x46 3x43 20.00234.03NoNo099
512x46 3x42 20.15033.28267NoYes099
523x42 3x45 29.95316.34833YesNo099
533x45 4x46 30.3715.477NoNo098
544x42 4x46 30.51214.935YesNo088
554x42 I2 38.0244.17933YesYes388
56b.l17x5 b.l17x6 67.06863.28867NoYes069
57b.l17x5 b.l19x2 66.34513.08967NoYes069
58b.l17x3 b.l19x2 45.44295.418YesYes499
59b.b19x4 b.l17x3 24.78326.208YesYes489
60b.b19x4 b.b20x6 18.91175.665YesYes486
61b.b17x7 b.b20x6 47.50968.82433YesYes486
62b.b17x7 b.b21x1 39.1064.02033YesYes487
63b.1x19 b.b21x1 31.64886.232NoYes027
64b.1x15 b.1x19 24.73732.837YesNo042
65b.1x11 b.1x15 20.89392.02067NoYes064
66b.b20x4 b.l17x3 19.667217.4527YesYes489
67b.b20x4 b.b20x6 37.80384.13233YesYes486
68b.b20x2 b.l19x2 20.16539.20233NoYes069
69b.b20x2 b.b20x4 19.66385.563NoYes068
70b.1x11 g.h1x11 20.12493.71633NoNo069
71b.l26x5 g.ctx4 11.70116.59867NoNo057
72g.ctx3 g.ctx4 11.41984.40067YesNo097
73b.b2x5 b.b3x2 10.708910.554YesNo775
74b.b3x2 b.b4x6 93.09784.63167NoYes759
75b.b3x4 b.b4x6 46.90444.48767NoYes099
76b.l26x3 b.l26x5 11.08857.486NoNo075
77b.l26x1 b.l26x3 11.17696.26433NoNo777
78b.b2x5 b.l26x1 11.738811.1603YesNo777
79b.b16x5 b.l14x6 12.56816.04333NoNo053
80b.b16x7 b.l14x6 10.7733.66333NoNo093
81b.l21x7 b.l23x1 10.68613.78767NoYes056
82b.l21x7 b.l23x2 10.33776.01633NoNo058
83b.1x10 g.h1x11 18.58651.98433NoNo089
84b.1x10 g.h1x12 10.25351.645NoNo086
85b.b2x3 b.b3x2 82.35263.768NoNo765
86b.b3x4 b.l1x3 47.83177.205NoYes099
87b.b4x4 b.b4x6 46.778712.7617NoYes789
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
3x29E25.683670NoYes9721
3x30E25.922330NoYes6721
3x33E26.8242YesYes9721
3x33E2x524.3442YesYes9822
4x60E24.148670NoYes8721
4x61E23.828670NoYes8721
4x64E29.8682NoYes6721
E2E239.6492YesYes7711
5x39E210.83872NoYes7721
E2E2x524.562332YesYes7812
5x39E2x524.9152NoYes7822
NTNT20.44932YesYes0022
E2NT14.64472YesYes7012
1x29E24.2480NoYes0721
3x26E22.8820NoYes9721
5x38E22.2820NoYes5721
2x60E22.159672NoYes9721
E2Lig1.8472YesNo7010
4x65E20.9286670NoYes0721
5x37Lig0.7230NoNo6010

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
100.00Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
25.00Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
25.00Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
25.00Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
20.00Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
20.00Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
16.67Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
16.67Single5N2RPSB-365N2R-A2A-PSB-36-Na
16.67Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
16.67Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
16.67Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
16.67Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
16.67Single8PWNTheophylline8PWN-A2A-Theophylline
16.67Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
15.38Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
15.38Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
14.29Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
14.29Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
14.29Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
14.29Single8A2OTheophylline8A2O-A2A-Theophylline-Na
14.29Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
14.29Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
14.29Consensusp2y_offOrthosteric Ligandp2y1_off
13.33Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
12.50Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
12.50Single3OE6IT1t3OE6-CXCR4-IT1t
12.50Single4XNWMRS25004XNW-P2Y1-MRS2500
12.50Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
12.50Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
12.50Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
12.50Single6ME5Agomelatine6ME5-MT1-Agomelatine
12.50Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
12.50Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
12.50Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
12.50Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
12.50Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
12.50Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
12.50Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
12.50Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
12.50Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
12.50Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
12.50Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
12.50Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
12.50Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
12.50Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
12.50Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
12.50Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
11.11Single3OE9IT1t3OE9-CXCR4-IT1t
11.11Single4O9RCyclopamine4O9R-SMO-Cyclopamine
11.11Single5L7IVismodegib5L7I-SMO-Vismodegib
11.11Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
11.11Single6LI0C176LI0-GPR52-C17
11.11Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
11.11Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
11.11Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
11.11Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
11.11Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
11.11Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
11.11Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
11.11Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
11.11Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
11.11Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
11.11Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
11.11Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
11.11Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
11.11Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
11.11Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
11.11Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
11.11Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
11.11Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
11.11Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
11.11Single8K5BNiacin8K5B-HCA2-Niacin
11.11Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
11.11Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
11.11Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
11.11Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
11.11Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
11.11Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
11.11Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
11.11Single9B9Y7DY9B9Y-CB1-7DY
11.11Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.11Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
11.11Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
11.11Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
11.11Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
11.11Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
11.11Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
11.11Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
11.11Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
11.11Consensusgq_nucleotideOrthosteric Ligandgq_p2y
11.11Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
10.53Single5WF5UK-4320975WF5-A2A-UK-432097
10.00Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
10.00Single3ODUIT1t3ODU-CXCR4-IT1t
10.00Single3PWHZM-2413853PWH-A2A-ZM-241385
10.00Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
10.00Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
10.00Single4BWBNeurotensin4BWB-NTS1-Neurotensin
10.00Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
10.00Single4QINSAG1.54QIN-SMO-SAG1.5
10.00Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
10.00Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
10.00Single5U09Taranabant5U09-CB1-Taranabant
10.00Single5ZKQABT-4915ZKQ-PAF-ABT-491
10.00Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
10.00Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
10.00Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
10.00Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
10.00Single6ME2Ramelteon6ME2-MT1-Ramelteon
10.00Single6ME9Ramelteon6ME9-MT2-Ramelteon
10.00Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
10.00Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
10.00Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
10.00Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
10.00Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
10.00Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
10.00Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
10.00Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
10.00Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
10.00Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
10.00Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
10.00Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
10.00Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
10.00Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
10.00Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
10.00Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
10.00Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
10.00Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
10.00Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
10.00Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single8GNGIstradefylline8GNG-A2A-Istradefylline
10.00Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
10.00Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
10.00Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
10.00Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
10.00Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
10.00Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
10.00Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
10.00Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
10.00Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
10.00Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
10.00Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
10.00Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
10.00Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
10.00Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
10.00Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
10.00Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
10.00Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
10.00Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
10.00Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
10.00Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
10.00Single9H2XA1IR19H2X-A2A-A1IR1-Na
10.00Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
10.00Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
10.00Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
10.00Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
10.00Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
10.00Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
10.00Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
10.00Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
10.00Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
9.52Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
9.52Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
9.09Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
9.09Single2YDOAdenosine2YDO-A2A-Adenosine
9.09Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
9.09Single5IU7Q274563465IU7-A2A-Q27456346-Na
9.09Single5IUBQ274563445IUB-A2A-Q27456344-Na
9.09Single5JTBZM-2413855JTB-A2A-ZM-241385
9.09Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
9.09Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
9.09Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
9.09Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
9.09Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
9.09Single5UVIZM-2413855UVI-A2A-ZM-241385
9.09Single6AQFZM-2413856AQF-A2A-ZM-241385
9.09Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
9.09Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
9.09Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
9.09Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
9.09Single6MH8ZM-2413856MH8-A2A-ZM-241385
9.09Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
9.09Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
9.09Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
9.09Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
9.09Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
9.09Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
9.09Single7AROLUF58337ARO-A2A-LUF5833-Na
9.09Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
9.09Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
9.09Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
9.09Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
9.09Single7F61PF-036547467F61-H3-PF-03654746
9.09Single7T32ZM-2413857T32-A2A-ZM-241385
9.09Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
9.09Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
9.09Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
9.09Single7VV6C48/807VV6-MRGPRX2-C48/80
9.09Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
9.09Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
9.09Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
9.09Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
9.09Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
9.09Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
9.09Single8IHKAcifran8IHK-HCA3-Acifran
9.09Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
9.09Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
9.09Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
9.09Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
9.09Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
9.09Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
9.09Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
9.09Single8K5CAcipimox8K5C-HCA2-Acipimox
9.09Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
9.09Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
9.09Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
9.09Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
9.09Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
9.09Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
9.09Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
9.09Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
9.09Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
9.09Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
9.09Single9BA0A1AKN9BA0-CB1-A1AKN
9.09Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
9.09Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
9.09Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
9.09Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
9.09Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
9.09Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
9.09Consensusa2_offOrthosteric Liganda2a_off
9.09Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
9.09Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
9.09Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
9.09Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
9.09Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
9.09Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
9.09Consensushca_onOrthosteric Ligandhca2_on
9.09Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
9.09Consensusopsins_offOrthosteric Ligandrhodopsin_off
9.09Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
9.09Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
9.09Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
9.09Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
9.09Consensussensory_offOrthosteric Ligandopsins_off
9.09Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
8.70Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
8.70Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
8.70Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
8.33Single3EMLZM-2413853EML-A2A-ZM-241385
8.33Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
8.33Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
8.33Single4QIMANTA XV4QIM-SMO-ANTA XV
8.33Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
8.33Single5IU8Q274563475IU8-A2A-Q27456347-Na
8.33Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
8.33Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
8.33Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
8.33Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
8.33Single5T04Neurotensin5T04-NTS1-Neurotensin
8.33Single5TGZAM65385TGZ-CB1-AM6538
8.33Single5UENDU1725UEN-A1-DU172
8.33Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
8.33Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
8.33Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
8.33Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
8.33Single6IIVDaltroban6IIV-TXA2-Daltroban
8.33Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
8.33Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
8.33Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
8.33Single6S0LZM-2413856S0L-A2A-ZM-241385
8.33Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
8.33Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
8.33Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
8.33Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
8.33Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
8.33Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
8.33Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
8.33Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
8.33Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
8.33Single7PYRPSB-21157PYR-A2A-PSB-2115
8.33Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
8.33Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
8.33Single7V3ZCP559407V3Z-CB1-CP55940
8.33Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
8.33Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
8.33Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
8.33Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
8.33Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
8.33Single8CU6LJ-45178CU6-A2A-LJ-4517
8.33Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
8.33Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.33Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
8.33Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
8.33Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
8.33Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
8.33Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
8.33Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
8.33Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
8.33Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
8.33Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
8.33Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
8.33Single8T1WCVN4248T1W-GPR6-CVN424
8.33Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
8.33Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
8.33Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
8.33Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
8.33Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
8.33Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
8.33Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
8.33Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
8.33Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
8.33Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
8.33Single9CHXS-Carazolol9CHX-β2-S-Carazolol
8.33Single9H37A1IR09H37-A2A-A1IR0-Na
8.33Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
8.33Single9IYAONO-97105319IYA-GPR55-ONO-9710531
8.33Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
8.33Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
8.33Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
8.33Consensusa3_onOrthosteric Liganda3a_on
8.33Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
8.33Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
8.33Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
8.33Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
8.33Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
8.33Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
8.33Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
8.33Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
8.33Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
8.33Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
8.33Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
8.33Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
8.33Consensushca_on_gpOrthosteric Ligandhca2_on_gp
8.33Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
8.33Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
8.33Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
8.33Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
8.00Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
8.00Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
7.69Single4JKVTaladegib4JKV-SMO-Taladegib
7.69Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
7.69Single5IUAQ274563485IUA-A2A-Q27456348-Na
7.69Single5N2SPSB365N2S-A1-PSB36
7.69Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
7.69Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
7.69Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
7.69Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
7.69Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
7.69Single6D26Fevipiprant6D26-DP2-Fevipiprant
7.69Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
7.69Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
7.69Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
7.69Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
7.69Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
7.69Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
7.69Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
7.69Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
7.69Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
7.69Single6S0QZM-2413856S0Q-A2A-ZM-241385
7.69Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
7.69Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
7.69Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
7.69Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
7.69Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
7.69Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
7.69Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
7.69Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
7.69Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
7.69Single7SINNPS-21437SIN-CaS-NPS-2143
7.69Single7SINNPS-21437SIN-CaS-NPS-2143
7.69Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
7.69Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
7.69Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
7.69Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
7.69Single7W41PD1762527W41-BB2-PD176252
7.69Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
7.69Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
7.69Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.69Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
7.69Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
7.69Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
7.69Single8GNEKW-63568GNE-A2A-KW-6356-Na
7.69Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
7.69Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
7.69Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
7.69Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
7.69Single8JXSPF-61428JXS-D1-PF-6142
7.69Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
7.69Single8QOTNanobody-E8QOT-μ-Nanobody-E
7.69Single8S4DCMF-0198S4D-Apelin-CMF-019
7.69Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
7.69Single8TF5Oleic acid8TF5-GPR6-Oleic acid
7.69Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
7.69Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
7.69Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
7.69Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
7.69Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
7.69Single9B9ZA1AKO9B9Z-CB1-A1AKO
7.69Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
7.69Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
7.69Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
7.69Single9EHSLUF76029EHS-A3A-LUF7602
7.69Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
7.69Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
7.69Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
7.69Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
7.69Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
7.69Consensusa3_on_gpOrthosteric Liganda3a_on_gp
7.69Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
7.69Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
7.69Consensusadenosine_offOrthosteric Liganda1_off a2_off
7.69Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
7.69Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
7.69Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
7.69Consensusbombesin_offOrthosteric Ligandbb2_off
7.69Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
7.69Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
7.69Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
7.69Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
7.69Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
7.69Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
7.69Consensusdp_offOrthosteric Liganddp2_off
7.69Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
7.69Consensusep_offOrthosteric Ligandep4_off
7.69Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
7.69Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
7.69Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
7.69Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
7.69Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
7.69Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
7.69Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
7.69Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
7.69Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
7.69Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.69Consensustrace-amine_onOrthosteric Ligandta1_on
7.41Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
7.41Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
7.14Single2YDVNECA2YDV-A2A-NECA
7.14Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
7.14Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
7.14Single4BV0Neurotensin4BV0-NTS1-Neurotensin
7.14Single4UHRCGS216804UHR-A2A-CGS21680
7.14Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
7.14Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
7.14Single5G53NECA5G53-A2A-NECA-Gs
7.14Single5TZRMK86665TZR-FFA1-MK8666
7.14Single5V56TC1145V56-SMO-TC114
7.14Single5V57TC1145V57-SMO-TC114
7.14Single5XR8AM8415XR8-CB1-AM841
7.14Single5XRAAM115425XRA-CB1-AM11542
7.14Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
7.14Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
7.14Single6J21Aprepitant6J21-NK1-Aprepitant
7.14Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
7.14Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
7.14Single6OS1TRV0266OS1-AT1-TRV026
7.14Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
7.14Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
7.14Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
7.14Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
7.14Single7F1TMIP-1a7F1T-CCR5-MIP-1a
7.14Single7FEECP559407FEE-CB1-CP55940-ZCZ011
7.14Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
7.14Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
7.14Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
7.14Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
7.14Single7PX4PSB-21137PX4-A2A-PSB-2113
7.14Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
7.14Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
7.14Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
7.14Single7TUYGSK682753A7TUY-GPR183-GSK682753A
7.14Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
7.14Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
7.14Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
7.14Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
7.14Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
7.14Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
7.14Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
7.14Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
7.14Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
7.14Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
7.14Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
7.14Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
7.14Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
7.14Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
7.14Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
7.14Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
7.14Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
7.14Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
7.14Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
7.14Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
7.14Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
7.14Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
7.14Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
7.14Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
7.14Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
7.14Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
7.14Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
7.14Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
7.14Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
7.14Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
7.14Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
7.14Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
7.14Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
7.14Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
7.14Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
7.14Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
7.14Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
7.14Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
7.14Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
7.14Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
7.14Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
7.14Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
7.14Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
7.14Consensusa2_onOrthosteric Liganda2b_on
7.14Consensusa2_on_gpOrthosteric Liganda2b_on_gp
7.14Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
7.14Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
7.14Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
7.14Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
7.14Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
7.14Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
7.14Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
7.14Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
7.14Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
7.14Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
7.14Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
7.14Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
7.14Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
7.14Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
7.14Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
7.14Consensuslpa_onOrthosteric Ligandlpa1_on
7.14Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
7.14Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Consensusneurotensin_onOrthosteric Ligandnts1_on
7.14Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
7.14Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
7.14Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
7.14Consensusrelaxin_onOrthosteric Ligandrxfp4_on
7.14Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
7.14Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.14Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
6.90Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
6.67Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
6.67Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
6.67Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
6.67Single4N4WSANT-14N4W-SMO-SANT-1
6.67Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
6.67Single4PY02MeSATP4PY0-P2Y12-2MeSATP
6.67Single4XEENeurotensin4XEE-NTS1-Neurotensin
6.67Single4XESNeurotensin4XES-NTS1-Neurotensin
6.67Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
6.67Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
6.67Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
6.67Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
6.67Single6IIURamatroban6IIU-TXA2-Ramatroban
6.67Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
6.67Single6KQICP559406KQI-CB1-CP55940-Org27569
6.67Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
6.67Single6OS2TRV0266OS2-AT1-TRV026
6.67Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
6.67Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
6.67Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
6.67Single6YVRNTS8-136YVR-NTS1-NTS8-13
6.67Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
6.67Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
6.67Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
6.67Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
6.67Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
6.67Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
6.67Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
6.67Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
6.67Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
6.67Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
6.67Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.67Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
6.67Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
6.67Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
6.67Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.67Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
6.67Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
6.67Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
6.67Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
6.67Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
6.67Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
6.67Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
6.67Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
6.67Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
6.67Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
6.67Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
6.67Single8JWY2-1188JWY-A2A-2-118
6.67Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
6.67Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
6.67Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
6.67Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
6.67Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
6.67Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single8XQJJN2418XQJ-Apelin-JN241
6.67Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
6.67Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
6.67Single8XWACXCL18XWA-CXCR2-CXCL1
6.67Single8XWMCXCL68XWM-CXCR2-CXCL6
6.67Single8XWSCXCL58XWS-CXCR2-CXCL5
6.67Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
6.67Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
6.67Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
6.67Single9DGIZ85267113509DGI-CB1-Z8526711350
6.67Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.67Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
6.67Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
6.67Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
6.67Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
6.67Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
6.67Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
6.67Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
6.67Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
6.67Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
6.67Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
6.67Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
6.67Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
6.67Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
6.67Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
6.67Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
6.67Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
6.67Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
6.67Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
6.67Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
6.67Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
6.67Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
6.67Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
6.67Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
6.67Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
6.67Consensuslpa_offOrthosteric Ligandlpa1_off
6.67Consensuslpl_offOrthosteric Ligands1p_off lpa_off
6.67Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
6.67Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
6.67Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
6.67Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
6.67Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
6.45Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
6.25Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
6.25Single4BUONeurotensin4BUO-NTS1-Neurotensin
6.25Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
6.25Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
6.25Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
6.25Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
6.25Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
6.25Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
6.25Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
6.25Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
6.25Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
6.25Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
6.25Single7EZCUKA7EZC-A2A-UKA
6.25Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
6.25Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
6.25Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
6.25Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
6.25Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
6.25Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
6.25Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
6.25Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
6.25Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
6.25Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
6.25Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
6.25Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
6.25Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
6.25Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
6.25Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
6.25Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
6.25Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
6.25Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
6.25Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
6.25Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
6.25Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
6.25Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
6.25Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
6.25Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
6.25Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
6.25Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
6.25Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single8XVUCXCL28XVU-CXCR2-CXCL2
6.25Single8XWFCXCL38XWF-CXCR2-CXCL3
6.25Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
6.25Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
6.25Single8ZPLHF511168ZPL-CXCR4-HF51116
6.25Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
6.25Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
6.25Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.25Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
6.25Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
6.25Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
6.25Consensuscck_onOrthosteric Ligandccka_on cckb_on
6.25Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
6.25Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
6.25Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
6.25Consensuschemerin_onOrthosteric Ligandcml1_on
6.25Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
6.25Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
6.25Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.25Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.25Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
6.25Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
6.25Consensusprostanoid_offOrthosteric Ligandep_off dp_off
6.25Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
6.25Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
6.25Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single3NY9ICI118-5513NY9-β2-ICI118-551
5.88Single4UG2CGS216804UG2-A2A-CGS21680
5.88Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
5.88Single5WF6UK-4320975WF6-A2A-UK-432097
5.88Single5ZTYAM102575ZTY-CB2-AM10257
5.88Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
5.88Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
5.88Single6KNMJN241-96KNM-Apelin-JN241-9
5.88Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
5.88Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
5.88Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
5.88Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
5.88Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
5.88Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
5.88Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
5.88Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
5.88Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
5.88Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.88Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
5.88Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
5.88Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
5.88Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
5.88Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
5.88Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
5.88Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
5.88Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
5.88Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
5.88Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
5.88Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
5.88Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
5.88Single8QJ2pN1628QJ2-MC4-pN162-Gs
5.88Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
5.88Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
5.88Single8XQJJN2418XQJ-Apelin-JN241
5.88Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
5.88Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
5.88Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
5.88Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
5.88Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
5.88Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
5.88Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
5.88Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
5.88Single9JF4PD1683689JF4-BB1-PD168368
5.88Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
5.88Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
5.88Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
5.88Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
5.88Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
5.88Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
5.88Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
5.88Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
5.88Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
5.88Consensuskisspeptin_onOrthosteric Ligandkiss1_on
5.88Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
5.88Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
5.56Single4XT1Fractalkine4XT1-US28-Fractalkine
5.56Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
5.56Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
5.56Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
5.56Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
5.56Single7F8XNN90567F8X-CCKA-NN9056
5.56Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
5.56Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
5.56Single7QA8Peptide7QA8-STE2-Peptide
5.56Single7QA8Peptide7QA8-STE2-Peptide
5.56Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
5.56Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
5.56Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
5.56Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
5.56Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
5.56Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
5.56Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
5.56Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
5.56Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
5.56Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
5.56Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.56Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
5.56Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
5.56Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
5.56Single8IEBA1LYA8IEB-GPR156-A1LYA
5.56Single8IEIA1LYA8IEI-GPR156-A1LYA
5.56Single8IEIA1LYA8IEI-GPR156-A1LYA
5.56Single8IEPA1LYA8IEP-GPR156-A1LYA
5.56Single8IEPA1LYA8IEP-GPR156-A1LYA
5.56Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
5.56Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
5.56Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
5.56Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
5.56Single8WDTphotoNECA8WDT-A2A-photoNECA
5.56Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.56Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
5.56Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
5.56Single8XWNCXCL88XWN-CXCR2-CXCL8
5.56Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
5.56Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
5.56Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
5.56Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.56Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
5.56Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
5.56Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
5.56Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
5.56Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
5.56Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
5.56Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
5.56Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
5.56Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
5.56Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
5.56Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
5.56Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
5.56Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
5.56Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
5.56Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
5.56Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
5.56Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
5.56Consensuslpl_onOrthosteric Ligands1p_on lpa_on
5.56Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
5.56Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
5.56Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
5.56Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
5.56Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
5.56Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
5.26Single3QAKUK-4320973QAK-A2A-UK-432097
5.26Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
5.26Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
5.26Single6HLOAprepitant6HLO-NK1-Aprepitant
5.26Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
5.26Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
5.26Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
5.26Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
5.26Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
5.26Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
5.26Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
5.26Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
5.26Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
5.26Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
5.26Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
5.26Single7XNACYN1548067XNA-SST2-CYN154806
5.26Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
5.26Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
5.26Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
5.26Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single8IEBA1LYA8IEB-GPR156-A1LYA
5.26Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
5.26Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
5.26Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
5.26Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
5.26Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
5.26Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
5.26Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
5.26Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
5.26Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
5.26Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
5.26Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
5.26Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
5.26Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
5.26Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
5.26Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
5.26Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
5.26Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
5.26Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
5.26Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
5.26Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
5.26Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
5.26Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
5.26Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
5.00Single3OE0CVX153OE0-CXCR4-CVX15
5.00Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
5.00Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
5.00Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
5.00Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
5.00Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
5.00Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
5.00Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
5.00Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
5.00Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
5.00Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
5.00Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
5.00Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
5.00Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
5.00Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
5.00Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
5.00Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
5.00Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
5.00Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
5.00Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
5.00Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
5.00Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
5.00Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
5.00Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
5.00Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.00Consensusangiotensin_onOrthosteric Ligandat1_on
5.00Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
5.00Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
5.00Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
5.00Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
5.00Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
5.00Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
5.00Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
5.00Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
5.00Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
5.00Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
5.00Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
5.00Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
5.00Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
5.00Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
5.00Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
5.00Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
5.00Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
5.00Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
5.00Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
5.00Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
4.76Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
4.76Single6JODAngiotensin II6JOD-AT2-Angiotensin II
4.76Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
4.76Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
4.76Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
4.76Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
4.76Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
4.76Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
4.76Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
4.76Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
4.76Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
4.76Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
4.76Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
4.76Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
4.76Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
4.76Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
4.76Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
4.76Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
4.76Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
4.76Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
4.76Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
4.76Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
4.76Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
4.76Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
4.76Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
4.76Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
4.76Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
4.76Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
4.76Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
4.76Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
4.76Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
4.76Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
4.76Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
4.76Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
4.76Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
4.76Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
4.76Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
4.76Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
4.76Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
4.76Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
4.76Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
4.76Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
4.76Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
4.76Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
4.76Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
4.76Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
4.76Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
4.76Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
4.76Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
4.76Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
4.76Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
4.55Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
4.55Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
4.55Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
4.55Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
4.55Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
4.55Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
4.55Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
4.55Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
4.55Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
4.55Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
4.55Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
4.55Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
4.55Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
4.55Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
4.55Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
4.55Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
4.55Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.55Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
4.55Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
4.55Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
4.55Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
4.55Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
4.55Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
4.55Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
4.55Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
4.55Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
4.55Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single8ZRTET-18ZRT-ETB-ET-1
4.55Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
4.55Consensuscalcitonin_onOrthosteric Ligandctlike_on
4.55Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
4.55Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
4.55Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
4.55Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
4.55Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
4.55Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
4.55Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
4.55Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
4.55Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
4.55Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
4.55Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
4.55Consensuspac_onOrthosteric Ligandpac1_on
4.55Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
4.55Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
4.35Single4XT3Fractalkine4XT3-US28-Fractalkine
4.35Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
4.35Single6FJ3PTH6FJ3-PTH1-PTH
4.35Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
4.35Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
4.35Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
4.35Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
4.35Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
4.35Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
4.35Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
4.35Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
4.35Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
4.35Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
4.35Single7SK3CXCL127SK3-ACKR3-CXCL12
4.35Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
4.35Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
4.35Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
4.35Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
4.35Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
4.35Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
4.35Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
4.35Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
4.35Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
4.35Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
4.35Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
4.35Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
4.35Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
4.35Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
4.35Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
4.35Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
4.35Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
4.35Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
4.35Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
4.35Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
4.35Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
4.35Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
4.35Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
4.35Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
4.35Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
4.35Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
4.35Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
4.35Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
4.35Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
4.17Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
4.17Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
4.17Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
4.17Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
4.17Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
4.17Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
4.17Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
4.17Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
4.17Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
4.17Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
4.17Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
4.17Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
4.17Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
4.17Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
4.17Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
4.17Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
4.17Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
4.17Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
4.17Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
4.17Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
4.17Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
4.17Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
4.17Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
4.17Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
4.17Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
4.17Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
4.17Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
4.17Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
4.17Single9KDFRES-701-39KDF-ETB-RES-701-3
4.17Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
4.17Consensusglp_onOrthosteric Ligandglp1_on glp2_on
4.17Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
4.17Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
4.17Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
4.17Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
4.17Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
4.17Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
4.00Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
4.00Single6IGLIRL16206IGL-ETB-IRL1620
4.00Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
4.00Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
4.00Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
4.00Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
4.00Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
4.00Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
4.00Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
4.00Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
4.00Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
4.00Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
4.00Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
4.00Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
4.00Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
4.00Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
4.00Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
4.00Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
4.00Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
4.00Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
4.00Single8IY6Endothelin-18IY6-ETB-Endothelin-1
4.00Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
4.00Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
4.00Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
4.00Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
4.00Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
4.00Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
4.00Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
4.00Consensusbradykinin_onOrthosteric Ligandbk2_on
4.00Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
4.00Consensusendothelin_onOrthosteric Ligandetb_on eta_on
4.00Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
4.00Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
4.00Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
4.00Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
4.00Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
4.00Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
4.00Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
3.85Single5GLHEndothelin-15GLH-ETB-Endothelin-1
3.85Single6IGKEndothelin-36IGK-ETB-Endothelin-3
3.85Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
3.85Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
3.85Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
3.85Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
3.85Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
3.85Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
3.85Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
3.85Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
3.85Consensusbombesin_onOrthosteric Ligandbb2_on
3.85Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
3.85Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
3.85Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
3.85Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
3.85Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
3.85Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
3.85Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
3.85Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
3.85Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
3.70Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
3.70Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
3.70Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
3.70Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
3.70Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
3.70Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
3.70Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
3.70Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
3.70Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
3.70Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
3.70Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
3.70Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
3.70Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
3.57Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
3.57Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
3.57Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
3.57Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
3.57Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
3.57Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
3.57Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.57Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
3.57Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
3.57Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
3.45Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
3.45Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
3.45Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
3.45Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
3.45Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
3.45Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
3.45Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
3.45Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.45Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
3.45Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
3.33Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
3.33Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
3.33Consensuspth_onOrthosteric Ligandpth1_on pth2_on
3.23Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
3.23Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
3.12Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
3.12Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
3.03Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
2.94Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
2.94Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
2.78Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
2.70Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1

Consensus Members
Id Members
adgrg_on_gp adgrg2_on_gp
adgrg4_on_gp
adgrf_on_gp adgrf1_on_gp
adgrl_on_gp adgrl3_on_gp
adgre_on_gp adgre5_on_gp
adgrd_on_gp adgrd1_on_gp
Net Summary
Imin 3.08467
Number of Linked Nodes 918
Number of Links 1050
Number of Hubs 148
Number of Links mediated by Hubs 613
Number of Communities 20
Number of Nodes involved in Communities 183
Number of Links involved in Communities 246
Path Summary
Number Of Nodes in MetaPath 88
Number Of Links MetaPath 87
Number of Shortest Paths 2610833
Length Of Smallest Path 3
Average Path Length 31.2963
Length of Longest Path 58
Minimum Path Strength 0.256667
Average Path Strength 5.86588
Maximum Path Strength 23.0308
Minimum Path Correlation 0.701667
Average Path Correlation 0.968832
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 1.92308
Average % Of Corr. Nodes 32.5084
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 45.8388
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following differences:
Id1st Network2nd Network
class-b1_class-b2_diff_on_gpclass-b1_on_gpclass-b2_on_gp
This network is also present in following consensuses:
IdComponents
class-b1_class-b2_cons_on_gpclass-b1_on_gp
class-b2_on_gp



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