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Show: Click this button to access the corresponding database entry page.
PDB: PDB code of the receptor used to compute the network and a direct link to the corresponding entry in the Protein Data Bank.
Class: Receptor Class.
SubFamily: Receptor Sub Family.
Type: Receptor Type.
Subtype: Receptor SubType.
Species: Organism.
Orthosteric Ligand: Name of the orthosteric ligand, if present.
Other Ligand(s): Name of other allosteric ligands, if present.
Protein Partners: G Protein, Arrestin or Kinase coupled to a given receptor.
Resolution: Structure resolution.
Date: Deposition date.
DOI: DOI and link of the corresponding paper.
Show | PDB | Class | SubFamily | Type | SubType | Species | Orthosteric Ligand | Other Ligand(s) | Protein Partners | Resolution | Date | DOI |
---|---|---|---|---|---|---|---|---|---|---|---|---|
9L3Z | A | Protein | Chemerin | CML1 | Homo sapiens | LRH7-C2 | - | - | 3.9 | 2025-03-12 | doi.org/10.1093/procel/pwae073 | |
9L3W | A | Protein | Chemerin | CML1 | Homo sapiens | Retinoic acid receptor responder protein 2 | - | Gi1/β1/γ2 | 3.5 | 2025-03-12 | doi.org/10.1093/procel/pwae073 | |
9L3W (No Gprot) | A | Protein | Chemerin | CML1 | Homo sapiens | Retinoic acid receptor responder protein 2 | - | 3.5 | 2025-03-12 | doi.org/10.1093/procel/pwae073 | ||
9L3Y | A | Protein | Chemerin | CML2 | Homo sapiens | Retinoic acid receptor responder protein 2 | - | Gi1/β1/γ2 | 3.6 | 2025-03-12 | doi.org/10.1093/procel/pwae073 | |
9L3Y (No Gprot) | A | Protein | Chemerin | CML2 | Homo sapiens | Retinoic acid receptor responder protein 2 | - | 3.6 | 2025-03-12 | doi.org/10.1093/procel/pwae073 | ||
9EAJ | A | Peptide | Angiotensin | AT1 | Homo sapiens | - | Nanobody AT209 | - | 3.2 | 2025-03-05 | To be published | |
9EAH | A | Peptide | Angiotensin | AT1 | Homo sapiens | Olmesartan | Nanobody AT209 | - | 3.1 | 2025-03-05 | To be published | |
8YU7 | A | Protein | Chemokine | CXCR4 | Homo sapiens | - | - | - | 3.01 | 2025-03-05 | 10.1016/j.celrep.2025.115255 | |
8YU7 (Multimeric) | A | Protein | Chemokine | CXCR4 | Homo sapiens | - | - | 3.01 | 2025-03-05 | 10.1016/j.celrep.2025.115255 | ||
9B65 | A | Lipid | Cannabinoid | CB1 | Homo sapiens | KCA | - | Gi1/β1/γ2 | 3.03 | 2025-03-05 | 10.1038/s41586-025-08618-7 | |
9B65 (No Gprot) | A | Lipid | Cannabinoid | CB1 | Homo sapiens | KCA | - | 3.03 | 2025-03-05 | 10.1038/s41586-025-08618-7 | ||
9II3 | C | Aminoacid | Metabotropic Glutamate | mGlu3; mGlu3 | Homo sapiens | Glutamate | - | Arrestin2 | 3.9 | 2025-03-05 | doi.org/10.1038/s41589-025-01858-8 | |
9II2 | C | Aminoacid | Metabotropic Glutamate | mGlu3; mGlu3 | Homo sapiens | Glutamate | - | Arrestin2 | 3.7 | 2025-03-05 | doi.org/10.1038/s41589-025-01858-8 | |
9GE3 | A | Orphan | Orphan | GPR55 | Homo sapiens | Lysophosphatidylinositol | - | chim(CtGi1-G13)/β1/γ2 | 2.87 | 2025-03-05 | doi.org/10.1038/s41467-025-57204-y | |
9GE3 (No Gprot) | A | Orphan | Orphan | GPR55 | Homo sapiens | Lysophosphatidylinositol | - | 2.87 | 2025-03-05 | doi.org/10.1038/s41467-025-57204-y | ||
9GE2 | A | Orphan | Orphan | GPR55 | Homo sapiens | ML184 | Cholesterol | chim(CtGi1-G13)/β1/γ2 | 2.51 | 2025-03-05 | doi.org/10.1038/s41467-025-57204-y | |
9GE2 (No Gprot) | A | Orphan | Orphan | GPR55 | Homo sapiens | ML184 | Cholesterol | 2.51 | 2025-03-05 | doi.org/10.1038/s41467-025-57204-y | ||
9B54 | A | Lipid | Cannabinoid | CB1 | Homo sapiens | A1AIW | - | Gi1/β1/γ2 | 2.86 | 2025-03-05 | 10.1038/s41586-025-08618-7 | |
9B54 (No Gprot) | A | Lipid | Cannabinoid | CB1 | Homo sapiens | A1AIW | - | 2.86 | 2025-03-05 | 10.1038/s41586-025-08618-7 | ||
8ZFE | A | Orphan | Orphan | GPR4 | Mus musculus | - | - | - | 2.56 | 2025-02-26 | 10.1016/j.cell.2024.12.001 | |
8ZFD | A | Orphan | Orphan | GPR4 | Mus musculus | - | - | - | 2.56 | 2025-02-26 | 10.1016/j.cell.2024.12.001 | |
8ZFB | A | Orphan | Orphan | GPR4 | Xenopus tropicalis | - | - | - | 3.78 | 2025-02-26 | 10.1016/j.cell.2024.12.001 | |
8ZF7 | A | Orphan | Orphan | GPR4 | Xenopus tropicalis | - | - | - | 3.15 | 2025-02-26 | 10.1016/j.cell.2024.12.001 | |
9JVG | A | Orphan | Orphan | GPR4 | Mus musculus | - | - | chim(NtGi1-Gs)/β1/γ2 | 2.76 | 2025-02-26 | 10.1016/j.cell.2024.12.001 | |
9JVG (No Gprot) | A | Orphan | Orphan | GPR4 | Mus musculus | - | - | 2.76 | 2025-02-26 | 10.1016/j.cell.2024.12.001 | ||
8ZFC | A | Orphan | Orphan | GPR4 | Mus musculus | - | - | chim(NtGi1-Gs)/β1/γ2 | 2.68 | 2025-02-26 | 10.1016/j.cell.2024.12.001 | |
8ZFC (No Gprot) | A | Orphan | Orphan | GPR4 | Mus musculus | - | - | 2.68 | 2025-02-26 | 10.1016/j.cell.2024.12.001 | ||
8ZFA | A | Orphan | Orphan | GPR4 | Xenopus tropicalis | - | - | chim(NtGi1-Gs)/β1/γ2 | 2.96 | 2025-02-26 | 10.1016/j.cell.2024.12.001 | |
8ZFA (No Gprot) | A | Orphan | Orphan | GPR4 | Xenopus tropicalis | - | - | 2.96 | 2025-02-26 | 10.1016/j.cell.2024.12.001 | ||
8ZF9 | A | Orphan | Orphan | GPR4 | Mus musculus | - | - | chim(NtGi1-Gs)/β1/γ2 | 2.56 | 2025-02-26 | 10.1016/j.cell.2024.12.001 | |
8ZF9 (No Gprot) | A | Orphan | Orphan | GPR4 | Mus musculus | - | - | 2.56 | 2025-02-26 | 10.1016/j.cell.2024.12.001 | ||
8ZF6 | A | Orphan | Orphan | GPR4 | Xenopus tropicalis | - | - | chim(NtGi1-Gs)/β1/γ2 | 2.98 | 2025-02-26 | 10.1016/j.cell.2024.12.001 | |
8ZF6 (No Gprot) | A | Orphan | Orphan | GPR4 | Xenopus tropicalis | - | - | 2.98 | 2025-02-26 | 10.1016/j.cell.2024.12.001 | ||
8ZD1 | A | Orphan | Orphan | GPR4 | Xenopus tropicalis | - | - | chim(NtGi1-Gs)/β1/γ2 | 2.6 | 2025-02-26 | 10.1016/j.cell.2024.12.001 | |
8ZD1 (No Gprot) | A | Orphan | Orphan | GPR4 | Xenopus tropicalis | - | - | 2.6 | 2025-02-26 | 10.1016/j.cell.2024.12.001 | ||
8ZF4 | A | Orphan | Orphan | GPR4 | Xenopus tropicalis | - | - | - | 3.05 | 2025-02-26 | 10.1016/j.cell.2024.12.001 | |
9MQL | A | Peptide | Opioid | κ | Homo sapiens | Isoquinuclidine | - | - | 2.96 | 2025-02-12 | 10.1101/2025.01.09.632033 | |
9MQK | A | Peptide | Opioid | κ | Homo sapiens | Isoquinuclidine | - | - | 3.18 | 2025-02-12 | 10.1101/2025.01.09.632033 | |
9MQJ | A | Peptide | Opioid | μ | Homo sapiens | Isoquinuclidine | - | - | 3.23 | 2025-02-12 | 10.1101/2025.01.09.632033 | |
9MQI | A | Peptide | Opioid | μ | Homo sapiens | Isoquinuclidine | - | - | 3.3 | 2025-02-12 | 10.1101/2025.01.09.632033 | |
9MQH | A | Peptide | Opioid | μ | Homo sapiens | - | - | - | 3.9 | 2025-02-12 | 10.1101/2025.01.09.632033 | |
8Y51 | A | Peptide | Bombesin | BB3 | Homo sapiens | - | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.3 | 2025-02-12 | To be published | |
8Y51 (No Gprot) | A | Peptide | Bombesin | BB3 | Homo sapiens | - | - | 3.3 | 2025-02-12 | To be published | ||
9IV2 | B2 | Adhesion | Adhesion | ADGRD1 | Homo sapiens | 5α-DHT | - | chim(NtGi1-Gs)/β1/γ2 | 3.53 | 2025-02-12 | doi.org/10.1016/j.cell.2025.01.006 | |
9IV2 (No Gprot) | B2 | Adhesion | Adhesion | ADGRD1 | Homo sapiens | 5α-DHT | - | 3.53 | 2025-02-12 | doi.org/10.1016/j.cell.2025.01.006 | ||
9IV1 | B2 | Adhesion | Adhesion | ADGRD1 | Homo sapiens | 5α-DHT | - | chim(NtGi1-Gs)/β1/γ2 | 2.98 | 2025-02-12 | doi.org/10.1016/j.cell.2025.01.006 | |
9IV1 (No Gprot) | B2 | Adhesion | Adhesion | ADGRD1 | Homo sapiens | 5α-DHT | - | 2.98 | 2025-02-12 | doi.org/10.1016/j.cell.2025.01.006 | ||
8X9U | B2 | Adhesion | Adhesion | ADGRD1 | Homo sapiens | Metenolone | - | chim(NtGi1-Gs)/β1/γ2 | 2.88 | 2025-02-12 | doi.org/10.1016/j.cell.2025.01.006 | |
8X9U (No Gprot) | B2 | Adhesion | Adhesion | ADGRD1 | Homo sapiens | Metenolone | - | 2.88 | 2025-02-12 | doi.org/10.1016/j.cell.2025.01.006 | ||
8X9T | B2 | Adhesion | Adhesion | ADGRD1 | Homo sapiens | AP503 | - | chim(NtGi1-Gs)/β1/γ2 | 2.75 | 2025-02-12 | doi.org/10.1016/j.cell.2025.01.006 | |
8X9T (No Gprot) | B2 | Adhesion | Adhesion | ADGRD1 | Homo sapiens | AP503 | - | 2.75 | 2025-02-12 | doi.org/10.1016/j.cell.2025.01.006 | ||
8X9S | B2 | Adhesion | Adhesion | ADGRD1 | Homo sapiens | 5α-DHT | - | chim(NtGi1-Gs)/β1/γ2 | 3.49 | 2025-02-12 | doi.org/10.1016/j.cell.2025.01.006 | |
8X9S (No Gprot) | B2 | Adhesion | Adhesion | ADGRD1 | Homo sapiens | 5α-DHT | - | 3.49 | 2025-02-12 | doi.org/10.1016/j.cell.2025.01.006 | ||
8Y01 | A | Sensory | Opsins | Opsin1MW | Homo sapiens | Retinal | - | Gi1/β1/γ2 | 2.48 | 2025-02-12 | To be published | |
8Y01 (No Gprot) | A | Sensory | Opsins | Opsin1MW | Homo sapiens | Retinal | - | 2.48 | 2025-02-12 | To be published | ||
8YJP | C | Orphan | Orphan | GPR156 | Homo sapiens | - | - | - | 3.09 | 2025-02-05 | doi.org/10.1038/s41467-024-54681-5 | |
8Y63 | A | Peptide | Formylpeptide | FPR2-ALX | Homo sapiens | C20:0 Ceramide | - | Gi1/β1/γ2 | 3.2 | 2025-02-05 | To be published | |
8Y63 (No Gprot) | A | Peptide | Formylpeptide | FPR2-ALX | Homo sapiens | C20:0 Ceramide | - | 3.2 | 2025-02-05 | To be published | ||
8Y62 | A | Peptide | Formylpeptide | FPR2-ALX | Homo sapiens | C16:0 Ceramide | - | Gi1/β1/γ2 | 3.2 | 2025-02-05 | To be published | |
8Y62 (No Gprot) | A | Peptide | Formylpeptide | FPR2-ALX | Homo sapiens | C16:0 Ceramide | - | 3.2 | 2025-02-05 | To be published | ||
8YK0 | C | Orphan | Orphan | GPR156 | Homo sapiens | - | - | Gi3/β1/γ2 | 2.4 | 2025-02-05 | doi.org/10.1038/s41467-024-54681-5 | |
8YK0 (No Gprot) | C | Orphan | Orphan | GPR156 | Homo sapiens | - | - | 2.4 | 2025-02-05 | doi.org/10.1038/s41467-024-54681-5 | ||
9K27 | A | Peptide | Prolactin-releasing peptide | PrRP | Homo sapiens | PrRP31 | - | chim(NtGi1-Gq)/β1/γ2 | 2.68 | 2025-01-29 | To be published | |
9K27 (No Gprot) | A | Peptide | Prolactin-releasing peptide | PrRP | Homo sapiens | PrRP31 | - | 2.68 | 2025-01-29 | To be published | ||
9K26 | A | Peptide | Prolactin-releasing peptide | PrRP | Homo sapiens | PrRP31 | - | Gi1/β1/γ2 | 3 | 2025-01-29 | To be published | |
9K26 (No Gprot) | A | Peptide | Prolactin-releasing peptide | PrRP | Homo sapiens | PrRP31 | - | 3 | 2025-01-29 | To be published | ||
9FUP | A | Nucleotide | Adenosine | A2A | Homo sapiens | Istradefylline | Na | - | 2.5 | 2025-01-22 | doi.org/10.1038/s42004-024-01404-y | |
8Z74 | A | Peptide | Apelin | Apelin | Homo sapiens | Agonistic antibody | - | - | 3.01 | 2025-01-22 | 10.1038/s41467-024-55555-6 | |
8XQJ | A | Peptide | Apelin | Apelin | Homo sapiens | JN241 | - | - | 2.95 | 2025-01-22 | doi.org/10.1038/s41467-024-55555-6 | |
8XQI | A | Peptide | Apelin | Apelin | Homo sapiens | - | - | - | 3.25 | 2025-01-22 | doi.org/10.1038/s41467-024-55555-6 | |
9BI6 | A | Orphan | Orphan | GPR68 | Homo sapiens | - | - | chim(Gs-CtGq)/β1/γ2 | 2.9 | 2025-01-22 | doi.org/10.1016/j.cell.2024.11.036 | |
9BI6 (No Gprot) | A | Orphan | Orphan | GPR68 | Homo sapiens | - | - | 2.9 | 2025-01-22 | doi.org/10.1016/j.cell.2024.11.036 | ||
8JSR | A | Peptide | Ghrelin | Ghrelin | Homo sapiens | Anamorelin | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.9 | 2025-01-22 | doi.org/10.1038/s41594-024-01481-6 | |
8JSR (No Gprot) | A | Peptide | Ghrelin | Ghrelin | Homo sapiens | Anamorelin | - | 2.9 | 2025-01-22 | doi.org/10.1038/s41594-024-01481-6 | ||
9J31 | A | Orphan | Orphan | GPR4 | Danio rerio | - | - | chim(NtGi1-Gs)/β1/γ2 | 3.05 | 2025-01-22 | doi.org/10.1038/s41467-025-55901-2 | |
9J31 (No Gprot) | A | Orphan | Orphan | GPR4 | Danio rerio | - | - | 3.05 | 2025-01-22 | doi.org/10.1038/s41467-025-55901-2 | ||
8ZFZ | A | Orphan | Orphan | GPR4 | Danio rerio | - | - | chim(NtGi1-Gs)/β1/γ2 | 3.3 | 2025-01-22 | doi.org/10.1038/s41467-025-55901-2 | |
8ZFZ (No Gprot) | A | Orphan | Orphan | GPR4 | Danio rerio | - | - | 3.3 | 2025-01-22 | doi.org/10.1038/s41467-025-55901-2 | ||
8Z7J | A | Peptide | Apelin | Apelin | Homo sapiens | Agonistic antibody | - | Gi1/β1/γ2 | 3.12 | 2025-01-22 | 10.1038/s41467-024-55555-6 | |
8Z7J (No Gprot) | A | Peptide | Apelin | Apelin | Homo sapiens | Agonistic antibody | - | 3.12 | 2025-01-22 | 10.1038/s41467-024-55555-6 | ||
8XQF | A | Peptide | Apelin | Apelin | Homo sapiens | Apelin-13 | - | Gi1/β1/γ2 | 3.13 | 2025-01-22 | doi.org/10.1038/s41467-024-55555-6 | |
8XQF (No Gprot) | A | Peptide | Apelin | Apelin | Homo sapiens | Apelin-13 | - | 3.13 | 2025-01-22 | doi.org/10.1038/s41467-024-55555-6 | ||
8XQE | A | Peptide | Apelin | Apelin | Homo sapiens | Apelin-13 | - | Gi1/β1/γ2 | 3.48 | 2025-01-22 | doi.org/10.1038/s41467-024-55555-6 | |
8XQE (No Gprot) | A | Peptide | Apelin | Apelin | Homo sapiens | Apelin-13 | - | 3.48 | 2025-01-22 | doi.org/10.1038/s41467-024-55555-6 | ||
8ZJG | A | Protein | Chemerin | CML1 | Homo sapiens | Chemerin | - | Gi1/β1/γ2 | 3.18 | 2025-01-22 | doi.org/10.1038/s42003-024-07228-9 | |
8ZJG (No Gprot) | A | Protein | Chemerin | CML1 | Homo sapiens | Chemerin | - | 3.18 | 2025-01-22 | doi.org/10.1038/s42003-024-07228-9 | ||
9BHL | A | Orphan | Orphan | GPR65 | Homo sapiens | - | - | Gs/β1 | 2.8 | 2025-01-22 | doi.org/10.1016/j.cell.2024.11.036 | |
9BHL (No Gprot) | A | Orphan | Orphan | GPR65 | Homo sapiens | - | - | 2.8 | 2025-01-22 | doi.org/10.1016/j.cell.2024.11.036 | ||
9BHM | A | Orphan | Orphan | GPR68 | Homo sapiens | - | - | Gs/β1 | 2.9 | 2025-01-22 | doi.org/10.1016/j.cell.2024.11.036 | |
9BHM (No Gprot) | A | Orphan | Orphan | GPR68 | Homo sapiens | - | - | 2.9 | 2025-01-22 | doi.org/10.1016/j.cell.2024.11.036 | ||
9BIP | A | Orphan | Orphan | GPR4 | Homo sapiens | - | - | Gs/β1/γ2 | 2.8 | 2025-01-22 | doi.org/10.1016/j.cell.2024.11.036 | |
9BIP (No Gprot) | A | Orphan | Orphan | GPR4 | Homo sapiens | - | - | 2.8 | 2025-01-22 | doi.org/10.1016/j.cell.2024.11.036 | ||
8XWS | A | Protein | Chemokine | CXCR2 | Homo sapiens | CXCL5 | - | - | 3.06 | 2025-01-15 | To be published | |
8XWN | A | Protein | Chemokine | CXCR2 | Homo sapiens | CXCL8 | - | - | 3.29 | 2025-01-15 | To be published | |
8XWM | A | Protein | Chemokine | CXCR2 | Homo sapiens | CXCL6 | - | - | 3.71 | 2025-01-15 | To be published | |
8XWF | A | Protein | Chemokine | CXCR2 | Homo sapiens | CXCL3 | - | - | 3.65 | 2025-01-15 | To be published | |
8XWA | A | Protein | Chemokine | CXCR2 | Homo sapiens | CXCL1 | - | - | 3.48 | 2025-01-15 | To be published | |
8XVU | A | Protein | Chemokine | CXCR2 | Homo sapiens | CXCL2 | - | - | 3.09 | 2025-01-15 | To be published | |
8XUM | A | Orphan | Orphan | LGR4 | Homo sapiens | R-spondin-2 | - | - | 2.9 | 2025-01-15 | To be published | |
8XT9 | A | Orphan | Orphan | LGR4 | Homo sapiens | - | - | - | 3.1 | 2025-01-15 | To be published | |
9ITB | A | Lipid | Lysophospholipid | LPA6 | Homo sapiens | LPA | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.89 | 2025-01-15 | doi.org/10.1073/pnas.2415426122 | |
9ITB (No Gprot) | A | Lipid | Lysophospholipid | LPA6 | Homo sapiens | LPA | - | 2.89 | 2025-01-15 | doi.org/10.1073/pnas.2415426122 | ||
9ITE | A | Lipid | Lysophospholipid | LPA6 | Homo sapiens | LPA | - | chim(NtGi2-G13)/β1/γ2 | 3.06 | 2025-01-15 | doi.org/10.1073/pnas.2415426122 | |
9ITE (No Gprot) | A | Lipid | Lysophospholipid | LPA6 | Homo sapiens | LPA | - | 3.06 | 2025-01-15 | doi.org/10.1073/pnas.2415426122 | ||
9D61 | A | Peptide | Opioid | κ | Homo sapiens | JDTic | - | Gi1/β1/γ2 | 3.58 | 2025-01-15 | doi.org/10.1038/s41589-024-01812-0 | |
9D61 (No Gprot) | A | Peptide | Opioid | κ | Homo sapiens | JDTic | - | 3.58 | 2025-01-15 | doi.org/10.1038/s41589-024-01812-0 | ||
8VVG | A | Peptide | Opioid | κ | Homo sapiens | GB18 | - | Gi1/β1/γ2 | 3.3 | 2025-01-15 | doi.org/10.1038/s41589-024-01812-0 | |
8VVG (No Gprot) | A | Peptide | Opioid | κ | Homo sapiens | GB18 | - | 3.3 | 2025-01-15 | doi.org/10.1038/s41589-024-01812-0 | ||
8VVF | A | Peptide | Opioid | κ | Homo sapiens | JDTic | - | Gi1/β1/γ2 | 3 | 2025-01-15 | doi.org/10.1038/s41589-024-01812-0 | |
8VVF (No Gprot) | A | Peptide | Opioid | κ | Homo sapiens | JDTic | - | 3 | 2025-01-15 | doi.org/10.1038/s41589-024-01812-0 | ||
8VVE | A | Peptide | Opioid | κ | Homo sapiens | norBNI | - | Gi1/β1/γ2 | 3.3 | 2025-01-15 | doi.org/10.1038/s41589-024-01812-0 | |
8VVE (No Gprot) | A | Peptide | Opioid | κ | Homo sapiens | norBNI | - | 3.3 | 2025-01-15 | doi.org/10.1038/s41589-024-01812-0 | ||
8JZP | A | Peptide | Complement Peptide | C5a1 | Homo sapiens | C5A anaphylatoxin | - | Go/β1/γ2 | 3.54 | 2025-01-15 | To be published | |
8JZP (No Gprot) | A | Peptide | Complement Peptide | C5a1 | Homo sapiens | C5A anaphylatoxin | - | 3.54 | 2025-01-15 | To be published | ||
8XXX | A | Protein | Chemokine | CXCR2 | Homo sapiens | CXCL6 | - | Go/β1/γ2 | 3.17 | 2025-01-15 | To be published | |
8XXX (No Gprot) | A | Protein | Chemokine | CXCR2 | Homo sapiens | CXCL6 | - | 3.17 | 2025-01-15 | To be published | ||
8XXR | A | Protein | Chemokine | CXCR2 | Homo sapiens | - | - | Go/β1/γ2 | 3.17 | 2025-01-15 | To be published | |
8XXR (No Gprot) | A | Protein | Chemokine | CXCR2 | Homo sapiens | - | - | 3.17 | 2025-01-15 | To be published | ||
8XXH | A | Protein | Chemokine | CXCR2 | Homo sapiens | CXCL2 | - | Go/β1/γ2 | 2.8 | 2025-01-15 | To be published | |
8XXH (No Gprot) | A | Protein | Chemokine | CXCR2 | Homo sapiens | CXCL2 | - | 2.8 | 2025-01-15 | To be published | ||
8XX7 | A | Protein | Chemokine | CXCR2 | Homo sapiens | CXCL5 | - | Go/β1/γ2 | 3.32 | 2025-01-15 | To be published | |
8XX7 (No Gprot) | A | Protein | Chemokine | CXCR2 | Homo sapiens | CXCL5 | - | 3.32 | 2025-01-15 | To be published | ||
8XX6 | A | Protein | Chemokine | CXCR2 | Homo sapiens | CXCL8 | - | Go/β1/γ2 | 2.99 | 2025-01-15 | To be published | |
8XX6 (No Gprot) | A | Protein | Chemokine | CXCR2 | Homo sapiens | CXCL8 | - | 2.99 | 2025-01-15 | To be published | ||
8XX3 | A | Protein | Chemokine | CXCR2 | Homo sapiens | CXCL3 | - | Go/β1/γ2 | 3.38 | 2025-01-15 | To be published | |
8XX3 (No Gprot) | A | Protein | Chemokine | CXCR2 | Homo sapiens | CXCL3 | - | 3.38 | 2025-01-15 | To be published | ||
8XWV | A | Protein | Chemokine | CXCR2 | Homo sapiens | CXCL1 | - | Go/β1/γ2 | 3.07 | 2025-01-15 | To be published | |
8XWV (No Gprot) | A | Protein | Chemokine | CXCR2 | Homo sapiens | CXCL1 | - | 3.07 | 2025-01-15 | To be published | ||
8RWX | A | Nucleotide | Adenosine | A2A | Homo sapiens | StilSwitch3 | Na | - | 3.05 | 2025-01-08 | doi.org/10.1038/s41467-024-55109-w | |
8RWI | A | Nucleotide | Adenosine | A2A | Homo sapiens | StilSwitch2 | Na | - | 2.8 | 2025-01-08 | doi.org/10.1038/s41467-024-55109-w | |
8RWH | A | Nucleotide | Adenosine | A2A | Homo sapiens | StilSwitch2 | Na | - | 2.45 | 2025-01-08 | doi.org/10.1038/s41467-024-55109-w | |
8RWE | A | Nucleotide | Adenosine | A2A | Homo sapiens | StilSwitch4 | Na | - | 2.2 | 2025-01-08 | doi.org/10.1038/s41467-024-55109-w | |
8RWD | A | Nucleotide | Adenosine | A2A | Homo sapiens | StilSwitch3 | Na | - | 2.05 | 2025-01-08 | doi.org/10.1038/s41467-024-55109-w | |
8RWC | A | Nucleotide | Adenosine | A2A | Homo sapiens | StilSwitch2 | Na | - | 2.31 | 2025-01-08 | doi.org/10.1038/s41467-024-55109-w | |
8RW7 | A | Nucleotide | Adenosine | A2A | Homo sapiens | StilSwitch1 | Na | - | 2.25 | 2025-01-08 | doi.org/10.1038/s41467-024-55109-w | |
8RW4 | A | Nucleotide | Adenosine | A2A | Homo sapiens | AzoSwitch2 | Na | - | 2.2 | 2025-01-08 | doi.org/10.1038/s41467-024-55109-w | |
8RW0 | A | Nucleotide | Adenosine | A2A | Homo sapiens | Istradefylline | Na | - | 1.94 | 2025-01-08 | 10.1038/s41467-024-55109-w | |
8RVW | A | Nucleotide | Adenosine | A2A | Homo sapiens | StilSwitch3 | Na | - | 2.65 | 2025-01-08 | doi.org/10.1038/s41467-024-55109-w | |
9IZG | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | NKP | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.04 | 2025-01-01 | 10.1016/j.jsb.2024.108164 | |
9IZG (No Gprot) | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | NKP | - | 3.04 | 2025-01-01 | 10.1016/j.jsb.2024.108164 | ||
9IY8 | A | Orphan | Orphan | GPR55 | Homo sapiens | - | - | chim(NtGi1-G13)/β1/γ2 | 3.01 | 2025-01-01 | doi.org/10.1038/s41422-024-01046-8 | |
9IY8 (No Gprot) | A | Orphan | Orphan | GPR55 | Homo sapiens | - | - | 3.01 | 2025-01-01 | doi.org/10.1038/s41422-024-01046-8 | ||
9IZH | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | LPA | - | chim(NtGi2-G13)/β1/γ2 | 3.04 | 2025-01-01 | doi.org/10.1016/j.jsb.2024.108164 | |
9IZH (No Gprot) | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | LPA | - | 3.04 | 2025-01-01 | doi.org/10.1016/j.jsb.2024.108164 | ||
8XML | A | Protein | Chemokine | CCR8 | Homo sapiens | - | - | Gi1/β1/γ2 | 2.58 | 2025-01-01 | To be published | |
8XML (No Gprot) | A | Protein | Chemokine | CCR8 | Homo sapiens | - | - | 2.58 | 2025-01-01 | To be published | ||
8UGW | A | Nucleotide | Adenosine | A2A | Homo sapiens | PubChem 3086599 | - | - | 3.9 | 2024-12-18 | doi.org/10.1038/s41557-024-01719-2 | |
8JEF | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA3 | Homo sapiens | (3S)-3-hydroxyoctanoic acid | - | Gi1/β1/γ2 | 2.96 | 2024-12-18 | doi.org/10.1016/j.celrep.2024.114895 | |
8JEF (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA3 | Homo sapiens | (3S)-3-hydroxyoctanoic acid | - | 2.96 | 2024-12-18 | doi.org/10.1016/j.celrep.2024.114895 | ||
9DQJ | A | Orphan | Orphan | MRGPRD | Homo sapiens | EP-3945 | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.9 | 2024-12-11 | 10.1016/j.celrep.2024.114942 | |
9DQJ (No Gprot) | A | Orphan | Orphan | MRGPRD | Homo sapiens | EP-3945 | - | 2.9 | 2024-12-11 | 10.1016/j.celrep.2024.114942 | ||
9DQH | A | Orphan | Orphan | MRGPRD | Homo sapiens | EP-2825 | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.92 | 2024-12-11 | 10.1016/j.celrep.2024.114942 | |
9DQH (No Gprot) | A | Orphan | Orphan | MRGPRD | Homo sapiens | EP-2825 | - | 2.92 | 2024-12-11 | 10.1016/j.celrep.2024.114942 | ||
9K1C | A | Lipid | Free Fatty Acid | FFA1 | Homo sapiens | - | DHA | Gi1/β1/γ2 | 3.2 | 2024-12-11 | 10.1016/j.celrep.2024.115024 | |
9K1C (No Gprot) | A | Lipid | Free Fatty Acid | FFA1 | Homo sapiens | - | DHA | 3.2 | 2024-12-11 | 10.1016/j.celrep.2024.115024 | ||
9K1D | A | Lipid | Free Fatty Acid | FFA2 | Homo sapiens | Butanoic acid | Cholesterol | Gi1/β1/γ2 | 3.34 | 2024-12-11 | 10.1016/j.celrep.2024.115024 | |
9K1D (No Gprot) | A | Lipid | Free Fatty Acid | FFA2 | Homo sapiens | Butanoic acid | Cholesterol | 3.34 | 2024-12-11 | 10.1016/j.celrep.2024.115024 | ||
9AST | A | Protein | Chemokine | XCR1 | Homo sapiens | Lymphotactin | - | Gi1/β1/γ2 | 3.07 | 2024-12-11 | 10.1073/pnas.2405732121 | |
9AST (No Gprot) | A | Protein | Chemokine | XCR1 | Homo sapiens | Lymphotactin | - | 3.07 | 2024-12-11 | 10.1073/pnas.2405732121 | ||
8YIC | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | SAR247799 | - | Gi1/β1/γ2 | 3.47 | 2024-12-11 | To be published | |
8YIC (No Gprot) | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | SAR247799 | - | 3.47 | 2024-12-11 | To be published | ||
9IYB | A | Lipid | Prostanoid | DP2 | Homo sapiens | Prostaglandin | A1D5Q | Gi1/β1/γ2 | 2.82 | 2024-12-04 | 10.1073/pnas.2403304121 | |
9IYB (No Gprot) | A | Lipid | Prostanoid | DP2 | Homo sapiens | Prostaglandin | A1D5Q | 2.82 | 2024-12-04 | 10.1073/pnas.2403304121 | ||
8S4D | A | Peptide | Apelin | Apelin | Homo sapiens | CMF-019 | - | - | 2.58 | 2024-12-04 | doi.org/10.1038/s41467-024-55381-w | |
8TF5 | A | Orphan | Orphan | GPR6 | Homo sapiens | Oleic acid | - | - | 2.1 | 2024-12-04 | 10.2210/pdb8TF5/pdb | |
8T1W | A | Orphan | Orphan | GPR6 | Homo sapiens | CVN424 | - | - | 3.49 | 2024-12-04 | 10.1126/scisignal.ado8741 | |
8T1V | A | Orphan | Orphan | GPR6 | Homo sapiens | PubChem 118310209 | Na | - | 2.6 | 2024-12-04 | 10.1126/scisignal.ado8741 | |
8XXV | A | Lipid | Prostanoid | DP2 | Homo sapiens | Indomethacin | A1D5Q | Gi1/β1/γ2 | 2.33 | 2024-12-04 | doi.org/10.1073/pnas.2403304121 | |
8XXV (No Gprot) | A | Lipid | Prostanoid | DP2 | Homo sapiens | Indomethacin | A1D5Q | 2.33 | 2024-12-04 | doi.org/10.1073/pnas.2403304121 | ||
8XXU | A | Lipid | Prostanoid | DP2 | Homo sapiens | - | A1D5Q | Gi1/β1/γ2 | 2.54 | 2024-12-04 | doi.org/10.1073/pnas.2403304121 | |
8XXU (No Gprot) | A | Lipid | Prostanoid | DP2 | Homo sapiens | - | A1D5Q | 2.54 | 2024-12-04 | doi.org/10.1073/pnas.2403304121 | ||
8TYW | A | Orphan | Orphan | GPR6 | Homo sapiens | - | - | Gs/β1/γ2 | 3.43 | 2024-12-04 | 10.2210/pdb8TF5/pdb | |
8TYW (No Gprot) | A | Orphan | Orphan | GPR6 | Homo sapiens | - | - | 3.43 | 2024-12-04 | 10.2210/pdb8TF5/pdb | ||
8Y69 | A | Orphan | Orphan | LGR4 | Homo sapiens | R-spondin-2 | Cholesterol | ZNRF3 | 3.38 | 2024-12-04 | To be published | |
8XFT | A | Orphan | Orphan | LGR4 | Homo sapiens | R-spondin-2 | - | ZNRF3 | 3.24 | 2024-12-04 | To be published | |
8XFS | A | Orphan | Orphan | LGR4 | Homo sapiens | R-spondin-2 | - | ZNRF3 | 3.2 | 2024-12-04 | To be published | |
8XFP | A | Orphan | Orphan | LGR4 | Homo sapiens | R-spondin-2 | - | ZNRF3 | 3.21 | 2024-12-04 | To be published | |
8RQL | T2 | Sensory | Taste2 | TAS2R14 | Homo sapiens | Flufenamic acid | Flufenamic acid | chim(NtGi1-Gt3)/β1/γ2 | 3.03 | 2024-11-27 | 10.1038/s41467-024-54157-6 | |
8RQL (No Gprot) | T2 | Sensory | Taste2 | TAS2R14 | Homo sapiens | Flufenamic acid | Flufenamic acid | 3.03 | 2024-11-27 | 10.1038/s41467-024-54157-6 | ||
9J5V | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | CpY | - | Gi1/β1/γ2 | 2.86 | 2024-11-27 | 10.1038/s42003-024-07152-y | |
9J5V (No Gprot) | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | CpY | - | 2.86 | 2024-11-27 | 10.1038/s42003-024-07152-y | ||
8WGD | C | Aminoacid | Metabotropic Glutamate | mGlu4; mGlu2 | Homo sapiens | WAG/WA6 | - | - | 4.45 | 2024-11-27 | To be published | |
8WGC | C | Aminoacid | Metabotropic Glutamate | mGlu4; mGlu2 | Homo sapiens | LY379268 | - | - | 5.95 | 2024-11-27 | To be published | |
8WG9 | C | Aminoacid | Metabotropic Glutamate | mGlu4; mGlu2 | Homo sapiens | (2S)-2-amino-4-phosphonobutanoic acid | - | - | 4.46 | 2024-11-27 | To be published | |
8Y45 | A | Peptide | Opioid | δ | Homo sapiens | ADL5859 | - | Gi2/β1/γ2 | 3.45 | 2024-11-27 | doi.org/10.1038/s41467-024-52601-1 | |
8Y45 (No Gprot) | A | Peptide | Opioid | δ | Homo sapiens | ADL5859 | - | 3.45 | 2024-11-27 | doi.org/10.1038/s41467-024-52601-1 | ||
9BA0 | A | Lipid | Cannabinoid | CB1 | Homo sapiens | A1AKN | - | - | 3.13 | 2024-11-20 | 10.1038/s41467-024-54206-0 | |
9B9Z | A | Lipid | Cannabinoid | CB1 | Homo sapiens | A1AKO | - | - | 3.3 | 2024-11-20 | 10.1038/s41467-024-54206-0 | |
8JEI | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCAR3 | Homo sapiens | 3-nitro-4-(propylamino)benzoic acid | - | Gi1/β1/γ2 | 2.73 | 2024-11-20 | 10.2210/pdb8JEI/pdb | |
8JEI (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCAR3 | Homo sapiens | 3-nitro-4-(propylamino)benzoic acid | - | 2.73 | 2024-11-20 | 10.2210/pdb8JEI/pdb | ||
9B9Y | A | Lipid | Cannabinoid | CB1 | Homo sapiens | 7DY | - | - | 3.5 | 2024-11-20 | 10.1038/s41467-024-54206-0 | |
8X3L | A | Lipid | Cannabinoid | CB2 | Homo sapiens | XWD | - | Gi1/β1/γ2 | 3.13 | 2024-11-20 | To be published | |
8X3L (No Gprot) | A | Lipid | Cannabinoid | CB2 | Homo sapiens | XWD | - | 3.13 | 2024-11-20 | To be published | ||
8P15 | A | Sensory | Opsin | Rhodopsin | Bos taurus | - | - | Gi1/β1/γT1 | 5.9 | 2024-11-20 | To be published | |
8P15 (No Gprot) | A | Sensory | Opsin | Rhodopsin | Bos taurus | - | - | 5.9 | 2024-11-20 | To be published | ||
8P13 | A | Sensory | Opsin | Rhodopsin | Bos taurus | - | - | Gi1/β1/γT1 | 5.2 | 2024-11-20 | To be published | |
8P13 (No Gprot) | A | Sensory | Opsin | Rhodopsin | Bos taurus | - | - | 5.2 | 2024-11-20 | To be published | ||
8P12 | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | - | Gi1/β1/γT1 | 3.21 | 2024-11-20 | To be published | |
8P12 (No Gprot) | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | - | 3.21 | 2024-11-20 | To be published | ||
9CHV | A | Amine | Adrenergic | β2 | Homo sapiens | - | - | - | 3.95 | 2024-11-13 | 10.1073/pnas.2414544121 | |
9CHU | A | Amine | Adrenergic | β2 | Homo sapiens | Noradrenaline | - | - | 3.49 | 2024-11-13 | 10.1073/pnas.2414544121 | |
9IVM | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | GLP-1 (Truncated) | LSN3318839 | chim(NtGi1-Gs)/β2/γ2 | 3.22 | 2024-11-13 | 10.1016/j.apsb.2024.09.002 | |
9IVM (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | GLP-1 (Truncated) | LSN3318839 | 3.22 | 2024-11-13 | 10.1016/j.apsb.2024.09.002 | ||
9CHX | A | Amine | Adrenergic | β2 | Homo sapiens | S-Carazolol | - | - | 3.5 | 2024-11-13 | 10.1073/pnas.2414544121 | |
8WWN | A | Peptide | Melanin Concentrating Hormone | MCH1 | Homo sapiens | MCH | - | Gi1/β1/γ2 | 2.65 | 2024-11-13 | To be published | |
8WWN (No Gprot) | A | Peptide | Melanin Concentrating Hormone | MCH1 | Homo sapiens | MCH | - | 2.65 | 2024-11-13 | To be published | ||
8WWM | A | Peptide | Melanin Concentrating Hormone | MCH1 | Homo sapiens | MCH | - | Gi1/β1/γ2 | 2.81 | 2024-11-13 | To be published | |
8WWM (No Gprot) | A | Peptide | Melanin Concentrating Hormone | MCH1 | Homo sapiens | MCH | - | 2.81 | 2024-11-13 | To be published | ||
8WWL | A | Peptide | Melanin Concentrating Hormone | MCH1 | Homo sapiens | MCH | - | Gi1/β1/γ2 | 2.78 | 2024-11-13 | To be published | |
8WWL (No Gprot) | A | Peptide | Melanin Concentrating Hormone | MCH1 | Homo sapiens | MCH | - | 2.78 | 2024-11-13 | To be published | ||
8WWK | A | Peptide | Melanin Concentrating Hormone | MCH1 | Homo sapiens | MCH | - | Gi1/β1/γ2 | 2.61 | 2024-11-13 | To be published | |
8WWK (No Gprot) | A | Peptide | Melanin Concentrating Hormone | MCH1 | Homo sapiens | MCH | - | 2.61 | 2024-11-13 | To be published | ||
8WWJ | A | Peptide | Melanin Concentrating Hormone | MCH1 | Homo sapiens | - | - | Gi1/β1/γ2 | 3.03 | 2024-11-13 | To be published | |
8WWJ (No Gprot) | A | Peptide | Melanin Concentrating Hormone | MCH1 | Homo sapiens | - | - | 3.03 | 2024-11-13 | To be published | ||
8WWI | A | Peptide | Melanin Concentrating Hormone | MCH1 | Homo sapiens | - | - | Gi1/β1/γ2 | 3.43 | 2024-11-13 | To be published | |
8WWI (No Gprot) | A | Peptide | Melanin Concentrating Hormone | MCH1 | Homo sapiens | - | - | 3.43 | 2024-11-13 | To be published | ||
8WWH | A | Peptide | Melanin Concentrating Hormone | MCH1 | Homo sapiens | - | - | Gi1/β1/γ2 | 2.84 | 2024-11-13 | To be published | |
8WWH (No Gprot) | A | Peptide | Melanin Concentrating Hormone | MCH1 | Homo sapiens | - | - | 2.84 | 2024-11-13 | To be published | ||
8XYD | A | Lipid | Platelet Activating Factor | PAF | Homo sapiens | Platelet Activating Factor | - | Gi1/β1/γ2 | 2.9 | 2024-11-13 | 10.1016/j.celrep.2024.114422 | |
8XYD (No Gprot) | A | Lipid | Platelet Activating Factor | PAF | Homo sapiens | Platelet Activating Factor | - | 2.9 | 2024-11-13 | 10.1016/j.celrep.2024.114422 | ||
8YH6 | A | Nucleotide | Adenosine | A3A | Homo sapiens | Namodenoson | - | Gi1/β1/γ2 | 3.62 | 2024-11-06 | doi.org/10.1038/s41467-024-53473-1 | |
8YH6 (No Gprot) | A | Nucleotide | Adenosine | A3A | Homo sapiens | Namodenoson | - | 3.62 | 2024-11-06 | doi.org/10.1038/s41467-024-53473-1 | ||
8YH5 | A | Nucleotide | Adenosine | A3A | Homo sapiens | Riboprine | - | Gi1/β1/γ2 | 3.66 | 2024-11-06 | doi.org/10.1038/s41467-024-53473-1 | |
8YH5 (No Gprot) | A | Nucleotide | Adenosine | A3A | Homo sapiens | Riboprine | - | 3.66 | 2024-11-06 | doi.org/10.1038/s41467-024-53473-1 | ||
8YH3 | A | Nucleotide | Adenosine | A3A | Homo sapiens | N-methyladenosine | - | Gi1/β1/γ2 | 3.4 | 2024-11-06 | doi.org/10.1038/s41467-024-53473-1 | |
8YH3 (No Gprot) | A | Nucleotide | Adenosine | A3A | Homo sapiens | N-methyladenosine | - | 3.4 | 2024-11-06 | doi.org/10.1038/s41467-024-53473-1 | ||
8YH2 | A | Nucleotide | Adenosine | A3A | Homo sapiens | Adenosine | - | Gi1/β1/γ2 | 3.27 | 2024-11-06 | doi.org/10.1038/s41467-024-53473-1 | |
8YH2 (No Gprot) | A | Nucleotide | Adenosine | A3A | Homo sapiens | Adenosine | - | 3.27 | 2024-11-06 | doi.org/10.1038/s41467-024-53473-1 | ||
8KEX | A | Orphan | Orphan | MRGPRX4 | Homo sapiens | DCA-3P | - | - | 3.2 | 2024-11-06 | doi.org/10.1016/j.cell.2024.10.001 | |
8K4S | A | Orphan | Orphan | MRGPRX4 | Homo sapiens | DCA-3P | - | chim(NtGi1L-Gs-CtGq)/β1/γ2 | 2.9 | 2024-11-06 | doi.org/10.1016/j.cell.2024.10.001 | |
8K4S (No Gprot) | A | Orphan | Orphan | MRGPRX4 | Homo sapiens | DCA-3P | - | 2.9 | 2024-11-06 | doi.org/10.1016/j.cell.2024.10.001 | ||
8YH0 | A | Nucleotide | Adenosine | A3A | Homo sapiens | NECA | - | Gi1/β1/γ2 | 2.86 | 2024-11-06 | doi.org/10.1038/s41467-024-53473-1 | |
8YH0 (No Gprot) | A | Nucleotide | Adenosine | A3A | Homo sapiens | NECA | - | 2.86 | 2024-11-06 | doi.org/10.1038/s41467-024-53473-1 | ||
8UXY | O1 | Odorant receptors | Odorant family 51 | consOR1 | Homo sapiens | L-menthol | - | Gs/β1/γ2 | 3.3 | 2024-10-30 | doi.org/10.1038/s41586-024-08126-0 | |
8UXY (No Gprot) | O1 | Odorant receptors | Odorant family 51 | consOR1 | Homo sapiens | L-menthol | - | 3.3 | 2024-10-30 | doi.org/10.1038/s41586-024-08126-0 | ||
8UY0 | O2 | Odorant receptors | Odorant family 2 | consOR2 | Homo sapiens | S-carvone | - | Gs/β1/γ2 | 3.2 | 2024-10-30 | doi.org/10.1038/s41586-024-08126-0 | |
8UY0 (No Gprot) | O2 | Odorant receptors | Odorant family 2 | consOR2 | Homo sapiens | S-carvone | - | 3.2 | 2024-10-30 | doi.org/10.1038/s41586-024-08126-0 | ||
8UYQ | O2 | Odorant receptors | Odorant family 4 | consOR4 | Homo sapiens | 2-methylthiazoline | - | Gs/β1/γ2 | 3.5 | 2024-10-30 | doi.org/10.1038/s41586-024-08126-0 | |
8UYQ (No Gprot) | O2 | Odorant receptors | Odorant family 4 | consOR4 | Homo sapiens | 2-methylthiazoline | - | 3.5 | 2024-10-30 | doi.org/10.1038/s41586-024-08126-0 | ||
8UXV | O1 | Odorant receptors | Odorant family 51 | consOR51 | Homo sapiens | - | - | Gs/β1/γ2 | 3.2 | 2024-10-30 | doi.org/10.1038/s41586-024-08126-0 | |
8UXV (No Gprot) | O1 | Odorant receptors | Odorant family 51 | consOR51 | Homo sapiens | - | - | 3.2 | 2024-10-30 | doi.org/10.1038/s41586-024-08126-0 | ||
8WVY | A | Orphan | Orphan | LGR4 | Homo sapiens | Norrin | - | - | 3.29 | 2024-10-30 | To be published | |
8WVW | A | Orphan | Orphan | LGR4 | Homo sapiens | - | - | - | 3.53 | 2024-10-30 | To be published | |
8WVV | A | Orphan | Orphan | LGR4 | Homo sapiens | - | - | - | 3.35 | 2024-10-30 | To be published | |
8XGS | A | Peptide | Kisspeptin | Kiss1 | Homo sapiens | Metastin | - | chim(NtGi1-Gq)/β1/γ2 | 2.95 | 2024-10-30 | doi.org/10.1126/sciadv.adn7771 | |
8XGS (No Gprot) | A | Peptide | Kisspeptin | Kiss1 | Homo sapiens | Metastin | - | 2.95 | 2024-10-30 | doi.org/10.1126/sciadv.adn7771 | ||
8XGO | A | Peptide | Kisspeptin | Kiss1 | Homo sapiens | TAK448 | - | chim(NtGi1-Gq)/β1/γ2 | 2.68 | 2024-10-30 | doi.org/10.1126/sciadv.adn7771 | |
8XGO (No Gprot) | A | Peptide | Kisspeptin | Kiss1 | Homo sapiens | TAK448 | - | 2.68 | 2024-10-30 | doi.org/10.1126/sciadv.adn7771 | ||
8XGU | A | Peptide | Kisspeptin | Kiss1 | Homo sapiens | TAK448 | - | Gi1/β1/γ2 | 3 | 2024-10-30 | doi.org/10.1126/sciadv.adn7771 | |
8XGU (No Gprot) | A | Peptide | Kisspeptin | Kiss1 | Homo sapiens | TAK448 | - | 3 | 2024-10-30 | doi.org/10.1126/sciadv.adn7771 | ||
9EPR | A | Sensory | Opsins | Rhodopsin | Hasarius adansoni | Retinal | - | Gi1/β1/γ2 | 4.9 | 2024-10-30 | doi.org/10.1038/s41467-024-53208-2 | |
9EPR (No Gprot) | A | Sensory | Opsins | Rhodopsin | Hasarius adansoni | Retinal | - | 4.9 | 2024-10-30 | doi.org/10.1038/s41467-024-53208-2 | ||
8WGB | C | Aminoacid | Metabotropic Glutamate | mGlu4; mGlu2 | Homo sapiens | Glutammate | W9R | Gi3/β1/γ2 | 3.7 | 2024-10-30 | doi.org/10.1038/s41467-024-54744-7 | |
8WGB (No Gprot) | C | Aminoacid | Metabotropic Glutamate | mGlu4; mGlu2 | Homo sapiens | Glutammate | W9R | 3.7 | 2024-10-30 | doi.org/10.1038/s41467-024-54744-7 | ||
8VHF | A | Lipid | GPR119 | GPR119 | Homo sapiens | MBX-2982 | - | Gs/β1/γ2 | 3.51 | 2024-10-30 | doi.org/10.1016/j.str.2024.10.004 | |
8VHF (No Gprot) | A | Lipid | GPR119 | GPR119 | Homo sapiens | MBX-2982 | - | 3.51 | 2024-10-30 | doi.org/10.1016/j.str.2024.10.004 | ||
8WVU | A | Orphan | Orphan | LGR4 | Homo sapiens | R-spondin-1 | - | RNF43 | 3.61 | 2024-10-30 | To be published | |
8WVX | A | Orphan | Orphan | LGR4 | Homo sapiens | Norrin | - | - | 3.32 | 2024-10-30 | To be published | |
9EPQ | A | Sensory | Opsins | Rhodopsin | Hasarius adansoni | 11,20-Ethanoretinal | - | chim(Gi1-CtGq)/β1/γ2 | 4.15 | 2024-10-23 | 10.1038/s41467-024-53208-2 | |
9EPQ (No Gprot) | A | Sensory | Opsins | Rhodopsin | Hasarius adansoni | 11,20-Ethanoretinal | - | 4.15 | 2024-10-23 | 10.1038/s41467-024-53208-2 | ||
9EPP | A | Sensory | Opsins | Rhodopsin | Hasarius adansoni | 11,20-Ethanoretinal | - | chim(Gi1-CtGq)/β1/γ2 | 4.06 | 2024-10-23 | 10.1038/s41467-024-53208-2 | |
9EPP (No Gprot) | A | Sensory | Opsins | Rhodopsin | Hasarius adansoni | 11,20-Ethanoretinal | - | 4.06 | 2024-10-23 | 10.1038/s41467-024-53208-2 | ||
8YNA | A | Amine | Histamine | H4 | Homo sapiens | Immepip | - | Gi1/β1/γ | 2.63 | 2024-10-16 | 10.2210/pdb8YN7/pdb | |
8YNA (No Gprot) | A | Amine | Histamine | H4 | Homo sapiens | Immepip | - | 2.63 | 2024-10-16 | 10.2210/pdb8YN7/pdb | ||
8YN8 | A | Amine | Histamine | H3 | Homo sapiens | Proxyfan | - | Go1/β1/γ2 | 2.77 | 2024-10-16 | 10.2210/pdb8YN7/pdb | |
8YN8 (No Gprot) | A | Amine | Histamine | H3 | Homo sapiens | Proxyfan | - | 2.77 | 2024-10-16 | 10.2210/pdb8YN7/pdb | ||
8YN7 | A | Amine | Histamine | H3 | Homo sapiens | Immethridine | - | Go1/β1/γ2 | 2.77 | 2024-10-16 | 10.2210/pdb8YN7/pdb | |
8YN7 (No Gprot) | A | Amine | Histamine | H3 | Homo sapiens | Immethridine | - | 2.77 | 2024-10-16 | 10.2210/pdb8YN7/pdb | ||
9JR3 | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | PTH | - | chim(NtGi1L-Gs-CtGq)/β1/γ2 | 2.8 | 2024-10-16 | To be published | |
9JR3 (No Gprot) | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | PTH | - | 2.8 | 2024-10-16 | To be published | ||
9JR2 | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | PTH | - | chim(NtGi1L-Gs-CtGq)/β1/γ2 | 2.8 | 2024-10-16 | To be published | |
9JR2 (No Gprot) | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | PTH | - | 2.8 | 2024-10-16 | To be published | ||
9JKQ | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | METH | - | Gs/β1/γ2 | 2.66 | 2024-10-16 | doi.org/10.1021/acs.jmedchem.4c01961 | |
9JKQ (No Gprot) | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | METH | - | 2.66 | 2024-10-16 | doi.org/10.1021/acs.jmedchem.4c01961 | ||
9GYO | A | Steroid | Bile acid | GPBA | Homo sapiens | P395 | - | chim(NtGi1-Gs)/β1/γ2 | 2.5 | 2024-10-09 | To be published | |
9GYO (No Gprot) | A | Steroid | Bile acid | GPBA | Homo sapiens | P395 | - | 2.5 | 2024-10-09 | To be published | ||
8YN2 | A | Amine | Histamine | H1 | Homo sapiens | Histamine | - | chim(NtGi1L-Gs-CtGq)/β1/γ2 | 2.66 | 2024-10-09 | doi.org/10.1038/s41467-024-52585-y | |
8YN2 (No Gprot) | A | Amine | Histamine | H1 | Homo sapiens | Histamine | - | 2.66 | 2024-10-09 | doi.org/10.1038/s41467-024-52585-y | ||
8YN4 | A | Amine | Histamine | H2 | Homo sapiens | Histamine | - | chim(NtGi1L-Gs-CtGq)/β1/γ2 | 2.97 | 2024-10-09 | doi.org/10.1038/s41467-024-52585-y | |
8YN4 (No Gprot) | A | Amine | Histamine | H2 | Homo sapiens | Histamine | - | 2.97 | 2024-10-09 | doi.org/10.1038/s41467-024-52585-y | ||
8YN6 | A | Amine | Histamine | H3 | Homo sapiens | Imetit | - | Gi1/β1/γ2 | 2.77 | 2024-10-09 | doi.org/10.1038/s41467-024-52585-y | |
8YN6 (No Gprot) | A | Amine | Histamine | H3 | Homo sapiens | Imetit | - | 2.77 | 2024-10-09 | doi.org/10.1038/s41467-024-52585-y | ||
8YN5 | A | Amine | Histamine | H3 | Homo sapiens | Histamine | - | Gi1/β1/γ2 | 2.7 | 2024-10-09 | doi.org/10.1038/s41467-024-52585-y | |
8YN5 (No Gprot) | A | Amine | Histamine | H3 | Homo sapiens | Histamine | - | 2.7 | 2024-10-09 | doi.org/10.1038/s41467-024-52585-y | ||
8YN9 | A | Amine | Histamine | H4 | Homo sapiens | Histamine | - | Gi1/β1/γ2 | 2.3 | 2024-10-09 | doi.org/10.1038/s41467-024-52585-y | |
8YN9 (No Gprot) | A | Amine | Histamine | H4 | Homo sapiens | Histamine | - | 2.3 | 2024-10-09 | doi.org/10.1038/s41467-024-52585-y | ||
8YN3 | A | Amine | Histamine | H2 | Homo sapiens | Histamine | - | Gs/β1/γ2 | 2.56 | 2024-10-09 | doi.org/10.1038/s41467-024-52585-y | |
8YN3 (No Gprot) | A | Amine | Histamine | H2 | Homo sapiens | Histamine | - | 2.56 | 2024-10-09 | doi.org/10.1038/s41467-024-52585-y | ||
9C2F | C | Ion | Calcium Sensing | CaS | Homo sapiens | Ca | Ca; Ca; Tryptophan; '6218; PO4 | - | 2.8 | 2024-10-02 | 10.1126/science.ado1868 | |
9C1P | C | Ion | Calcium Sensing | CaS | Homo sapiens | Ca | Ca; Tryptophan; '6218; PO4 | - | 2.8 | 2024-10-02 | 10.1126/science.ado1868 | |
8ZRT | A | Peptide | Endothelin | ETB | Homo sapiens | ET-1 | - | - | 3.62 | 2024-10-02 | doi.org/10.1038/s42003-024-06905-z | |
9EPO | F | Protein | Frizzled | FZD7 | Homo sapiens | - | - | - | 1.9 | 2024-10-02 | To be published | |
9EW2 | F | Protein | Frizzled | FZD7 | Homo sapiens | - | - | Gs/β1/γ2 | 3.2 | 2024-10-02 | To be published | |
9EW2 (No Gprot) | F | Protein | Frizzled | FZD7 | Homo sapiens | - | - | 3.2 | 2024-10-02 | To be published | ||
8WJX | A | Nucleotide | P2Y | P2Y1 | Homo sapiens | ADP | - | chim(Gs-CtGq)/β1/γ2 | 3.2 | 2024-10-02 | To be published | |
8WJX (No Gprot) | A | Nucleotide | P2Y | P2Y1 | Homo sapiens | ADP | - | 3.2 | 2024-10-02 | To be published | ||
8XWQ | A | Peptide | Endothelin | ETB | Homo sapiens | Endothelin-1 | - | Gi1/β1/γ2 | 4.6 | 2024-10-02 | doi.org/10.1038/s42003-024-06905-z | |
8XWQ (No Gprot) | A | Peptide | Endothelin | ETB | Homo sapiens | Endothelin-1 | - | 4.6 | 2024-10-02 | doi.org/10.1038/s42003-024-06905-z | ||
8XWP | A | Peptide | Endothelin | ETB | Homo sapiens | Endothelin-1 | - | Gi1/β1/γ2 | 3.21 | 2024-10-02 | doi.org/10.1038/s42003-024-06905-z | |
8XWP (No Gprot) | A | Peptide | Endothelin | ETB | Homo sapiens | Endothelin-1 | - | 3.21 | 2024-10-02 | doi.org/10.1038/s42003-024-06905-z | ||
8ZPT | A | Peptide | Prolactin-releasing peptide | PrRP | Homo sapiens | PrRP20 | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.96 | 2024-09-25 | doi.org/10.1038/s41421-024-00724-6 | |
8ZPT (No Gprot) | A | Peptide | Prolactin-releasing peptide | PrRP | Homo sapiens | PrRP20 | - | 2.96 | 2024-09-25 | doi.org/10.1038/s41421-024-00724-6 | ||
8ZPS | A | Peptide | Prolactin-releasing peptide | PrRP | Homo sapiens | PrRP20 | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.97 | 2024-09-25 | doi.org/10.1038/s41421-024-00724-6 | |
8ZPS (No Gprot) | A | Peptide | Prolactin-releasing peptide | PrRP | Homo sapiens | PrRP20 | - | 2.97 | 2024-09-25 | doi.org/10.1038/s41421-024-00724-6 | ||
8QJ2 | A | Peptide | Melanocortin | MC4 | Homo sapiens | pN162 | - | Gs | 3.4 | 2024-09-25 | To be published | |
8QJ2 (No Gprot) | A | Peptide | Melanocortin | MC4 | Homo sapiens | pN162 | - | 3.4 | 2024-09-25 | To be published | ||
9F34 | A | Amine | Dopamine | D3 | Homo sapiens | FOB02-04A | - | Go1/β1/γ2 | 3.05 | 2024-09-18 | 10.1038/s41467-024-51993-4 | |
9F34 (No Gprot) | A | Amine | Dopamine | D3 | Homo sapiens | FOB02-04A | - | 3.05 | 2024-09-18 | 10.1038/s41467-024-51993-4 | ||
9F33 | A | Amine | Dopamine | D3 | Homo sapiens | FOB02-04A | - | Go1/β1/γ2 | 3.05 | 2024-09-18 | 10.1038/s41467-024-51993-4 | |
9F33 (No Gprot) | A | Amine | Dopamine | D3 | Homo sapiens | FOB02-04A | - | 3.05 | 2024-09-18 | 10.1038/s41467-024-51993-4 | ||
8IRJ | C | Orphan | Orphan | GPR179 | Homo sapiens | - | - | - | 3.49 | 2024-09-18 | To be published | |
8XOR | A | Peptide | Proteinase-activated | PAR1 | Homo sapiens | - | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3 | 2024-09-18 | doi.org/10.1038/s41422-024-00997-2 | |
8XOR (No Gprot) | A | Peptide | Proteinase-activated | PAR1 | Homo sapiens | - | - | 3 | 2024-09-18 | doi.org/10.1038/s41422-024-00997-2 | ||
8YW4 | B1 | Peptide | Glucagon | GIP | Homo sapiens | Retatrutide | - | chim(NtGi1-Gs)/β1/γ22 | 3.26 | 2024-09-18 | doi.org/10.1038/s41421-024-00700-0 | |
8YW4 (No Gprot) | B1 | Peptide | Glucagon | GIP | Homo sapiens | Retatrutide | - | 3.26 | 2024-09-18 | doi.org/10.1038/s41421-024-00700-0 | ||
8XOS | A | Peptide | Proteinase-activated | PAR1 | Homo sapiens | - | - | Gi1/β1/γ2 | 3.2 | 2024-09-18 | doi.org/10.1038/s41422-024-00997-2 | |
8XOS (No Gprot) | A | Peptide | Proteinase-activated | PAR1 | Homo sapiens | - | - | 3.2 | 2024-09-18 | doi.org/10.1038/s41422-024-00997-2 | ||
8YW3 | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Retatrutide | - | Gs/β1/γ2 | 2.68 | 2024-09-18 | doi.org/10.1038/s41421-024-00700-0 | |
8YW3 (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Retatrutide | - | 2.68 | 2024-09-18 | doi.org/10.1038/s41421-024-00700-0 | ||
8YW5 | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | Retatrutide | - | Gs/β1/γ2 | 2.84 | 2024-09-18 | doi.org/10.1038/s41421-024-00700-0 | |
8YW5 (No Gprot) | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | Retatrutide | - | 2.84 | 2024-09-18 | doi.org/10.1038/s41421-024-00700-0 | ||
9BQJ | A | Peptide | Opioid | μ | Mus musculus | RO76 | - | Gi1/β1/γ2 | 3.3 | 2024-09-11 | 10.1021/acscentsci.4c00525 | |
9BQJ (No Gprot) | A | Peptide | Opioid | μ | Mus musculus | RO76 | - | 3.3 | 2024-09-11 | 10.1021/acscentsci.4c00525 | ||
8WMA | F | Protein | Frizzled | FZD4 | Homo sapiens | DVL-2 | - | - | 3.47 | 2024-09-11 | doi.org/10.1038/s41467-024-52174-z | |
8WM9 | F | Protein | Frizzled | FZD4 | Homo sapiens | DVL-2 | - | - | 3.53 | 2024-09-11 | doi.org/10.1038/s41467-024-52174-z | |
9IMA | C | Orphan | Orphan | GPRC5D | Homo sapiens | Talquetamab | - | - | 2.65 | 2024-09-11 | doi.org/10.1016/j.jmb.2024.168748 | |
8Y53 | A | Peptide | Bombesin | BB3 | Homo sapiens | MK5046 | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.93 | 2024-09-11 | doi.org/10.1016/j.celrep.2024.114511 | |
8Y53 (No Gprot) | A | Peptide | Bombesin | BB3 | Homo sapiens | MK5046 | - | 2.93 | 2024-09-11 | doi.org/10.1016/j.celrep.2024.114511 | ||
8Y52 | A | Peptide | Bombesin | BB3 | Homo sapiens | BA1 | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.9 | 2024-09-11 | 10.1016/j.celrep.2024.114511 | |
8Y52 (No Gprot) | A | Peptide | Bombesin | BB3 | Homo sapiens | BA1 | - | 2.9 | 2024-09-11 | 10.1016/j.celrep.2024.114511 | ||
9CBM | A | Amine | Adrenergic | α2a | Homo sapiens | Dexmedetomidine | - | Gi1/β1/γ2 | 3.2 | 2024-09-11 | doi.org/10.1038/s12276-024-01296-x | |
9CBM (No Gprot) | A | Amine | Adrenergic | α2a | Homo sapiens | Dexmedetomidine | - | 3.2 | 2024-09-11 | doi.org/10.1038/s12276-024-01296-x | ||
9CBL | A | Amine | Adrenergic | α2a | Homo sapiens | Epinephrine | - | Gi1/β1/γ2 | 2.8 | 2024-09-11 | doi.org/10.1038/s12276-024-01296-x | |
9CBL (No Gprot) | A | Amine | Adrenergic | α2a | Homo sapiens | Epinephrine | - | 2.8 | 2024-09-11 | doi.org/10.1038/s12276-024-01296-x | ||
8WP1 | A | Alicarboxylic acid | Succinate | Succinate | Homo sapiens | Cis-Epoxysuccinic acid | - | Gi1/β1/γ2 | 3.15 | 2024-09-11 | doi.org/10.1016/j.celrep.2024.114381 | |
8WP1 (No Gprot) | A | Alicarboxylic acid | Succinate | Succinate | Homo sapiens | Cis-Epoxysuccinic acid | - | 3.15 | 2024-09-11 | doi.org/10.1016/j.celrep.2024.114381 | ||
8WOG | A | Alicarboxylic acid | Succinate | Succinate | Homo sapiens | Succinic acid | - | Gi1/β1/γ2 | 2.97 | 2024-09-11 | doi.org/10.1016/j.celrep.2024.114381 | |
8WOG (No Gprot) | A | Alicarboxylic acid | Succinate | Succinate | Homo sapiens | Succinic acid | - | 2.97 | 2024-09-11 | doi.org/10.1016/j.celrep.2024.114381 | ||
8JXS | A | Amine | Dopamine | D1 | Homo sapiens | PF-6142 | - | - | 3 | 2024-09-04 | doi.org/10.1016/j.neuron.2024.07.003 | |
8JXR | A | Amine | Dopamine | D1 | Homo sapiens | LSD | - | - | 3.57 | 2024-09-04 | doi.org/10.1016/j.neuron.2024.07.003 | |
8QW4 | F | Protein | Frizzled | FZD3 | Homo sapiens | - | - | - | 2.9 | 2024-09-04 | doi.org/10.1038/s41467-024-51451-1 | |
8ZMG | A | Amine | 5-Hydroxytryptamine | 5-HT2A | Homo sapiens | Pimavanserin | - | - | 3.4 | 2024-08-28 | 10.1021/acs.jmedchem.4c01244 | |
8ZMF | A | Amine | 5-Hydroxytryptamine | 5-HT2C | Homo sapiens | A1L10 | - | - | 3.6 | 2024-08-28 | 10.1021/acs.jmedchem.4c01244 | |
8XVL | A | Peptide | Endothelin | ETA | Homo sapiens | Zibotentan | - | - | 3.22 | 2024-08-28 | doi.org/10.1038/s41421-024-00705-9 | |
8XVK | A | Peptide | Endothelin | ETA | Homo sapiens | Ambrisentan | - | - | 3.21 | 2024-08-28 | doi.org/10.1038/s41421-024-00705-9 | |
8XVJ | A | Peptide | Endothelin | ETA | Homo sapiens | Macitentan | - | - | 3.26 | 2024-08-28 | doi.org/10.1038/s41421-024-00705-9 | |
8XVI | A | Peptide | Endothelin | ETA | Homo sapiens | Endothelin-1 | - | chim(Gs-CtGq)/β1/γ2 | 3.32 | 2024-08-28 | doi.org/10.1038/s41421-024-00705-9 | |
8XVI (No Gprot) | A | Peptide | Endothelin | ETA | Homo sapiens | Endothelin-1 | - | 3.32 | 2024-08-28 | doi.org/10.1038/s41421-024-00705-9 | ||
8XVH | A | Peptide | Endothelin | ETB | Homo sapiens | Endothelin-1 | - | chim(Gs-CtGq)/β1/γ2 | 3.26 | 2024-08-28 | doi.org/10.1038/s41421-024-00705-9 | |
8XVH (No Gprot) | A | Peptide | Endothelin | ETB | Homo sapiens | Endothelin-1 | - | 3.26 | 2024-08-28 | doi.org/10.1038/s41421-024-00705-9 | ||
8XVE | A | Peptide | Endothelin | ETB | Homo sapiens | BQ3020 | - | chim(Gs-CtGq)/β1/γ2 | 3 | 2024-08-28 | doi.org/10.1038/s41421-024-00705-9 | |
8XVE (No Gprot) | A | Peptide | Endothelin | ETB | Homo sapiens | BQ3020 | - | 3 | 2024-08-28 | doi.org/10.1038/s41421-024-00705-9 | ||
9IJE | A | Amine | Adrenergic | β3 | Homo sapiens | Epinephrine | - | chim(NtGi1-Gs)/β1/γ2 | 2.34 | 2024-08-21 | doi.org/10.1002/cplu.202400288 | |
9IJE (No Gprot) | A | Amine | Adrenergic | β3 | Homo sapiens | Epinephrine | - | 2.34 | 2024-08-21 | doi.org/10.1002/cplu.202400288 | ||
9IJD | A | Amine | Adrenergic | β3 | Homo sapiens | Carazolol | - | chim(NtGi1-Gs)/β1/γ2 | 2.76 | 2024-08-21 | doi.org/10.1002/cplu.202400288 | |
9IJD (No Gprot) | A | Amine | Adrenergic | β3 | Homo sapiens | Carazolol | - | 2.76 | 2024-08-21 | doi.org/10.1002/cplu.202400288 | ||
8XGM | A | Protein | Chemerin | CML2 | Homo sapiens | Chemerin | - | Gi1/β1/γ2 | 3.29 | 2024-08-21 | To be published | |
8XGM (No Gprot) | A | Protein | Chemerin | CML2 | Homo sapiens | Chemerin | - | 3.29 | 2024-08-21 | To be published | ||
8JJP | A | Protein | Chemerin | CML2 | Homo sapiens | Chemerin | - | Gi1/β1/γ2 | 2.9 | 2024-08-21 | To be published | |
8JJP (No Gprot) | A | Protein | Chemerin | CML2 | Homo sapiens | Chemerin | - | 2.9 | 2024-08-21 | To be published | ||
8U02 | A | Amine | Dopamine | D2 | Homo sapiens | L-Dopamine | - | Go/β1/γ2 | 3.28 | 2024-08-21 | doi.org/10.1038/s41467-024-50964-z | |
8U02 (No Gprot) | A | Amine | Dopamine | D2 | Homo sapiens | L-Dopamine | - | 3.28 | 2024-08-21 | doi.org/10.1038/s41467-024-50964-z | ||
8TZQ | A | Amine | Dopamine | D2 | Homo sapiens | L-Dopamine | - | Go/β1/γ2 | 3.2 | 2024-08-21 | doi.org/10.1038/s41467-024-50964-z | |
8TZQ (No Gprot) | A | Amine | Dopamine | D2 | Homo sapiens | L-Dopamine | - | 3.2 | 2024-08-21 | doi.org/10.1038/s41467-024-50964-z | ||
8WKZ | A | Peptide | Melanocortin | MC4 | Homo sapiens | SBL-MC-31 | - | - | 3.3 | 2024-08-07 | doi.org/10.1021/acs.jmedchem.3c01822 | |
8WKY | A | Peptide | Melanocortin | MC4 | Homo sapiens | PG-934 | - | - | 2.9 | 2024-08-07 | doi.org/10.1021/acs.jmedchem.3c01822 | |
8ZFJ | A | Orphan | Orphan | GPR4 | Danio rerio | - | - | chim(NtGi1-Gs)/β1/γ2 | 3.1 | 2024-08-07 | To be published | |
8ZFJ (No Gprot) | A | Orphan | Orphan | GPR4 | Danio rerio | - | - | 3.1 | 2024-08-07 | To be published | ||
8JPS | A | Protein | Chemokine | ACKR1 | Homo sapiens | CCL7 | - | - | 3.65 | 2024-07-31 | 10.1016/j.cell.2024.07.005 | |
8TRD | C | Aminoacid | Metabotropic Glutamate | mGlu3; mGlu3 | Rattus norvegicus | LY341495 | - | - | 3.4 | 2024-07-31 | To be published | |
8TRC | C | Aminoacid | Metabotropic Glutamate | mGlu3; mGlu3 | Rattus norvegicus | LY341495 | - | - | 3.3 | 2024-07-31 | 10.1101/2023.08.13.552748 | |
8TR2 | C | Aminoacid | Metabotropic Glutamate | mGlu3; mGlu3 | Rattus norvegicus | Ca; LY379268 | Ca | - | 3.5 | 2024-07-31 | 10.1101/2023.08.13.552748 | |
8TR0 | C | Aminoacid | Metabotropic Glutamate | mGlu3; mGlu3 | Rattus norvegicus | LY341495 | - | - | 3.2 | 2024-07-31 | 10.1101/2023.08.13.552748 | |
8TQB | C | Aminoacid | Metabotropic Glutamate | mGlu3; mGlu3 | Rattus norvegicus | Ca; PAM VU6023326 | Ca | - | 3.3 | 2024-07-31 | 10.1101/2023.08.13.552748 | |
8KGG | A | Nucleotide | P2Y | P2Y10 | Homo sapiens | LPS | - | chim(NtGi2-G13)/β1/γ2 | 3.06 | 2024-07-31 | To be published | |
8KGG (No Gprot) | A | Nucleotide | P2Y | P2Y10 | Homo sapiens | LPS | - | 3.06 | 2024-07-31 | To be published | ||
8K6O | A | Peptide | Neuropeptide Y | Y1 | Homo sapiens | Pro-neuropeptide-Y | - | Gi2/β1/γ1 | 3.3 | 2024-07-31 | To be published | |
8K6O (No Gprot) | A | Peptide | Neuropeptide Y | Y1 | Homo sapiens | Pro-neuropeptide-Y | - | 3.3 | 2024-07-31 | To be published | ||
8K6M | A | Peptide | Neuropeptide Y | Y1 | Homo sapiens | Neuropeptide-Y | - | Gi2/β1/γ1 | 3.3 | 2024-07-31 | To be published | |
8K6M (No Gprot) | A | Peptide | Neuropeptide Y | Y1 | Homo sapiens | Neuropeptide-Y | - | 3.3 | 2024-07-31 | To be published | ||
8K6N | A | Peptide | Neuropeptide Y | Y2 | Homo sapiens | Pro-neuropeptide-Y | - | Gi2/β1/γ1 | 3.2 | 2024-07-31 | To be published | |
8K6N (No Gprot) | A | Peptide | Neuropeptide Y | Y2 | Homo sapiens | Pro-neuropeptide-Y | - | 3.2 | 2024-07-31 | To be published | ||
8ZSV | A | Amine | Trace Amine Receptors | TA1 | Mus musculus | RO5263397 | - | chim(NtGi1-Gs)/β1/γ2 | 2.96 | 2024-07-24 | 10.1016/j.celrep.2024.114505 | |
8ZSV (No Gprot) | A | Amine | Trace Amine Receptors | TA1 | Mus musculus | RO5263397 | - | 2.96 | 2024-07-24 | 10.1016/j.celrep.2024.114505 | ||
8ZSS | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | RO5263397 | - | chim(NtGi1-Gs)/β1/γ2 | 3.07 | 2024-07-24 | 10.1016/j.celrep.2024.114505 | |
8ZSS (No Gprot) | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | RO5263397 | - | 3.07 | 2024-07-24 | 10.1016/j.celrep.2024.114505 | ||
8ZSP | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | LSD | - | chim(NtGi1L-Gs-CtGq)/β1/γ2 | 3.14 | 2024-07-24 | 10.1016/j.celrep.2024.114505 | |
8ZSP (No Gprot) | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | LSD | - | 3.14 | 2024-07-24 | 10.1016/j.celrep.2024.114505 | ||
8ZSJ | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | - | - | chim(NtGi1L-Gs-CtGq)/β1/γ2 | 2.8 | 2024-07-24 | 10.1016/j.celrep.2024.114505 | |
8ZSJ (No Gprot) | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | - | - | 2.8 | 2024-07-24 | 10.1016/j.celrep.2024.114505 | ||
8K4P | A | Other | Unclassified | KSHV | Human gammaherpesvirus 8 | - | - | Gi1/β1/γ1 | 2.81 | 2024-07-24 | To be published | |
8K4P (No Gprot) | A | Other | Unclassified | KSHV | Human gammaherpesvirus 8 | - | - | 2.81 | 2024-07-24 | To be published | ||
8K4O | A | Other | Unclassified | KSHV | Human gammaherpesvirus 8 | CXCL1 | - | Gi1/β1/γ1 | 3.01 | 2024-07-24 | To be published | |
8K4O (No Gprot) | A | Other | Unclassified | KSHV | Human gammaherpesvirus 8 | CXCL1 | - | 3.01 | 2024-07-24 | To be published | ||
9BJK | A | Peptide | Opioid | μ | Mus musculus | Naloxone | NAM | - | 3.26 | 2024-07-17 | 10.1038/s41586-024-07587-7 | |
8W1V | A | Amine | Adrenergic | β2 | Homo sapiens | PubChem 171716265 | - | - | 3 | 2024-07-17 | doi.org/10.1021/acs.jmedchem.4c00578 | |
8W1V (Multimeric) | A | Amine | Adrenergic | β2 | Homo sapiens | PubChem 171716265 | - | 3 | 2024-07-17 | doi.org/10.1021/acs.jmedchem.4c00578 | ||
8K3Z | A | Protein | Chemokine | CXCR4 | Homo sapiens | CXCL12 | - | Gi1/β1/γ1 | 2.81 | 2024-07-17 | To be published | |
8K3Z (No Gprot) | A | Protein | Chemokine | CXCR4 | Homo sapiens | CXCL12 | - | 2.81 | 2024-07-17 | To be published | ||
8ZQE | A | Orphan | Orphan | GPR15 | Homo sapiens | GPR15L(C11) | - | Gi1/β1/γ1 | 2.9 | 2024-07-10 | 10.1038/s41421-024-00698-5 | |
8ZQE (No Gprot) | A | Orphan | Orphan | GPR15 | Homo sapiens | GPR15L(C11) | - | 2.9 | 2024-07-10 | 10.1038/s41421-024-00698-5 | ||
8ZCJ | A | Peptide | Somatostatin | SST5 | Homo sapiens | Pasireotide | - | Gi1/β1/γ1 | 3.09 | 2024-07-10 | 10.1038/s41401-024-01314-8 | |
8ZCJ (No Gprot) | A | Peptide | Somatostatin | SST5 | Homo sapiens | Pasireotide | - | 3.09 | 2024-07-10 | 10.1038/s41401-024-01314-8 | ||
8ZBE | A | Peptide | Somatostatin | SST5 | Homo sapiens | Octreotide | - | Gi1/β1/γ1 | 3.24 | 2024-07-10 | 10.1038/s41401-024-01314-8 | |
8ZBE (No Gprot) | A | Peptide | Somatostatin | SST5 | Homo sapiens | Octreotide | - | 3.24 | 2024-07-10 | 10.1038/s41401-024-01314-8 | ||
8XQT | T2 | Sensory | Taste2 | TAS2R14 | Homo sapiens | Cholesterol | Cholesterol | Gi1/β1/γ1 | 2.94 | 2024-07-10 | 10.1038/s41586-024-07569-9 | |
8XQT (No Gprot) | T2 | Sensory | Taste2 | TAS2R14 | Homo sapiens | Cholesterol | Cholesterol | 2.94 | 2024-07-10 | 10.1038/s41586-024-07569-9 | ||
8XQS | T2 | Sensory | Taste2 | TAS2R14 | Homo sapiens | Cholesterol | Flufenamic acid | Gi1/β1/γ1 | 3.3 | 2024-07-10 | 10.1038/s41586-024-07569-9 | |
8XQS (No Gprot) | T2 | Sensory | Taste2 | TAS2R14 | Homo sapiens | Cholesterol | Flufenamic acid | 3.3 | 2024-07-10 | 10.1038/s41586-024-07569-9 | ||
8XQO | T2 | Sensory | Taste2 | TAS2R14 | Homo sapiens | Cholesterol | Aristolochic acid A | Gi1/β1/γ1 | 2.77 | 2024-07-10 | 10.1038/s41586-024-07569-9 | |
8XQO (No Gprot) | T2 | Sensory | Taste2 | TAS2R14 | Homo sapiens | Cholesterol | Aristolochic acid A | 2.77 | 2024-07-10 | 10.1038/s41586-024-07569-9 | ||
8XQN | T2 | Sensory | Taste2 | TAS2R14 | Homo sapiens | Cholesterol | Aristolochic acid A | Gi1/β1/γ1 | 3.05 | 2024-07-10 | 10.1038/s41586-024-07569-9 | |
8XQN (No Gprot) | T2 | Sensory | Taste2 | TAS2R14 | Homo sapiens | Cholesterol | Aristolochic acid A | 3.05 | 2024-07-10 | 10.1038/s41586-024-07569-9 | ||
8XQR | T2 | Sensory | Taste2 | TAS2R14 | Homo sapiens | - | Flufenamic acid | Gt3/β1/γ1 | 3.2 | 2024-07-10 | 10.1038/s41586-024-07569-9 | |
8XQR (No Gprot) | T2 | Sensory | Taste2 | TAS2R14 | Homo sapiens | - | Flufenamic acid | 3.2 | 2024-07-10 | 10.1038/s41586-024-07569-9 | ||
8XQP | T2 | Sensory | Taste2 | TAS2R14 | Homo sapiens | Cholesterol | Aristolochic acid A | Gt3/β1/γ1 | 3.29 | 2024-07-10 | 10.1038/s41586-024-07569-9 | |
8XQP (No Gprot) | T2 | Sensory | Taste2 | TAS2R14 | Homo sapiens | Cholesterol | Aristolochic acid A | 3.29 | 2024-07-10 | 10.1038/s41586-024-07569-9 | ||
8XQL | T2 | Sensory | Taste2 | TAS2R14 | Homo sapiens | Cholesterol | Aristolochic acid A | Gt3/β1/γ1 | 2.99 | 2024-07-10 | 10.1038/s41586-024-07569-9 | |
8XQL (No Gprot) | T2 | Sensory | Taste2 | TAS2R14 | Homo sapiens | Cholesterol | Aristolochic acid A | 2.99 | 2024-07-10 | 10.1038/s41586-024-07569-9 | ||
8YZK | C | Orphan | Orphan | GPRC5D | Homo sapiens | - | - | - | 3.4 | 2024-07-03 | 10.1038/s41467-024-49625-y | |
8ZJE | A | Peptide | Kisspeptin | Kiss1 | Homo sapiens | TAK-448 | - | chim(NtGi1-Gq)/β1/γ1 | 3.07 | 2024-07-03 | To be published | |
8ZJE (No Gprot) | A | Peptide | Kisspeptin | Kiss1 | Homo sapiens | TAK-448 | - | 3.07 | 2024-07-03 | To be published | ||
8ZJD | A | Peptide | Kisspeptin | Kiss1 | Homo sapiens | Kisspeptin-10 | - | chim(NtGi1-Gq)/β1/γ1 | 3.06 | 2024-07-03 | To be published | |
8ZJD (No Gprot) | A | Peptide | Kisspeptin | Kiss1 | Homo sapiens | Kisspeptin-10 | - | 3.06 | 2024-07-03 | To be published | ||
8XIP | A | Peptide | Somatostatin | SST1 | Homo sapiens | Pasireotide | - | chim(NtGi1-Gs-CtGi1)/β1/γ2 | 3.29 | 2024-07-03 | doi.org/10.1073/pnas.2400298121 | |
8XIP (No Gprot) | A | Peptide | Somatostatin | SST1 | Homo sapiens | Pasireotide | - | 3.29 | 2024-07-03 | doi.org/10.1073/pnas.2400298121 | ||
8XIO | A | Peptide | Somatostatin | SST1 | Homo sapiens | L797591 | - | chim(NtGi1-Gs-CtGi1)/β1/γ2 | 2.65 | 2024-07-03 | doi.org/10.1073/pnas.2400298121 | |
8XIO (No Gprot) | A | Peptide | Somatostatin | SST1 | Homo sapiens | L797591 | - | 2.65 | 2024-07-03 | doi.org/10.1073/pnas.2400298121 | ||
8XIR | A | Peptide | Somatostatin | SST3 | Homo sapiens | Pasireotide | - | chim(NtGi1-Gs-CtGi1)/β1/γ2 | 2.52 | 2024-07-03 | doi.org/10.1073/pnas.2400298121 | |
8XIR (No Gprot) | A | Peptide | Somatostatin | SST3 | Homo sapiens | Pasireotide | - | 2.52 | 2024-07-03 | doi.org/10.1073/pnas.2400298121 | ||
8XIQ | A | Peptide | Somatostatin | SST3 | Homo sapiens | L796778 | - | chim(NtGi1-Gs-CtGi1)/β1/γ2 | 2.71 | 2024-07-03 | doi.org/10.1073/pnas.2400298121 | |
8XIQ (No Gprot) | A | Peptide | Somatostatin | SST3 | Homo sapiens | L796778 | - | 2.71 | 2024-07-03 | doi.org/10.1073/pnas.2400298121 | ||
8ZH8 | A | Peptide | P518 | QRFP | Homo sapiens | QRF-Amide | - | Gq/β1/γ1 | 3.19 | 2024-07-03 | 10.1038/s41467-024-49030-5 | |
8ZH8 (No Gprot) | A | Peptide | P518 | QRFP | Homo sapiens | QRF-Amide | - | 3.19 | 2024-07-03 | 10.1038/s41467-024-49030-5 | ||
9ERX | A | Lipid | Cannabinoid | CB1 | Homo sapiens | D9-THC analog | - | Gi1/β1/γ2 | 2.9 | 2024-06-26 | 10.21203/rs.3.rs-4277209/v1 | |
9ERX (No Gprot) | A | Lipid | Cannabinoid | CB1 | Homo sapiens | D9-THC analog | - | 2.9 | 2024-06-26 | 10.21203/rs.3.rs-4277209/v1 | ||
8ZRK | A | Lipid | GPR119 | GPR119 | Homo sapiens | GSK-1292263 | - | Gs/β1/γ2 | 2.82 | 2024-06-19 | To be published | |
8ZRK (No Gprot) | A | Lipid | GPR119 | GPR119 | Homo sapiens | GSK-1292263 | - | 2.82 | 2024-06-19 | To be published | ||
8ZR5 | A | Lipid | GPR119 | GPR119 | Homo sapiens | Firuglipel | - | Gs/β1/γ2 | 3.31 | 2024-06-19 | To be published | |
8ZR5 (No Gprot) | A | Lipid | GPR119 | GPR119 | Homo sapiens | Firuglipel | - | 3.31 | 2024-06-19 | To be published | ||
8RLN | A | Nucleotide | Adenosine | A2A | Homo sapiens | LUF5834 | - | - | 2.43 | 2024-06-19 | doi.org/10.1021/acsptsci.4c00051 | |
8WST | A | Peptide | Melanin Concentrating Hormone | MCH2 | Homo sapiens | Pro-MCH | - | chim(NtGi1L-Gs-CtGq)/β1/γ2 | 2.4 | 2024-06-19 | 10.1038/s41421-024-00679-8 | |
8WST (No Gprot) | A | Peptide | Melanin Concentrating Hormone | MCH2 | Homo sapiens | Pro-MCH | - | 2.4 | 2024-06-19 | 10.1038/s41421-024-00679-8 | ||
8WZ2 | A | Peptide | P518 | QRFP | Homo sapiens | Orexigenic Neuropeptide QRFP | - | chim(NtGi1L-Gs-CtGq)/β1/γ2 | 2.73 | 2024-06-19 | 10.1038/s41421-024-00670-3 | |
8WZ2 (No Gprot) | A | Peptide | P518 | QRFP | Homo sapiens | Orexigenic Neuropeptide QRFP | - | 2.73 | 2024-06-19 | 10.1038/s41421-024-00670-3 | ||
8WSS | A | Peptide | Melanin Concentrating Hormone | MCH1 | Homo sapiens | Pro-MCH | - | Gi1/β1/γ1 | 3.01 | 2024-06-19 | 10.1038/s41421-024-00679-8 | |
8WSS (No Gprot) | A | Peptide | Melanin Concentrating Hormone | MCH1 | Homo sapiens | Pro-MCH | - | 3.01 | 2024-06-19 | 10.1038/s41421-024-00679-8 | ||
8X8N | A | Peptide | Somatostatin | SST5 | Homo sapiens | Octreotide | - | chim(NtGi1-Gs-CtGi1)/β1/γ2 | 2.9 | 2024-06-12 | To be published | |
8X8N (No Gprot) | A | Peptide | Somatostatin | SST5 | Homo sapiens | Octreotide | - | 2.9 | 2024-06-12 | To be published | ||
8X8L | A | Peptide | Somatostatin | SST5 | Homo sapiens | Cortistatin | - | chim(NtGi1-Gs-CtGi1)/β1/γ2 | 2.7 | 2024-06-12 | To be published | |
8X8L (No Gprot) | A | Peptide | Somatostatin | SST5 | Homo sapiens | Cortistatin | - | 2.7 | 2024-06-12 | To be published | ||
8YUT | A | Amine | Histamine | H2 | Homo sapiens | Amthamine | - | Gs/β1/γ2 | 2.7 | 2024-06-05 | 10.1002/advs.202310120 | |
8YUT (No Gprot) | A | Amine | Histamine | H2 | Homo sapiens | Amthamine | - | 2.7 | 2024-06-05 | 10.1002/advs.202310120 | ||
8IKH | A | Lipid | Cannabinoid | CB1 | Homo sapiens | - | Q2L | Gi1/β1/γ1 | 3.3 | 2024-06-05 | 10.1073/pnas.2321532121 | |
8IKH (No Gprot) | A | Lipid | Cannabinoid | CB1 | Homo sapiens | - | Q2L | 3.3 | 2024-06-05 | 10.1073/pnas.2321532121 | ||
8IKG | A | Lipid | Cannabinoid | CB1 | Homo sapiens | - | Q2B | Gi1/β1/γ1 | 3.4 | 2024-06-05 | 10.1073/pnas.2321532121 | |
8IKG (No Gprot) | A | Lipid | Cannabinoid | CB1 | Homo sapiens | - | Q2B | 3.4 | 2024-06-05 | 10.1073/pnas.2321532121 | ||
8YUU | A | Amine | Histamine | H3 | Homo sapiens | Histamine | - | Gi1/β1/γ1 | 2.7 | 2024-06-05 | doi.org/10.1002/advs.202310120 | |
8YUU (No Gprot) | A | Amine | Histamine | H3 | Homo sapiens | Histamine | - | 2.7 | 2024-06-05 | doi.org/10.1002/advs.202310120 | ||
8V6U | A | Amine | 5-Hydroxytryptamine | 5-HT2A | Homo sapiens | PubChem 171392456 | - | chim(NtGi2-Gs-CtGq)/β1/γ2 | 3 | 2024-05-29 | 10.1126/science.adn6354 | |
8V6U (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT2A | Homo sapiens | PubChem 171392456 | - | 3 | 2024-05-29 | 10.1126/science.adn6354 | ||
8UWL | A | Amine | 5-Hydroxytryptamine | 5-HT2A | Homo sapiens | Lisuride | - | chim(NtGi2-Gs-CtGq)/β1/γ2 | 2.8 | 2024-05-29 | 10.1126/science.adn6354 | |
8UWL (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT2A | Homo sapiens | Lisuride | - | 2.8 | 2024-05-29 | 10.1126/science.adn6354 | ||
8PKM | A | Amine | 5-Hydroxytryptamine | 5-HT1A | Homo sapiens | Befiradol | t7m | Gi1/β1/γ1 | 2.9 | 2024-05-29 | To be published | |
8PKM (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT1A | Homo sapiens | Befiradol | t7m | 2.9 | 2024-05-29 | To be published | ||
8PJK | A | Amine | 5-Hydroxytryptamine | 5-HT1A | Homo sapiens | ST171 | t7m | Gi1/β1/γ1 | 2.4 | 2024-05-29 | To be published | |
8PJK (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT1A | Homo sapiens | ST171 | t7m | 2.4 | 2024-05-29 | To be published | ||
8YKX | A | Alicarboxylic acid | Succinate | Succinate | Homo sapiens | Maleic acid | - | Gi1/β1/γ1 | 2.69 | 2024-05-29 | 10.1038/s41422-024-00984-7 | |
8YKX (No Gprot) | A | Alicarboxylic acid | Succinate | Succinate | Homo sapiens | Maleic acid | - | 2.69 | 2024-05-29 | 10.1038/s41422-024-00984-7 | ||
8YKW | A | Alicarboxylic acid | Succinate | Succinate | Homo sapiens | Succinic acid | - | Gi1/β1/γ1 | 2.75 | 2024-05-29 | 10.1038/s41422-024-00984-7 | |
8YKW (No Gprot) | A | Alicarboxylic acid | Succinate | Succinate | Homo sapiens | Succinic acid | - | 2.75 | 2024-05-29 | 10.1038/s41422-024-00984-7 | ||
8YKV | A | Alicarboxylic acid | Succinate | Succinate | Homo sapiens | PubChem 137553168 | - | Gi1/β1/γ2 | 2.48 | 2024-05-29 | doi.org/10.1038/s41422-024-00984-7 | |
8YKV (No Gprot) | A | Alicarboxylic acid | Succinate | Succinate | Homo sapiens | PubChem 137553168 | - | 2.48 | 2024-05-29 | doi.org/10.1038/s41422-024-00984-7 | ||
8K9L | A | Peptide | Opioid | μ | Homo sapiens | Damgo | VV9 | Gi3/β1/γ1 | 3.05 | 2024-05-29 | 10.1038/s41467-024-47792-6 | |
8K9L (No Gprot) | A | Peptide | Opioid | μ | Homo sapiens | Damgo | VV9 | 3.05 | 2024-05-29 | 10.1038/s41467-024-47792-6 | ||
8K9K | A | Peptide | Opioid | μ | Homo sapiens | Damgo | - | Gi3/β1/γ1 | 2.98 | 2024-05-29 | 10.1038/s41467-024-47792-6 | |
8K9K (No Gprot) | A | Peptide | Opioid | μ | Homo sapiens | Damgo | - | 2.98 | 2024-05-29 | 10.1038/s41467-024-47792-6 | ||
8YRG | A | Orphan | Orphan | MRGPRX4 | Homo sapiens | Fospropofol | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.14 | 2024-05-22 | 10.1126/scitranslmed.adk8198 | |
8YRG (No Gprot) | A | Orphan | Orphan | MRGPRX4 | Homo sapiens | Fospropofol | - | 3.14 | 2024-05-22 | 10.1126/scitranslmed.adk8198 | ||
8TH4 | A | Peptide | Angiotensin | AT1 | Homo sapiens | Losartan | AT118-L Nanobody | - | 3.3 | 2024-05-22 | 10.1038/s41589-024-01620-6 | |
8TH3 | A | Peptide | Angiotensin | AT1 | Homo sapiens | - | AT118-H Nanobody | - | 3 | 2024-05-22 | 10.1038/s41589-024-01620-6 | |
8JPP | A | Alicarboxylic acid | Succinate | Succinate | Homo sapiens | Succinic acid | - | chim(Gs-CtGq)/β1/γ1 | 3.2 | 2024-05-22 | 10.1038/s41422-024-00968-7 | |
8JPP (No Gprot) | A | Alicarboxylic acid | Succinate | Succinate | Homo sapiens | Succinic acid | - | 3.2 | 2024-05-22 | 10.1038/s41422-024-00968-7 | ||
9BKK | A | Peptide | Cholecystokinin | CCKA | Homo sapiens | Cholecystokinin-8 | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.51 | 2024-05-22 | To be published | |
9BKK (No Gprot) | A | Peptide | Cholecystokinin | CCKA | Homo sapiens | Cholecystokinin-8 | - | 2.51 | 2024-05-22 | To be published | ||
9BKJ | A | Peptide | Cholecystokinin | CCKA | Homo sapiens | Cholecystokinin-8 | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.59 | 2024-05-22 | To be published | |
9BKJ (No Gprot) | A | Peptide | Cholecystokinin | CCKA | Homo sapiens | Cholecystokinin-8 | - | 2.59 | 2024-05-22 | To be published | ||
8JPN | A | Alicarboxylic acid | Succinate | Succinate | Homo sapiens | Cis-Epoxysuccinic acid | - | Gi1/β1/γ1 | 2.9 | 2024-05-22 | 10.1038/s41422-024-00968-7 | |
8JPN (No Gprot) | A | Alicarboxylic acid | Succinate | Succinate | Homo sapiens | Cis-Epoxysuccinic acid | - | 2.9 | 2024-05-22 | 10.1038/s41422-024-00968-7 | ||
8Z1E | A | Orphan | Orphan | UL78 | Human herpesvirus 5 | - | - | - | 3.12 | 2024-05-15 | 10.1038/s41421-024-00684-x | |
8Z1E (Multimeric) | A | Orphan | Orphan | UL78 | Human herpesvirus 5 | - | - | 3.12 | 2024-05-15 | 10.1038/s41421-024-00684-x | ||
8XBG | A | Orphan | Orphan | GPR34 | Homo sapiens | S3E-LysoPS | - | - | 3.43 | 2024-05-15 | 10.1038/s41467-024-45046-z | |
8FYX | A | Amine | 5-Hydroxytryptamine | 5-HT1A | Homo sapiens | Buspirone | - | Gi1/β1/γ1 | 2.72 | 2024-05-15 | 10.1038/s41586-024-07403-2 | |
8FYX (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT1A | Homo sapiens | Buspirone | - | 2.72 | 2024-05-15 | 10.1038/s41586-024-07403-2 | ||
8FYT | A | Amine | 5-Hydroxytryptamine | 5-HT1A | Homo sapiens | LSD | - | Gi1/β1/γ1 | 2.64 | 2024-05-15 | 10.1038/s41586-024-07403-2 | |
8FYT (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT1A | Homo sapiens | LSD | - | 2.64 | 2024-05-15 | 10.1038/s41586-024-07403-2 | ||
8FYL | A | Amine | 5-Hydroxytryptamine | 5-HT1A | Homo sapiens | Vilazodone | - | Gi1/β1/γ1 | 2.94 | 2024-05-15 | 10.1038/s41586-024-07403-2 | |
8FYL (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT1A | Homo sapiens | Vilazodone | - | 2.94 | 2024-05-15 | 10.1038/s41586-024-07403-2 | ||
8FYE | A | Amine | 5-Hydroxytryptamine | 5-HT1A | Homo sapiens | 4-F,5-MeO-PyrT | - | Gi1/β1/γ1 | 2.85 | 2024-05-15 | 10.1038/s41586-024-07403-2 | |
8FYE (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT1A | Homo sapiens | 4-F,5-MeO-PyrT | - | 2.85 | 2024-05-15 | 10.1038/s41586-024-07403-2 | ||
8FY8 | A | Amine | 5-Hydroxytryptamine | 5-HT1A | Homo sapiens | 5-MeO-DMT | - | Gi1/β1/γ1 | 2.79 | 2024-05-15 | 10.1038/s41586-024-07403-2 | |
8FY8 (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT1A | Homo sapiens | 5-MeO-DMT | - | 2.79 | 2024-05-15 | 10.1038/s41586-024-07403-2 | ||
8XBE | A | Orphan | Orphan | GPR34 | Homo sapiens | S3E-LysoPS | - | Gi1/β1/γ1 | 3.4 | 2024-05-15 | 10.1038/s41467-024-45046-z | |
8XBE (No Gprot) | A | Orphan | Orphan | GPR34 | Homo sapiens | S3E-LysoPS | - | 3.4 | 2024-05-15 | 10.1038/s41467-024-45046-z | ||
8UH3 | A | Amine | 5-Hydroxytryptamine | 5-HT1E | Homo sapiens | Setiptiline | - | Gi1/β1/γ1 | 3.31 | 2024-05-01 | 10.1126/sciadv.adk4855 | |
8UH3 (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT1E | Homo sapiens | Setiptiline | - | 3.31 | 2024-05-01 | 10.1126/sciadv.adk4855 | ||
8UGY | A | Amine | 5-Hydroxytryptamine | 5-HT1E | Homo sapiens | Mianserin | - | Gi1/β1/γ1 | 3.31 | 2024-05-01 | 10.1126/sciadv.adk4855 | |
8UGY (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT1E | Homo sapiens | Mianserin | - | 3.31 | 2024-05-01 | 10.1126/sciadv.adk4855 | ||
8X17 | A | Nucleotide | Adenosine | A3A | Homo sapiens | Namodenoson | - | Gi1/β1/γ2 | 3.19 | 2024-04-24 | 10.1038/s41467-024-47207-6 | |
8X17 (No Gprot) | A | Nucleotide | Adenosine | A3A | Homo sapiens | Namodenoson | - | 3.19 | 2024-04-24 | 10.1038/s41467-024-47207-6 | ||
8X16 | A | Nucleotide | Adenosine | A3A | Homo sapiens | Piclidenoson | - | Gi1/β1/γ2 | 3.29 | 2024-04-24 | 10.1038/s41467-024-47207-6 | |
8X16 (No Gprot) | A | Nucleotide | Adenosine | A3A | Homo sapiens | Piclidenoson | - | 3.29 | 2024-04-24 | 10.1038/s41467-024-47207-6 | ||
8YY8 | F | Protein | Frizzled | FZD7 | Homo sapiens | - | - | Gs/β1/γ2 | 3.22 | 2024-04-24 | 10.1038/s41422-021-00525-6 | |
8YY8 (No Gprot) | F | Protein | Frizzled | FZD7 | Homo sapiens | - | - | 3.22 | 2024-04-24 | 10.1038/s41422-021-00525-6 | ||
9AUC | B1 | Peptide | Calcitonin | CT (AMY1) | Homo sapiens | Calcitonin gene-related peptide-1 | - | Gs/β1/γ2; RAMP1 | 2.4 | 2024-04-24 | 10.1021/acs.biochem.4c00114 | |
9AUC (No Gprot) | B1 | Peptide | Calcitonin | CT (AMY1) | Homo sapiens | Calcitonin gene-related peptide-1 | - | 2.4 | 2024-04-24 | 10.1021/acs.biochem.4c00114 | ||
9AXF | C | Ion | Calcium Sensing | CaS | Homo sapiens | Ca | Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4 | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.5 | 2024-04-17 | 10.1038/s41586-024-07331-1 | |
9AXF (No Gprot) | C | Ion | Calcium Sensing | CaS | Homo sapiens | Ca | Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4 | 3.5 | 2024-04-17 | 10.1038/s41586-024-07331-1 | ||
9ASB | C | Ion | Calcium Sensing | CaS | Homo sapiens | Ca | Ca; Ca; Cyclomethyltryptophan; 9IG; PO4 | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.4 | 2024-04-17 | 10.1038/s41586-024-07331-1 | |
9ASB (No Gprot) | C | Ion | Calcium Sensing | CaS | Homo sapiens | Ca | Ca; Ca; Cyclomethyltryptophan; 9IG; PO4 | 3.4 | 2024-04-17 | 10.1038/s41586-024-07331-1 | ||
9AVG | C | Ion | Calcium Sensing | CaS | Homo sapiens | Ca | Ca; Ca; Cyclomethyltryptophan; 9IG; PO4 | chim(NtGi1-Gs)/β1/γ2 | 3.6 | 2024-04-17 | 10.1038/s41586-024-07331-1 | |
9AVG (No Gprot) | C | Ion | Calcium Sensing | CaS | Homo sapiens | Ca | Ca; Ca; Cyclomethyltryptophan; 9IG; PO4 | 3.6 | 2024-04-17 | 10.1038/s41586-024-07331-1 | ||
9AYF | C | Ion | Calcium Sensing | CaS | Homo sapiens | Ca | Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4 | Gi1/β1/γ2 | 3.6 | 2024-04-17 | 10.1038/s41586-024-07331-1 | |
9AYF (No Gprot) | C | Ion | Calcium Sensing | CaS | Homo sapiens | Ca | Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4 | 3.6 | 2024-04-17 | 10.1038/s41586-024-07331-1 | ||
8J23 | A | Lipid | Free Fatty Acid | FFA2 | Homo sapiens | - | - | Gi1/β1/γ2 | 3.2 | 2024-04-17 | To be published | |
8J23 (No Gprot) | A | Lipid | Free Fatty Acid | FFA2 | Homo sapiens | - | - | 3.2 | 2024-04-17 | To be published | ||
9AVL | C | Ion | Calcium Sensing | CaS | Homo sapiens | Ca | Ca; Ca; Cyclomethyltryptophan; 9IG; PO4 | Gi3/β2/γ2 | 3.8 | 2024-04-17 | 10.1038/s41586-024-07331-1 | |
9AVL (No Gprot) | C | Ion | Calcium Sensing | CaS | Homo sapiens | Ca | Ca; Ca; Cyclomethyltryptophan; 9IG; PO4 | 3.8 | 2024-04-17 | 10.1038/s41586-024-07331-1 | ||
8XOG | A | Orphan | Orphan | GPR30 | Homo sapiens | - | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.9 | 2024-04-10 | To be published | |
8XOG (No Gprot) | A | Orphan | Orphan | GPR30 | Homo sapiens | - | - | 2.9 | 2024-04-10 | To be published | ||
8XOJ | A | Orphan | Orphan | GPR30 | Homo sapiens | - | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.1 | 2024-04-10 | To be published | |
8XOJ (No Gprot) | A | Orphan | Orphan | GPR30 | Homo sapiens | - | - | 3.1 | 2024-04-10 | To be published | ||
8XOI | A | Orphan | Orphan | GPR30 | Homo sapiens | - | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.2 | 2024-04-10 | To be published | |
8XOI (No Gprot) | A | Orphan | Orphan | GPR30 | Homo sapiens | - | - | 3.2 | 2024-04-10 | To be published | ||
8XOH | A | Orphan | Orphan | GPR30 | Homo sapiens | - | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.2 | 2024-04-10 | To be published | |
8XOH (No Gprot) | A | Orphan | Orphan | GPR30 | Homo sapiens | - | - | 3.2 | 2024-04-10 | To be published | ||
8XOF | A | Orphan | Orphan | GPR30 | Homo sapiens | Lys05 | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.6 | 2024-04-10 | doi.org/10.1038/s41422-024-00963-y | |
8XOF (No Gprot) | A | Orphan | Orphan | GPR30 | Homo sapiens | Lys05 | - | 2.6 | 2024-04-10 | doi.org/10.1038/s41422-024-00963-y | ||
8IZ4 | A | Orphan | Orphan | GPR34 | Homo sapiens | Lysophosphatidylserine | - | Gi1/β1/γ2 | 2.94 | 2024-04-10 | To be published | |
8IZ4 (No Gprot) | A | Orphan | Orphan | GPR34 | Homo sapiens | Lysophosphatidylserine | - | 2.94 | 2024-04-10 | To be published | ||
8RQQ | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | Na | - | 2.37 | 2024-04-03 | doi.org/10.1021/acs.cgd.4c00087 | |
8X2K | A | Orphan | Orphan | GPR3 | Homo sapiens | Oleic monoethanolamide | - | chim(NtGi1-Gs)/β1/γ2 | 3.03 | 2024-04-03 | To be published | |
8X2K (No Gprot) | A | Orphan | Orphan | GPR3 | Homo sapiens | Oleic monoethanolamide | - | 3.03 | 2024-04-03 | To be published | ||
8J6L | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | Niacin | - | Gi1/β1/γ2 | 3.05 | 2024-04-03 | 10.1016/j.celrep.2023.113406 | |
8J6L (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | Niacin | - | 3.05 | 2024-04-03 | 10.1016/j.celrep.2023.113406 | ||
8J6I | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | MK6892 | - | Gi1/β1/γ2 | 2.92 | 2024-04-03 | 10.1016/j.celrep.2023.113406 | |
8J6I (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | MK6892 | - | 2.92 | 2024-04-03 | 10.1016/j.celrep.2023.113406 | ||
8IU2 | A | Sensory | Opsins | Opsin1LW | Homo sapiens | Retinal | - | Gi1/β1/γ2 | 3.35 | 2024-03-27 | To be published | |
8IU2 (No Gprot) | A | Sensory | Opsins | Opsin1LW | Homo sapiens | Retinal | - | 3.35 | 2024-03-27 | To be published | ||
8IYX | A | Orphan | Orphan | GPR34 | Homo sapiens | YL-365 | - | - | 3.34 | 2024-03-20 | 10.1073/pnas.2308435120 | |
8WU1 | A | Lipid | Cannabinoid | CB1 | Homo sapiens | PubChem 119025665 | - | Arrestin2 | 3.2 | 2024-03-20 | To be published | |
8XZJ | A | Peptide | Apelin | Apelin | Homo sapiens | WN353 | - | Gi1/β1/γ2 | 3 | 2024-03-20 | 10.1016/j.cell.2024.02.004 | |
8XZJ (No Gprot) | A | Peptide | Apelin | Apelin | Homo sapiens | WN353 | - | 3 | 2024-03-20 | 10.1016/j.cell.2024.02.004 | ||
8XZI | A | Peptide | Apelin | Apelin | Homo sapiens | CMF-019 | - | Gi1/β1/γ2 | 2.7 | 2024-03-20 | doi.org/10.1016/j.cell.2024.02.004 | |
8XZI (No Gprot) | A | Peptide | Apelin | Apelin | Homo sapiens | CMF-019 | - | 2.7 | 2024-03-20 | doi.org/10.1016/j.cell.2024.02.004 | ||
8XZH | A | Peptide | Apelin | Apelin | Homo sapiens | MM07 | - | Gi1/β1/γ2 | 2.06 | 2024-03-20 | 10.1016/j.cell.2024.02.004 | |
8XZH (No Gprot) | A | Peptide | Apelin | Apelin | Homo sapiens | MM07 | - | 2.06 | 2024-03-20 | 10.1016/j.cell.2024.02.004 | ||
8XZG | A | Peptide | Apelin | Apelin | Homo sapiens | Apelin-13 | - | Gi1/β1/γ2 | 3.2 | 2024-03-20 | 10.1016/j.cell.2024.02.004 | |
8XZG (No Gprot) | A | Peptide | Apelin | Apelin | Homo sapiens | Apelin-13 | - | 3.2 | 2024-03-20 | 10.1016/j.cell.2024.02.004 | ||
8XZF | A | Peptide | Apelin | Apelin | Homo sapiens | WN561 | - | Gi1/β1/γ2 | 3 | 2024-03-20 | 10.1016/j.cell.2024.02.004 | |
8XZF (No Gprot) | A | Peptide | Apelin | Apelin | Homo sapiens | WN561 | - | 3 | 2024-03-20 | 10.1016/j.cell.2024.02.004 | ||
8JXX | A | Amine | Histamine | H4 | Homo sapiens | Clobenpropit | - | Gi1/β1/γ2 | 3.06 | 2024-03-20 | 10.1038/s41467-024-46840-5 | |
8JXX (No Gprot) | A | Amine | Histamine | H4 | Homo sapiens | Clobenpropit | - | 3.06 | 2024-03-20 | 10.1038/s41467-024-46840-5 | ||
8JXW | A | Amine | Histamine | H4 | Homo sapiens | VUF6884 | - | Gi1/β1/γ2 | 3.01 | 2024-03-20 | 10.1038/s41467-024-46840-5 | |
8JXW (No Gprot) | A | Amine | Histamine | H4 | Homo sapiens | VUF6884 | - | 3.01 | 2024-03-20 | 10.1038/s41467-024-46840-5 | ||
8JXV | A | Amine | Histamine | H4 | Homo sapiens | Clozapine | - | Gi1/β1/γ2 | 3.21 | 2024-03-20 | 10.1038/s41467-024-46840-5 | |
8JXV (No Gprot) | A | Amine | Histamine | H4 | Homo sapiens | Clozapine | - | 3.21 | 2024-03-20 | 10.1038/s41467-024-46840-5 | ||
8JXT | A | Amine | Histamine | H4 | Homo sapiens | Histamine | PO4 | Gi1/β1/γ2 | 3.07 | 2024-03-20 | 10.1038/s41467-024-46840-5 | |
8JXT (No Gprot) | A | Amine | Histamine | H4 | Homo sapiens | Histamine | PO4 | 3.07 | 2024-03-20 | 10.1038/s41467-024-46840-5 | ||
8U4T | A | Protein | Chemokine | CXCR4 | Homo sapiens | REGN7663-Fab | - | - | 3.38 | 2024-03-13 | doi.org/10.1038/s41594-024-01397-1 | |
8U4T (Multimeric) | A | Protein | Chemokine | CXCR4 | Homo sapiens | REGN7663-Fab | - | 3.38 | 2024-03-13 | doi.org/10.1038/s41594-024-01397-1 | ||
8U4S | A | Protein | Chemokine | CXCR4 | Homo sapiens | REGN7663-Fab | - | - | 3.35 | 2024-03-13 | doi.org/10.1038/s41594-024-01397-1 | |
8U4S (Multimeric) | A | Protein | Chemokine | CXCR4 | Homo sapiens | REGN7663-Fab | - | 3.35 | 2024-03-13 | doi.org/10.1038/s41594-024-01397-1 | ||
8U4R | A | Protein | Chemokine | CXCR4 | Homo sapiens | REGN7663-Fab | Cholesterol | - | 3.1 | 2024-03-13 | 10.1101/2024.02.09.579708 | |
8U4Q | A | Protein | Chemokine | CXCR4 | Homo sapiens | REGN7663-Fab | Cholesterol | Gi1/β1/γ2 | 3.36 | 2024-03-13 | 10.1101/2024.02.09.579708 | |
8U4Q (No Gprot) | A | Protein | Chemokine | CXCR4 | Homo sapiens | REGN7663-Fab | Cholesterol | 3.36 | 2024-03-13 | 10.1101/2024.02.09.579708 | ||
8U4P | A | Protein | Chemokine | CXCR4 | Homo sapiens | AMD3100 | Cholesterol | Gi1/β1/γ2 | 3.15 | 2024-03-13 | 10.1101/2024.02.09.579708 | |
8U4P (No Gprot) | A | Protein | Chemokine | CXCR4 | Homo sapiens | AMD3100 | Cholesterol | 3.15 | 2024-03-13 | 10.1101/2024.02.09.579708 | ||
8U4O | A | Protein | Chemokine | CXCR4 | Homo sapiens | CXCL12 | Cholesterol | Gi1/β1/γ2 | 3.29 | 2024-03-13 | 10.1101/2024.02.09.579708 | |
8U4O (No Gprot) | A | Protein | Chemokine | CXCR4 | Homo sapiens | CXCL12 | Cholesterol | 3.29 | 2024-03-13 | 10.1101/2024.02.09.579708 | ||
8U4N | A | Protein | Chemokine | CXCR4 | Homo sapiens | - | Cholesterol | Gi1/β1/γ2 | 2.72 | 2024-03-13 | 10.1101/2024.02.09.579708 | |
8U4N (No Gprot) | A | Protein | Chemokine | CXCR4 | Homo sapiens | - | Cholesterol | 2.72 | 2024-03-13 | 10.1101/2024.02.09.579708 | ||
8GH1 | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | - | 4.1 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GH0 | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | - | 4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GGZ | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | - | 3.9 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GGY | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | - | 3.9 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GGX | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | - | 3.6 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GGW | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | - | 3.6 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GGV | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | - | 3.5 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GGU | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | - | 3.4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GGT | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | - | 3.5 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GGS | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | - | 3.5 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GGR | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | - | 3.4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GGQ | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | - | 3.4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GGP | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | - | 3.2 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GGO | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | - | 3.2 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GGN | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | - | 3.3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GGM | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | - | 3.2 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GGL | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | - | 3.2 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GGK | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | - | 3.3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GGJ | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | - | 3.5 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GGI | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | - | 3.5 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8WG8 | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | - | Peptide | chim(NtGi1-Gs)/β1/γ2 | 2.71 | 2024-03-06 | 10.1038/s41421-024-00649-0 | |
8WG8 (No Gprot) | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | - | Peptide | 2.71 | 2024-03-06 | 10.1038/s41421-024-00649-0 | ||
8JHN | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | MMF | - | Go/β1/γ2 | 3.75 | 2024-03-06 | 10.1038/s41467-024-46239-2 | |
8JHN (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | MMF | - | 3.75 | 2024-03-06 | 10.1038/s41467-024-46239-2 | ||
8JER | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | Acipimox | - | Go/β1/γ2 | 3.45 | 2024-03-06 | 10.1038/s41467-024-46239-2 | |
8JER (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | Acipimox | - | 3.45 | 2024-03-06 | 10.1038/s41467-024-46239-2 | ||
8IYW | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | GSK256073 | - | Go/β1/γ2 | 3.45 | 2024-03-06 | 10.1038/s41467-024-46239-2 | |
8IYW (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | GSK256073 | - | 3.45 | 2024-03-06 | 10.1038/s41467-024-46239-2 | ||
8IYH | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | MK6892 | - | Go/β1/γ2 | 3.3 | 2024-03-06 | 10.1038/s41467-024-46239-2 | |
8IYH (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | MK6892 | - | 3.3 | 2024-03-06 | 10.1038/s41467-024-46239-2 | ||
8IY9 | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | Niacin | - | Go/β1/γ2 | 3.37 | 2024-03-06 | 10.1038/s41467-024-46239-2 | |
8IY9 (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | Niacin | - | 3.37 | 2024-03-06 | 10.1038/s41467-024-46239-2 | ||
8UO4 | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP; Mg | Gs/β1/γ2 | 4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8UO4 (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP; Mg | 4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8UO3 | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP; Mg | Gs/β1/γ2 | 3.5 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8UO3 (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP; Mg | 3.5 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8UO2 | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.6 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8UO2 (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.6 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8UO1 | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP; Mg | Gs/β1/γ2 | 3.6 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8UO1 (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP; Mg | 3.6 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8UO0 | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.5 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8UO0 (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.5 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8UNZ | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.8 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8UNZ (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.8 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8UNY | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.6 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8UNY (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.6 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8UNX | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.6 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8UNX (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.6 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8UNW | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8UNW (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8UNV | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8UNV (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8UNU | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.5 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8UNU (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.5 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8UNT | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8UNT (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8UNS | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8UNS (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8UNR | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8UNR (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8UNQ | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8UNQ (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8UNP | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8UNP (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8UNO | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8UNO (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8UNN | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8UNN (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8UNM | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8UNM (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8UNL | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8UNL (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GGF | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.6 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GGF (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.6 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GGE | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.5 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GGE (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.5 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GGC | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GGC (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GGB | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.5 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GGB (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.5 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GGA | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.5 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GGA (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.5 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GG9 | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GG9 (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GG8 | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GG8 (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GG7 | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GG7 (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GG6 | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GG6 (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GG5 | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.2 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GG5 (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.2 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GG4 | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.2 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GG4 (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.2 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GG3 | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.1 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GG3 (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.1 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GG2 | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GG2 (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GG1 | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GG1 (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GG0 | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 2.9 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GG0 (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 2.9 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GFZ | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GFZ (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GFY | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GFY (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GFX | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GFX (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GFW | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GFW (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GFV | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | Gs/β1/γ2 | 3.1 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GFV (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | GTP | 3.1 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GEJ | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | Gs/β1/γ2 | 4.2 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GEJ (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | 4.2 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GEI | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | Gs/β1/γ2 | 4.1 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GEI (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | 4.1 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GEH | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | Gs/β1/γ2 | 4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GEH (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | 4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GEG | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | Gs/β1/γ2 | 3.8 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GEG (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | 3.8 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GEF | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | Gs/β1/γ2 | 3.8 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GEF (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | 3.8 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GEE | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | Gs/β1/γ2 | 3.7 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GEE (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | 3.7 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GED | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | Gs/β1/γ2 | 3.5 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GED (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | 3.5 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GEC | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | Gs/β1/γ2 | 3.5 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GEC (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | 3.5 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GEB | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | Gs/β1/γ2 | 3.6 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GEB (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | 3.6 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GEA | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | Gs/β1/γ2 | 3.5 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GEA (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | 3.5 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GE9 | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | Gs/β1/γ2 | 3.5 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GE9 (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | 3.5 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GE8 | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | Gs/β1/γ2 | 3.4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GE8 (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | 3.4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GE7 | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | Gs/β1/γ2 | 3.4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GE7 (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | 3.4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GE6 | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | Gs/β1/γ2 | 3.4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GE6 (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | 3.4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GE4 | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | Gs/β1/γ2 | 3.3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GE4 (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | 3.3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GE3 | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | Gs/β1/γ2 | 3.3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GE3 (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | 3.3 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GE1 | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | Gs/β1/γ2 | 3.4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GE1 (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | 3.4 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8GDZ | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | Gs/β1/γ2 | 3.5 | 2024-03-06 | 10.1038/s41586-024-07153-1 | |
8GDZ (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | 3.5 | 2024-03-06 | 10.1038/s41586-024-07153-1 | ||
8WA3 | B1 | Peptide | Glucagon | GIP | Homo sapiens | - | - | Gs/β1/γ2 | 2.86 | 2024-03-06 | 10.1038/s41421-024-00649-0 | |
8WA3 (No Gprot) | B1 | Peptide | Glucagon | GIP | Homo sapiens | - | - | 2.86 | 2024-03-06 | 10.1038/s41421-024-00649-0 | ||
8WG7 | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | - | - | Gs/β1/γ2 | 2.54 | 2024-03-06 | 10.1038/s41421-024-00649-0 | |
8WG7 (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | - | - | 2.54 | 2024-03-06 | 10.1038/s41421-024-00649-0 | ||
8U8F | A | Orphan | Orphan | GPR3 | Homo sapiens | Palmitic Acid | - | Gs/β1/γ2 | 3.49 | 2024-03-06 | 10.1021/acs.biochem.3c00647 | |
8U8F (No Gprot) | A | Orphan | Orphan | GPR3 | Homo sapiens | Palmitic Acid | - | 3.49 | 2024-03-06 | 10.1021/acs.biochem.3c00647 | ||
8POK | A | Amine | Histamine | H2 | Homo sapiens | Histamine | - | Gs/β1/γ2 | 3.4 | 2024-03-06 | 10.1038/s41467-024-46096-z | |
8POK (No Gprot) | A | Amine | Histamine | H2 | Homo sapiens | Histamine | - | 3.4 | 2024-03-06 | 10.1038/s41467-024-46096-z | ||
8X7A | A | Lipid | Prostanoid | I2 | Homo sapiens | Treprostinil | - | Gs/β1/γ2 | 2.56 | 2024-03-06 | 10.1126/sciadv.adk5184 | |
8X7A (No Gprot) | A | Lipid | Prostanoid | I2 | Homo sapiens | Treprostinil | - | 2.56 | 2024-03-06 | 10.1126/sciadv.adk5184 | ||
8X79 | A | Lipid | Prostanoid | I2 | Homo sapiens | MRE-269 | - | Gs/β1/γ2 | 2.41 | 2024-03-06 | 10.1126/sciadv.adk5184 | |
8X79 (No Gprot) | A | Lipid | Prostanoid | I2 | Homo sapiens | MRE-269 | - | 2.41 | 2024-03-06 | 10.1126/sciadv.adk5184 | ||
8JBF | A | Peptide | Tachykinin | NK3 | Homo sapiens | Senktide | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3 | 2024-02-28 | 10.1038/s41421-023-00564-w | |
8JBF (No Gprot) | A | Peptide | Tachykinin | NK3 | Homo sapiens | Senktide | - | 3 | 2024-02-28 | 10.1038/s41421-023-00564-w | ||
8JT8 | A | Amine | 5-Hydroxytryptamine | 5-HT2A | Homo sapiens | (R)-IHCH-7179 | - | - | 2.7 | 2024-02-28 | To be published | |
8WRZ | A | Lipid | Cannabinoid | CB1 | Homo sapiens | PubChem 102336704 | - | Arrestin2 | 3.6 | 2024-02-28 | 10.1093/procel/pwad055 | |
8XJK | A | Lipid | Prostanoid | FP-alpha | Homo sapiens | Cloprosetnol | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.63 | 2024-02-28 | doi.org/10.1016/j.celrep.2024.113893 | |
8XJK (No Gprot) | A | Lipid | Prostanoid | FP-alpha | Homo sapiens | Cloprosetnol | - | 2.63 | 2024-02-28 | doi.org/10.1016/j.celrep.2024.113893 | ||
8XJO | A | Lipid | Prostanoid | TP | Homo sapiens | U46619 | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.11 | 2024-02-28 | To be published | |
8XJO (No Gprot) | A | Lipid | Prostanoid | TP | Homo sapiens | U46619 | - | 3.11 | 2024-02-28 | To be published | ||
8XJN | A | Lipid | Prostanoid | TP | Homo sapiens | Cloprosetnol | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.06 | 2024-02-28 | doi.org/10.1016/j.celrep.2024.113893 | |
8XJN (No Gprot) | A | Lipid | Prostanoid | TP | Homo sapiens | Cloprosetnol | - | 3.06 | 2024-02-28 | doi.org/10.1016/j.celrep.2024.113893 | ||
8XJM | A | Lipid | Prostanoid | FP-alpha | Homo sapiens | Latanoprost | - | chim(NtGi2-Gs-CtGq)/β1/γ2 | 2.85 | 2024-02-28 | To be published | |
8XJM (No Gprot) | A | Lipid | Prostanoid | FP-alpha | Homo sapiens | Latanoprost | - | 2.85 | 2024-02-28 | To be published | ||
8XJL | A | Lipid | Prostanoid | FP-alpha | Homo sapiens | PGF2-α | - | chim(NtGi2-Gs-CtGq)/β1/γ2 | 2.77 | 2024-02-28 | To be published | |
8XJL (No Gprot) | A | Lipid | Prostanoid | FP-alpha | Homo sapiens | PGF2-α | - | 2.77 | 2024-02-28 | To be published | ||
8JT6 | A | Amine | 5-Hydroxytryptamine | 5-HT1A | Homo sapiens | (R)-IHCH-7179 | - | Gi1/β1/γ2 | 3 | 2024-02-28 | To be published | |
8JT6 (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT1A | Homo sapiens | (R)-IHCH-7179 | - | 3 | 2024-02-28 | To be published | ||
8GAG | A | Lipid | Cannabinoid | CB1 | Homo sapiens | PubChem 170838490 | - | Gi1/β1/γ2 | 3.3 | 2024-02-28 | To be published | |
8GAG (No Gprot) | A | Lipid | Cannabinoid | CB1 | Homo sapiens | PubChem 170838490 | - | 3.3 | 2024-02-28 | To be published | ||
8SMV | A | Orphan | Orphan | GPR161 | Homo sapiens | - | - | Gs/β1/γ2 | 2.74 | 2024-02-21 | 10.1038/s41594-024-01223-8 | |
8SMV (No Gprot) | A | Orphan | Orphan | GPR161 | Homo sapiens | - | - | 2.74 | 2024-02-21 | 10.1038/s41594-024-01223-8 | ||
8IKJ | B2 | Adhesion | Adhesion | ADGRE5 | Homo sapiens | - | - | - | 3.2 | 2024-02-14 | 10.1016/j.molcel.2023.12.020 | |
8IEP | C | Orphan | Orphan | GPR156 | Homo sapiens | A1LYA | - | - | 2.61 | 2024-02-14 | doi.org/10.1038/s41594-024-01224-7 | |
8IEI | C | Orphan | Orphan | GPR156 | Homo sapiens | A1LYA | - | - | 2.62 | 2024-02-14 | doi.org/10.1038/s41594-024-01224-7 | |
8IEB | C | Orphan | Orphan | GPR156 | Homo sapiens | A1LYA | - | - | 3.03 | 2024-02-14 | doi.org/10.1038/s41594-024-01224-7 | |
8K8J | A | Lipid | Cannabinoid | CB1 | Homo sapiens | Fenofibrate | - | chim(Gs-CtGq)/β1/γ2 | 2.88 | 2024-02-14 | 10.1002/advs.202306311 | |
8K8J (No Gprot) | A | Lipid | Cannabinoid | CB1 | Homo sapiens | Fenofibrate | - | 2.88 | 2024-02-14 | 10.1002/advs.202306311 | ||
8WW2 | A | Orphan | Orphan | GPR3 | Homo sapiens | - | - | chim(NtGi1-Gs)/β1/γ2 | 2.79 | 2024-02-14 | 10.1038/s41422-024-00932-5 | |
8WW2 (No Gprot) | A | Orphan | Orphan | GPR3 | Homo sapiens | - | - | 2.79 | 2024-02-14 | 10.1038/s41422-024-00932-5 | ||
8IED | C | Orphan | Orphan | GPR156 | Homo sapiens | A1LYA | - | Go/β1/γ2 | 3.33 | 2024-02-14 | doi.org/10.1038/s41594-024-01224-7 | |
8IED (No Gprot) | C | Orphan | Orphan | GPR156 | Homo sapiens | A1LYA | - | 3.33 | 2024-02-14 | doi.org/10.1038/s41594-024-01224-7 | ||
8SZF | C | Ion | Calcium Sensing | CaS | Homo sapiens | - | Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW | - | 2.8 | 2024-02-07 | 10.1038/s41586-024-07055-2 | |
8SZG | C | Ion | Calcium Sensing | CaS | Homo sapiens | - | Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW | chim(NtGi1-Gq)/β1/γ2 | 3.6 | 2024-02-07 | 10.1038/s41586-024-07055-2 | |
8SZG (No Gprot) | C | Ion | Calcium Sensing | CaS | Homo sapiens | - | Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW | 3.6 | 2024-02-07 | 10.1038/s41586-024-07055-2 | ||
8JBH | A | Peptide | Tachykinin | NK3 | Homo sapiens | Substance-P | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.9 | 2024-02-07 | doi.org/10.1038/s41421-023-00564-w | |
8JBH (No Gprot) | A | Peptide | Tachykinin | NK3 | Homo sapiens | Substance-P | - | 2.9 | 2024-02-07 | doi.org/10.1038/s41421-023-00564-w | ||
8JBG | A | Peptide | Tachykinin | NK3 | Homo sapiens | Neurokinin-B | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.8 | 2024-02-07 | doi.org/10.1038/s41421-023-00564-w | |
8JBG (No Gprot) | A | Peptide | Tachykinin | NK3 | Homo sapiens | Neurokinin-B | - | 2.8 | 2024-02-07 | doi.org/10.1038/s41421-023-00564-w | ||
8SZH | C | Ion | Calcium Sensing | CaS | Homo sapiens | - | Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW | Gi1/β1/γ2 | 3.1 | 2024-02-07 | 10.1038/s41586-024-07055-2 | |
8SZH (No Gprot) | C | Ion | Calcium Sensing | CaS | Homo sapiens | - | Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW | 3.1 | 2024-02-07 | 10.1038/s41586-024-07055-2 | ||
8KFZ | A | Protein | Chemokine | CCR8 | Homo sapiens | - | - | Gi1/β1/γ2 | 3.3 | 2024-02-07 | 10.1126/sciadv.adj7500 | |
8KFZ (No Gprot) | A | Protein | Chemokine | CCR8 | Homo sapiens | - | - | 3.3 | 2024-02-07 | 10.1126/sciadv.adj7500 | ||
8KFY | A | Protein | Chemokine | CCR8 | Homo sapiens | ZK-756326 | - | Gi1/β1/γ2 | 3.06 | 2024-02-07 | 10.1126/sciadv.adj7500 | |
8KFY (No Gprot) | A | Protein | Chemokine | CCR8 | Homo sapiens | ZK-756326 | - | 3.06 | 2024-02-07 | 10.1126/sciadv.adj7500 | ||
8KFX | A | Protein | Chemokine | CCR8 | Homo sapiens | LMD-009 | - | Gi1/β1/γ2 | 2.96 | 2024-02-07 | 10.1126/sciadv.adj7500 | |
8KFX (No Gprot) | A | Protein | Chemokine | CCR8 | Homo sapiens | LMD-009 | - | 2.96 | 2024-02-07 | 10.1126/sciadv.adj7500 | ||
8I7W | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | GSK256073 | - | Gi1/β1/γ2 | 3.39 | 2024-02-07 | 10.1038/s41467-023-42764-8 | |
8I7W (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | GSK256073 | - | 3.39 | 2024-02-07 | 10.1038/s41467-023-42764-8 | ||
8I7V | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | Acipimox | - | Gi1/β1/γ2 | 2.77 | 2024-02-07 | 10.1038/s41467-023-42764-8 | |
8I7V (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | Acipimox | - | 2.77 | 2024-02-07 | 10.1038/s41467-023-42764-8 | ||
8SZI | C | Ion | Calcium Sensing | CaS | Homo sapiens | - | Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW | Gi3/β1/γ2 | 3.5 | 2024-02-07 | 10.1038/s41586-024-07055-2 | |
8SZI (No Gprot) | C | Ion | Calcium Sensing | CaS | Homo sapiens | - | Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW | 3.5 | 2024-02-07 | 10.1038/s41586-024-07055-2 | ||
8IQ6 | A | Lipid | Prostanoid | FP-alpha | Homo sapiens | Latanoprost | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.4 | 2024-01-31 | 10.1038/s41467-023-43922-8 | |
8IQ6 (No Gprot) | A | Lipid | Prostanoid | FP-alpha | Homo sapiens | Latanoprost | - | 3.4 | 2024-01-31 | 10.1038/s41467-023-43922-8 | ||
8IQ4 | A | Lipid | Prostanoid | FP-alpha | Homo sapiens | Carboprost | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.7 | 2024-01-31 | 10.1038/s41467-023-43922-8 | |
8IQ4 (No Gprot) | A | Lipid | Prostanoid | FP-alpha | Homo sapiens | Carboprost | - | 2.7 | 2024-01-31 | 10.1038/s41467-023-43922-8 | ||
8IKL | B2 | Adhesion | Adhesion | ADGRE5 | Homo sapiens | - | - | chim(NtGi1L-G13)/β1/γ2 | 2.33 | 2024-01-24 | 10.1016/j.molcel.2023.12.020 | |
8IKL (No Gprot) | B2 | Adhesion | Adhesion | ADGRE5 | Homo sapiens | - | - | 2.33 | 2024-01-24 | 10.1016/j.molcel.2023.12.020 | ||
8T3V | A | Lipid | Free Fatty Acid | FFA1 | Homo sapiens | Docosa-4,7,10,13,16,19-Hexaenoic acid | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 3.39 | 2024-01-24 | 10.1126/sciadv.adj2384 | |
8T3V (No Gprot) | A | Lipid | Free Fatty Acid | FFA1 | Homo sapiens | Docosa-4,7,10,13,16,19-Hexaenoic acid | - | 3.39 | 2024-01-24 | 10.1126/sciadv.adj2384 | ||
8T3S | A | Lipid | Free Fatty Acid | FFA2 | Homo sapiens | Butyric acid | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 3.07 | 2024-01-24 | 10.1126/sciadv.adj2384 | |
8T3S (No Gprot) | A | Lipid | Free Fatty Acid | FFA2 | Homo sapiens | Butyric acid | - | 3.07 | 2024-01-24 | 10.1126/sciadv.adj2384 | ||
8T3Q | A | Lipid | Free Fatty Acid | FFA4 | Homo sapiens | Docosa-4,7,10,13,16,19-Hexaenoic acid | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 3.14 | 2024-01-24 | 10.1126/sciadv.adj2384 | |
8T3Q (No Gprot) | A | Lipid | Free Fatty Acid | FFA4 | Homo sapiens | Docosa-4,7,10,13,16,19-Hexaenoic acid | - | 3.14 | 2024-01-24 | 10.1126/sciadv.adj2384 | ||
8J24 | A | Lipid | Free Fatty Acid | FFA2 | Homo sapiens | Acetic acid | - | Gi1/β1/γ2 | 2.6 | 2024-01-24 | 10.1038/s41422-023-00914-z | |
8J24 (No Gprot) | A | Lipid | Free Fatty Acid | FFA2 | Homo sapiens | Acetic acid | - | 2.6 | 2024-01-24 | 10.1038/s41422-023-00914-z | ||
8J22 | A | Lipid | Free Fatty Acid | FFA2 | Homo sapiens | TUG-1375 | - | Gi1/β1/γ2 | 3.2 | 2024-01-24 | 10.1038/s41422-023-00914-z | |
8J22 (No Gprot) | A | Lipid | Free Fatty Acid | FFA2 | Homo sapiens | TUG-1375 | - | 3.2 | 2024-01-24 | 10.1038/s41422-023-00914-z | ||
8J21 | A | Lipid | Free Fatty Acid | FFA3 | Homo sapiens | Butyric acid | - | Gi1/β1/γ2 | 3.3 | 2024-01-24 | 10.1038/s41422-023-00914-z | |
8J21 (No Gprot) | A | Lipid | Free Fatty Acid | FFA3 | Homo sapiens | Butyric acid | - | 3.3 | 2024-01-24 | 10.1038/s41422-023-00914-z | ||
8J20 | A | Lipid | Free Fatty Acid | FFA3 | Homo sapiens | Valeric acid | AR420626 | Gi1/β1/γ2 | 3.2 | 2024-01-24 | 10.1038/s41422-023-00914-z | |
8J20 (No Gprot) | A | Lipid | Free Fatty Acid | FFA3 | Homo sapiens | Valeric acid | AR420626 | 3.2 | 2024-01-24 | 10.1038/s41422-023-00914-z | ||
8WDT | A | Nucleotide | Adenosine | A2A | Homo sapiens | photoNECA | - | - | 3.34 | 2024-01-17 | doi.org/10.1016/j.bbrc.2023.149393 | |
8J9O | F | Protein | Frizzled | FZD1 | Homo sapiens | - | - | - | 3.4 | 2024-01-17 | 10.1038/s41421-023-00627-y | |
8JHC | F | Protein | Frizzled | FZD3 | Homo sapiens | - | - | - | 3.3 | 2024-01-17 | 10.1038/s41421-023-00627-y | |
8JH7 | F | Protein | Frizzled | FZD6 | Homo sapiens | - | - | - | 3.2 | 2024-01-17 | 10.1038/s41421-023-00627-y | |
8X64 | A | Amine | Histamine | H1 | Homo sapiens | Desloratadine | - | - | 3.4 | 2024-01-17 | 10.1038/s41467-023-44477-4 | |
8X63 | A | Amine | Histamine | H1 | Homo sapiens | Mepyramine | - | - | 3.2 | 2024-01-17 | 10.1038/s41467-023-44477-4 | |
8X5Y | A | Amine | Histamine | H1 | Homo sapiens | Astemizole | - | - | 3 | 2024-01-17 | 10.1038/s41467-023-44477-4 | |
8X5X | A | Amine | Histamine | H1 | Homo sapiens | - | - | - | 3.5 | 2024-01-17 | 10.1038/s41467-023-44477-4 | |
8J9N | F | Protein | Frizzled | FZD1 | Homo sapiens | - | - | chim(Gs-CtGq)/β1/γ2 | 3.5 | 2024-01-17 | 10.1038/s41421-023-00627-y | |
8J9N (No Gprot) | F | Protein | Frizzled | FZD1 | Homo sapiens | - | - | 3.5 | 2024-01-17 | 10.1038/s41421-023-00627-y | ||
8T3O | A | Lipid | Free Fatty Acid | FFA4 | Homo sapiens | TUG-891 | 2Y5 | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 3.06 | 2024-01-17 | 10.1126/sciadv.adj2384 | |
8T3O (No Gprot) | A | Lipid | Free Fatty Acid | FFA4 | Homo sapiens | TUG-891 | 2Y5 | 3.06 | 2024-01-17 | 10.1126/sciadv.adj2384 | ||
8JHI | F | Protein | Frizzled | FZD3 | Homo sapiens | - | - | chim(NtGsXLas-Gs)/β1/γ2 | 3.2 | 2024-01-17 | 10.1038/s41421-023-00627-y | |
8JHI (No Gprot) | F | Protein | Frizzled | FZD3 | Homo sapiens | - | - | 3.2 | 2024-01-17 | 10.1038/s41421-023-00627-y | ||
8JHB | F | Protein | Frizzled | FZD6 | Homo sapiens | - | - | chim(NtGsXLas-Gs)/β1/γ2 | 3.3 | 2024-01-17 | 10.1038/s41421-023-00627-y | |
8JHB (No Gprot) | F | Protein | Frizzled | FZD6 | Homo sapiens | - | - | 3.3 | 2024-01-17 | 10.1038/s41421-023-00627-y | ||
8JGF | A | Orphan | Orphan | MRGPRX1 | Homo sapiens | BAM8-22 | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.7 | 2024-01-10 | 10.1038/s41467-023-40705-z | |
8JGF (No Gprot) | A | Orphan | Orphan | MRGPRX1 | Homo sapiens | BAM8-22 | - | 2.7 | 2024-01-10 | 10.1038/s41467-023-40705-z | ||
8J6J | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | GSK256073 | - | Gi1/β1/γ2 | 2.8 | 2024-01-10 | 10.1016/j.celrep.2023.113406 | |
8J6J (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | GSK256073 | - | 2.8 | 2024-01-10 | 10.1016/j.celrep.2023.113406 | ||
8JGG | A | Orphan | Orphan | MRGPRX1 | Homo sapiens | BAM8-22 | - | Gi1/β1/γ2 | 3 | 2024-01-10 | 10.1038/s41467-023-40705-z | |
8JGG (No Gprot) | A | Orphan | Orphan | MRGPRX1 | Homo sapiens | BAM8-22 | - | 3 | 2024-01-10 | 10.1038/s41467-023-40705-z | ||
8JGB | A | Orphan | Orphan | MRGPRX1 | Homo sapiens | Conorfamide-Tx2 | - | Gi1/β1/γ2 | 2.84 | 2024-01-10 | 10.1038/s41467-023-40705-z | |
8JGB (No Gprot) | A | Orphan | Orphan | MRGPRX1 | Homo sapiens | Conorfamide-Tx2 | - | 2.84 | 2024-01-10 | 10.1038/s41467-023-40705-z | ||
8UHB | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | RO5256390 | - | Gs/β1/γ2 | 3.35 | 2024-01-10 | 10.1038/s41467-023-44601-4 | |
8UHB (No Gprot) | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | RO5256390 | - | 3.35 | 2024-01-10 | 10.1038/s41467-023-44601-4 | ||
8W8S | A | Orphan | Orphan | GPR101 | Homo sapiens | - | AA-14 | - | 3.3 | 2024-01-03 | 10.1038/s41589-023-01456-6 | |
8W8R | A | Orphan | Orphan | GPR101 | Homo sapiens | - | AA-14 | chim(NtGi1-Gs)/β1/γ2 | 3.3 | 2024-01-03 | 10.1038/s41589-023-01456-6 | |
8W8R (No Gprot) | A | Orphan | Orphan | GPR101 | Homo sapiens | - | AA-14 | 3.3 | 2024-01-03 | 10.1038/s41589-023-01456-6 | ||
8GDC | A | Lipid | Prostanoid | EP3 | Homo sapiens | PGE2 | - | Gi1/β1/γ2 | 3.5 | 2024-01-03 | 10.1073/pnas.2216329120 | |
8GDC (No Gprot) | A | Lipid | Prostanoid | EP3 | Homo sapiens | PGE2 | - | 3.5 | 2024-01-03 | 10.1073/pnas.2216329120 | ||
8GCP | A | Lipid | Prostanoid | EP4 | Homo sapiens | PGE2 | - | Gi1/β1/γ2 | 3.1 | 2024-01-03 | 10.1073/pnas.2216329120 | |
8GCP (No Gprot) | A | Lipid | Prostanoid | EP4 | Homo sapiens | PGE2 | - | 3.1 | 2024-01-03 | 10.1073/pnas.2216329120 | ||
8GCM | A | Lipid | Prostanoid | EP4 | Homo sapiens | L902688 | - | Gi1/β1/γ2 | 3.5 | 2024-01-03 | 10.1073/pnas.2216329120 | |
8GCM (No Gprot) | A | Lipid | Prostanoid | EP4 | Homo sapiens | L902688 | - | 3.5 | 2024-01-03 | 10.1073/pnas.2216329120 | ||
8IJD | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | MK6892 | - | Gi1/β1/γ2 | 3.25 | 2024-01-03 | 10.1038/s41421-023-00610-7 | |
8IJD (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | MK6892 | - | 3.25 | 2024-01-03 | 10.1038/s41421-023-00610-7 | ||
8IJB | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | Acipimox | - | Gi1/β1/γ2 | 3.23 | 2024-01-03 | 10.1038/s41421-023-00610-7 | |
8IJB (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | Acipimox | - | 3.23 | 2024-01-03 | 10.1038/s41421-023-00610-7 | ||
8IJA | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | Niacin | - | Gi1/β1/γ2 | 2.69 | 2024-01-03 | 10.1038/s41421-023-00610-7 | |
8IJA (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | Niacin | - | 2.69 | 2024-01-03 | 10.1038/s41421-023-00610-7 | ||
8IJ3 | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | - | - | Gi1/β1/γ2 | 3.28 | 2024-01-03 | 10.1038/s41421-023-00610-7 | |
8IJ3 (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | - | - | 3.28 | 2024-01-03 | 10.1038/s41421-023-00610-7 | ||
8GDB | A | Lipid | Prostanoid | EP4 | Homo sapiens | PGE2 | - | Gs/β1/γ2 | 3.1 | 2024-01-03 | 10.1073/pnas.2216329120 | |
8GDB (No Gprot) | A | Lipid | Prostanoid | EP4 | Homo sapiens | PGE2 | - | 3.1 | 2024-01-03 | 10.1073/pnas.2216329120 | ||
8GDA | A | Lipid | Prostanoid | EP4 | Homo sapiens | L902688 | - | Gs/β1/γ2 | 3.3 | 2024-01-03 | 10.1073/pnas.2216329120 | |
8GDA (No Gprot) | A | Lipid | Prostanoid | EP4 | Homo sapiens | L902688 | - | 3.3 | 2024-01-03 | 10.1073/pnas.2216329120 | ||
8GD9 | A | Lipid | Prostanoid | EP4 | Homo sapiens | Rivenprost | - | Gs/β1/γ2 | 3.2 | 2024-01-03 | 10.1073/pnas.2216329120 | |
8GD9 (No Gprot) | A | Lipid | Prostanoid | EP4 | Homo sapiens | Rivenprost | - | 3.2 | 2024-01-03 | 10.1073/pnas.2216329120 | ||
8W8Q | A | Orphan | Orphan | GPR101 | Homo sapiens | - | - | Gs/β1/γ2 | 2.89 | 2024-01-03 | 10.1038/s41589-023-01456-6 | |
8W8Q (No Gprot) | A | Orphan | Orphan | GPR101 | Homo sapiens | - | - | 2.89 | 2024-01-03 | 10.1038/s41589-023-01456-6 | ||
8XBI | A | Orphan | Orphan | GPR34 | Homo sapiens | S3E-LysoPS | - | - | 3.06 | 2023-12-27 | To be published | |
8QOT | A | Peptide | Opioid | μ | Mus musculus | Nanobody-E | - | - | 3.2 | 2023-12-27 | 10.1101/2023.12.06.570395 | |
8WCC | A | Amine | Trace Amine Receptors | TA1 | Mus musculus | Cyclohexylammonium Ion | - | - | 3.04 | 2023-12-27 | 10.1016/j.cell.2023.10.014 | |
8WCB | A | Amine | Trace Amine Receptors | TA1 | Mus musculus | Cyclohexylammonium Ion | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.1 | 2023-12-27 | 10.1016/j.cell.2023.10.014 | |
8WCB (No Gprot) | A | Amine | Trace Amine Receptors | TA1 | Mus musculus | Cyclohexylammonium Ion | - | 3.1 | 2023-12-27 | 10.1016/j.cell.2023.10.014 | ||
8WC9 | A | Amine | Trace Amine Receptors | TA1 | Mus musculus | ZH8651 | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.2 | 2023-12-27 | 10.1016/j.cell.2023.10.014 | |
8WC9 (No Gprot) | A | Amine | Trace Amine Receptors | TA1 | Mus musculus | ZH8651 | - | 3.2 | 2023-12-27 | 10.1016/j.cell.2023.10.014 | ||
8WCA | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | 2-Phenylethylamine | - | chim(NtGi1-Gs)/β1/γ2 | 3.48 | 2023-12-27 | 10.1016/j.cell.2023.10.014 | |
8WCA (No Gprot) | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | 2-Phenylethylamine | - | 3.48 | 2023-12-27 | 10.1016/j.cell.2023.10.014 | ||
8WC8 | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | ZH8651 | - | chim(NtGi1-Gs)/β1/γ2 | 2.9 | 2023-12-27 | 10.1016/j.cell.2023.10.014 | |
8WC8 (No Gprot) | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | ZH8651 | - | 2.9 | 2023-12-27 | 10.1016/j.cell.2023.10.014 | ||
8WC7 | A | Amine | Trace Amine Receptors | TA1 | Mus musculus | ZH8667 | - | chim(NtGi1-Gs)/β1/γ2 | 3.1 | 2023-12-27 | 10.1016/j.cell.2023.10.014 | |
8WC7 (No Gprot) | A | Amine | Trace Amine Receptors | TA1 | Mus musculus | ZH8667 | - | 3.1 | 2023-12-27 | 10.1016/j.cell.2023.10.014 | ||
8WC6 | A | Amine | Trace Amine Receptors | TA1 | Mus musculus | 2-Phenylethylamine | - | chim(NtGi1-Gs)/β1/γ2 | 3.2 | 2023-12-27 | 10.1016/j.cell.2023.10.014 | |
8WC6 (No Gprot) | A | Amine | Trace Amine Receptors | TA1 | Mus musculus | 2-Phenylethylamine | - | 3.2 | 2023-12-27 | 10.1016/j.cell.2023.10.014 | ||
8WC5 | A | Amine | Trace Amine Receptors | TA1 | Mus musculus | Tetramethylammonium Ion | - | chim(NtGi1-Gs)/β1/γ2 | 3.3 | 2023-12-27 | 10.1016/j.cell.2023.10.014 | |
8WC5 (No Gprot) | A | Amine | Trace Amine Receptors | TA1 | Mus musculus | Tetramethylammonium Ion | - | 3.3 | 2023-12-27 | 10.1016/j.cell.2023.10.014 | ||
8WC4 | A | Amine | Trace Amine Receptors | TA1 | Mus musculus | ZH8651 | - | chim(NtGi1-Gs)/β1/γ2 | 3.1 | 2023-12-27 | 10.1016/j.cell.2023.10.014 | |
8WC4 (No Gprot) | A | Amine | Trace Amine Receptors | TA1 | Mus musculus | ZH8651 | - | 3.1 | 2023-12-27 | 10.1016/j.cell.2023.10.014 | ||
8WC3 | A | Amine | Trace Amine Receptors | TA1 | Mus musculus | SEP-363856 | - | chim(NtGi1-Gs)/β1/γ2 | 3 | 2023-12-27 | 10.1016/j.cell.2023.10.014 | |
8WC3 (No Gprot) | A | Amine | Trace Amine Receptors | TA1 | Mus musculus | SEP-363856 | - | 3 | 2023-12-27 | 10.1016/j.cell.2023.10.014 | ||
8XBH | A | Orphan | Orphan | GPR34 | Homo sapiens | S3E-LysoPS | - | Gi1/β1/γ2 | 2.83 | 2023-12-27 | To be published | |
8XBH (No Gprot) | A | Orphan | Orphan | GPR34 | Homo sapiens | S3E-LysoPS | - | 2.83 | 2023-12-27 | To be published | ||
8HJ1 | A | Orphan | Orphan | GPR21 | Homo sapiens | - | - | Gs/β1/γ2 | 3.27 | 2023-12-27 | 10.1038/s41467-023-35882-w | |
8HJ1 (No Gprot) | A | Orphan | Orphan | GPR21 | Homo sapiens | - | - | 3.27 | 2023-12-27 | 10.1038/s41467-023-35882-w | ||
8HN1 | A | Amine | Adrenergic | Alpha1A | Homo sapiens | Toxin AdTx1 | - | - | 2.9 | 2023-12-20 | To be published | |
8TLM | A | Protein | Chemokine | CCR8 | Homo sapiens | Anti-murine CCR8 antibody | - | - | 3.9 | 2023-12-20 | 10.1038/s41467-023-43601-8 | |
8W77 | O1 | Odorant receptors | Odorant family 52 | OR52C | Homo sapiens | - | - | - | 3.61 | 2023-12-20 | 10.1038/s41467-023-43983-9 | |
8J46 | O1 | Odorant receptors | Odorant family 52 | OR52C | Homo sapiens | - | - | - | 3.66 | 2023-12-20 | 10.1038/s41467-023-43983-9 | |
8U1U | A | Protein | Chemokine | CCR8 | Homo sapiens | CCL1 | - | Gi1/β1/γ2 | 3.1 | 2023-12-20 | 10.1038/s41467-023-43601-8 | |
8U1U (No Gprot) | A | Protein | Chemokine | CCR8 | Homo sapiens | CCL1 | - | 3.1 | 2023-12-20 | 10.1038/s41467-023-43601-8 | ||
8HOC | A | Amine | Histamine | H4 | Homo sapiens | Imetit | - | Gi1/β1/γ2 | 3 | 2023-12-20 | To be published | |
8HOC (No Gprot) | A | Amine | Histamine | H4 | Homo sapiens | Imetit | - | 3 | 2023-12-20 | To be published | ||
8HN8 | A | Amine | Histamine | H4 | Homo sapiens | Histamine | - | Gi1/β1/γ2 | 3 | 2023-12-20 | To be published | |
8HN8 (No Gprot) | A | Amine | Histamine | H4 | Homo sapiens | Histamine | - | 3 | 2023-12-20 | To be published | ||
8HTI | O1 | Odorant receptors | Odorant family 52 | OR52C | Homo sapiens | Ocatnoic acid | - | Gs/β1/γ2 | 2.97 | 2023-12-20 | 10.1038/s41467-023-43983-9 | |
8HTI (No Gprot) | O1 | Odorant receptors | Odorant family 52 | OR52C | Homo sapiens | Ocatnoic acid | - | 2.97 | 2023-12-20 | 10.1038/s41467-023-43983-9 | ||
8IA7 | A | Peptide | Cholecystokinin | CCKB | Homo sapiens | Cholecystokinin-8 | - | chim(NtGi1L-Gq)/β1/γ2 | 3.1 | 2023-12-06 | 10.1038/s41421-022-00420-3 | |
8IA7 (No Gprot) | A | Peptide | Cholecystokinin | CCKB | Homo sapiens | Cholecystokinin-8 | - | 3.1 | 2023-12-06 | 10.1038/s41421-022-00420-3 | ||
8J6R | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | MK6892 | - | Gi1/β1/γ2 | 2.76 | 2023-12-06 | 10.1038/s41467-023-43537-z | |
8J6R (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | MK6892 | - | 2.76 | 2023-12-06 | 10.1038/s41467-023-43537-z | ||
8J6Q | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | β-Hydroxybutyrate | Compound 9n | Gi1/β1/γ2 | 2.6 | 2023-12-06 | 10.1038/s41467-023-43537-z | |
8J6Q (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | β-Hydroxybutyrate | Compound 9n | 2.6 | 2023-12-06 | 10.1038/s41467-023-43537-z | ||
8J6P | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | Niacin | Compound 9n | Gi1/β1/γ2 | 2.55 | 2023-12-06 | 10.1038/s41467-023-43537-z | |
8J6P (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | Niacin | Compound 9n | 2.55 | 2023-12-06 | 10.1038/s41467-023-43537-z | ||
8FEG | A | Peptide | Opioid | κ | Homo sapiens | (DNCP)-β-Naloxamine | - | Gi1/β1/γ2 | 2.54 | 2023-12-06 | 10.1038/s41467-023-43718-w | |
8FEG (No Gprot) | A | Peptide | Opioid | κ | Homo sapiens | (DNCP)-β-Naloxamine | - | 2.54 | 2023-12-06 | 10.1038/s41467-023-43718-w | ||
8K2W | A | Protein | Chemokine | CXCR3 | Homo sapiens | AMG487 | - | - | 3 | 2023-11-29 | 10.1038/s41594-023-01175-5 | |
8HNN | A | Protein | Chemokine | CXCR3 | Homo sapiens | SCH546738 | - | - | 3.6 | 2023-11-29 | 10.1038/s41594-023-01175-5 | |
8K2X | A | Protein | Chemokine | CXCR3 | Homo sapiens | CXCL10 | - | Gi1/β1/γ2 | 3.2 | 2023-11-29 | 10.1038/s41594-023-01175-5 | |
8K2X (No Gprot) | A | Protein | Chemokine | CXCR3 | Homo sapiens | CXCL10 | - | 3.2 | 2023-11-29 | 10.1038/s41594-023-01175-5 | ||
8HNM | A | Protein | Chemokine | CXCR3 | Homo sapiens | VUF11222 | - | Gi1/β1/γ2 | 2.94 | 2023-11-29 | 10.1038/s41594-023-01175-5 | |
8HNM (No Gprot) | A | Protein | Chemokine | CXCR3 | Homo sapiens | VUF11222 | - | 2.94 | 2023-11-29 | 10.1038/s41594-023-01175-5 | ||
8HNL | A | Protein | Chemokine | CXCR3 | Homo sapiens | PS372424 | - | Gi1/β1/γ2 | 2.98 | 2023-11-29 | 10.1038/s41594-023-01175-5 | |
8HNL (No Gprot) | A | Protein | Chemokine | CXCR3 | Homo sapiens | PS372424 | - | 2.98 | 2023-11-29 | 10.1038/s41594-023-01175-5 | ||
8HNK | A | Protein | Chemokine | CXCR3 | Homo sapiens | CXCL11 | - | Gi1/β1/γ2 | 3.01 | 2023-11-29 | 10.1038/s41594-023-01175-5 | |
8HNK (No Gprot) | A | Protein | Chemokine | CXCR3 | Homo sapiens | CXCL11 | - | 3.01 | 2023-11-29 | 10.1038/s41594-023-01175-5 | ||
8K5D | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | GSK256073 | - | - | 3.74 | 2023-11-22 | 10.1038/s41467-023-42764-8 | |
8K5C | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | Acipimox | - | - | 3.13 | 2023-11-22 | 10.1038/s41467-023-42764-8 | |
8K5B | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | Niacin | - | - | 3.43 | 2023-11-22 | 10.1038/s41467-023-42764-8 | |
8WPG | C | Ion | Calcium Sensing | CaS | Homo sapiens | - | Tryptophan; Cinacalcet; PO4; Ca | - | 2.7 | 2023-11-22 | 10.1038/s41422-023-00892-2 | |
8W8A | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | RO5256390 | - | chim(NtGi1L-Gs)/β1/γ2 | 2.8 | 2023-11-22 | 10.1038/s41586-023-06775-1 | |
8W8A (No Gprot) | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | RO5256390 | - | 2.8 | 2023-11-22 | 10.1038/s41586-023-06775-1 | ||
8W89 | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | PEA | - | chim(NtGi1L-Gs)/β1/γ2 | 3 | 2023-11-22 | 10.1038/s41586-023-06775-1 | |
8W89 (No Gprot) | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | PEA | - | 3 | 2023-11-22 | 10.1038/s41586-023-06775-1 | ||
8W87 | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | METH | - | chim(NtGi1L-Gs)/β1/γ2 | 2.8 | 2023-11-22 | 10.1038/s41586-023-06775-1 | |
8W87 (No Gprot) | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | METH | - | 2.8 | 2023-11-22 | 10.1038/s41586-023-06775-1 | ||
8WPU | C | Ion | Calcium Sensing | CaS | Homo sapiens | - | Tryptophan; Cinacalcet; PO4; Ca | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 3.1 | 2023-11-22 | 10.1038/s41422-023-00892-2 | |
8WPU (No Gprot) | C | Ion | Calcium Sensing | CaS | Homo sapiens | - | Tryptophan; Cinacalcet; PO4; Ca | 3.1 | 2023-11-22 | 10.1038/s41422-023-00892-2 | ||
8W8B | A | Amine | 5-Hydroxytryptamine | 5-HT1A | Homo sapiens | SEP-363856 | - | Gi1/β1/γ2 | 3 | 2023-11-22 | 10.1038/s41586-023-06775-1 | |
8W8B (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT1A | Homo sapiens | SEP-363856 | - | 3 | 2023-11-22 | 10.1038/s41586-023-06775-1 | ||
8W88 | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | SEP-363856 | - | Gs/β1/γ2 | 2.6 | 2023-11-22 | 10.1038/s41586-023-06775-1 | |
8W88 (No Gprot) | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | SEP-363856 | - | 2.6 | 2023-11-22 | 10.1038/s41586-023-06775-1 | ||
8JSO | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | AMPH | - | chim(NtGi1-Gs)/β1/γ2 | 3.4 | 2023-11-15 | 10.1038/s41586-023-06804-z | |
8JSO (No Gprot) | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | AMPH | - | 3.4 | 2023-11-15 | 10.1038/s41586-023-06804-z | ||
8JLR | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | A77636 | - | chim(NtGi1-Gs)/β1/γ2 | 3 | 2023-11-15 | 10.1038/s41586-023-06804-z | |
8JLR (No Gprot) | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | A77636 | - | 3 | 2023-11-15 | 10.1038/s41586-023-06804-z | ||
8JLK | A | Amine | Trace Amine Receptors | TA1 | Mus musculus | Ulotaront | - | chim(NtGi1-Gs)/β1/γ2 | 3.22 | 2023-11-15 | 10.1038/s41586-023-06804-z | |
8JLK (No Gprot) | A | Amine | Trace Amine Receptors | TA1 | Mus musculus | Ulotaront | - | 3.22 | 2023-11-15 | 10.1038/s41586-023-06804-z | ||
8JLJ | A | Amine | Trace Amine Receptors | TA1 | Mus musculus | T1AM | - | chim(NtGi1-Gs)/β1/γ2 | 3.1 | 2023-11-15 | 10.1038/s41586-023-06804-z | |
8JLJ (No Gprot) | A | Amine | Trace Amine Receptors | TA1 | Mus musculus | T1AM | - | 3.1 | 2023-11-15 | 10.1038/s41586-023-06804-z | ||
8JSP | A | Amine | 5-Hydroxytryptamine | 5-HT1A | Homo sapiens | Ulotaront | - | Gi1/β1/γ2 | 3.65 | 2023-11-15 | 10.1038/s41586-023-06804-z | |
8JSP (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT1A | Homo sapiens | Ulotaront | - | 3.65 | 2023-11-15 | 10.1038/s41586-023-06804-z | ||
8U26 | A | Peptide | Tachykinin | NK1 | Homo sapiens | Protachykinin-1 | - | Gs/β1/γ2 | 2.5 | 2023-11-15 | 10.1038/s41592-023-02082-9 | |
8U26 (No Gprot) | A | Peptide | Tachykinin | NK1 | Homo sapiens | Protachykinin-1 | - | 2.5 | 2023-11-15 | 10.1038/s41592-023-02082-9 | ||
8JLQ | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | Fenoldopam | - | Gs/β1/γ2 | 2.84 | 2023-11-15 | 10.1038/s41586-023-06804-z | |
8JLQ (No Gprot) | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | Fenoldopam | - | 2.84 | 2023-11-15 | 10.1038/s41586-023-06804-z | ||
8JLP | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | Ralmitaront | - | Gs/β1/γ2 | 3.23 | 2023-11-15 | 10.1038/s41586-023-06804-z | |
8JLP (No Gprot) | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | Ralmitaront | - | 3.23 | 2023-11-15 | 10.1038/s41586-023-06804-z | ||
8JLO | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | Ulotaront | - | Gs/β1/γ2 | 3.52 | 2023-11-15 | 10.1038/s41586-023-06804-z | |
8JLO (No Gprot) | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | Ulotaront | - | 3.52 | 2023-11-15 | 10.1038/s41586-023-06804-z | ||
8JLN | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | T1AM | - | Gs/β1/γ2 | 3.24 | 2023-11-15 | 10.1038/s41586-023-06804-z | |
8JLN (No Gprot) | A | Amine | Trace Amine Receptors | TA1 | Homo sapiens | T1AM | - | 3.24 | 2023-11-15 | 10.1038/s41586-023-06804-z | ||
8JIS | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Peptide-15 | - | chim(NtGi1-Gs)/β1/γ2 | 2.46 | 2023-11-08 | 10.1073/pnas.2303696120 | |
8JIS (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Peptide-15 | - | 2.46 | 2023-11-08 | 10.1073/pnas.2303696120 | ||
8WRB | A | Orphan | Orphan | GPR34 | Homo sapiens | Lysophosphatidylserine | - | Gi1/β1/γ2 | 2.91 | 2023-11-08 | 10.1371/journal.pbio.3002387 | |
8WRB (No Gprot) | A | Orphan | Orphan | GPR34 | Homo sapiens | Lysophosphatidylserine | - | 2.91 | 2023-11-08 | 10.1371/journal.pbio.3002387 | ||
8SG1 | A | Protein | Chemerin | CML1 | Homo sapiens | Chemerin-9 | - | Gi1/β1/γ2 | 2.94 | 2023-11-01 | 10.1371/journal.pbio.3002188 | |
8SG1 (No Gprot) | A | Protein | Chemerin | CML1 | Homo sapiens | Chemerin-9 | - | 2.94 | 2023-11-01 | 10.1371/journal.pbio.3002188 | ||
8G05 | A | Orphan | Orphan | GPR84 | Homo sapiens | 6-OAU | - | Gi1/β1/γ2 | 3 | 2023-11-01 | 10.1038/s41467-023-41201-0 | |
8G05 (No Gprot) | A | Orphan | Orphan | GPR84 | Homo sapiens | 6-OAU | - | 3 | 2023-11-01 | 10.1038/s41467-023-41201-0 | ||
8IZB | A | Orphan | Orphan | GPR174 | Homo sapiens | Lysophosphatidylserine | - | Gs/β1/γ2 | 3.06 | 2023-11-01 | 10.1371/journal.pbio.3002387 | |
8IZB (No Gprot) | A | Orphan | Orphan | GPR174 | Homo sapiens | Lysophosphatidylserine | - | 3.06 | 2023-11-01 | 10.1371/journal.pbio.3002387 | ||
7YFD | A | Amine | Histamine | H4 | Homo sapiens | Imetit | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.1 | 2023-10-25 | 10.1038/s41467-023-42260-z | |
7YFD (No Gprot) | A | Amine | Histamine | H4 | Homo sapiens | Imetit | - | 3.1 | 2023-10-25 | 10.1038/s41467-023-42260-z | ||
7YFC | A | Amine | Histamine | H4 | Homo sapiens | Histamine | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3 | 2023-10-25 | 10.1038/s41467-023-42260-z | |
7YFC (No Gprot) | A | Amine | Histamine | H4 | Homo sapiens | Histamine | - | 3 | 2023-10-25 | 10.1038/s41467-023-42260-z | ||
8K4N | A | Orphan | Orphan | GPR34 | Homo sapiens | VF0 | - | Gi1/β1/γ2 | 2.83 | 2023-10-25 | To be published | |
8K4N (No Gprot) | A | Orphan | Orphan | GPR34 | Homo sapiens | VF0 | - | 2.83 | 2023-10-25 | To be published | ||
8E0G | A | Peptide | Opioid | μ | Mus musculus | BU72 | - | - | 2.1 | 2023-10-18 | 10.1186/s12915-023-01689-w | |
8J6D | A | Peptide | Complement Peptide | C3aB | Homo sapiens | EP141 | - | Go/β1/γ2 | 3.1 | 2023-10-18 | 10.1016/j.cell.2023.09.020 | |
8J6D (No Gprot) | A | Peptide | Complement Peptide | C3aB | Homo sapiens | EP141 | - | 3.1 | 2023-10-18 | 10.1016/j.cell.2023.09.020 | ||
8JZZ | A | Peptide | Complement Peptide | C5a1 | Homo sapiens | C5a-desArg | - | Go/β1/γ2 | 3.31 | 2023-10-18 | 10.1016/j.cell.2023.09.020 | |
8JZZ (No Gprot) | A | Peptide | Complement Peptide | C5a1 | Homo sapiens | C5a-desArg | - | 3.31 | 2023-10-18 | 10.1016/j.cell.2023.09.020 | ||
8I9A | A | Peptide | Complement Peptide | C3aB | Homo sapiens | EP54 | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.57 | 2023-10-18 | 10.1016/j.cell.2023.09.020 | |
8I9A (No Gprot) | A | Peptide | Complement Peptide | C3aB | Homo sapiens | EP54 | - | 3.57 | 2023-10-18 | 10.1016/j.cell.2023.09.020 | ||
8I9S | A | Peptide | Complement Peptide | C3aB | Homo sapiens | - | - | Go/β1/γ2 | 3.26 | 2023-10-18 | 10.1016/j.cell.2023.09.020 | |
8I9S (No Gprot) | A | Peptide | Complement Peptide | C3aB | Homo sapiens | - | - | 3.26 | 2023-10-18 | 10.1016/j.cell.2023.09.020 | ||
8I9L | A | Peptide | Complement Peptide | C3aB | Homo sapiens | C3a anaphylatoxin | - | Go/β1/γ2 | 3.18 | 2023-10-18 | 10.1016/j.cell.2023.09.020 | |
8I9L (No Gprot) | A | Peptide | Complement Peptide | C3aB | Homo sapiens | C3a anaphylatoxin | - | 3.18 | 2023-10-18 | 10.1016/j.cell.2023.09.020 | ||
8I97 | A | Peptide | Complement Peptide | C3aB | Homo sapiens | - | - | Go/β1/γ2 | 3.1 | 2023-10-18 | 10.1016/j.cell.2023.09.020 | |
8I97 (No Gprot) | A | Peptide | Complement Peptide | C3aB | Homo sapiens | - | - | 3.1 | 2023-10-18 | 10.1016/j.cell.2023.09.020 | ||
8I95 | A | Peptide | Complement Peptide | C3aB | Homo sapiens | EP54 | - | Go/β1/γ2 | 2.88 | 2023-10-18 | 10.1016/j.cell.2023.09.020 | |
8I95 (No Gprot) | A | Peptide | Complement Peptide | C3aB | Homo sapiens | EP54 | - | 2.88 | 2023-10-18 | 10.1016/j.cell.2023.09.020 | ||
8IA2 | A | Peptide | Complement Peptide | C5a1 | Homo sapiens | C5a anaphylatoxin | - | Go/β1/γ2 | 3.21 | 2023-10-18 | 10.1016/j.cell.2023.09.020 | |
8IA2 (No Gprot) | A | Peptide | Complement Peptide | C5a1 | Homo sapiens | C5a anaphylatoxin | - | 3.21 | 2023-10-18 | 10.1016/j.cell.2023.09.020 | ||
8HPT | A | Peptide | Complement Peptide | C5a1 | Mus musculus | C5a anaphylatoxin C-terminal peptide | - | Go/β1/γ2 | 3.39 | 2023-10-18 | 10.1016/j.cell.2023.09.020 | |
8HPT (No Gprot) | A | Peptide | Complement Peptide | C5a1 | Mus musculus | C5a anaphylatoxin C-terminal peptide | - | 3.39 | 2023-10-18 | 10.1016/j.cell.2023.09.020 | ||
8ITM | B1 | Peptide | Glucagon | GIP | Homo sapiens | - | - | Gs/β1/γ2 | 3.13 | 2023-10-18 | 10.1073/pnas.2306145120 | |
8ITM (No Gprot) | B1 | Peptide | Glucagon | GIP | Homo sapiens | - | - | 3.13 | 2023-10-18 | 10.1073/pnas.2306145120 | ||
8ITL | B1 | Peptide | Glucagon | GIP | Homo sapiens | - | - | Gs/β1/γ2 | 3.23 | 2023-10-18 | 10.1073/pnas.2306145120 | |
8ITL (No Gprot) | B1 | Peptide | Glucagon | GIP | Homo sapiens | - | - | 3.23 | 2023-10-18 | 10.1073/pnas.2306145120 | ||
8HVI | A | Orphan | Orphan | GPR132 | Homo sapiens | NOX-6-7 | - | Gi1/β1/γ2 | 3.04 | 2023-10-11 | 0.1038/s42255-023-00899-4 | |
8HVI (No Gprot) | A | Orphan | Orphan | GPR132 | Homo sapiens | NOX-6-7 | - | 3.04 | 2023-10-11 | 0.1038/s42255-023-00899-4 | ||
8HQN | A | Orphan | Orphan | GPR132 | Homo sapiens | 9-S-HODE | - | Gi1/β1/γ2 | 3 | 2023-10-11 | 0.1038/s42255-023-00899-4 | |
8HQN (No Gprot) | A | Orphan | Orphan | GPR132 | Homo sapiens | 9-S-HODE | - | 3 | 2023-10-11 | 0.1038/s42255-023-00899-4 | ||
8HQM | A | Orphan | Orphan | GPR132 | Homo sapiens | NPGLY | - | Gi1/β1/γ2 | 2.95 | 2023-10-11 | 0.1038/s42255-023-00899-4 | |
8HQM (No Gprot) | A | Orphan | Orphan | GPR132 | Homo sapiens | NPGLY | - | 2.95 | 2023-10-11 | 0.1038/s42255-023-00899-4 | ||
8HQE | A | Orphan | Orphan | GPR132 | Homo sapiens | - | - | Gi1/β1/γ2 | 2.97 | 2023-10-11 | 0.1038/s42255-023-00899-4 | |
8HQE (No Gprot) | A | Orphan | Orphan | GPR132 | Homo sapiens | - | - | 2.97 | 2023-10-11 | 0.1038/s42255-023-00899-4 | ||
8H2G | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | Niacin | - | Gi1/β1/γ2 | 3.01 | 2023-10-11 | To be published | |
8H2G (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | Niacin | - | 3.01 | 2023-10-11 | To be published | ||
8TB7 | A | Orphan | Orphan | GPR61 | Homo sapiens | - | PubChem 168510218 | - | 2.94 | 2023-10-04 | 10.1038/s41467-023-41646-3 | |
8TB0 | A | Orphan | Orphan | GPR61 | Homo sapiens | - | - | chim(NtGi1-Gs)/β1/γ2 | 3.47 | 2023-10-04 | 10.1038/s41467-023-41646-3 | |
8TB0 (No Gprot) | A | Orphan | Orphan | GPR61 | Homo sapiens | - | - | 3.47 | 2023-10-04 | 10.1038/s41467-023-41646-3 | ||
8JZ7 | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | MK6892 | - | Gi1/β1/γ2 | 2.6 | 2023-10-04 | 10.1038/s41392-023-01625-y | |
8JZ7 (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | MK6892 | - | 2.6 | 2023-10-04 | 10.1038/s41392-023-01625-y | ||
8IOC | A | Peptide | Melanocortin | MC3 | Homo sapiens | γ-MSH | Ca | chim(NtGi1-Gs)/β1/γ2 | 2.86 | 2023-09-20 | 10.1038/s41421-023-00586-4 | |
8IOC (No Gprot) | A | Peptide | Melanocortin | MC3 | Homo sapiens | γ-MSH | Ca | 2.86 | 2023-09-20 | 10.1038/s41421-023-00586-4 | ||
8IOD | A | Peptide | Melanocortin | MC5 | Homo sapiens | PG-901 | Ca | chim(NtGi1-Gs)/β1/γ2 | 2.59 | 2023-09-20 | 10.1038/s41421-023-00586-4 | |
8IOD (No Gprot) | A | Peptide | Melanocortin | MC5 | Homo sapiens | PG-901 | Ca | 2.59 | 2023-09-20 | 10.1038/s41421-023-00586-4 | ||
8INR | A | Peptide | Melanocortin | MC5 | Homo sapiens | α-MSH | Ca | chim(NtGi1-Gs)/β1/γ2 | 2.73 | 2023-09-20 | 10.1038/s41421-023-00586-4 | |
8INR (No Gprot) | A | Peptide | Melanocortin | MC5 | Homo sapiens | α-MSH | Ca | 2.73 | 2023-09-20 | 10.1038/s41421-023-00586-4 | ||
8GTM | B1 | Peptide | Corticotropin Releasing Factor | CRF1 | Homo sapiens | - | BMK-C203 | - | 2.6 | 2023-09-13 | 10.1038/s12276-023-01082-1 | |
8GTI | B1 | Peptide | Corticotropin Releasing Factor | CRF1 | Homo sapiens | - | BMK-C205 | - | 2.2 | 2023-09-13 | 10.1038/s12276-023-01082-1 | |
8GTG | B1 | Peptide | Corticotropin Releasing Factor | CRF1 | Homo sapiens | - | BMK-I152 | - | 2.75 | 2023-09-13 | 10.1038/s12276-023-01082-1 | |
8IHB | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | GSK256073 | - | Gi1/β1/γ2 | 2.85 | 2023-09-13 | 10.1038/s41467-023-41650-7 | |
8IHB (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | GSK256073 | - | 2.85 | 2023-09-13 | 10.1038/s41467-023-41650-7 | ||
8FX5 | A | Amine | Acetylcholine (muscarinic) | M4 | Homo sapiens | Xanomeline | Xanomeline | Gi1/β1/γ2 | 2.45 | 2023-09-13 | 10.1038/s41467-023-41199-5 | |
8FX5 (No Gprot) | A | Amine | Acetylcholine (muscarinic) | M4 | Homo sapiens | Xanomeline | Xanomeline | 2.45 | 2023-09-13 | 10.1038/s41467-023-41199-5 | ||
8JMT | B2 | Adhesion | Adhesion | ADGRL3 | Homo sapiens | - | - | - | 3.3 | 2023-09-06 | 10.1038/s41589-023-01389-0 | |
8JIR | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | SAR425899 | - | chim(NtGi1-Gs)/β1/γ2 | 2.57 | 2023-09-06 | 10.1073/pnas.2303696120 | |
8JIR (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | SAR425899 | - | 2.57 | 2023-09-06 | 10.1073/pnas.2303696120 | ||
8JIP | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | MEDI0382 | - | chim(NtGi1-Gs)/β1/γ2 | 2.85 | 2023-09-06 | 10.1073/pnas.2303696120 | |
8JIP (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | MEDI0382 | - | 2.85 | 2023-09-06 | 10.1073/pnas.2303696120 | ||
8JIM | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | MMF | - | Gi1/β1/γ2 | 2.98 | 2023-09-06 | 10.1016/j.molcel.2023.07.030 | |
8JIM (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | MMF | - | 2.98 | 2023-09-06 | 10.1016/j.molcel.2023.07.030 | ||
8JIL | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | Niacin | - | Gi1/β1/γ2 | 3.5 | 2023-09-06 | 10.1016/j.molcel.2023.07.030 | |
8JIL (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | Niacin | - | 3.5 | 2023-09-06 | 10.1016/j.molcel.2023.07.030 | ||
8JII | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | Niacin | Compound 9n | Gi1/β1/γ2 | 3.17 | 2023-09-06 | 10.1016/j.molcel.2023.07.030 | |
8JII (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | Niacin | Compound 9n | 3.17 | 2023-09-06 | 10.1016/j.molcel.2023.07.030 | ||
8JHY | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | - | Compound 9n | Gi1/β1/γ2 | 2.87 | 2023-09-06 | 10.1016/j.molcel.2023.07.030 | |
8JHY (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | - | Compound 9n | 2.87 | 2023-09-06 | 10.1016/j.molcel.2023.07.030 | ||
8JIT | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | MEDI0382 | - | Gs/β1/γ2 | 2.91 | 2023-09-06 | 10.1073/pnas.2303696120 | |
8JIT (No Gprot) | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | MEDI0382 | - | 2.91 | 2023-09-06 | 10.1073/pnas.2303696120 | ||
8A2P | A | Nucleotide | Adenosine | A2A | Homo sapiens | LUAA47070 | Na | - | 3.5 | 2023-08-30 | 10.1107/S1600576723006428 | |
8A2O | A | Nucleotide | Adenosine | A2A | Homo sapiens | Theophylline | Na | - | 3.45 | 2023-08-30 | 10.1107/S1600576723006428 | |
8IHK | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA3 | Homo sapiens | Acifran | - | - | 3.21 | 2023-08-30 | 10.1038/s41467-023-41650-7 | |
8FD1 | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | - | - | 4.25 | 2023-08-30 | 10.1038/s41467-023-40911-9 | |
8FD1 (Multimeric) | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | - | 4.25 | 2023-08-30 | 10.1038/s41467-023-40911-9 | ||
8FD0 | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | - | - | 3.71 | 2023-08-30 | 10.1038/s41467-023-40911-9 | |
8FD0 (Multimeric) | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | - | 3.71 | 2023-08-30 | 10.1038/s41467-023-40911-9 | ||
8FCZ | A | Sensory | Opsins | Rhodopsin | Bos taurus | 11-cis-Retinal | - | - | 3.7 | 2023-08-30 | 10.1038/s41467-023-40911-9 | |
8FCZ (Multimeric) | A | Sensory | Opsins | Rhodopsin | Bos taurus | 11-cis-Retinal | - | 3.7 | 2023-08-30 | 10.1038/s41467-023-40911-9 | ||
8IHI | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | Acifran | - | Gi1/β1/γ2 | 3.11 | 2023-08-30 | 10.1038/s41467-023-41650-7 | |
8IHI (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | Acifran | - | 3.11 | 2023-08-30 | 10.1038/s41467-023-41650-7 | ||
8IHH | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | LUF6283 | - | Gi1/β1/γ2 | 3.06 | 2023-08-30 | 10.1038/s41467-023-41650-7 | |
8IHH (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | LUF6283 | - | 3.06 | 2023-08-30 | 10.1038/s41467-023-41650-7 | ||
8IHF | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | MK6892 | - | Gi1/β1/γ2 | 2.97 | 2023-08-30 | 10.1038/s41467-023-41650-7 | |
8IHF (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | MK6892 | - | 2.97 | 2023-08-30 | 10.1038/s41467-023-41650-7 | ||
8IHJ | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA3 | Homo sapiens | Acifran | - | Gi1/β1/γ2 | 3.07 | 2023-08-30 | 10.1038/s41467-023-41650-7 | |
8IHJ (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA3 | Homo sapiens | Acifran | - | 3.07 | 2023-08-30 | 10.1038/s41467-023-41650-7 | ||
8JWZ | A | Nucleotide | Adenosine | A2A | Homo sapiens | AB928 | Na | - | 2.37 | 2023-08-16 | 10.1007/s11427-023-2459-8 | |
8JWY | A | Nucleotide | Adenosine | A2A | Homo sapiens | 2-118 | - | - | 2.33 | 2023-08-16 | 10.1007/s11427-023-2459-8 | |
8IY6 | A | Peptide | Endothelin | ETB | Homo sapiens | Endothelin-1 | - | - | 3.13 | 2023-08-16 | 10.7554/eLife.85821 | |
8JRV | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | Glucagon | - | Arrestin2 | 3.3 | 2023-08-16 | 10.1038/s41586-023-06420-x | |
8JRU | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | - | - | Arrestin2 | 3.5 | 2023-08-16 | 10.1038/s41586-023-06420-x | |
8THL | A | Amine | Adrenergic | Alpha1A | Homo sapiens | Epinephrine | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 3.1 | 2023-08-16 | 10.1038/s41467-023-40524-2 | |
8THL (No Gprot) | A | Amine | Adrenergic | Alpha1A | Homo sapiens | Epinephrine | - | 3.1 | 2023-08-16 | 10.1038/s41467-023-40524-2 | ||
8THK | A | Amine | Adrenergic | Alpha1A | Homo sapiens | A61603 | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 2.6 | 2023-08-16 | 10.1038/s41467-023-40524-2 | |
8THK (No Gprot) | A | Amine | Adrenergic | Alpha1A | Homo sapiens | A61603 | - | 2.6 | 2023-08-16 | 10.1038/s41467-023-40524-2 | ||
8IY5 | A | Peptide | Endothelin | ETB | Homo sapiens | Endothelin-1 | - | Gi1/β1/γ2 | 2.8 | 2023-08-16 | 10.7554/eLife.85821 | |
8IY5 (No Gprot) | A | Peptide | Endothelin | ETB | Homo sapiens | Endothelin-1 | - | 2.8 | 2023-08-16 | 10.7554/eLife.85821 | ||
8JPF | A | Peptide | Neurotensin | NTS1 | Homo sapiens | Neurotensin | PubChem 118610427 | - | 3.02 | 2023-08-09 | 10.1038/s41586-023-06395-9 | |
8H0P | A | Peptide | Bombesin | BB1 | Homo sapiens | NMB30 | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.15 | 2023-08-09 | 10.1038/s41422-022-00743-6 | |
8H0P (No Gprot) | A | Peptide | Bombesin | BB1 | Homo sapiens | NMB30 | - | 3.15 | 2023-08-09 | 10.1038/s41422-022-00743-6 | ||
8H0Q | A | Peptide | Bombesin | BB2 | Homo sapiens | Gastrin Releasing Peptide | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.3 | 2023-08-09 | 10.1038/s41422-022-00743-6 | |
8H0Q (No Gprot) | A | Peptide | Bombesin | BB2 | Homo sapiens | Gastrin Releasing Peptide | - | 3.3 | 2023-08-09 | 10.1038/s41422-022-00743-6 | ||
8JPC | A | Peptide | Neurotensin | NTS1 | Homo sapiens | Neurotensin-(8-13) | PubChem 118610427; GDP; Mg | Gq; GRK2 | 3.07 | 2023-08-09 | 10.1038/s41586-023-06395-9 | |
8JPC (No Gprot) | A | Peptide | Neurotensin | NTS1 | Homo sapiens | Neurotensin-(8-13) | PubChem 118610427; GDP; Mg | 3.07 | 2023-08-09 | 10.1038/s41586-023-06395-9 | ||
8JPB | A | Peptide | Neurotensin | NTS1 | Homo sapiens | Neurotensin-(8-13) | PubChem 118610427; GDP; Mg | Gq; GRK2 | 3.07 | 2023-08-09 | 10.1038/s41586-023-06395-9 | |
8JPB (No Gprot) | A | Peptide | Neurotensin | NTS1 | Homo sapiens | Neurotensin-(8-13) | PubChem 118610427; GDP; Mg | 3.07 | 2023-08-09 | 10.1038/s41586-023-06395-9 | ||
8PM2 | A | Amine | Trace Amine Receptors | TA7 | Mus musculus | DMCH | - | Gs/β1/γ2 | 2.92 | 2023-08-09 | doi.org/10.1101/2023.07.07.547762 | |
8PM2 (No Gprot) | A | Amine | Trace Amine Receptors | TA7 | Mus musculus | DMCH | - | 2.92 | 2023-08-09 | doi.org/10.1101/2023.07.07.547762 | ||
8JR9 | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | - | PCO371 | chim(NtGi1-Gs)/β1/γ2 | 2.57 | 2023-08-02 | 10.1038/s41586-023-06467-w | |
8JR9 (No Gprot) | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | - | PCO371 | 2.57 | 2023-08-02 | 10.1038/s41586-023-06467-w | ||
8F0J | B1 | Peptide | Calcitonin | CT | Homo sapiens | Pramlintide Analogue San45 | - | Gs/β1/γ2 | 2 | 2023-08-02 | 10.1038/s41589-023-01393-4 | |
8F0J (No Gprot) | B1 | Peptide | Calcitonin | CT | Homo sapiens | Pramlintide Analogue San45 | - | 2 | 2023-08-02 | 10.1038/s41589-023-01393-4 | ||
8F2B | B1 | Peptide | Calcitonin | CT (AMY3) | Homo sapiens | Pramlintide Analogue San45 | - | Gs/β1/γ2; RAMP3 | 2 | 2023-08-02 | 10.1038/s41589-023-01393-4 | |
8F2B (No Gprot) | B1 | Peptide | Calcitonin | CT (AMY3) | Homo sapiens | Pramlintide Analogue San45 | - | 2 | 2023-08-02 | 10.1038/s41589-023-01393-4 | ||
8F2A | B1 | Peptide | Calcitonin | CT (AMY3) | Homo sapiens | Pramlintide Analogue San385 | - | Gs/β1/γ2; RAMP3 | 2.2 | 2023-08-02 | 10.1038/s41589-023-01393-4 | |
8F2A (No Gprot) | B1 | Peptide | Calcitonin | CT (AMY3) | Homo sapiens | Pramlintide Analogue San385 | - | 2.2 | 2023-08-02 | 10.1038/s41589-023-01393-4 | ||
8F0K | B1 | Peptide | Calcitonin | CT (AMY3) | Homo sapiens | Pramlintide Analogue San385 | - | Gs/β1/γ2; RAMP3 | 1.9 | 2023-08-02 | 10.1038/s41589-023-01393-4 | |
8F0K (No Gprot) | B1 | Peptide | Calcitonin | CT (AMY3) | Homo sapiens | Pramlintide Analogue San385 | - | 1.9 | 2023-08-02 | 10.1038/s41589-023-01393-4 | ||
8IC0 | A | Protein | Chemokine | CXCR1 | Homo sapiens | Interleukin-8 | - | Gi1/β1/γ2 | 3.41 | 2023-07-19 | 10.1038/s41467-023-39799-2 | |
8IC0 (No Gprot) | A | Protein | Chemokine | CXCR1 | Homo sapiens | Interleukin-8 | - | 3.41 | 2023-07-19 | 10.1038/s41467-023-39799-2 | ||
8C9W | A | Nucleotide | Adenosine | A2A | Homo sapiens | Etrumadenant | - | - | 2.11 | 2023-07-12 | 10.1038/s42004-023-00894-6 | |
7YDJ | B2 | Adhesion | Adhesion | ADGRE5 | Homo sapiens | - | - | chim(NtGi1-G12)/β1/γ2 | 3.03 | 2023-07-12 | To be published | |
7YDJ (No Gprot) | B2 | Adhesion | Adhesion | ADGRE5 | Homo sapiens | - | - | 3.03 | 2023-07-12 | To be published | ||
7YDM | B2 | Adhesion | Adhesion | ADGRE5 | Homo sapiens | - | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.89 | 2023-07-12 | 10.1016/j.chembiol.2023.08.003 | |
7YDM (No Gprot) | B2 | Adhesion | Adhesion | ADGRE5 | Homo sapiens | - | - | 2.89 | 2023-07-12 | 10.1016/j.chembiol.2023.08.003 | ||
8IUM | A | Lipid | Prostanoid | FP-alpha | Homo sapiens | Tafluprost acid | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.14 | 2023-07-12 | 10.1038/s41467-023-38411-x | |
8IUM (No Gprot) | A | Lipid | Prostanoid | FP-alpha | Homo sapiens | Tafluprost acid | - | 3.14 | 2023-07-12 | 10.1038/s41467-023-38411-x | ||
8IUL | A | Lipid | Prostanoid | FP-alpha | Homo sapiens | Latanoprost | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.78 | 2023-07-12 | 10.1038/s41467-023-38411-x | |
8IUL (No Gprot) | A | Lipid | Prostanoid | FP-alpha | Homo sapiens | Latanoprost | - | 2.78 | 2023-07-12 | 10.1038/s41467-023-38411-x | ||
8IUK | A | Lipid | Prostanoid | FP-alpha | Homo sapiens | PGF2-α | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.67 | 2023-07-12 | 10.1038/s41467-023-38411-x | |
8IUK (No Gprot) | A | Lipid | Prostanoid | FP-alpha | Homo sapiens | PGF2-α | - | 2.67 | 2023-07-12 | 10.1038/s41467-023-38411-x | ||
7YDP | B2 | Adhesion | Adhesion | ADGRE5 | Homo sapiens | - | - | chim(NtGi1-Gs)/β1/γ2 | 3.1 | 2023-07-12 | 10.1016/j.chembiol.2023.08.003 | |
7YDP (No Gprot) | B2 | Adhesion | Adhesion | ADGRE5 | Homo sapiens | - | - | 3.1 | 2023-07-12 | 10.1016/j.chembiol.2023.08.003 | ||
7YDH | B2 | Adhesion | Adhesion | ADGRE5 | Homo sapiens | - | - | chim(NtGi2-G13)/β1/γ2 | 3.1 | 2023-07-12 | 10.1016/j.chembiol.2023.08.003 | |
7YDH (No Gprot) | B2 | Adhesion | Adhesion | ADGRE5 | Homo sapiens | - | - | 3.1 | 2023-07-12 | 10.1016/j.chembiol.2023.08.003 | ||
7YMJ | A | Amine | Adrenergic | Alpha1A | Homo sapiens | Tamsulosin | - | - | 3.35 | 2023-07-05 | 10.1038/s41467-023-39310-x | |
7YMH | A | Amine | Adrenergic | Alpha1A | Homo sapiens | Norepinephrine | - | chim(Gs-CtGq) | 3.52 | 2023-07-05 | 10.1038/s41467-023-39310-x | |
7YMH (No Gprot) | A | Amine | Adrenergic | Alpha1A | Homo sapiens | Norepinephrine | - | 3.52 | 2023-07-05 | 10.1038/s41467-023-39310-x | ||
7YM8 | A | Amine | Adrenergic | Alpha1A | Homo sapiens | Oxymetazoline | - | chim(Gs-CtGq) | 2.92 | 2023-07-05 | 10.1038/s41467-023-39310-x | |
7YM8 (No Gprot) | A | Amine | Adrenergic | Alpha1A | Homo sapiens | Oxymetazoline | - | 2.92 | 2023-07-05 | 10.1038/s41467-023-39310-x | ||
7Y36 | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | Teriparatide | - | Gs/β1/γ2 | 2.8 | 2023-07-05 | To be published | |
7Y36 (No Gprot) | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | Teriparatide | - | 2.8 | 2023-07-05 | To be published | ||
7Y35 | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | Abaloparatide | - | Gs/β1/γ2 | 2.9 | 2023-07-05 | To be published | |
7Y35 (No Gprot) | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | Abaloparatide | - | 2.9 | 2023-07-05 | To be published | ||
8JLZ | A | Amine | 5-Hydroxytryptamine | 5-HT6 | Homo sapiens | ST1936 | - | Gs/β1/γ2 | 3.09 | 2023-06-28 | 10.1016/j.bbrc.2023.05.126 | |
8JLZ (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT6 | Homo sapiens | ST1936 | - | 3.09 | 2023-06-28 | 10.1016/j.bbrc.2023.05.126 | ||
8JD2 | C | Aminoacid | Metabotropic Glutamate | mGlu2; mGlu3 | Homo sapiens | Glutamate | - | - | 2.8 | 2023-06-21 | 10.1038/s41422-023-00830-2 | |
8JD1 | C | Aminoacid | Metabotropic Glutamate | mGlu2; mGlu3 | Homo sapiens | Glutamate | - | - | 3.7 | 2023-06-21 | 10.1038/s41422-023-00830-2 | |
8JD0 | C | Aminoacid | Metabotropic Glutamate | mGlu2; mGlu3 | Homo sapiens | Glutamate | NAM563 | - | 3.3 | 2023-06-21 | 10.1038/s41422-023-00830-2 | |
8JCZ | C | Aminoacid | Metabotropic Glutamate | mGlu2; mGlu3 | Homo sapiens | LY341495 | - | - | 3 | 2023-06-21 | 10.1038/s41422-023-00830-2 | |
8JCY | C | Aminoacid | Metabotropic Glutamate | mGlu2; mGlu3 | Homo sapiens | LY341495 | - | - | 2.9 | 2023-06-21 | 10.1038/s41422-023-00830-2 | |
8JCX | C | Aminoacid | Metabotropic Glutamate | mGlu2; mGlu3 | Homo sapiens | LY341495 | - | - | 3 | 2023-06-21 | 10.1038/s41422-023-00830-2 | |
8JCW | C | Aminoacid | Metabotropic Glutamate | mGlu2; mGlu3 | Homo sapiens | LY341495 | - | - | 3 | 2023-06-21 | 10.1038/s41422-023-00830-2 | |
8JCV | C | Aminoacid | Metabotropic Glutamate | mGlu2; mGlu3 | Homo sapiens | LY341495 | - | - | 3.4 | 2023-06-21 | 10.1038/s41422-023-00830-2 | |
8JCU | C | Aminoacid | Metabotropic Glutamate | mGlu2; mGlu3 | Homo sapiens | LY341495 | - | - | 2.8 | 2023-06-21 | 10.1038/s41422-023-00830-2 | |
8JD4 | C | Aminoacid | Metabotropic Glutamate | mGlu2; mGlu4 | Homo sapiens | Glutamate | - | - | 2.9 | 2023-06-21 | 10.1038/s41422-023-00830-2 | |
8H4L | A | Lipid | Free Fatty Acid | FFA4 | Homo sapiens | Doconexent | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.07 | 2023-06-21 | 10.1038/s41422-023-00835-x | |
8H4L (No Gprot) | A | Lipid | Free Fatty Acid | FFA4 | Homo sapiens | Doconexent | - | 3.07 | 2023-06-21 | 10.1038/s41422-023-00835-x | ||
8H4K | A | Lipid | Free Fatty Acid | FFA4 | Homo sapiens | GW9508 | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.1 | 2023-06-21 | 10.1038/s41422-023-00835-x | |
8H4K (No Gprot) | A | Lipid | Free Fatty Acid | FFA4 | Homo sapiens | GW9508 | - | 3.1 | 2023-06-21 | 10.1038/s41422-023-00835-x | ||
8H4I | A | Lipid | Free Fatty Acid | FFA4 | Homo sapiens | Doconexent | - | chim(NtGi1-Gs)/β1/γ2 | 3.06 | 2023-06-21 | 10.1038/s41422-023-00835-x | |
8H4I (No Gprot) | A | Lipid | Free Fatty Acid | FFA4 | Homo sapiens | Doconexent | - | 3.06 | 2023-06-21 | 10.1038/s41422-023-00835-x | ||
8IYS | A | Lipid | Free Fatty Acid | FFA4 | Homo sapiens | TUG-891 | GDP | chim(NtGi1L-Gq)/β1/γ2 | 2.95 | 2023-06-21 | 10.1038/s41422-023-00835-x | |
8IYS (No Gprot) | A | Lipid | Free Fatty Acid | FFA4 | Homo sapiens | TUG-891 | GDP | 2.95 | 2023-06-21 | 10.1038/s41422-023-00835-x | ||
8J1A | A | Orphan | Orphan | GPR84 | Homo sapiens | - | - | Gi1/β1/γ2 | 3.24 | 2023-06-21 | 10.1038/s41467-023-38985-6 | |
8J1A (No Gprot) | A | Orphan | Orphan | GPR84 | Homo sapiens | - | - | 3.24 | 2023-06-21 | 10.1038/s41467-023-38985-6 | ||
8J19 | A | Orphan | Orphan | GPR84 | Homo sapiens | LY237 | - | Gi1/β1/γ2 | 3.23 | 2023-06-21 | 10.1038/s41467-023-38985-6 | |
8J19 (No Gprot) | A | Orphan | Orphan | GPR84 | Homo sapiens | LY237 | - | 3.23 | 2023-06-21 | 10.1038/s41467-023-38985-6 | ||
8J18 | A | Orphan | Orphan | GPR84 | Homo sapiens | (3R)-3-Hydroxydodecanoic acid | - | Gi1/β1/γ2 | 2.89 | 2023-06-21 | 10.1038/s41467-023-38985-6 | |
8J18 (No Gprot) | A | Orphan | Orphan | GPR84 | Homo sapiens | (3R)-3-Hydroxydodecanoic acid | - | 2.89 | 2023-06-21 | 10.1038/s41467-023-38985-6 | ||
8JD3 | C | Aminoacid | Metabotropic Glutamate | mGlu2; mGlu3 | Homo sapiens | Glutamate | HZR; PEF | Gi1/β1/γ2 | 3.3 | 2023-06-21 | 10.1038/s41422-023-00830-2 | |
8JD3 (No Gprot) | C | Aminoacid | Metabotropic Glutamate | mGlu2; mGlu3 | Homo sapiens | Glutamate | HZR; PEF | 3.3 | 2023-06-21 | 10.1038/s41422-023-00830-2 | ||
8JD5 | C | Aminoacid | Metabotropic Glutamate | mGlu2; mGlu4 | Homo sapiens | Glutamate | BQI; HZE; PEF | Gi1/β1/γ2 | 3.6 | 2023-06-21 | 10.1038/s41422-023-00830-2 | |
8JD5 (No Gprot) | C | Aminoacid | Metabotropic Glutamate | mGlu2; mGlu4 | Homo sapiens | Glutamate | BQI; HZE; PEF | 3.6 | 2023-06-21 | 10.1038/s41422-023-00830-2 | ||
8JD6 | C | Aminoacid | Metabotropic Glutamate | mGlu4; mGlu4 | Homo sapiens | Phosphoserine | N-(3-chlorophenyl)pyridine-2-carboxamide | Gi3/β1/γ2 | 3.4 | 2023-06-21 | 10.1038/s41422-023-00830-2 | |
8JD6 (No Gprot) | C | Aminoacid | Metabotropic Glutamate | mGlu4; mGlu4 | Homo sapiens | Phosphoserine | N-(3-chlorophenyl)pyridine-2-carboxamide | 3.4 | 2023-06-21 | 10.1038/s41422-023-00830-2 | ||
8HMP | A | Orphan | Orphan | GPR52 | Homo sapiens | - | C17 | Gs/β1/γ2 | 2.77 | 2023-06-21 | 10.1002/mco2.260 | |
8HMP (No Gprot) | A | Orphan | Orphan | GPR52 | Homo sapiens | - | C17 | 2.77 | 2023-06-21 | 10.1002/mco2.260 | ||
8GW8 | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | - | KHF | Gs/β1/γ2 | 2.9 | 2023-06-14 | 10.1038/s41586-023-06169-3 | |
8GW8 (No Gprot) | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | - | KHF | 2.9 | 2023-06-14 | 10.1038/s41586-023-06169-3 | ||
8IRU | A | Amine | Dopamine | D4 | Homo sapiens | Rotigotine | - | chim(NtGi1-Gs-CtGi1)/β1/γ2 | 3.2 | 2023-06-07 | 10.1038/s41422-023-00808-0 | |
8IRU (No Gprot) | A | Amine | Dopamine | D4 | Homo sapiens | Rotigotine | - | 3.2 | 2023-06-07 | 10.1038/s41422-023-00808-0 | ||
8IRV | A | Amine | Dopamine | D5 | Homo sapiens | Rotigotine | - | chim(NtGi1-Gs)/β1/γ2 | 3.1 | 2023-06-07 | 10.1038/s41422-023-00808-0 | |
8IRV (No Gprot) | A | Amine | Dopamine | D5 | Homo sapiens | Rotigotine | - | 3.1 | 2023-06-07 | 10.1038/s41422-023-00808-0 | ||
8IRS | A | Amine | Dopamine | D2 | Homo sapiens | Rotigotine | - | Gi1/β1/γ2 | 3 | 2023-06-07 | 10.1038/s41422-023-00808-0 | |
8IRS (No Gprot) | A | Amine | Dopamine | D2 | Homo sapiens | Rotigotine | - | 3 | 2023-06-07 | 10.1038/s41422-023-00808-0 | ||
8IRT | A | Amine | Dopamine | D3 | Homo sapiens | Rotigotine | - | Gi1/β1/γ2 | 2.7 | 2023-06-07 | 10.1038/s41422-023-00808-0 | |
8IRT (No Gprot) | A | Amine | Dopamine | D3 | Homo sapiens | Rotigotine | - | 2.7 | 2023-06-07 | 10.1038/s41422-023-00808-0 | ||
8IRR | A | Amine | Dopamine | D1 | Homo sapiens | Rotigotine | - | Gs/β1/γ2 | 3.2 | 2023-06-07 | 10.1038/s41422-023-00808-0 | |
8IRR (No Gprot) | A | Amine | Dopamine | D1 | Homo sapiens | Rotigotine | - | 3.2 | 2023-06-07 | 10.1038/s41422-023-00808-0 | ||
7Y3G | A | Orphan | Orphan | GPR12 | Homo sapiens | - | - | Gs/β1/γ2 | 2.77 | 2023-06-07 | 10.1016/j.scib.2022.12.023 | |
7Y3G (No Gprot) | A | Orphan | Orphan | GPR12 | Homo sapiens | - | - | 2.77 | 2023-06-07 | 10.1016/j.scib.2022.12.023 | ||
7XXH | A | Nucleotide | P2Y | P2Y1 | Homo sapiens | 2MeSADP | - | chim(NtGi1-G11)/β1/γ2 | 2.9 | 2023-06-07 | 10.1093/procel/pwac025 | |
7XXH (No Gprot) | A | Nucleotide | P2Y | P2Y1 | Homo sapiens | 2MeSADP | - | 2.9 | 2023-06-07 | 10.1093/procel/pwac025 | ||
7XXI | A | Nucleotide | P2Y | P2Y12 | Homo sapiens | 2MeSADP | - | Gi2/β1/γ2 | 3 | 2023-06-07 | 10.1093/procel/pwac025 | |
7XXI (No Gprot) | A | Nucleotide | P2Y | P2Y12 | Homo sapiens | 2MeSADP | - | 3 | 2023-06-07 | 10.1093/procel/pwac025 | ||
8CIC | A | Nucleotide | Adenosine | A2A | Homo sapiens | Etrumadenant | Na | - | 2.1 | 2023-05-31 | 10.1038/s42004-023-00894-6 | |
8IWM | A | Orphan | Orphan | TA9 | Mus musculus | 2-Phenylethylamine | - | - | 3.17 | 2023-05-31 | 10.1038/s41586-023-06106-4 | |
8IWE | A | Orphan | Orphan | TA9 | Mus musculus | Spermidine | - | - | 3.4 | 2023-05-31 | 10.1038/s41586-023-06106-4 | |
8HJ5 | A | Orphan | Orphan | MRGPRX1 | Homo sapiens | PubChem 139030531 | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3 | 2023-05-31 | 10.1371/journal.pbio.3001975 | |
8HJ5 (No Gprot) | A | Orphan | Orphan | MRGPRX1 | Homo sapiens | PubChem 139030531 | - | 3 | 2023-05-31 | 10.1371/journal.pbio.3001975 | ||
7XWO | A | Peptide | Tachykinin | NK2 | Homo sapiens | Neurokinin-A | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.7 | 2023-05-31 | 10.1038/s41421-022-00437-8 | |
7XWO (No Gprot) | A | Peptide | Tachykinin | NK2 | Homo sapiens | Neurokinin-A | - | 2.7 | 2023-05-31 | 10.1038/s41421-022-00437-8 | ||
8IW9 | A | Orphan | Orphan | TA9 | Mus musculus | - | - | chim(NtGi1-Gs)/β1/γ2 | 3.08 | 2023-05-31 | 10.1038/s41586-023-06106-4 | |
8IW9 (No Gprot) | A | Orphan | Orphan | TA9 | Mus musculus | - | - | 3.08 | 2023-05-31 | 10.1038/s41586-023-06106-4 | ||
8IW7 | A | Orphan | Orphan | TA9 | Mus musculus | 2-Phenylethylamine | - | chim(NtGi1-Gs)/β1/γ2 | 2.97 | 2023-05-31 | 10.1038/s41586-023-06106-4 | |
8IW7 (No Gprot) | A | Orphan | Orphan | TA9 | Mus musculus | 2-Phenylethylamine | - | 2.97 | 2023-05-31 | 10.1038/s41586-023-06106-4 | ||
8IW4 | A | Orphan | Orphan | TA9 | Mus musculus | Spermidine | - | chim(NtGi1-Gs)/β1/γ2 | 3.49 | 2023-05-31 | 10.1038/s41586-023-06106-4 | |
8IW4 (No Gprot) | A | Orphan | Orphan | TA9 | Mus musculus | Spermidine | - | 3.49 | 2023-05-31 | 10.1038/s41586-023-06106-4 | ||
8IW1 | A | Orphan | Orphan | TA9 | Mus musculus | - | - | chim(NtGi1-Gs)/β1/γ2 | 3.4 | 2023-05-31 | 10.1038/s41586-023-06106-4 | |
8IW1 (No Gprot) | A | Orphan | Orphan | TA9 | Mus musculus | - | - | 3.4 | 2023-05-31 | 10.1038/s41586-023-06106-4 | ||
8ITF | A | Orphan | Orphan | TA9 | Mus musculus | DMCHA | - | chim(NtGi1-Gs)/β1/γ2 | 3.46 | 2023-05-31 | 10.1038/s41586-023-06106-4 | |
8ITF (No Gprot) | A | Orphan | Orphan | TA9 | Mus musculus | DMCHA | - | 3.46 | 2023-05-31 | 10.1038/s41586-023-06106-4 | ||
8EJK | A | Lipid | Free Fatty Acid | FFA1 | Homo sapiens | TAK-875 | - | chim(NtGi1L-Gs-CtGq)/β1/γ2 | 3.4 | 2023-05-24 | 10.1073/pnas.2219569120 | |
8EJK (No Gprot) | A | Lipid | Free Fatty Acid | FFA1 | Homo sapiens | TAK-875 | - | 3.4 | 2023-05-24 | 10.1073/pnas.2219569120 | ||
8EJC | A | Lipid | Free Fatty Acid | FFA1 | Homo sapiens | TAK-875 | - | chim(NtGi1L-Gs-CtGq)/β1/γ2 | 3 | 2023-05-24 | 10.1073/pnas.2219569120 | |
8EJC (No Gprot) | A | Lipid | Free Fatty Acid | FFA1 | Homo sapiens | TAK-875 | - | 3 | 2023-05-24 | 10.1073/pnas.2219569120 | ||
8EIT | A | Lipid | Free Fatty Acid | FFA1 | Homo sapiens | Doconexent | - | chim(NtGi1L-Gs-CtGq)/β1/γ2 | 2.8 | 2023-05-24 | 10.1073/pnas.2219569120 | |
8EIT (No Gprot) | A | Lipid | Free Fatty Acid | FFA1 | Homo sapiens | Doconexent | - | 2.8 | 2023-05-24 | 10.1073/pnas.2219569120 | ||
8IA8 | A | Peptide | Complement Peptide | C3aB | Homo sapiens | E7 peptide | - | Gi1/β1/γ2 | 2.86 | 2023-05-24 | To be published | |
8IA8 (No Gprot) | A | Peptide | Complement Peptide | C3aB | Homo sapiens | E7 peptide | - | 2.86 | 2023-05-24 | To be published | ||
8GHV | A | Lipid | Cannabinoid | CB1 | Homo sapiens | AMG315 | - | Gi1/β1/γ2 | 2.8 | 2023-05-24 | 10.1038/s41467-023-37864-4 | |
8GHV (No Gprot) | A | Lipid | Cannabinoid | CB1 | Homo sapiens | AMG315 | - | 2.8 | 2023-05-24 | 10.1038/s41467-023-37864-4 | ||
7Y1F | A | Peptide | Opioid | κ | Homo sapiens | Dynorphin | - | Gi1/β1/γ2 | 3.3 | 2023-05-24 | 10.1093/procel/pwac033 | |
7Y1F (No Gprot) | A | Peptide | Opioid | κ | Homo sapiens | Dynorphin | - | 3.3 | 2023-05-24 | 10.1093/procel/pwac033 | ||
7TRS | A | Amine | Acetylcholine (muscarinic) | M4 | Homo sapiens | Acetylcholine | - | Gi1/β1/γ2 | 2.8 | 2023-05-17 | 10.2139/ssrn.4034884 | |
7TRS (No Gprot) | A | Amine | Acetylcholine (muscarinic) | M4 | Homo sapiens | Acetylcholine | - | 2.8 | 2023-05-17 | 10.2139/ssrn.4034884 | ||
7TRQ | A | Amine | Acetylcholine (muscarinic) | M4 | Homo sapiens | Iperoxo | VU0467154 | Gi1/β1/γ2 | 2.5 | 2023-05-17 | 10.2139/ssrn.4034884 | |
7TRQ (No Gprot) | A | Amine | Acetylcholine (muscarinic) | M4 | Homo sapiens | Iperoxo | VU0467154 | 2.5 | 2023-05-17 | 10.2139/ssrn.4034884 | ||
7TRP | A | Amine | Acetylcholine (muscarinic) | M4 | Homo sapiens | Iperoxo | LY2033298 | Gi1/β1/γ2 | 2.4 | 2023-05-17 | 10.2139/ssrn.4034884 | |
7TRP (No Gprot) | A | Amine | Acetylcholine (muscarinic) | M4 | Homo sapiens | Iperoxo | LY2033298 | 2.4 | 2023-05-17 | 10.2139/ssrn.4034884 | ||
7TRK | A | Amine | Acetylcholine (muscarinic) | M4 | Homo sapiens | Iperoxo | - | Gi1/β1/γ2 | 2.8 | 2023-05-17 | 10.2139/ssrn.4034884 | |
7TRK (No Gprot) | A | Amine | Acetylcholine (muscarinic) | M4 | Homo sapiens | Iperoxo | - | 2.8 | 2023-05-17 | 10.2139/ssrn.4034884 | ||
8G2Y | B2 | Adhesion | Adhesion | ADGRF1 | Homo sapiens | - | LPC | chim(Gs-CtGq)/β1/γ2 | 3.44 | 2023-05-10 | 10.1038/s41467-023-38083-7 | |
8G2Y (No Gprot) | B2 | Adhesion | Adhesion | ADGRF1 | Homo sapiens | - | LPC | 3.44 | 2023-05-10 | 10.1038/s41467-023-38083-7 | ||
8HK3 | A | Peptide | Complement Peptide | C3aB | Homo sapiens | - | - | Gi1/β1/γ2 | 3.2 | 2023-05-10 | 10.1038/s41589-023-01339-w | |
8HK3 (No Gprot) | A | Peptide | Complement Peptide | C3aB | Homo sapiens | - | - | 3.2 | 2023-05-10 | 10.1038/s41589-023-01339-w | ||
8HK2 | A | Peptide | Complement Peptide | C3aB | Homo sapiens | C3a anaphylatoxin | - | Gi1/β1/γ2 | 2.9 | 2023-05-10 | 10.1038/s41589-023-01339-w | |
8HK2 (No Gprot) | A | Peptide | Complement Peptide | C3aB | Homo sapiens | C3a anaphylatoxin | - | 2.9 | 2023-05-10 | 10.1038/s41589-023-01339-w | ||
8HK5 | A | Peptide | Complement Peptide | C5a1 | Homo sapiens | Complement C5 | - | Gi1/β1/γ2 | 3 | 2023-05-10 | 10.1038/s41589-023-01339-w | |
8HK5 (No Gprot) | A | Peptide | Complement Peptide | C5a1 | Homo sapiens | Complement C5 | - | 3 | 2023-05-10 | 10.1038/s41589-023-01339-w | ||
8GUT | A | Lipid | Cannabinoid | CB2 | Homo sapiens | LEI-102 | - | Gi1/β1/γ2 | 2.98 | 2023-05-10 | 10.1038/s41467-023-37112-9 | |
8GUT (No Gprot) | A | Lipid | Cannabinoid | CB2 | Homo sapiens | LEI-102 | - | 2.98 | 2023-05-10 | 10.1038/s41467-023-37112-9 | ||
8GUS | A | Lipid | Cannabinoid | CB2 | Homo sapiens | HU-308 | - | Gi1/β1/γ2 | 2.97 | 2023-05-10 | 10.1038/s41467-023-37112-9 | |
8GUS (No Gprot) | A | Lipid | Cannabinoid | CB2 | Homo sapiens | HU-308 | - | 2.97 | 2023-05-10 | 10.1038/s41467-023-37112-9 | ||
8GUR | A | Lipid | Cannabinoid | CB2 | Homo sapiens | CP55,940 | - | Gi1/β1/γ2 | 2.84 | 2023-05-10 | 10.1038/s41467-023-37112-9 | |
8GUR (No Gprot) | A | Lipid | Cannabinoid | CB2 | Homo sapiens | CP55,940 | - | 2.84 | 2023-05-10 | 10.1038/s41467-023-37112-9 | ||
8GUQ | A | Lipid | Cannabinoid | CB2 | Homo sapiens | Olorinab | - | Gi1/β1/γ2 | 3.08 | 2023-05-10 | 10.1038/s41467-023-37112-9 | |
8GUQ (No Gprot) | A | Lipid | Cannabinoid | CB2 | Homo sapiens | Olorinab | - | 3.08 | 2023-05-10 | 10.1038/s41467-023-37112-9 | ||
7XY7 | A | Nucleotide | Adenosine | A2B | Homo sapiens | NECA | - | chim(NtGi1-Gs)/β1/γ2 | 3.26 | 2023-05-03 | 10.1126/sciadv.add3709 | |
7XY7 (No Gprot) | A | Nucleotide | Adenosine | A2B | Homo sapiens | NECA | - | 3.26 | 2023-05-03 | 10.1126/sciadv.add3709 | ||
7XY6 | A | Nucleotide | Adenosine | A2B | Homo sapiens | BAY 60-6583 | - | chim(NtGi1-Gs)/β1/γ2 | 2.99 | 2023-05-03 | 10.1126/sciadv.add3709 | |
7XY6 (No Gprot) | A | Nucleotide | Adenosine | A2B | Homo sapiens | BAY 60-6583 | - | 2.99 | 2023-05-03 | 10.1126/sciadv.add3709 | ||
8DZR | A | Peptide | Opioid | κ | Homo sapiens | GR89,696 | - | chim(NtGi2-Gt3)/β1/γ2 | 2.61 | 2023-05-03 | 10.1038/s41586-023-06030-7 | |
8DZR (No Gprot) | A | Peptide | Opioid | κ | Homo sapiens | GR89,696 | - | 2.61 | 2023-05-03 | 10.1038/s41586-023-06030-7 | ||
8DZS | A | Peptide | Opioid | κ | Homo sapiens | GR89,696 | - | chim(NtGi2-Gz)/β1/γ2 | 2.65 | 2023-05-03 | 10.1038/s41586-023-06030-7 | |
8DZS (No Gprot) | A | Peptide | Opioid | κ | Homo sapiens | GR89,696 | - | 2.65 | 2023-05-03 | 10.1038/s41586-023-06030-7 | ||
8DZP | A | Peptide | Opioid | κ | Homo sapiens | momSalB | - | Gi1/β1/γ2 | 2.71 | 2023-05-03 | 10.1038/s41586-023-06030-7 | |
8DZP (No Gprot) | A | Peptide | Opioid | κ | Homo sapiens | momSalB | - | 2.71 | 2023-05-03 | 10.1038/s41586-023-06030-7 | ||
7XJJ | A | Peptide | Galanin | GAL1 | Homo sapiens | Galanin | - | Go/β1/γ2 | 3.3 | 2023-05-03 | 10.1073/pnas.2121465119 | |
7XJJ (No Gprot) | A | Peptide | Galanin | GAL1 | Homo sapiens | Galanin | - | 3.3 | 2023-05-03 | 10.1073/pnas.2121465119 | ||
8DZQ | A | Peptide | Opioid | κ | Homo sapiens | momSalB | - | Go/β1/γ2 | 2.82 | 2023-05-03 | 10.1038/s41586-023-06030-7 | |
8DZQ (No Gprot) | A | Peptide | Opioid | κ | Homo sapiens | momSalB | - | 2.82 | 2023-05-03 | 10.1038/s41586-023-06030-7 | ||
7XKA | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Epinephrine | - | - | 3.1 | 2023-04-26 | 10.1038/s41467-023-37808-y | |
7XK9 | A | Amine | Adrenergic | β2 | Homo sapiens | Constrained Isoproterenol | Na | - | 3.4 | 2023-04-26 | doi.org/10.1038/s41467-023-37808-y | |
8FLU | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | Long-Acting PTH | - | Gs/β1/γ2 | 2.76 | 2023-04-26 | 10.1016/j.str.2023.04.002 | |
8FLU (No Gprot) | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | Long-Acting PTH | - | 2.76 | 2023-04-26 | 10.1016/j.str.2023.04.002 | ||
8FLT | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | M-PTH(1-14) | - | Gs/β1/γ2 | 3.03 | 2023-04-26 | 10.1016/j.str.2023.04.002 | |
8FLT (No Gprot) | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | M-PTH(1-14) | - | 3.03 | 2023-04-26 | 10.1016/j.str.2023.04.002 | ||
8FLS | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | Abaloparatide | - | Gs/β1/γ2 | 3.09 | 2023-04-26 | 10.1016/j.str.2023.04.002 | |
8FLS (No Gprot) | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | Abaloparatide | - | 3.09 | 2023-04-26 | 10.1016/j.str.2023.04.002 | ||
8FLR | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | PTHrP(1-36) | - | Gs/β1/γ2 | 2.94 | 2023-04-26 | 10.1016/j.str.2023.04.002 | |
8FLR (No Gprot) | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | PTHrP(1-36) | - | 2.94 | 2023-04-26 | 10.1016/j.str.2023.04.002 | ||
8FLQ | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | PTH | - | Gs/β1/γ2 | 2.55 | 2023-04-26 | 10.1016/j.str.2023.04.002 | |
8FLQ (No Gprot) | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | PTH | - | 2.55 | 2023-04-26 | 10.1016/j.str.2023.04.002 | ||
7YKD | A | Protein | Chemerin | CML1 | Homo sapiens | Chemerin-9 | - | Gi1/β1/γ2 | 2.81 | 2023-04-19 | 10.1073/pnas.2214324120 | |
7YKD (No Gprot) | A | Protein | Chemerin | CML1 | Homo sapiens | Chemerin-9 | - | 2.81 | 2023-04-19 | 10.1073/pnas.2214324120 | ||
8G94 | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | - | CD69 | Gi1/β1/γ2 | 3.15 | 2023-04-19 | 10.7554/eLife.88204 | |
8G94 (No Gprot) | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | - | CD69 | 3.15 | 2023-04-19 | 10.7554/eLife.88204 | ||
7YAE | A | Peptide | Somatostatin | SST2 | Homo sapiens | Octreotide | - | Gi1/β1/γ2 | 3.37 | 2023-04-19 | 10.1038/s41467-023-36673-z | |
7YAE (No Gprot) | A | Peptide | Somatostatin | SST2 | Homo sapiens | Octreotide | - | 3.37 | 2023-04-19 | 10.1038/s41467-023-36673-z | ||
7YAC | A | Peptide | Somatostatin | SST2 | Homo sapiens | Paltusotine | - | Gi1/β1/γ2 | 3.24 | 2023-04-19 | 10.1038/s41467-023-36673-z | |
7YAC (No Gprot) | A | Peptide | Somatostatin | SST2 | Homo sapiens | Paltusotine | - | 3.24 | 2023-04-19 | 10.1038/s41467-023-36673-z | ||
7ZLY | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | - | - | - | 2.7 | 2023-04-12 | 10.1038/s41467-023-37177-6 | |
7ZL9 | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | - | - | - | 2.7 | 2023-04-12 | 10.1038/s41467-023-37177-6 | |
8IBV | A | Peptide | Motilin | Motilin | Homo sapiens | Motilin | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.19 | 2023-04-12 | 10.1126/sciadv.ade9020 | |
8IBV (No Gprot) | A | Peptide | Motilin | Motilin | Homo sapiens | Motilin | - | 3.19 | 2023-04-12 | 10.1126/sciadv.ade9020 | ||
8IBU | A | Peptide | Motilin | Motilin | Homo sapiens | Erythromycin-A | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.51 | 2023-04-12 | 10.1126/sciadv.ade9020 | |
8IBU (No Gprot) | A | Peptide | Motilin | Motilin | Homo sapiens | Erythromycin-A | - | 3.51 | 2023-04-12 | 10.1126/sciadv.ade9020 | ||
8FU6 | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | Glucagon derivative ZP3780 | - | Gs/β1/γ2 | 2.9 | 2023-04-12 | 10.1016/j.cell.2023.02.028 | |
8FU6 (No Gprot) | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | Glucagon derivative ZP3780 | - | 2.9 | 2023-04-12 | 10.1016/j.cell.2023.02.028 | ||
7YIT | A | Peptide | Opioid | κ | Homo sapiens | Nalfurafine | - | - | 3.3 | 2023-04-12 | 10.1038/s41467-023-37041-7 | |
8A6E | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | - | 1.8 | 2023-03-29 | 10.1038/s41586-023-05863-6 | |
8A6D | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | - | 1.8 | 2023-03-29 | 10.1038/s41586-023-05863-6 | |
8A6C | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | - | 1.8 | 2023-03-29 | 10.1038/s41586-023-05863-6 | |
7ZBE | A | Sensory | Opsins | Rhodopsin | Bos taurus | 11-cis-Retinal | - | - | 1.8 | 2023-03-29 | 10.1038/s41586-023-05863-6 | |
7ZBC | A | Sensory | Opsins | Rhodopsin | Bos taurus | 11-cis-Retinal | - | - | 1.8 | 2023-03-29 | 10.1038/s41586-023-05863-6 | |
8FN1 | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | Neurotensin/Neuromedin-N | - | chim(NtGi1-Go)/β1/γ2 | 2.88 | 2023-03-29 | 10.1021/acs.biochem.3c00029 | |
8FN1 (No Gprot) | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | Neurotensin/Neuromedin-N | - | 2.88 | 2023-03-29 | 10.1021/acs.biochem.3c00029 | ||
8FN0 | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | Neurotensin/Neuromedin-N | PubChem 118610427 | chim(NtGi1-Go)/β1/γ2 | 2.89 | 2023-03-29 | 10.1021/acs.biochem.3c00029 | |
8FN0 (No Gprot) | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | Neurotensin/Neuromedin-N | PubChem 118610427 | 2.89 | 2023-03-29 | 10.1021/acs.biochem.3c00029 | ||
7YS6 | A | Amine | 5-Hydroxytryptamine | 5-HT6 | Homo sapiens | Serotonin | - | chim(NtGi1-Gs)/β1/γ2 | 3 | 2023-03-29 | 10.1073/pnas.2209917120 | |
7YS6 (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT6 | Homo sapiens | Serotonin | - | 3 | 2023-03-29 | 10.1073/pnas.2209917120 | ||
8FMZ | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | Neurotensin/Neuromedin-N | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 2.59 | 2023-03-29 | 10.1021/acs.biochem.3c00029 | |
8FMZ (No Gprot) | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | Neurotensin/Neuromedin-N | - | 2.59 | 2023-03-29 | 10.1021/acs.biochem.3c00029 | ||
7F6G | A | Peptide | Angiotensin | AT1 | Homo sapiens | SAR1-AngII | - | Gq/β1/γ2 | 2.9 | 2023-03-29 | 10.15252/embj.2022112940 | |
7F6G (No Gprot) | A | Peptide | Angiotensin | AT1 | Homo sapiens | SAR1-AngII | - | 2.9 | 2023-03-29 | 10.15252/embj.2022112940 | ||
8I2H | A | Protein | Glycoprotein Hormone | FSH | Homo sapiens | - | - | - | 6 | 2023-03-22 | 10.1038/s41467-023-36170-3 | |
8F76 | O1 | Odorant receptors | Odorant family 51 | OR51E2 | Homo sapiens | Propanoic acid | - | Gs/β1/γ2 | 3.1 | 2023-03-22 | 10.1038/s41586-023-05798-y | |
8F76 (No Gprot) | O1 | Odorant receptors | Odorant family 51 | OR51E2 | Homo sapiens | Propanoic acid | - | 3.1 | 2023-03-22 | 10.1038/s41586-023-05798-y | ||
8GNG | A | Nucleotide | Adenosine | A2A | Homo sapiens | Istradefylline | - | - | 3.2 | 2023-03-22 | 10.1124/molpharm.122.000633 | |
8GNE | A | Nucleotide | Adenosine | A2A | Homo sapiens | KW-6356 | Na | - | 2.3 | 2023-03-22 | 10.1124/molpharm.122.000633 | |
8HCQ | A | Peptide | Endothelin | ETA | Homo sapiens | Endothelin-1 | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.01 | 2023-03-22 | 10.1038/s41467-023-36998-9 | |
8HCQ (No Gprot) | A | Peptide | Endothelin | ETA | Homo sapiens | Endothelin-1 | - | 3.01 | 2023-03-22 | 10.1038/s41467-023-36998-9 | ||
8HCX | A | Peptide | Endothelin | ETB | Homo sapiens | Endothelin-1 | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 3.5 | 2023-03-22 | 10.1038/s41467-023-36998-9 | |
8HCX (No Gprot) | A | Peptide | Endothelin | ETB | Homo sapiens | Endothelin-1 | - | 3.5 | 2023-03-22 | 10.1038/s41467-023-36998-9 | ||
8HBD | A | Peptide | Endothelin | ETB | Homo sapiens | IRL1620 | - | Gi1/β1/γ2 | 2.99 | 2023-03-22 | 10.1038/s41467-023-36998-9 | |
8HBD (No Gprot) | A | Peptide | Endothelin | ETB | Homo sapiens | IRL1620 | - | 2.99 | 2023-03-22 | 10.1038/s41467-023-36998-9 | ||
7YOO | A | Peptide | Neuropeptide Y | Y2 | Homo sapiens | Neuropeptide-Y | - | Gi1/β1/γ2 | 3.11 | 2023-03-22 | 10.1016/j.str.2022.11.010 | |
7YOO (No Gprot) | A | Peptide | Neuropeptide Y | Y2 | Homo sapiens | Neuropeptide-Y | - | 3.11 | 2023-03-22 | 10.1016/j.str.2022.11.010 | ||
7YON | A | Peptide | Neuropeptide Y | Y2 | Homo sapiens | Peptide-YY(3-36) | - | Gi1/β1/γ2 | 2.95 | 2023-03-22 | 10.1016/j.str.2022.11.010 | |
7YON (No Gprot) | A | Peptide | Neuropeptide Y | Y2 | Homo sapiens | Peptide-YY(3-36) | - | 2.95 | 2023-03-22 | 10.1016/j.str.2022.11.010 | ||
8ID9 | A | Lipid | Free Fatty Acid | FFA4 | Homo sapiens | Eicosapentaenoic acid | - | Gi1/β1/γ2 | 3 | 2023-03-15 | 10.1126/science.add6220 | |
8ID9 (No Gprot) | A | Lipid | Free Fatty Acid | FFA4 | Homo sapiens | Eicosapentaenoic acid | - | 3 | 2023-03-15 | 10.1126/science.add6220 | ||
8ID8 | A | Lipid | Free Fatty Acid | FFA4 | Homo sapiens | TUG-891 | - | Gi1/β1/γ2 | 3 | 2023-03-15 | 10.1126/science.add6220 | |
8ID8 (No Gprot) | A | Lipid | Free Fatty Acid | FFA4 | Homo sapiens | TUG-891 | - | 3 | 2023-03-15 | 10.1126/science.add6220 | ||
8ID6 | A | Lipid | Free Fatty Acid | FFA4 | Homo sapiens | Oleic acid | - | Gi1/β1/γ2 | 2.8 | 2023-03-15 | 10.1126/science.add6220 | |
8ID6 (No Gprot) | A | Lipid | Free Fatty Acid | FFA4 | Homo sapiens | Oleic acid | - | 2.8 | 2023-03-15 | 10.1126/science.add6220 | ||
8ID4 | A | Lipid | Free Fatty Acid | FFA4 | Homo sapiens | Linoleic acid | - | Gi1/β1/γ2 | 3.1 | 2023-03-15 | 10.1126/science.add6220 | |
8ID4 (No Gprot) | A | Lipid | Free Fatty Acid | FFA4 | Homo sapiens | Linoleic acid | - | 3.1 | 2023-03-15 | 10.1126/science.add6220 | ||
8ID3 | A | Lipid | Free Fatty Acid | FFA4 | Homo sapiens | 9-Hydroxystearic acid | - | Gi1/β1/γ2 | 3.1 | 2023-03-15 | 10.1126/science.add6220 | |
8ID3 (No Gprot) | A | Lipid | Free Fatty Acid | FFA4 | Homo sapiens | 9-Hydroxystearic acid | - | 3.1 | 2023-03-15 | 10.1126/science.add6220 | ||
8HJ2 | A | Orphan | Orphan | GPR21 | Homo sapiens | - | - | chim(Gs-CtG15)/β1/γ2 | 3.8 | 2023-03-15 | 10.1038/s41467-023-35882-w | |
8HJ2 (No Gprot) | A | Orphan | Orphan | GPR21 | Homo sapiens | - | - | 3.8 | 2023-03-15 | 10.1038/s41467-023-35882-w | ||
8HJ0 | A | Orphan | Orphan | GPR21 | Homo sapiens | - | - | chim(Gs-CtG15)/β1/γ2 | 3.12 | 2023-03-15 | 10.1038/s41467-023-35882-w | |
8HJ0 (No Gprot) | A | Orphan | Orphan | GPR21 | Homo sapiens | - | - | 3.12 | 2023-03-15 | 10.1038/s41467-023-35882-w | ||
8HIX | A | Orphan | Orphan | GPR21 | Homo sapiens | - | - | Gs/β1/γ2 | 3.12 | 2023-03-15 | 10.1038/s41467-023-35882-w | |
8HIX (No Gprot) | A | Orphan | Orphan | GPR21 | Homo sapiens | - | - | 3.12 | 2023-03-15 | 10.1038/s41467-023-35882-w | ||
8HS2 | A | Orphan | Orphan | GPR20 | Homo sapiens | Fab046 | - | - | 3.08 | 2023-03-08 | 10.1038/s41421-023-00520-8 | |
8HSC | A | Orphan | Orphan | GPR20 | Homo sapiens | Fab046 | - | Gi1/β1/γ2 | 3.22 | 2023-03-08 | 10.1038/s41421-023-00520-8 | |
8HSC (No Gprot) | A | Orphan | Orphan | GPR20 | Homo sapiens | Fab046 | - | 3.22 | 2023-03-08 | 10.1038/s41421-023-00520-8 | ||
8HS3 | A | Orphan | Orphan | GPR20 | Homo sapiens | - | - | Gi1/β1/γ2 | 3.14 | 2023-03-08 | 10.1038/s41421-023-00520-8 | |
8HS3 (No Gprot) | A | Orphan | Orphan | GPR20 | Homo sapiens | - | - | 3.14 | 2023-03-08 | 10.1038/s41421-023-00520-8 | ||
8FYN | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | Na | - | 2 | 2023-03-08 | 10.1038/s41467-023-36733-4 | |
8G59 | A | Lipid | Free Fatty Acid | FFA4 | Homo sapiens | TUG-891 | - | chim(Gi1-CtGq)/β1/γ2 | 2.64 | 2023-03-08 | 10.1126/science.add6220 | |
8G59 (No Gprot) | A | Lipid | Free Fatty Acid | FFA4 | Homo sapiens | TUG-891 | - | 2.64 | 2023-03-08 | 10.1126/science.add6220 | ||
7W41 | A | Peptide | Bombesin | BB2 | Homo sapiens | PD176252 | - | - | 2.95 | 2023-02-22 | 10.1073/pnas.2216230120 | |
7W40 | A | Peptide | Bombesin | BB2 | Homo sapiens | Bombesin | - | chim(NtGi1L-Gq)/β1/γ2 | 3 | 2023-02-22 | 10.1073/pnas.2216230120 | |
7W40 (No Gprot) | A | Peptide | Bombesin | BB2 | Homo sapiens | Bombesin | - | 3 | 2023-02-22 | 10.1073/pnas.2216230120 | ||
7W3Z | A | Peptide | Bombesin | BB2 | Homo sapiens | Gastrin Releasing Peptide | - | chim(NtGi1L-Gq)/β1/γ2 | 3 | 2023-02-22 | 10.1073/pnas.2216230120 | |
7W3Z (No Gprot) | A | Peptide | Bombesin | BB2 | Homo sapiens | Gastrin Releasing Peptide | - | 3 | 2023-02-22 | 10.1073/pnas.2216230120 | ||
7XK2 | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | MK6892 | - | Gi1/β1/γ2 | 3.1 | 2023-02-22 | 10.1038/s41467-023-37177-6 | |
7XK2 (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | MK6892 | - | 3.1 | 2023-02-22 | 10.1038/s41467-023-37177-6 | ||
7XK8 | A | Peptide | Neuromedin U | NMUR2 | Homo sapiens | Neuromedin-U-25 | - | Gi1/β1/γ2 | 3.3 | 2023-02-22 | 10.1038/s41467-022-34814-4 | |
7XK8 (No Gprot) | A | Peptide | Neuromedin U | NMUR2 | Homo sapiens | Neuromedin-U-25 | - | 3.3 | 2023-02-22 | 10.1038/s41467-022-34814-4 | ||
7TMW | A | Peptide | Relaxin | RXFP1 | Homo sapiens | - | - | Gs/β1/γ2 | 3.2 | 2023-02-15 | 10.1101/2022.01.22.477343 | |
7TMW (No Gprot) | A | Peptide | Relaxin | RXFP1 | Homo sapiens | - | - | 3.2 | 2023-02-15 | 10.1101/2022.01.22.477343 | ||
7XV3 | A | Orphan | Orphan | GPR174 | Homo sapiens | Lysophosphatidylserine | - | chim(NtGi1-Gs)/β1/γ2 | 2.76 | 2023-02-15 | 10.1038/s41467-023-36575-0 | |
7XV3 (No Gprot) | A | Orphan | Orphan | GPR174 | Homo sapiens | Lysophosphatidylserine | - | 2.76 | 2023-02-15 | 10.1038/s41467-023-36575-0 | ||
8H8J | A | Orphan | Orphan | GPR35 | Homo sapiens | Lodoxamide | Ca | chim(NtGi1L-G13)/β1/γ2 | 3.2 | 2023-02-08 | 10.1038/s41421-022-00499-8 | |
8H8J (No Gprot) | A | Orphan | Orphan | GPR35 | Homo sapiens | Lodoxamide | Ca | 3.2 | 2023-02-08 | 10.1038/s41421-022-00499-8 | ||
7T96 | A | Amine | Acetylcholine (muscarinic) | M2 | Homo sapiens | Acetylcholine | LY2119620 | Go/β1/γ2 | 3.22 | 2023-01-25 | doi.org/10.1038/s41467-022-35726-z | |
7T96 (No Gprot) | A | Amine | Acetylcholine (muscarinic) | M2 | Homo sapiens | Acetylcholine | LY2119620 | 3.22 | 2023-01-25 | doi.org/10.1038/s41467-022-35726-z | ||
7XW9 | A | Peptide | Thyrotropin Releasing Hormone | TRH | Homo sapiens | TRH | - | chim(NtGi1L-Gs-CtGq)/β1/γ2 | 2.7 | 2022-12-28 | 10.1038/s41421-022-00477-0 | |
7XW9 (No Gprot) | A | Peptide | Thyrotropin Releasing Hormone | TRH | Homo sapiens | TRH | - | 2.7 | 2022-12-28 | 10.1038/s41421-022-00477-0 | ||
7WCN | A | Lipid | GPR119 | GPR119 | Homo sapiens | AR231453 | - | Gs/β1/γ2 | 2.87 | 2022-12-21 | 10.1038/s41467-022-34696-6 | |
7WCN (No Gprot) | A | Lipid | GPR119 | GPR119 | Homo sapiens | AR231453 | - | 2.87 | 2022-12-21 | 10.1038/s41467-022-34696-6 | ||
7WCM | A | Lipid | GPR119 | GPR119 | Homo sapiens | MBX-2982 | - | Gs/β1/γ2 | 2.33 | 2022-12-21 | 10.1038/s41467-022-34696-6 | |
7WCM (No Gprot) | A | Lipid | GPR119 | GPR119 | Homo sapiens | MBX-2982 | - | 2.33 | 2022-12-21 | 10.1038/s41467-022-34696-6 | ||
8HAO | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | PTH | - | chim(NtGi1-Gs)/β1/γ2 | 3.76 | 2022-12-21 | 10.1038/s41401-022-01032-z | |
8HAO (No Gprot) | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | PTH | - | 3.76 | 2022-12-21 | 10.1038/s41401-022-01032-z | ||
8HAF | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | PTHrP(1-36) | - | chim(NtGi1-Gs)/β1/γ2 | 3.25 | 2022-12-21 | 10.1038/s41401-022-01032-z | |
8HAF (No Gprot) | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | PTHrP(1-36) | - | 3.25 | 2022-12-21 | 10.1038/s41401-022-01032-z | ||
8HA0 | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | PTH | - | chim(NtGi1-Gs)/β1/γ2 | 2.62 | 2022-12-21 | 10.1038/s41401-022-01032-z | |
8HA0 (No Gprot) | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | PTH | - | 2.62 | 2022-12-21 | 10.1038/s41401-022-01032-z | ||
8F7S | A | Peptide | Opioid | δ | Homo sapiens | Deltorphin | - | Gi1/β1/γ2 | 3 | 2022-12-14 | 10.1016/j.cell.2022.12.026 | |
8F7S (No Gprot) | A | Peptide | Opioid | δ | Homo sapiens | Deltorphin | - | 3 | 2022-12-14 | 10.1016/j.cell.2022.12.026 | ||
8F7W | A | Peptide | Opioid | κ | Homo sapiens | Dynorphin | - | Gi1/β1/γ2 | 3.19 | 2022-12-14 | 10.1016/j.cell.2022.12.026 | |
8F7W (No Gprot) | A | Peptide | Opioid | κ | Homo sapiens | Dynorphin | - | 3.19 | 2022-12-14 | 10.1016/j.cell.2022.12.026 | ||
8F7R | A | Peptide | Opioid | μ | Homo sapiens | Endomorphin | - | Gi1/β1/γ2 | 3.28 | 2022-12-14 | 10.1016/j.cell.2022.12.026 | |
8F7R (No Gprot) | A | Peptide | Opioid | μ | Homo sapiens | Endomorphin | - | 3.28 | 2022-12-14 | 10.1016/j.cell.2022.12.026 | ||
8F7Q | A | Peptide | Opioid | μ | Homo sapiens | β-Endorphin | - | Gi1/β1/γ2 | 3.22 | 2022-12-14 | 10.1016/j.cell.2022.12.026 | |
8F7Q (No Gprot) | A | Peptide | Opioid | μ | Homo sapiens | β-Endorphin | - | 3.22 | 2022-12-14 | 10.1016/j.cell.2022.12.026 | ||
8F7X | A | Peptide | Opioid | NOP | Homo sapiens | Nociceptin | - | Gi1/β1/γ2 | 3.28 | 2022-12-14 | 10.1016/j.cell.2022.12.026 | |
8F7X (No Gprot) | A | Peptide | Opioid | NOP | Homo sapiens | Nociceptin | - | 3.28 | 2022-12-14 | 10.1016/j.cell.2022.12.026 | ||
7T2H | A | Peptide | Opioid | μ | Mus musculus | Lofentanil | - | Gi1/β1/γ2 | 2.5 | 2022-12-07 | 10.1038/s41589-022-01208-y | |
7T2H (No Gprot) | A | Peptide | Opioid | μ | Mus musculus | Lofentanil | - | 2.5 | 2022-12-07 | 10.1038/s41589-022-01208-y | ||
7T2G | A | Peptide | Opioid | μ | Mus musculus | Mitragynine Pseudoindoxyl | - | Gi1/β1/γ2 | 2.5 | 2022-12-07 | 10.1038/s41589-022-01208-y | |
7T2G (No Gprot) | A | Peptide | Opioid | μ | Mus musculus | Mitragynine Pseudoindoxyl | - | 2.5 | 2022-12-07 | 10.1038/s41589-022-01208-y | ||
7U2K | A | Peptide | Opioid | μ | Mus musculus | C6-guano | - | Gi1/β1/γ2 | 3.3 | 2022-12-07 | 10.1038/s41586-022-05588-y | |
7U2K (No Gprot) | A | Peptide | Opioid | μ | Mus musculus | C6-guano | - | 3.3 | 2022-12-07 | 10.1038/s41586-022-05588-y | ||
7XRR | A | Peptide | Orexin | OX2 | Homo sapiens | Lemborexant | - | - | 2.89 | 2022-11-23 | 10.1016/j.str.2022.11.001 | |
7TRY | B1 | Peptide | Corticotropin Releasing Factor | CRF2 | Homo sapiens | Urocortin | - | chim(NtGi1-G11)/β1/γ2 | 3.7 | 2022-11-09 | 10.1038/s41467-022-33851-3 | |
7TRY (No Gprot) | B1 | Peptide | Corticotropin Releasing Factor | CRF2 | Homo sapiens | Urocortin | - | 3.7 | 2022-11-09 | 10.1038/s41467-022-33851-3 | ||
7TS0 | B1 | Peptide | Corticotropin Releasing Factor | CRF2 | Homo sapiens | Urocortin | - | chim(NtGi1L-Go)/β1/γ2 | 2.8 | 2022-11-09 | 10.1038/s41467-022-33851-3 | |
7TS0 (No Gprot) | B1 | Peptide | Corticotropin Releasing Factor | CRF2 | Homo sapiens | Urocortin | - | 2.8 | 2022-11-09 | 10.1038/s41467-022-33851-3 | ||
7X10 | B2 | Adhesion | Adhesion | ADGRL3 | Mus musculus | - | - | chim(NtGi1-G12)/β1/γ2 | 2.93 | 2022-10-26 | 10.1016/j.molcel.2022.10.009 | |
7X10 (No Gprot) | B2 | Adhesion | Adhesion | ADGRL3 | Mus musculus | - | - | 2.93 | 2022-10-26 | 10.1016/j.molcel.2022.10.009 | ||
7WY5 | B2 | Adhesion | Adhesion | ADGRL3 | Mus musculus | - | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.83 | 2022-10-26 | 10.1016/j.molcel.2022.10.009 | |
7WY5 (No Gprot) | B2 | Adhesion | Adhesion | ADGRL3 | Mus musculus | - | - | 2.83 | 2022-10-26 | 10.1016/j.molcel.2022.10.009 | ||
7WY8 | B2 | Adhesion | Adhesion | ADGRL3 | Mus musculus | - | - | chim(NtGi1-Gs)/β1/γ2 | 2.83 | 2022-10-26 | 10.1016/j.molcel.2022.10.009 | |
7WY8 (No Gprot) | B2 | Adhesion | Adhesion | ADGRL3 | Mus musculus | - | - | 2.83 | 2022-10-26 | 10.1016/j.molcel.2022.10.009 | ||
7WYB | B2 | Adhesion | Adhesion | ADGRL3 | Mus musculus | - | - | Gi1/β1/γ2 | 2.97 | 2022-10-26 | 10.1016/j.molcel.2022.10.009 | |
7WYB (No Gprot) | B2 | Adhesion | Adhesion | ADGRL3 | Mus musculus | - | - | 2.97 | 2022-10-26 | 10.1016/j.molcel.2022.10.009 | ||
7Y27 | A | Peptide | Somatostatin | SST2 | Homo sapiens | Somatostatin-14 | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 3.48 | 2022-10-19 | 10.1038/s41589-022-01130-3 | |
7Y27 (No Gprot) | A | Peptide | Somatostatin | SST2 | Homo sapiens | Somatostatin-14 | - | 3.48 | 2022-10-19 | 10.1038/s41589-022-01130-3 | ||
7Y26 | A | Peptide | Somatostatin | SST2 | Homo sapiens | Octreotide | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 3.3 | 2022-10-19 | 10.1038/s41589-022-01130-3 | |
7Y26 (No Gprot) | A | Peptide | Somatostatin | SST2 | Homo sapiens | Octreotide | - | 3.3 | 2022-10-19 | 10.1038/s41589-022-01130-3 | ||
7Y24 | A | Peptide | Somatostatin | SST2 | Homo sapiens | Octreotide | - | Go/β1/γ2 | 3.25 | 2022-10-19 | 10.1038/s41589-022-01130-3 | |
7Y24 (No Gprot) | A | Peptide | Somatostatin | SST2 | Homo sapiens | Octreotide | - | 3.25 | 2022-10-19 | 10.1038/s41589-022-01130-3 | ||
7UL3 | A | Amine | Histamine | H2 | Homo sapiens | Famotidine | - | - | 3 | 2022-06-29 | doi.org/10.1038/s41594-022-00859-8 | |
7T11 | A | Peptide | Somatostatin | SST2 | Homo sapiens | Octreotide | - | Gi3/β1/γ2 | 2.7 | 2022-03-09 | doi.org/10.1038/s41594-022-00727-5 | |
7T11 (No Gprot) | A | Peptide | Somatostatin | SST2 | Homo sapiens | Octreotide | - | 2.7 | 2022-03-09 | doi.org/10.1038/s41594-022-00727-5 | ||
7T10 | A | Peptide | Somatostatin | SST2 | Homo sapiens | Somatostatin-14 | - | Gi3/β1/γ2 | 2.5 | 2022-03-09 | doi.org/10.1038/s41594-022-00727-5 | |
7T10 (No Gprot) | A | Peptide | Somatostatin | SST2 | Homo sapiens | Somatostatin-14 | - | 2.5 | 2022-03-09 | doi.org/10.1038/s41594-022-00727-5 | ||
7RKY | A | Other | Unclassified | US27 | Human betaherpesvirus 5 | - | GDP | Gi1/β1/γ2 | 3.8 | 2022-01-26 | doi.org/10.1126/sciadv.abl5442 | |
7RKY (No Gprot) | A | Other | Unclassified | US27 | Human betaherpesvirus 5 | - | GDP | 3.8 | 2022-01-26 | doi.org/10.1126/sciadv.abl5442 | ||
9EAI | A | Peptide | Angiotensin | AT1 | Homo sapiens | Losartan | Nanobody AT209 | - | 3.1 | 2025-03-05 | To be published | |
9JVM | A | Orphan | Orphan | GPR4 | Xenopus tropicalis | - | - | - | 2.36 | 2025-02-26 | 10.1016/j.cell.2024.12.001 | |
9JVH | A | Orphan | Orphan | GPR4 | Mus musculus | - | - | - | 2.76 | 2025-02-26 | 10.1016/j.cell.2024.12.001 | |
9IYA | A | Lipid | GPR55 | GPR55 | Homo sapiens | ONO-9710531 | - | - | 3.04 | 2025-01-01 | 10.1038/s41422-024-01046-8 | |
9IZF | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | NKP | - | Gi1/β1/γ2 | 3.14 | 2025-01-01 | 10.1016/j.jsb.2024.108164 | |
9IZF (No Gprot) | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | NKP | - | 3.14 | 2025-01-01 | 10.1016/j.jsb.2024.108164 | ||
8YNT | A | Peptide | Melanin Concentrating Hormone | MCH1 | Homo sapiens | SNAP-94847 | - | - | 3.43 | 2024-12-18 | 10.1038/s41421-024-00754-0 | |
8YNS | A | Peptide | Melanin Concentrating Hormone | MCH1 | Homo sapiens | SNAP-94847 | - | - | 3.33 | 2024-12-18 | 10.1038/s41421-024-00754-0 | |
9IVG | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | GLP-1 (Truncated) | - | chim(NtGi1-Gs)/β1/γ2 | 3 | 2024-11-27 | 10.1016/j.apsb.2024.09.002 | |
9IVG (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | GLP-1 (Truncated) | - | 3 | 2024-11-27 | 10.1016/j.apsb.2024.09.002 | ||
8ZX5 | A | Lipid | GPR55 | GPR55 | Homo sapiens | AM251 | - | chim(NtGi1-G13)/β1/γ2 | 2.85 | 2024-11-13 | 10.1038/s41422-024-01044-w | |
8ZX5 (No Gprot) | A | Lipid | GPR55 | GPR55 | Homo sapiens | AM251 | - | 2.85 | 2024-11-13 | 10.1038/s41422-024-01044-w | ||
8ZX4 | A | Lipid | GPR55 | GPR55 | Homo sapiens | Lysophosphatidylinositol | - | chim(NtGi1-G13)/β1/γ2 | 3.03 | 2024-11-13 | 10.1038/s41422-024-01044-w | |
8ZX4 (No Gprot) | A | Lipid | GPR55 | GPR55 | Homo sapiens | Lysophosphatidylinositol | - | 3.03 | 2024-11-13 | 10.1038/s41422-024-01044-w | ||
8YUV | A | Amine | Histamine | H3 | Homo sapiens | Immepip | - | Gi1/β1/γ2 | 3 | 2024-06-05 | 10.1002/advs.202310120 | |
8YUV (No Gprot) | A | Amine | Histamine | H3 | Homo sapiens | Immepip | - | 3 | 2024-06-05 | 10.1002/advs.202310120 | ||
8HMV | A | Orphan | Orphan | GPR21 | Homo sapiens | - | - | Gs/β1/γ2 | 2.91 | 2023-03-01 | 10.1002/mco2.205 | |
8HMV (No Gprot) | A | Orphan | Orphan | GPR21 | Homo sapiens | - | - | 2.91 | 2023-03-01 | 10.1002/mco2.205 | ||
8EA0 | A | Amine | Acetylcholine (muscarinic) | M3 | Homo sapiens | Iperoxo | - | - | 2.56 | 2022-11-30 | 10.1038/s41586-022-05489-0 | |
8E9X | A | Amine | Acetylcholine (muscarinic) | M4 | Homo sapiens | 2-Deoxycytidine | - | chim(NtGi1-Go)/β1/γ2 | 2.7 | 2022-11-30 | 10.1038/s41586-022-05489-0 | |
8E9X (No Gprot) | A | Amine | Acetylcholine (muscarinic) | M4 | Homo sapiens | 2-Deoxycytidine | - | 2.7 | 2022-11-30 | 10.1038/s41586-022-05489-0 | ||
8DWH | A | Orphan | Orphan | MRGPRX1 | Homo sapiens | PubChem 139030531 | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 3.25 | 2022-11-02 | 10.1038/s41589-022-01173-6 | |
8DWH (No Gprot) | A | Orphan | Orphan | MRGPRX1 | Homo sapiens | PubChem 139030531 | - | 3.25 | 2022-11-02 | 10.1038/s41589-022-01173-6 | ||
8DWG | A | Orphan | Orphan | MRGPRX1 | Homo sapiens | Proenkephalin-A | ML382 | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 2.71 | 2022-11-02 | 10.1038/s41589-022-01173-6 | |
8DWG (No Gprot) | A | Orphan | Orphan | MRGPRX1 | Homo sapiens | Proenkephalin-A | ML382 | 2.71 | 2022-11-02 | 10.1038/s41589-022-01173-6 | ||
8DWC | A | Orphan | Orphan | MRGPRX1 | Homo sapiens | Proenkephalin-A | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 2.87 | 2022-11-02 | 10.1038/s41589-022-01173-6 | |
8DWC (No Gprot) | A | Orphan | Orphan | MRGPRX1 | Homo sapiens | Proenkephalin-A | - | 2.87 | 2022-11-02 | 10.1038/s41589-022-01173-6 | ||
8Y0H | A | Protein | Chemokine | CXCR3 | Homo sapiens | VUF11418 | - | - | 3.53 | 2025-02-26 | To be published | |
8XYI | A | Protein | Chemokine | CXCR3 | Homo sapiens | VUF10661 | - | - | 3.16 | 2025-02-26 | To be published | |
8XXY | A | Protein | Chemokine | CXCR3 | Homo sapiens | - | - | - | 3.68 | 2025-02-26 | To be published | |
8ZPN | A | Protein | Chemokine | CXCR4 | Homo sapiens | AMD3100 | Cholesterol | - | 3.31 | 2025-02-26 | To be published | |
8ZPM | A | Protein | Chemokine | CXCR4 | Homo sapiens | AMD070 | Cholesterol | - | 3.2 | 2025-02-26 | To be published | |
8ZPL | A | Protein | Chemokine | CXCR4 | Homo sapiens | HF51116 | Cholesterol | - | 3.01 | 2025-02-26 | To be published | |
8KIG | A | Peptide | Melanocortin | MC3 | Homo sapiens | SHU9119 | Ca | - | 3.1 | 2025-02-26 | 10.2210/pdb8KIG/pdb | |
9J1P | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | g1:Ox | - | chim(NtGi1-Gs)/β1/γ2 | 2.99 | 2025-02-26 | 10.1021/jacs.4c12808 | |
9J1P (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | g1:Ox | - | 2.99 | 2025-02-26 | 10.1021/jacs.4c12808 | ||
8UUJ | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Mus musculus | FCH-2296413 | - | Gi1/β1/γ2 | 2.62 | 2025-02-26 | 10.1016/j.cell.2024.11.001 | |
8UUJ (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Mus musculus | FCH-2296413 | - | 2.62 | 2025-02-26 | 10.1016/j.cell.2024.11.001 | ||
8UTD | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | MK1903 | - | Gi1/β1/γ2 | 3.24 | 2025-02-26 | 10.1016/j.cell.2024.11.001 | |
8UTD (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic Acid | HCA2 | Homo sapiens | MK1903 | - | 3.24 | 2025-02-26 | 10.1016/j.cell.2024.11.001 | ||
8Y0N | A | Protein | Chemokine | CXCR3 | Homo sapiens | VUF11418 | - | Go1/β1/γ2 | 3.07 | 2025-02-26 | To be published | |
8Y0N (No Gprot) | A | Protein | Chemokine | CXCR3 | Homo sapiens | VUF11418 | - | 3.07 | 2025-02-26 | To be published | ||
8XYK | A | Protein | Chemokine | CXCR3 | Homo sapiens | VUF10661 | - | Go1/β1/γ2 | 3.03 | 2025-02-26 | To be published | |
8XYK (No Gprot) | A | Protein | Chemokine | CXCR3 | Homo sapiens | VUF10661 | - | 3.03 | 2025-02-26 | To be published | ||
8XXZ | A | Protein | Chemokine | CXCR3 | Homo sapiens | - | - | Go1/β1/γ2 | 3.3 | 2025-02-26 | To be published | |
8XXZ (No Gprot) | A | Protein | Chemokine | CXCR3 | Homo sapiens | - | - | 3.3 | 2025-02-26 | To be published | ||
8X0H | C | Aminoacid | Metabotropic Glutamate | mGlu5; mGlu5 | Homo sapiens | Quisqualate | - | - | 4.1 | 2024-11-06 | doi.org/10.1038/s41467-024-55439-9 | |
8X0G | C | Aminoacid | Metabotropic Glutamate | mGlu5; mGlu5 | Homo sapiens | Quisqualate | - | - | 3 | 2024-11-06 | doi.org/10.1038/s41467-024-55439-9 | |
8X0F | C | Aminoacid | Metabotropic Glutamate | mGlu5; mGlu5 | Homo sapiens | Quisqualate | VU0424465 | - | 3.3 | 2024-11-06 | doi.org/10.1038/s41467-024-55439-9 | |
8X0E | C | Aminoacid | Metabotropic Glutamate | mGlu5; mGlu5 | Homo sapiens | Quisqualate | - | - | 3.4 | 2024-11-06 | doi.org/10.1038/s41467-024-55439-9 | |
8X0D | C | Aminoacid | Metabotropic Glutamate | mGlu5; mGlu5 | Homo sapiens | Quisqualate | VU0424465 | - | 3.5 | 2024-11-06 | doi.org/10.1038/s41467-024-55439-9 | |
8X0C | C | Aminoacid | Metabotropic Glutamate | mGlu5; mGlu5 | Homo sapiens | Quisqualate | VU0424465 | - | 3.2 | 2024-11-06 | doi.org/10.1038/s41467-024-55439-9 | |
8X0B | C | Aminoacid | Metabotropic Glutamate | mGlu5; mGlu5 | Homo sapiens | Quisqualate | VU0424465 | - | 3.1 | 2024-11-06 | doi.org/10.1038/s41467-024-55439-9 | |
9IQT | A | Alicarboxylic acid | Hydroxycarboxylic acid | HCA2 | Homo sapiens | Niacin | - | Gi1/β1/γ2 | 2.9 | 2024-10-02 | doi.org/10.1016/j.jmb.2024.168795 | |
9IQT (No Gprot) | A | Alicarboxylic acid | Hydroxycarboxylic acid | HCA2 | Homo sapiens | Niacin | - | 2.9 | 2024-10-02 | doi.org/10.1016/j.jmb.2024.168795 | ||
8PWN | A | Nucleotide | Adenosine | A2A | Homo sapiens | Theophylline | - | - | 2.75 | 2023-10-25 | 10.1038/s42004-023-01014-0 | |
8HQC | A | Peptide | Complement Peptide | C5a1 | Mus musculus | C5a anaphylatoxin | - | Go/β1/γ2 | 3.89 | 2023-10-18 | 10.1016/j.cell.2023.09.020 | |
8HQC (No Gprot) | A | Peptide | Complement Peptide | C5a1 | Mus musculus | C5a anaphylatoxin | - | 3.89 | 2023-10-18 | 10.1016/j.cell.2023.09.020 | ||
8TAO | C | Aminoacid | Metabotropic Glutamate | mGlu5; mGlu5 | Homo sapiens | Quisqualate | CDPPB | - | 2.9 | 2023-10-11 | 10.1101/2023.08.29.555158 | |
8T8M | C | Aminoacid | Metabotropic Glutamate | mGlu5; mGlu5 | Homo sapiens | Quisqualate | - | - | 3 | 2023-10-11 | 10.1101/2023.08.29.555158 | |
8T7H | C | Aminoacid | Metabotropic Glutamate | mGlu5; mGlu5 | Homo sapiens | Quisqualate | - | - | 3.3 | 2023-10-11 | 10.1101/2023.08.29.555158 | |
8T6J | C | Aminoacid | Metabotropic Glutamate | mGlu5; mGlu5 | Homo sapiens | - | CDPPB | - | 3.5 | 2023-10-11 | 10.1101/2023.08.29.555158 | |
8KH4 | A | Orphan | Orphan | GPR161 | Homo sapiens | - | - | Gs/β1/γ2 | 3.1 | 2023-10-11 | 10.1038/s41467-023-41654-3 | |
8KH4 (No Gprot) | A | Orphan | Orphan | GPR161 | Homo sapiens | - | - | 3.1 | 2023-10-11 | 10.1038/s41467-023-41654-3 | ||
8KH5 | A | Orphan | Orphan | GPR174 | Homo sapiens | Lysophosphatidylserine | - | Gs/β1/γ2 | 2.83 | 2023-10-11 | 10.1038/s41467-023-41654-3 | |
8KH5 (No Gprot) | A | Orphan | Orphan | GPR174 | Homo sapiens | Lysophosphatidylserine | - | 2.83 | 2023-10-11 | 10.1038/s41467-023-41654-3 | ||
8KGK | A | Orphan | Orphan | GPR61 | Homo sapiens | - | - | Gs/β1/γ2 | 3.16 | 2023-10-11 | 10.1038/s41467-023-41654-3 | |
8KGK (No Gprot) | A | Orphan | Orphan | GPR61 | Homo sapiens | - | - | 3.16 | 2023-10-11 | 10.1038/s41467-023-41654-3 | ||
8SAI | A | Orphan | Orphan | GPR34 | Homo sapiens | 1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine | - | Gi1/β1/γ2 | 3.27 | 2023-10-04 | 10.1073/pnas.2308435120 | |
8SAI (No Gprot) | A | Orphan | Orphan | GPR34 | Homo sapiens | 1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine | - | 3.27 | 2023-10-04 | 10.1073/pnas.2308435120 | ||
8JIU | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | SAR425899 | - | Gs/β1/γ2 | 2.76 | 2023-09-13 | 10.1073/pnas.2303696120 | |
8JIU (No Gprot) | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | SAR425899 | - | 2.76 | 2023-09-13 | 10.1073/pnas.2303696120 | ||
8JIQ | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | Peptide-15 | - | Gs/β1/γ2 | 3.4 | 2023-09-13 | 10.1073/pnas.2303696120 | |
8JIQ (No Gprot) | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | Peptide-15 | - | 3.4 | 2023-09-13 | 10.1073/pnas.2303696120 | ||
8JJO | A | Amine | Adrenergic | β2 | Homo sapiens | Alprenolol | - | - | 3.4 | 2023-09-06 | 10.1038/s41589-023-01389-0 | |
8JJL | A | Amine | Adrenergic | β2 | Homo sapiens | Olodaterol | - | - | 3.2 | 2023-09-06 | 10.1038/s41589-023-01389-0 | |
8JJ8 | A | Amine | Adrenergic | β2 | Homo sapiens | Formoterol | - | - | 3.2 | 2023-09-06 | 10.1038/s41589-023-01389-0 | |
8I2G | A | Protein | Glycoprotein Hormone | FSH | Homo sapiens | Glycoprotein hormones α chain | Compound 716340 | Gs/β1/γ2 | 2.8 | 2023-03-29 | 10.1038/s41467-023-36170-3 | |
8I2G (No Gprot) | A | Protein | Glycoprotein Hormone | FSH | Homo sapiens | Glycoprotein hormones α chain | Compound 716340 | 2.8 | 2023-03-29 | 10.1038/s41467-023-36170-3 | ||
7Y67 | A | Peptide | Complement Peptide | C5a1 | Homo sapiens | C089 peptide | - | Gi1/β1/γ2 | 2.8 | 2023-03-01 | 10.1038/s41422-023-00779-2 | |
7Y67 (No Gprot) | A | Peptide | Complement Peptide | C5a1 | Homo sapiens | C089 peptide | - | 2.8 | 2023-03-01 | 10.1038/s41422-023-00779-2 | ||
7Y66 | A | Peptide | Complement Peptide | C5a1 | Homo sapiens | BM213 | - | Gi1/β1/γ2 | 2.9 | 2023-03-01 | 10.1038/s41422-023-00779-2 | |
7Y66 (No Gprot) | A | Peptide | Complement Peptide | C5a1 | Homo sapiens | BM213 | - | 2.9 | 2023-03-01 | 10.1038/s41422-023-00779-2 | ||
7Y65 | A | Peptide | Complement Peptide | C5a1 | Homo sapiens | C5a peptide | - | Gi1/β1/γ2 | 3.2 | 2023-03-01 | 10.1038/s41422-023-00779-2 | |
7Y65 (No Gprot) | A | Peptide | Complement Peptide | C5a1 | Homo sapiens | C5a peptide | - | 3.2 | 2023-03-01 | 10.1038/s41422-023-00779-2 | ||
7Y64 | A | Peptide | Complement Peptide | C5a1 | Homo sapiens | C5a anaphylatoxin | - | Gi1/β1/γ2 | 2.9 | 2023-03-01 | 10.1038/s41422-023-00779-2 | |
7Y64 (No Gprot) | A | Peptide | Complement Peptide | C5a1 | Homo sapiens | C5a anaphylatoxin | - | 2.9 | 2023-03-01 | 10.1038/s41422-023-00779-2 | ||
7YK7 | A | Peptide | Relaxin | RXFP4 | Homo sapiens | DC591053 | - | Gi2/β1/γ2 | 2.75 | 2023-03-01 | 10.1038/s41467-023-36182-z | |
7YK7 (No Gprot) | A | Peptide | Relaxin | RXFP4 | Homo sapiens | DC591053 | - | 2.75 | 2023-03-01 | 10.1038/s41467-023-36182-z | ||
7YK6 | A | Peptide | Relaxin | RXFP4 | Homo sapiens | PubChem 138319674 | - | Gi2/β1/γ2 | 3.03 | 2023-03-01 | 10.1038/s41467-023-36182-z | |
7YK6 (No Gprot) | A | Peptide | Relaxin | RXFP4 | Homo sapiens | PubChem 138319674 | - | 3.03 | 2023-03-01 | 10.1038/s41467-023-36182-z | ||
7YJ4 | A | Peptide | Relaxin | RXFP4 | Homo sapiens | INSL5 | - | Gi2/β1/γ2 | 3.19 | 2023-03-01 | 10.1038/s41467-023-36182-z | |
7YJ4 (No Gprot) | A | Peptide | Relaxin | RXFP4 | Homo sapiens | INSL5 | - | 3.19 | 2023-03-01 | 10.1038/s41467-023-36182-z | ||
7T94 | A | Amine | Acetylcholine (muscarinic) | M2 | Homo sapiens | Acetylcholine | PubChem 57664406 | chim(NtGi1-Go)/β1/γ2 | 3.16 | 2023-01-25 | 10.1038/s41467-022-35726-z | |
7T94 (No Gprot) | A | Amine | Acetylcholine (muscarinic) | M2 | Homo sapiens | Acetylcholine | PubChem 57664406 | 3.16 | 2023-01-25 | 10.1038/s41467-022-35726-z | ||
7T90 | A | Amine | Acetylcholine (muscarinic) | M2 | Homo sapiens | Acetylcholine | - | chim(NtGi1-Go)/β1/γ2 | 3.32 | 2023-01-25 | 10.1038/s41467-022-35726-z | |
7T90 (No Gprot) | A | Amine | Acetylcholine (muscarinic) | M2 | Homo sapiens | Acetylcholine | - | 3.32 | 2023-01-25 | 10.1038/s41467-022-35726-z | ||
7T8X | A | Amine | Acetylcholine (muscarinic) | M2 | Homo sapiens | Acetylcholine | - | chim(NtGi1-Go)/β1/γ2 | 3.21 | 2023-01-25 | 10.1038/s41467-022-35726-z | |
7T8X (No Gprot) | A | Amine | Acetylcholine (muscarinic) | M2 | Homo sapiens | Acetylcholine | - | 3.21 | 2023-01-25 | 10.1038/s41467-022-35726-z | ||
8HDP | A | Nucleotide | Adenosine | A2B | Homo sapiens | Adenosine | - | Gs/β1/γ2 | 3.2 | 2023-01-18 | 10.1038/s41421-022-00503-1 | |
8HDP (No Gprot) | A | Nucleotide | Adenosine | A2B | Homo sapiens | Adenosine | - | 3.2 | 2023-01-18 | 10.1038/s41421-022-00503-1 | ||
8HDO | A | Nucleotide | Adenosine | A2B | Homo sapiens | BAY 60-6583 | - | Gs/β1/γ2 | 2.87 | 2023-01-18 | 10.1038/s41421-022-00503-1 | |
8HDO (No Gprot) | A | Nucleotide | Adenosine | A2B | Homo sapiens | BAY 60-6583 | - | 2.87 | 2023-01-18 | 10.1038/s41421-022-00503-1 | ||
8GY7 | A | Peptide | Melanocortin | MC2 | Homo sapiens | Corticotropin | Ca | chim(NtGi1-Gs)/β1/γ2; MRAP1 | 3.3 | 2023-01-11 | 10.1038/s41422-022-00751-6 | |
8GY7 (No Gprot) | A | Peptide | Melanocortin | MC2 | Homo sapiens | Corticotropin | Ca | 3.3 | 2023-01-11 | 10.1038/s41422-022-00751-6 | ||
8E9Z | A | Amine | Acetylcholine (muscarinic) | M3 | Homo sapiens | Iperoxo | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 2.69 | 2022-11-30 | 10.1038/s41586-022-05489-0 | |
8E9Z (No Gprot) | A | Amine | Acetylcholine (muscarinic) | M3 | Homo sapiens | Iperoxo | - | 2.69 | 2022-11-30 | 10.1038/s41586-022-05489-0 | ||
8E9Y | A | Amine | Acetylcholine (muscarinic) | M3 | Homo sapiens | Clozapine-N-oxide | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 2.79 | 2022-11-30 | 10.1038/s41586-022-05489-0 | |
8E9Y (No Gprot) | A | Amine | Acetylcholine (muscarinic) | M3 | Homo sapiens | Clozapine-N-oxide | - | 2.79 | 2022-11-30 | 10.1038/s41586-022-05489-0 | ||
8E9W | A | Amine | Acetylcholine (muscarinic) | M3 | Homo sapiens | 2-Deoxycytidine | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 2.69 | 2022-11-30 | 10.1038/s41586-022-05489-0 | |
8E9W (No Gprot) | A | Amine | Acetylcholine (muscarinic) | M3 | Homo sapiens | 2-Deoxycytidine | - | 2.69 | 2022-11-30 | 10.1038/s41586-022-05489-0 | ||
8E3X | B1 | Peptide | VIP and PACAP | PAC1 | Homo sapiens | PACAP27 | - | Gs/β1/γ2 | 2.3 | 2022-11-23 | 10.1038/s41467-022-34629-3 | |
8E3X (No Gprot) | B1 | Peptide | VIP and PACAP | PAC1 | Homo sapiens | PACAP27 | - | 2.3 | 2022-11-23 | 10.1038/s41467-022-34629-3 | ||
8E3Z | B1 | Peptide | VIP and PACAP | VPAC1 | Homo sapiens | VIP | - | Gs/β1/γ2 | 2.7 | 2022-11-23 | 10.1038/s41467-022-34629-3 | |
8E3Z (No Gprot) | B1 | Peptide | VIP and PACAP | VPAC1 | Homo sapiens | VIP | - | 2.7 | 2022-11-23 | 10.1038/s41467-022-34629-3 | ||
8E3Y | B1 | Peptide | VIP and PACAP | VPAC1 | Homo sapiens | PACAP27 | - | Gs/β1/γ2 | 2.3 | 2022-11-23 | 10.1038/s41467-022-34629-3 | |
8E3Y (No Gprot) | B1 | Peptide | VIP and PACAP | VPAC1 | Homo sapiens | PACAP27 | - | 2.3 | 2022-11-23 | 10.1038/s41467-022-34629-3 | ||
8EFQ | A | Peptide | Opioid | μ | Homo sapiens | Damgo | - | Gi1/β1/γ2 | 3.3 | 2022-11-09 | 10.1016/j.cell.2022.09.041 | |
8EFQ (No Gprot) | A | Peptide | Opioid | μ | Homo sapiens | Damgo | - | 3.3 | 2022-11-09 | 10.1016/j.cell.2022.09.041 | ||
8EFO | A | Peptide | Opioid | μ | Homo sapiens | PZM21 | - | Gi1/β1/γ2 | 2.8 | 2022-11-09 | 10.1016/j.cell.2022.09.041 | |
8EFO (No Gprot) | A | Peptide | Opioid | μ | Homo sapiens | PZM21 | - | 2.8 | 2022-11-09 | 10.1016/j.cell.2022.09.041 | ||
8EFL | A | Peptide | Opioid | μ | Homo sapiens | SR17018 | - | Gi1/β1/γ2 | 3.2 | 2022-11-09 | 10.1016/j.cell.2022.09.041 | |
8EFL (No Gprot) | A | Peptide | Opioid | μ | Homo sapiens | SR17018 | - | 3.2 | 2022-11-09 | 10.1016/j.cell.2022.09.041 | ||
8EFB | A | Peptide | Opioid | μ | Homo sapiens | Oliceridine | - | Gi1/β1/γ2 | 3.2 | 2022-11-09 | 10.1016/j.cell.2022.09.041 | |
8EFB (No Gprot) | A | Peptide | Opioid | μ | Homo sapiens | Oliceridine | - | 3.2 | 2022-11-09 | 10.1016/j.cell.2022.09.041 | ||
8EF6 | A | Peptide | Opioid | μ | Homo sapiens | Morphine | - | Gi1/β1/γ2 | 3.2 | 2022-11-09 | 10.1016/j.cell.2022.09.041 | |
8EF6 (No Gprot) | A | Peptide | Opioid | μ | Homo sapiens | Morphine | - | 3.2 | 2022-11-09 | 10.1016/j.cell.2022.09.041 | ||
8EF5 | A | Peptide | Opioid | μ | Homo sapiens | Fentanyl | - | Gi1/β1/γ2 | 3.3 | 2022-11-09 | 10.1016/j.cell.2022.09.041 | |
8EF5 (No Gprot) | A | Peptide | Opioid | μ | Homo sapiens | Fentanyl | - | 3.3 | 2022-11-09 | 10.1016/j.cell.2022.09.041 | ||
7PP1 | A | Nucleotide | P2Y | P2Y12 | Homo sapiens | Selatogrel | - | - | 2.78 | 2022-11-02 | 10.1016/j.bcp.2022.115291 | |
7F61 | A | Amine | Histamine | H3 | Homo sapiens | PF-03654746 | Cholesterol | - | 2.6 | 2022-10-26 | 10.1038/s41467-022-33880-y | |
7WZ4 | A | Orphan | Orphan | GPR88 | Homo sapiens | - | - | Gi1/β1/γ2 | 3 | 2022-10-26 | 10.1038/s41467-022-30081-5 | |
7WZ4 (No Gprot) | A | Orphan | Orphan | GPR88 | Homo sapiens | - | - | 3 | 2022-10-26 | 10.1038/s41467-022-30081-5 | ||
7XP6 | T2 | Sensory | Taste2 | T2R46 | Homo sapiens | Strychnine | - | chim(Gs-CtGt3)/β1/γ2 | 3.01 | 2022-10-12 | 10.1126/science.abo1633 | |
7XP6 (No Gprot) | T2 | Sensory | Taste2 | T2R46 | Homo sapiens | Strychnine | - | 3.01 | 2022-10-12 | 10.1126/science.abo1633 | ||
7XP5 | T2 | Sensory | Taste2 | T2R46 | Homo sapiens | - | - | chim(Gs-CtGt3)/β1/γ2 | 3.08 | 2022-10-12 | 10.1126/science.abo1633 | |
7XP5 (No Gprot) | T2 | Sensory | Taste2 | T2R46 | Homo sapiens | - | - | 3.08 | 2022-10-12 | 10.1126/science.abo1633 | ||
7XP4 | T2 | Sensory | Taste2 | T2R46 | Homo sapiens | - | - | chim(Gs-CtGt3)/β1/γ2 | 3.01 | 2022-10-12 | 10.1126/science.abo1633 | |
7XP4 (No Gprot) | T2 | Sensory | Taste2 | T2R46 | Homo sapiens | - | - | 3.01 | 2022-10-12 | 10.1126/science.abo1633 | ||
7Y89 | A | Orphan | Orphan | GPR17 (CysLT) | Homo sapiens | - | - | Gi1/β1/γ2 | 3.02 | 2022-10-12 | 10.1002/mco2.159 | |
7Y89 (No Gprot) | A | Orphan | Orphan | GPR17 (CysLT) | Homo sapiens | - | - | 3.02 | 2022-10-12 | 10.1002/mco2.159 | ||
7YU4 | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | ONO-0740556 | - | - | 3.7 | 2022-10-05 | 10.1038/s41467-022-33121-2 | |
7YU8 | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | ONO-0740556 | - | Gi1/β1/γ2 | 5.6 | 2022-10-05 | 10.1038/s41467-022-33121-2 | |
7YU8 (No Gprot) | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | ONO-0740556 | - | 5.6 | 2022-10-05 | 10.1038/s41467-022-33121-2 | ||
7YU7 | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | ONO-0740556 | - | Gi1/β1/γ2 | 4.5 | 2022-10-05 | 10.1038/s41467-022-33121-2 | |
7YU7 (No Gprot) | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | ONO-0740556 | - | 4.5 | 2022-10-05 | 10.1038/s41467-022-33121-2 | ||
7YU6 | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | ONO-0740556 | - | Gi1/β1/γ2 | 3.9 | 2022-10-05 | 10.1038/s41467-022-33121-2 | |
7YU6 (No Gprot) | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | ONO-0740556 | - | 3.9 | 2022-10-05 | 10.1038/s41467-022-33121-2 | ||
7YU5 | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | ONO-0740556 | - | Gi1/β1/γ2 | 3.7 | 2022-10-05 | 10.1038/s41467-022-33121-2 | |
7YU5 (No Gprot) | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | ONO-0740556 | - | 3.7 | 2022-10-05 | 10.1038/s41467-022-33121-2 | ||
7YU3 | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | ONO-0740556 | - | Gi1/β1/γ2 | 3.5 | 2022-10-05 | 10.1038/s41467-022-33121-2 | |
7YU3 (No Gprot) | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | ONO-0740556 | - | 3.5 | 2022-10-05 | 10.1038/s41467-022-33121-2 | ||
7WZ7 | B2 | Adhesion | Adhesion | ADGRF1 | Homo sapiens | - | - | chim(NtGi1-G12)/β1/γ2 | 2.83 | 2022-09-28 | 10.1038/s41467-022-33173-4 | |
7WZ7 (No Gprot) | B2 | Adhesion | Adhesion | ADGRF1 | Homo sapiens | - | - | 2.83 | 2022-09-28 | 10.1038/s41467-022-33173-4 | ||
7WXU | B2 | Adhesion | Adhesion | ADGRF1 | Homo sapiens | - | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.85 | 2022-09-28 | 10.1038/s41467-022-33173-4 | |
7WXU (No Gprot) | B2 | Adhesion | Adhesion | ADGRF1 | Homo sapiens | - | - | 2.85 | 2022-09-28 | 10.1038/s41467-022-33173-4 | ||
7WXW | B2 | Adhesion | Adhesion | ADGRF1 | Homo sapiens | - | - | chim(NtGi1-Gs)/β1/γ2 | 2.84 | 2022-09-28 | 10.1038/s41467-022-33173-4 | |
7WXW (No Gprot) | B2 | Adhesion | Adhesion | ADGRF1 | Homo sapiens | - | - | 2.84 | 2022-09-28 | 10.1038/s41467-022-33173-4 | ||
7WY0 | B2 | Adhesion | Adhesion | ADGRF1 | Homo sapiens | - | - | chim(NtGi1L-G13)/β1/γ2 | 2.83 | 2022-09-28 | 10.1038/s41467-022-33173-4 | |
7WY0 (No Gprot) | B2 | Adhesion | Adhesion | ADGRF1 | Homo sapiens | - | - | 2.83 | 2022-09-28 | 10.1038/s41467-022-33173-4 | ||
7X2V | B2 | Adhesion | Adhesion | ADGRF1 | Homo sapiens | - | - | Gi1/β1/γ2 | 3.09 | 2022-09-28 | 10.1038/s41467-022-33173-4 | |
7X2V (No Gprot) | B2 | Adhesion | Adhesion | ADGRF1 | Homo sapiens | - | - | 3.09 | 2022-09-28 | 10.1038/s41467-022-33173-4 | ||
7VIH | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | CBP-307 | - | Gi1/β1/γ2 | 2.98 | 2022-09-28 | 10.1073/pnas.2117716119 | |
7VIH (No Gprot) | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | CBP-307 | - | 2.98 | 2022-09-28 | 10.1073/pnas.2117716119 | ||
7VIG | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | CBP-307 | - | Gi1/β1/γ2 | 2.89 | 2022-09-28 | 10.1073/pnas.2117716119 | |
7VIG (No Gprot) | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | CBP-307 | - | 2.89 | 2022-09-28 | 10.1073/pnas.2117716119 | ||
7VIF | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | S-FTY720-P | - | Gi1/β1/γ2 | 2.83 | 2022-09-28 | 10.1073/pnas.2117716119 | |
7VIF (No Gprot) | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | S-FTY720-P | - | 2.83 | 2022-09-28 | 10.1073/pnas.2117716119 | ||
7VIE | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | S1P | - | Gi1/β1/γ2 | 2.86 | 2022-09-28 | 10.1073/pnas.2117716119 | |
7VIE (No Gprot) | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | S1P | - | 2.86 | 2022-09-28 | 10.1073/pnas.2117716119 | ||
7W7E | A | Amine | Adrenergic | α2a | Homo sapiens | PubChem 164946676 | - | Go/β1/γ2 | 3.4 | 2022-09-28 | 10.1126/science.abn7065 | |
7W7E (No Gprot) | A | Amine | Adrenergic | α2a | Homo sapiens | PubChem 164946676 | - | 3.4 | 2022-09-28 | 10.1126/science.abn7065 | ||
7W6P | A | Amine | Adrenergic | α2a | Homo sapiens | N-pyridin-4-ylisoquinolin-4-amine | - | Go/β1/γ2 | 3.47 | 2022-09-28 | 10.1126/science.abn7065 | |
7W6P (No Gprot) | A | Amine | Adrenergic | α2a | Homo sapiens | N-pyridin-4-ylisoquinolin-4-amine | - | 3.47 | 2022-09-28 | 10.1126/science.abn7065 | ||
7SRQ | A | Amine | 5-Hydroxytryptamine | 5-HT2B | Homo sapiens | LSD | - | - | 2.7 | 2022-09-21 | 10.1016/j.neuron.2022.08.006 | |
7SRS | A | Amine | 5-Hydroxytryptamine | 5-HT2B | Homo sapiens | LSD | - | Arrestin2 | 3.3 | 2022-09-21 | 10.1016/j.neuron.2022.08.006 | |
7SRR | A | Amine | 5-Hydroxytryptamine | 5-HT2B | Homo sapiens | LSD | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 2.9 | 2022-09-21 | 10.1016/j.neuron.2022.08.006 | |
7SRR (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT2B | Homo sapiens | LSD | - | 2.9 | 2022-09-21 | 10.1016/j.neuron.2022.08.006 | ||
7VFX | A | Peptide | Formylpeptide | FPR1-ALX | Homo sapiens | fMLF | - | Gi1/β1/γ2 | 2.8 | 2022-09-21 | 10.1038/s41467-022-32822-y | |
7VFX (No Gprot) | A | Peptide | Formylpeptide | FPR1-ALX | Homo sapiens | fMLF | - | 2.8 | 2022-09-21 | 10.1038/s41467-022-32822-y | ||
7R0C | A | Peptide | Vasopressin and Oxytocin | V2 | Homo sapiens | AVP | - | Arrestin2 | 4.73 | 2022-09-14 | 10.1126/sciadv.abo7761 | |
7X5H | A | Amine | 5-Hydroxytryptamine | 5-HT5A | Homo sapiens | 5-CT | - | Gi1/β1/γ2 | 3.1 | 2022-09-14 | 10.1038/s41421-022-00412-3 | |
7X5H (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT5A | Homo sapiens | 5-CT | - | 3.1 | 2022-09-14 | 10.1038/s41421-022-00412-3 | ||
8CU7 | A | Nucleotide | Adenosine | A2A | Homo sapiens | LJ-4517 | Na | - | 2.05 | 2022-08-31 | 10.1021/acs.jmedchem.2c00462 | |
8CU6 | A | Nucleotide | Adenosine | A2A | Homo sapiens | LJ-4517 | - | - | 2.8 | 2022-08-31 | 10.1021/acs.jmedchem.2c00462 | |
7X1U | A | Peptide | Thyrotropin Releasing Hormone | TRH | Homo sapiens | TRH | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 3.19 | 2022-08-31 | 10.1038/s41422-022-00646-6 | |
7X1U (No Gprot) | A | Peptide | Thyrotropin Releasing Hormone | TRH | Homo sapiens | TRH | - | 3.19 | 2022-08-31 | 10.1038/s41422-022-00646-6 | ||
7X1T | A | Peptide | Thyrotropin Releasing Hormone | TRH | Homo sapiens | Taltirelin | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 3.26 | 2022-08-31 | 10.1038/s41422-022-00646-6 | |
7X1T (No Gprot) | A | Peptide | Thyrotropin Releasing Hormone | TRH | Homo sapiens | Taltirelin | - | 3.26 | 2022-08-31 | 10.1038/s41422-022-00646-6 | ||
7XAV | A | Peptide | Somatostatin | SST2 | Homo sapiens | Lanreotide | - | Gi1/β1/γ2 | 2.87 | 2022-08-31 | 10.1038/s41421-022-00405-2 | |
7XAV (No Gprot) | A | Peptide | Somatostatin | SST2 | Homo sapiens | Lanreotide | - | 2.87 | 2022-08-31 | 10.1038/s41421-022-00405-2 | ||
7XAU | A | Peptide | Somatostatin | SST2 | Homo sapiens | Octreotide | - | Gi1/β1/γ2 | 2.97 | 2022-08-31 | 10.1038/s41421-022-00405-2 | |
7XAU (No Gprot) | A | Peptide | Somatostatin | SST2 | Homo sapiens | Octreotide | - | 2.97 | 2022-08-31 | 10.1038/s41421-022-00405-2 | ||
7XAT | A | Peptide | Somatostatin | SST2 | Homo sapiens | Somatostatin-14 | - | Gi1/β1/γ2 | 2.85 | 2022-08-31 | 10.1038/s41421-022-00405-2 | |
7XAT (No Gprot) | A | Peptide | Somatostatin | SST2 | Homo sapiens | Somatostatin-14 | - | 2.85 | 2022-08-31 | 10.1038/s41421-022-00405-2 | ||
8DPI | A | Amine | 5-Hydroxytryptamine | 5-HT2C | Homo sapiens | Lorcaserin | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 3.4 | 2022-08-24 | 10.1016/j.celrep.2022.111211 | |
8DPI (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT2C | Homo sapiens | Lorcaserin | - | 3.4 | 2022-08-24 | 10.1016/j.celrep.2022.111211 | ||
8DPH | A | Amine | 5-Hydroxytryptamine | 5-HT2C | Homo sapiens | Lorcaserin | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 3.2 | 2022-08-24 | 10.1016/j.celrep.2022.111211 | |
8DPH (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT2C | Homo sapiens | Lorcaserin | - | 3.2 | 2022-08-24 | 10.1016/j.celrep.2022.111211 | ||
8DPG | A | Amine | 5-Hydroxytryptamine | 5-HT2C | Homo sapiens | Psilocin | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 3.6 | 2022-08-24 | 10.1016/j.celrep.2022.111211 | |
8DPG (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT2C | Homo sapiens | Psilocin | - | 3.6 | 2022-08-24 | 10.1016/j.celrep.2022.111211 | ||
8DPF | A | Amine | 5-Hydroxytryptamine | 5-HT2C | Homo sapiens | Lorcaserin | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 2.84 | 2022-08-24 | 10.1016/j.celrep.2022.111211 | |
8DPF (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT2C | Homo sapiens | Lorcaserin | - | 2.84 | 2022-08-24 | 10.1016/j.celrep.2022.111211 | ||
7XA3 | A | Protein | Chemokine | CCR2 | Homo sapiens | CCL2 | - | Gi1/β1/γ2 | 2.9 | 2022-08-24 | 10.1038/s41421-022-00403-4 | |
7XA3 (No Gprot) | A | Protein | Chemokine | CCR2 | Homo sapiens | CCL2 | - | 2.9 | 2022-08-24 | 10.1038/s41421-022-00403-4 | ||
7X9Y | A | Protein | Chemokine | CCR3 | Homo sapiens | - | - | Gi1/β1/γ2 | 3.1 | 2022-08-24 | 10.1038/s41421-022-00403-4 | |
7X9Y (No Gprot) | A | Protein | Chemokine | CCR3 | Homo sapiens | - | - | 3.1 | 2022-08-24 | 10.1038/s41421-022-00403-4 | ||
7YP7 | B2 | Adhesion | Adhesion | ADGRG2 | Mus musculus | - | - | Gs/β1/γ2 | 3.1 | 2022-08-24 | 10.1038/s41589-022-01084-6 | |
7YP7 (No Gprot) | B2 | Adhesion | Adhesion | ADGRG2 | Mus musculus | - | - | 3.1 | 2022-08-24 | 10.1038/s41589-022-01084-6 | ||
7XZ6 | A | Lipid | GPR119 | GPR119 | Homo sapiens | APD668 | - | Gs/β1/γ2 | 2.8 | 2022-08-24 | 10.1038/s41594-022-00816-5 | |
7XZ6 (No Gprot) | A | Lipid | GPR119 | GPR119 | Homo sapiens | APD668 | - | 2.8 | 2022-08-24 | 10.1038/s41594-022-00816-5 | ||
7XZ5 | A | Lipid | GPR119 | GPR119 | Homo sapiens | Lysophosphatidylcholine | - | Gs/β1/γ2 | 3.1 | 2022-08-24 | 10.1038/s41594-022-00816-5 | |
7XZ5 (No Gprot) | A | Lipid | GPR119 | GPR119 | Homo sapiens | Lysophosphatidylcholine | - | 3.1 | 2022-08-24 | 10.1038/s41594-022-00816-5 | ||
7XW5 | A | Protein | Glycoprotein Hormone | TSH | Homo sapiens | TSH | ML109 | Gs/β1/γ2 | 2.96 | 2022-08-24 | 10.1038/s41586-022-05173-3 | |
7XW5 (No Gprot) | A | Protein | Glycoprotein Hormone | TSH | Homo sapiens | TSH | ML109 | 2.96 | 2022-08-24 | 10.1038/s41586-022-05173-3 | ||
7XW7 | A | Protein | Glycoprotein Hormone | TSH | Homo sapiens | K1-70 | - | - | 5.5 | 2022-08-17 | 10.1038/s41586-022-05173-3 | |
7WU9 | A | Lipid | Prostanoid | EP3 | Homo sapiens | - | - | Gi1/β1/γ2 | 3.38 | 2022-08-17 | 10.1016/j.celrep.2022.111323 | |
7WU9 (No Gprot) | A | Lipid | Prostanoid | EP3 | Homo sapiens | - | - | 3.38 | 2022-08-17 | 10.1016/j.celrep.2022.111323 | ||
7XW6 | A | Protein | Glycoprotein Hormone | TSH | Homo sapiens | M22 Fab | ML109 | Gs/β1/γ2 | 2.78 | 2022-08-17 | 10.1038/s41586-022-05173-3 | |
7XW6 (No Gprot) | A | Protein | Glycoprotein Hormone | TSH | Homo sapiens | M22 Fab | ML109 | 2.78 | 2022-08-17 | 10.1038/s41586-022-05173-3 | ||
8DU3 | A | Nucleotide | Adenosine | A2A | Homo sapiens | PubChem 105526064 | - | - | 2.5 | 2022-08-10 | 10.1016/j.ejmech.2022.114620 | |
7T32 | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | - | - | 3.4 | 2022-08-10 | 10.1038/s41467-022-32125-2 | |
7YXA | A | Lipid | Lysophospholipid | S1P5 | Homo sapiens | ONO-5430608 | - | - | 2.2 | 2022-08-10 | 10.1038/s41467-022-32447-1 | |
7T9M | A | Protein | Glycoprotein Hormone | TSH | Homo sapiens | - | CS-17 Antibody | - | 3.1 | 2022-08-10 | 10.1038/s41586-022-05159-1 | |
7QVM | A | Peptide | Vasopressin and Oxytocin | OT | Homo sapiens | Oxytocin | - | chim(NtGi1-Go-CtGq)/β1/γ2 | 3.25 | 2022-08-10 | 10.1038/s41467-022-31325-0 | |
7QVM (No Gprot) | A | Peptide | Vasopressin and Oxytocin | OT | Homo sapiens | Oxytocin | - | 3.25 | 2022-08-10 | 10.1038/s41467-022-31325-0 | ||
7XKE | B2 | Adhesion | Adhesion | ADGRG2 | Mus musculus | β-Hydroxyandrosterone | - | chim(NtGi1-Gs)/β1/γ2 | 2.9 | 2022-08-10 | 10.1038/s41589-022-01084-6 | |
7XKE (No Gprot) | B2 | Adhesion | Adhesion | ADGRG2 | Mus musculus | β-Hydroxyandrosterone | - | 2.9 | 2022-08-10 | 10.1038/s41589-022-01084-6 | ||
7XKF | B2 | Adhesion | Adhesion | ADGRG2 | Mus musculus | β-Hydroxyandrosterone | - | Gs/β1/γ2 | 2.4 | 2022-08-10 | 10.1038/s41589-022-01084-6 | |
7XKF (No Gprot) | B2 | Adhesion | Adhesion | ADGRG2 | Mus musculus | β-Hydroxyandrosterone | - | 2.4 | 2022-08-10 | 10.1038/s41589-022-01084-6 | ||
7XKD | B2 | Adhesion | Adhesion | ADGRG2 | Mus musculus | β-Hydroxyandrosterone | - | Gs/β1/γ2 | 2.4 | 2022-08-10 | 10.1038/s41589-022-01084-6 | |
7XKD (No Gprot) | B2 | Adhesion | Adhesion | ADGRG2 | Mus musculus | β-Hydroxyandrosterone | - | 2.4 | 2022-08-10 | 10.1038/s41589-022-01084-6 | ||
8CXO | F | Protein | Frizzled | SMO | Mus musculus | - | - | - | 3.7 | 2022-08-03 | 10.1038/s41467-022-32125-2 | |
7XNA | A | Peptide | Somatostatin | SST2 | Homo sapiens | CYN154806 | - | - | 2.65 | 2022-08-03 | 10.1038/s41422-022-00679-x | |
7XN9 | A | Peptide | Somatostatin | SST2 | Homo sapiens | L-054,522 | - | - | 2.6 | 2022-08-03 | 10.1038/s41422-022-00679-x | |
7XMR | A | Peptide | Somatostatin | SST2 | Homo sapiens | Somatostatin-14 | - | Gi1/β1/γ2 | 3.1 | 2022-08-03 | 10.1038/s41422-022-00679-x | |
7XMR (No Gprot) | A | Peptide | Somatostatin | SST2 | Homo sapiens | Somatostatin-14 | - | 3.1 | 2022-08-03 | 10.1038/s41422-022-00679-x | ||
7XMT | A | Peptide | Somatostatin | SST4 | Homo sapiens | J-2156 | - | Gi1/β1/γ2 | 2.8 | 2022-08-03 | 10.1038/s41422-022-00679-x | |
7XMT (No Gprot) | A | Peptide | Somatostatin | SST4 | Homo sapiens | J-2156 | - | 2.8 | 2022-08-03 | 10.1038/s41422-022-00679-x | ||
7XMS | A | Peptide | Somatostatin | SST4 | Homo sapiens | Somatostatin-14 | - | Gi1/β1/γ2 | 2.9 | 2022-08-03 | 10.1038/s41422-022-00679-x | |
7XMS (No Gprot) | A | Peptide | Somatostatin | SST4 | Homo sapiens | Somatostatin-14 | - | 2.9 | 2022-08-03 | 10.1038/s41422-022-00679-x | ||
7VVO | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | PTH | - | Gs/β1/γ2 | 4.1 | 2022-08-03 | 10.1016/j.molcel.2022.07.003 | |
7VVO (No Gprot) | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | PTH | - | 4.1 | 2022-08-03 | 10.1016/j.molcel.2022.07.003 | ||
7VVN | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | PTH | - | Gs/β1/γ2 | 3.8 | 2022-08-03 | 10.1016/j.molcel.2022.07.003 | |
7VVN (No Gprot) | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | PTH | - | 3.8 | 2022-08-03 | 10.1016/j.molcel.2022.07.003 | ||
7VVM | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | PTH | - | Gs/β1/γ2 | 3.2 | 2022-08-03 | 10.1016/j.molcel.2022.07.003 | |
7VVM (No Gprot) | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | PTH | - | 3.2 | 2022-08-03 | 10.1016/j.molcel.2022.07.003 | ||
7VVL | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | PTH | - | Gs/β1/γ2 | 2.8 | 2022-08-03 | 10.1016/j.molcel.2022.07.003 | |
7VVL (No Gprot) | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | PTH | - | 2.8 | 2022-08-03 | 10.1016/j.molcel.2022.07.003 | ||
7VVK | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | PTH | - | Gs/β1/γ2 | 3.3 | 2022-08-03 | 10.1016/j.molcel.2022.07.003 | |
7VVK (No Gprot) | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | PTH | - | 3.3 | 2022-08-03 | 10.1016/j.molcel.2022.07.003 | ||
7VVJ | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | PTHrP(1-36) | - | Gs/β1/γ2 | 3.2 | 2022-08-03 | 10.1016/j.molcel.2022.07.003 | |
7VVJ (No Gprot) | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | PTHrP(1-36) | - | 3.2 | 2022-08-03 | 10.1016/j.molcel.2022.07.003 | ||
7UTZ | A | Protein | Glycoprotein Hormone | TSH | Homo sapiens | TR1402 | PubChem 644078 | Gs/β1/γ2 | 2.4 | 2022-08-03 | 10.1038/s41586-022-05159-1 | |
7UTZ (No Gprot) | A | Protein | Glycoprotein Hormone | TSH | Homo sapiens | TR1402 | PubChem 644078 | 2.4 | 2022-08-03 | 10.1038/s41586-022-05159-1 | ||
7T9N | A | Protein | Glycoprotein Hormone | TSH | Homo sapiens | M22 Fab | PubChem 644078 | Gs/β1/γ2 | 2.9 | 2022-08-03 | 10.1038/s41586-022-05159-1 | |
7T9N (No Gprot) | A | Protein | Glycoprotein Hormone | TSH | Homo sapiens | M22 Fab | PubChem 644078 | 2.9 | 2022-08-03 | 10.1038/s41586-022-05159-1 | ||
7T9I | A | Protein | Glycoprotein Hormone | TSH | Homo sapiens | TSH | - | Gs/β1/γ2 | 2.9 | 2022-08-03 | 10.1038/s41586-022-05159-1 | |
7T9I (No Gprot) | A | Protein | Glycoprotein Hormone | TSH | Homo sapiens | TSH | - | 2.9 | 2022-08-03 | 10.1038/s41586-022-05159-1 | ||
7SK9 | A | Protein | Chemokine | ACKR3 | Homo sapiens | - | CCX662 | - | 3.7 | 2022-07-27 | 10.1126/sciadv.abn8063 | |
7SK8 | A | Protein | Chemokine | ACKR3 | Homo sapiens | CXCL12 | CCX662 | - | 3.3 | 2022-07-27 | 10.1126/sciadv.abn8063 | |
7SK7 | A | Protein | Chemokine | ACKR3 | Homo sapiens | CXCL12 | CCX662 | - | 3.3 | 2022-07-27 | 10.1126/sciadv.abn8063 | |
7SK6 | A | Protein | Chemokine | ACKR3 | Homo sapiens | CXCL12_LRHQ | - | - | 4 | 2022-07-27 | 10.1126/sciadv.abn8063 | |
7SK5 | A | Protein | Chemokine | ACKR3 | Homo sapiens | CXCL12 | - | - | 4 | 2022-07-27 | 10.1126/sciadv.abn8063 | |
7SK4 | A | Protein | Chemokine | ACKR3 | Homo sapiens | CXCL12_LRHQ | - | - | 3.3 | 2022-07-27 | 10.1126/sciadv.abn8063 | |
7SK3 | A | Protein | Chemokine | ACKR3 | Homo sapiens | CXCL12 | - | - | 3.8 | 2022-07-27 | 10.1126/sciadv.abn8063 | |
7SUS | A | Peptide | Apelin | Apelin | Homo sapiens | PubChem 122701908 | - | - | 2.7 | 2022-07-27 | 10.1038/s41594-022-00797-5 | |
7XTA | A | Amine | 5-Hydroxytryptamine | 5-HT4 | Homo sapiens | Serotonin | - | Gi1/β1/γ2 | 3.2 | 2022-07-27 | 10.1016/j.molcel.2022.05.031 | |
7XTA (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT4 | Homo sapiens | Serotonin | - | 3.2 | 2022-07-27 | 10.1016/j.molcel.2022.05.031 | ||
7W0P | A | Peptide | Apelin | Apelin | Homo sapiens | Elabela | - | Gi1/β1/γ2 | 3.16 | 2022-07-27 | 10.1038/s41594-022-00797-5 | |
7W0P (No Gprot) | A | Peptide | Apelin | Apelin | Homo sapiens | Elabela | - | 3.16 | 2022-07-27 | 10.1038/s41594-022-00797-5 | ||
7W0O | A | Peptide | Apelin | Apelin | Homo sapiens | Elabela | - | Gi1/β1/γ2 | 3.78 | 2022-07-27 | 10.1038/s41594-022-00797-5 | |
7W0O (No Gprot) | A | Peptide | Apelin | Apelin | Homo sapiens | Elabela | - | 3.78 | 2022-07-27 | 10.1038/s41594-022-00797-5 | ||
7W0N | A | Peptide | Apelin | Apelin | Homo sapiens | Elabela | - | Gi1/β1/γ2 | 4.21 | 2022-07-27 | 10.1038/s41594-022-00797-5 | |
7W0N (No Gprot) | A | Peptide | Apelin | Apelin | Homo sapiens | Elabela | - | 4.21 | 2022-07-27 | 10.1038/s41594-022-00797-5 | ||
7W0M | A | Peptide | Apelin | Apelin | Homo sapiens | PubChem 122701908 | - | Gi1/β1/γ2 | 3.71 | 2022-07-27 | 10.1038/s41594-022-00797-5 | |
7W0M (No Gprot) | A | Peptide | Apelin | Apelin | Homo sapiens | PubChem 122701908 | - | 3.71 | 2022-07-27 | 10.1038/s41594-022-00797-5 | ||
7W0L | A | Peptide | Apelin | Apelin | Homo sapiens | PubChem 122701908 | - | Gi1/β1/γ2 | 3.57 | 2022-07-27 | 10.1038/s41594-022-00797-5 | |
7W0L (No Gprot) | A | Peptide | Apelin | Apelin | Homo sapiens | PubChem 122701908 | - | 3.57 | 2022-07-27 | 10.1038/s41594-022-00797-5 | ||
7XT9 | A | Amine | 5-Hydroxytryptamine | 5-HT4 | Homo sapiens | Serotonin | - | Gs/β1/γ2 | 3.2 | 2022-07-27 | 10.1016/j.molcel.2022.05.031 | |
7XT9 (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT4 | Homo sapiens | Serotonin | - | 3.2 | 2022-07-27 | 10.1016/j.molcel.2022.05.031 | ||
7XT8 | A | Amine | 5-Hydroxytryptamine | 5-HT4 | Homo sapiens | Serotonin | - | Gs/β1/γ2 | 3.1 | 2022-07-27 | 10.1016/j.molcel.2022.05.031 | |
7XT8 (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT4 | Homo sapiens | Serotonin | - | 3.1 | 2022-07-27 | 10.1016/j.molcel.2022.05.031 | ||
7XTB | A | Amine | 5-Hydroxytryptamine | 5-HT6 | Homo sapiens | Serotonin | - | Gs/β1/γ2 | 3.3 | 2022-07-27 | 10.1016/j.molcel.2022.05.031 | |
7XTB (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT6 | Homo sapiens | Serotonin | - | 3.3 | 2022-07-27 | 10.1016/j.molcel.2022.05.031 | ||
7XTC | A | Amine | 5-Hydroxytryptamine | 5-HT7 | Homo sapiens | 5-CT | - | Gs/β1/γ2 | 3.2 | 2022-07-27 | 10.1016/j.molcel.2022.05.031 | |
7XTC (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT7 | Homo sapiens | 5-CT | - | 3.2 | 2022-07-27 | 10.1016/j.molcel.2022.05.031 | ||
8DCS | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Cyanopindolol | - | Gs/β1/γ2 | 2.5 | 2022-07-27 | 10.1038/s41467-022-31823-1 | |
8DCS (No Gprot) | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Cyanopindolol | - | 2.5 | 2022-07-27 | 10.1038/s41467-022-31823-1 | ||
8DCR | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Dobutamine | - | Gs/β1/γ2 | 2.6 | 2022-07-27 | 10.1038/s41467-022-31823-1 | |
8DCR (No Gprot) | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Dobutamine | - | 2.6 | 2022-07-27 | 10.1038/s41467-022-31823-1 | ||
7UM4 | A | Amine | 5-Hydroxytryptamine | 5-HT5A | Homo sapiens | AS2674723 | - | - | 2.8 | 2022-07-20 | 10.1038/s41594-022-00796-6 | |
7Y14 | A | Orphan | Orphan | MRGPRD | Homo sapiens | β-Alanine | - | - | 3.2 | 2022-07-20 | 10.1038/s42003-022-03668-3 | |
7Y13 | A | Orphan | Orphan | MRGPRD | Homo sapiens | - | - | - | 3.1 | 2022-07-20 | 10.1038/s42003-022-03668-3 | |
7UM7 | A | Amine | 5-Hydroxytryptamine | 5-HT5A | Homo sapiens | Methylergometrine | - | chim(NtGi1-Go)/β1/γ2 | 2.75 | 2022-07-20 | 10.1038/s41594-022-00796-6 | |
7UM7 (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT5A | Homo sapiens | Methylergometrine | - | 2.75 | 2022-07-20 | 10.1038/s41594-022-00796-6 | ||
7UM6 | A | Amine | 5-Hydroxytryptamine | 5-HT5A | Homo sapiens | Lisuride | - | chim(NtGi1-Go)/β1/γ2 | 2.79 | 2022-07-20 | 10.1038/s41594-022-00796-6 | |
7UM6 (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT5A | Homo sapiens | Lisuride | - | 2.79 | 2022-07-20 | 10.1038/s41594-022-00796-6 | ||
7UM5 | A | Amine | 5-Hydroxytryptamine | 5-HT5A | Homo sapiens | 5-CT | - | chim(NtGi1-Go)/β1/γ2 | 2.73 | 2022-07-20 | 10.1038/s41594-022-00796-6 | |
7UM5 (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT5A | Homo sapiens | 5-CT | - | 2.73 | 2022-07-20 | 10.1038/s41594-022-00796-6 | ||
7XOW | A | Peptide | Cholecystokinin | CCKB | Homo sapiens | Gastrin | - | chim(NtGi1-Gq)/β1/γ2 | 3.1 | 2022-07-20 | 10.1038/s41421-022-00420-3 | |
7XOW (No Gprot) | A | Peptide | Cholecystokinin | CCKB | Homo sapiens | Gastrin | - | 3.1 | 2022-07-20 | 10.1038/s41421-022-00420-3 | ||
7Y15 | A | Orphan | Orphan | MRGPRD | Homo sapiens | - | - | Gi1/β1/γ2 | 2.9 | 2022-07-20 | 10.1038/s42003-022-03668-3 | |
7Y15 (No Gprot) | A | Orphan | Orphan | MRGPRD | Homo sapiens | - | - | 2.9 | 2022-07-20 | 10.1038/s42003-022-03668-3 | ||
7Y12 | A | Orphan | Orphan | MRGPRD | Homo sapiens | β-Alanine | - | Gi1/β1/γ2 | 3.1 | 2022-07-20 | 10.1038/s42003-022-03668-3 | |
7Y12 (No Gprot) | A | Orphan | Orphan | MRGPRD | Homo sapiens | β-Alanine | - | 3.1 | 2022-07-20 | 10.1038/s42003-022-03668-3 | ||
7XOV | A | Peptide | Cholecystokinin | CCKA | Homo sapiens | SR146131 | - | Gs/β1/γ2 | 3 | 2022-07-20 | 10.1038/s41421-022-00420-3 | |
7XOV (No Gprot) | A | Peptide | Cholecystokinin | CCKA | Homo sapiens | SR146131 | - | 3 | 2022-07-20 | 10.1038/s41421-022-00420-3 | ||
7XOU | A | Peptide | Cholecystokinin | CCKA | Homo sapiens | Cholecystokinin-8 | - | Gs/β1/γ2 | 3.2 | 2022-07-20 | 10.1038/s41421-022-00420-3 | |
7XOU (No Gprot) | A | Peptide | Cholecystokinin | CCKA | Homo sapiens | Cholecystokinin-8 | - | 3.2 | 2022-07-20 | 10.1038/s41421-022-00420-3 | ||
7XBD | A | Peptide | Galanin | GAL2 | Homo sapiens | Galanin | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 3.11 | 2022-07-13 | 10.1371/journal.pbio.3001714 | |
7XBD (No Gprot) | A | Peptide | Galanin | GAL2 | Homo sapiens | Galanin | - | 3.11 | 2022-07-13 | 10.1371/journal.pbio.3001714 | ||
7XBX | A | Protein | Chemokine | CX3CR1 | Homo sapiens | CX3CL1 | - | Gi1/β1/γ2 | 3.4 | 2022-07-13 | 10.1126/sciadv.abn8048 | |
7XBX (No Gprot) | A | Protein | Chemokine | CX3CR1 | Homo sapiens | CX3CL1 | - | 3.4 | 2022-07-13 | 10.1126/sciadv.abn8048 | ||
7XBW | A | Protein | Chemokine | CX3CR1 | Homo sapiens | - | - | Gi1/β1/γ2 | 2.8 | 2022-07-13 | 10.1126/sciadv.abn8048 | |
7XBW (No Gprot) | A | Protein | Chemokine | CX3CR1 | Homo sapiens | - | - | 2.8 | 2022-07-13 | 10.1126/sciadv.abn8048 | ||
7WJ5 | A | Peptide | Somatostatin | SST2 | Homo sapiens | Somatostatin-14 | - | Gi1/β1/γ2 | 3.72 | 2022-07-13 | 10.7554/eLife.76823 | |
7WJ5 (No Gprot) | A | Peptide | Somatostatin | SST2 | Homo sapiens | Somatostatin-14 | - | 3.72 | 2022-07-13 | 10.7554/eLife.76823 | ||
7RAN | A | Amine | 5-Hydroxytryptamine | 5-HT2A | Homo sapiens | PubChem 164575847 | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 3.45 | 2022-07-06 | 10.1038/s41586-022-05258-z | |
7RAN (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT2A | Homo sapiens | PubChem 164575847 | - | 3.45 | 2022-07-06 | 10.1038/s41586-022-05258-z | ||
7XTQ | A | Steroid | Bile Acid | GPBA | Homo sapiens | R399 | - | Gs/β1/γ2 | 3.2 | 2022-07-06 | 10.1073/pnas.2117054119 | |
7XTQ (No Gprot) | A | Steroid | Bile Acid | GPBA | Homo sapiens | R399 | - | 3.2 | 2022-07-06 | 10.1073/pnas.2117054119 | ||
7UL4 | A | Peptide | Opioid | μ | Mus musculus | Alvimopan | - | - | 2.8 | 2022-06-29 | 10.1038/s41594-022-00859-8 | |
7UL2 | A | Peptide | Neurotensin | NTS1 | Homo sapiens | SR48692 | Na | - | 2.4 | 2022-06-29 | 10.1038/s41594-022-00859-8 | |
7UL5 | A | Peptide | Somatostatin | SST2 | Homo sapiens | - | - | - | 3.1 | 2022-06-29 | 10.1038/s41594-022-00859-8 | |
7XJL | A | Peptide | Galanin | GAL2 | Homo sapiens | Spexin | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 3.5 | 2022-06-29 | 10.1073/pnas.2121465119 | |
7XJL (No Gprot) | A | Peptide | Galanin | GAL2 | Homo sapiens | Spexin | - | 3.5 | 2022-06-29 | 10.1073/pnas.2121465119 | ||
7XJK | A | Peptide | Galanin | GAL2 | Homo sapiens | Galanin | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 3.3 | 2022-06-29 | 10.1073/pnas.2121465119 | |
7XJK (No Gprot) | A | Peptide | Galanin | GAL2 | Homo sapiens | Galanin | - | 3.3 | 2022-06-29 | 10.1073/pnas.2121465119 | ||
7X2C | A | Amine | Dopamine | D1 | Homo sapiens | Fenoldopam | Fenoldopam | Gs/β1/γ2 | 3.2 | 2022-06-29 | 10.1038/s41467-022-30929-w | |
7X2C (No Gprot) | A | Amine | Dopamine | D1 | Homo sapiens | Fenoldopam | Fenoldopam | 3.2 | 2022-06-29 | 10.1038/s41467-022-30929-w | ||
7X8S | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | WB4-24 | - | Gs/β1/γ2 | 3.09 | 2022-06-29 | 10.1073/pnas.2200155119 | |
7X8S (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | WB4-24 | - | 3.09 | 2022-06-29 | 10.1073/pnas.2200155119 | ||
7X8R | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | BOC5 | - | Gs/β1/γ2 | 2.61 | 2022-06-29 | 10.1073/pnas.2200155119 | |
7X8R (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | BOC5 | - | 2.61 | 2022-06-29 | 10.1073/pnas.2200155119 | ||
7FEE | A | Lipid | Cannabinoid | CB1 | Homo sapiens | CP55940 | ZCZ011 | - | 2.7 | 2022-06-15 | 10.1038/s41589-022-01038-y | |
7ZI0 | F | Protein | Frizzled | SMO | Homo sapiens | SAG | Cholesterol | - | 3 | 2022-06-15 | 10.1126/sciadv.abm5563 | |
7WKD | A | Peptide | Thyrotropin Releasing Hormone | TRH | Homo sapiens | TRH | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.01 | 2022-06-15 | 10.1038/s41422-022-00641-x | |
7WKD (No Gprot) | A | Peptide | Thyrotropin Releasing Hormone | TRH | Homo sapiens | TRH | - | 3.01 | 2022-06-15 | 10.1038/s41422-022-00641-x | ||
7WV9 | A | Lipid | Cannabinoid | CB1 | Homo sapiens | CP55940 | ZCZ011 | Gi2/β1/γ2 | 3.36 | 2022-06-15 | 10.1038/s41589-022-01038-y | |
7WV9 (No Gprot) | A | Lipid | Cannabinoid | CB1 | Homo sapiens | CP55940 | ZCZ011 | 3.36 | 2022-06-15 | 10.1038/s41589-022-01038-y | ||
7X2F | A | Amine | Dopamine | D1 | Homo sapiens | Dopamine | Mevidalen | Gs/β1/γ2 | 3 | 2022-06-15 | 10.1038/s41467-022-30929-w | |
7X2F (No Gprot) | A | Amine | Dopamine | D1 | Homo sapiens | Dopamine | Mevidalen | 3 | 2022-06-15 | 10.1038/s41467-022-30929-w | ||
7X2D | A | Amine | Dopamine | D1 | Homo sapiens | Tavapadon | - | Gs/β1/γ2 | 3.3 | 2022-06-15 | 10.1038/s41467-022-30929-w | |
7X2D (No Gprot) | A | Amine | Dopamine | D1 | Homo sapiens | Tavapadon | - | 3.3 | 2022-06-15 | 10.1038/s41467-022-30929-w | ||
7F24 | A | Amine | Dopamine | D1 | Homo sapiens | Dopamine | GDP | Gs/β1/γ2 | 4.16 | 2022-06-15 | 10.1126/sciadv.abo4158 | |
7F24 (No Gprot) | A | Amine | Dopamine | D1 | Homo sapiens | Dopamine | GDP | 4.16 | 2022-06-15 | 10.1126/sciadv.abo4158 | ||
7F23 | A | Amine | Dopamine | D1 | Homo sapiens | Dopamine | GDP | Gs/β1/γ2 | 3.58 | 2022-06-15 | 10.1126/sciadv.abo4158 | |
7F23 (No Gprot) | A | Amine | Dopamine | D1 | Homo sapiens | Dopamine | GDP | 3.58 | 2022-06-15 | 10.1126/sciadv.abo4158 | ||
7F1Z | A | Amine | Dopamine | D1 | Homo sapiens | Dopamine | GDP | Gs/β1/γ2 | 3.46 | 2022-06-15 | 10.1126/sciadv.abo4158 | |
7F1Z (No Gprot) | A | Amine | Dopamine | D1 | Homo sapiens | Dopamine | GDP | 3.46 | 2022-06-15 | 10.1126/sciadv.abo4158 | ||
7F1O | A | Amine | Dopamine | D1 | Homo sapiens | Dopamine | GDP; Mg | Gs/β1/γ2 | 3.13 | 2022-06-15 | 10.1126/sciadv.abo4158 | |
7F1O (No Gprot) | A | Amine | Dopamine | D1 | Homo sapiens | Dopamine | GDP; Mg | 3.13 | 2022-06-15 | 10.1126/sciadv.abo4158 | ||
7F0T | A | Amine | Dopamine | D1 | Homo sapiens | Dopamine | - | Gs/β1/γ2 | 3.1 | 2022-06-15 | 10.1126/sciadv.abo4158 | |
7F0T (No Gprot) | A | Amine | Dopamine | D1 | Homo sapiens | Dopamine | - | 3.1 | 2022-06-15 | 10.1126/sciadv.abo4158 | ||
7S15 | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | PubChem 134611223 | - | - | 3.8 | 2022-06-08 | 10.1021/acs.jmedchem.1c01856 | |
7SR8 | A | Peptide | Orexin | OX2 | Homo sapiens | TAK-925 | - | chim(NtGi1L-Gs-CtGq)/β1/γ2 | 3.3 | 2022-06-08 | 10.1038/s41467-022-30601-3 | |
7SR8 (No Gprot) | A | Peptide | Orexin | OX2 | Homo sapiens | TAK-925 | - | 3.3 | 2022-06-08 | 10.1038/s41467-022-30601-3 | ||
7WIG | A | Peptide | Somatostatin | SST2 | Homo sapiens | L-054,264 | - | Gi1/β1/γ2 | 2.7 | 2022-06-01 | 10.1038/s41422-022-00669-z | |
7WIG (No Gprot) | A | Peptide | Somatostatin | SST2 | Homo sapiens | L-054,264 | - | 2.7 | 2022-06-01 | 10.1038/s41422-022-00669-z | ||
7WIC | A | Peptide | Somatostatin | SST2 | Homo sapiens | Somatostatin-14 | - | Gi1/β1/γ2 | 2.8 | 2022-06-01 | 10.1038/s41422-022-00669-z | |
7WIC (No Gprot) | A | Peptide | Somatostatin | SST2 | Homo sapiens | Somatostatin-14 | - | 2.8 | 2022-06-01 | 10.1038/s41422-022-00669-z | ||
7EUO | A | Peptide | Formylpeptide | FPR1-ALX | Homo sapiens | fMLF | - | Gi1/β1/γ2 | 2.9 | 2022-05-25 | 10.1038/s41467-022-32822-y | |
7EUO (No Gprot) | A | Peptide | Formylpeptide | FPR1-ALX | Homo sapiens | fMLF | - | 2.9 | 2022-05-25 | 10.1038/s41467-022-32822-y | ||
7SQO | A | Peptide | Orexin | OX2 | Homo sapiens | TAK-925 | - | Gi1/β1/γ2 | 3.17 | 2022-05-25 | 10.1038/s41467-022-30601-3 | |
7SQO (No Gprot) | A | Peptide | Orexin | OX2 | Homo sapiens | TAK-925 | - | 3.17 | 2022-05-25 | 10.1038/s41467-022-30601-3 | ||
7X9A | A | Peptide | Neuropeptide Y | Y1 | Homo sapiens | Neuropeptide-Y | - | Gi1/β1/γ2 | 3.2 | 2022-05-18 | 10.1126/sciadv.abm1232 | |
7X9A (No Gprot) | A | Peptide | Neuropeptide Y | Y1 | Homo sapiens | Neuropeptide-Y | - | 3.2 | 2022-05-18 | 10.1126/sciadv.abm1232 | ||
7X9B | A | Peptide | Neuropeptide Y | Y2 | Homo sapiens | Neuropeptide-Y | - | Gi1/β1/γ2 | 3.4 | 2022-05-18 | 10.1126/sciadv.abm1232 | |
7X9B (No Gprot) | A | Peptide | Neuropeptide Y | Y2 | Homo sapiens | Neuropeptide-Y | - | 3.4 | 2022-05-18 | 10.1126/sciadv.abm1232 | ||
7X9C | A | Peptide | Neuropeptide Y | Y4 | Homo sapiens | Pancreatic Hormone | - | Gi1/β1/γ2 | 3 | 2022-05-18 | 10.1126/sciadv.abm1232 | |
7X9C (No Gprot) | A | Peptide | Neuropeptide Y | Y4 | Homo sapiens | Pancreatic Hormone | - | 3 | 2022-05-18 | 10.1126/sciadv.abm1232 | ||
7WBJ | B1 | Peptide | VIP and PACAP | VPAC1 | Homo sapiens | PACAP27 | - | Gs/β1/γ2 | 3.42 | 2022-05-18 | 10.1038/s41467-022-30041-z | |
7WBJ (No Gprot) | B1 | Peptide | VIP and PACAP | VPAC1 | Homo sapiens | PACAP27 | - | 3.42 | 2022-05-18 | 10.1038/s41467-022-30041-z | ||
7VQX | B1 | Peptide | VIP and PACAP | VPAC1 | Homo sapiens | PACAP27 | - | Gs/β1/γ2 | 2.74 | 2022-05-18 | 10.1038/s41467-022-30041-z | |
7VQX (No Gprot) | B1 | Peptide | VIP and PACAP | VPAC1 | Homo sapiens | PACAP27 | - | 2.74 | 2022-05-18 | 10.1038/s41467-022-30041-z | ||
7EQ1 | B2 | Adhesion | Adhesion | ADGRG5 | Homo sapiens | - | - | chim(NtGi1-Gs)/β1/γ2 | 3.3 | 2022-05-11 | 10.1038/s41586-022-04619-y | |
7EQ1 (No Gprot) | B2 | Adhesion | Adhesion | ADGRG5 | Homo sapiens | - | - | 3.3 | 2022-05-11 | 10.1038/s41586-022-04619-y | ||
7V6A | A | Amine | Acetylcholine (muscarinic) | M4 | Homo sapiens | PubChem 9864275 | - | Gi1/β1/γ2 | 3.6 | 2022-05-11 | 10.1038/s41467-022-30595-y | |
7V6A (No Gprot) | A | Amine | Acetylcholine (muscarinic) | M4 | Homo sapiens | PubChem 9864275 | - | 3.6 | 2022-05-11 | 10.1038/s41467-022-30595-y | ||
7V69 | A | Amine | Acetylcholine (muscarinic) | M4 | Homo sapiens | - | - | Gi1/β1/γ2 | 3.4 | 2022-05-11 | 10.1038/s41467-022-30595-y | |
7V69 (No Gprot) | A | Amine | Acetylcholine (muscarinic) | M4 | Homo sapiens | - | - | 3.4 | 2022-05-11 | 10.1038/s41467-022-30595-y | ||
7V68 | A | Amine | Acetylcholine (muscarinic) | M4 | Homo sapiens | Iperoxo | PubChem 57664406 | Gi1/β1/γ2 | 3.4 | 2022-05-11 | 10.1038/s41467-022-30595-y | |
7V68 (No Gprot) | A | Amine | Acetylcholine (muscarinic) | M4 | Homo sapiens | Iperoxo | PubChem 57664406 | 3.4 | 2022-05-11 | 10.1038/s41467-022-30595-y | ||
7EPT | B2 | Adhesion | Adhesion | ADGRD1 | Homo sapiens | - | - | Gs/β1/γ2 | 3 | 2022-05-11 | 10.1038/s41586-022-04619-y | |
7EPT (No Gprot) | B2 | Adhesion | Adhesion | ADGRD1 | Homo sapiens | - | - | 3 | 2022-05-11 | 10.1038/s41586-022-04619-y | ||
7U2L | A | Peptide | Opioid | μ | Mus musculus | PubChem 163201242 | - | Gi1/β1/γ2 | 3.2 | 2022-05-04 | 10.1038/s41586-022-05588-y | |
7U2L (No Gprot) | A | Peptide | Opioid | μ | Mus musculus | PubChem 163201242 | - | 3.2 | 2022-05-04 | 10.1038/s41586-022-05588-y | ||
7XJI | A | Amine | Adrenergic | β3 | Canis lupus familiaris | Solabegron | - | Gs/β1/γ2 | 3.9 | 2022-05-04 | 10.1016/j.bbrc.2022.04.065 | |
7XJI (No Gprot) | A | Amine | Adrenergic | β3 | Canis lupus familiaris | Solabegron | - | 3.9 | 2022-05-04 | 10.1016/j.bbrc.2022.04.065 | ||
7XJH | A | Amine | Adrenergic | β3 | Canis lupus familiaris | Isoproterenol | - | Gs/β1/γ2 | 3.3 | 2022-05-04 | 10.1016/j.molcel.2021.06.024 | |
7XJH (No Gprot) | A | Amine | Adrenergic | β3 | Canis lupus familiaris | Isoproterenol | - | 3.3 | 2022-05-04 | 10.1016/j.molcel.2021.06.024 | ||
7WUI | B2 | Adhesion | Adhesion | ADGRG2 | Mus musculus | IP15 | - | chim(NtGi1-Gs)/β1/γ2 | 3.1 | 2022-04-27 | 10.1038/s41586-022-04590-8 | |
7WUI (No Gprot) | B2 | Adhesion | Adhesion | ADGRG2 | Mus musculus | IP15 | - | 3.1 | 2022-04-27 | 10.1038/s41586-022-04590-8 | ||
7WUJ | B2 | Adhesion | Adhesion | ADGRG4 | Homo sapiens | - | - | chim(NtGi1-Gs)/β1/γ2 | 3.3 | 2022-04-27 | 10.1038/s41586-022-04590-8 | |
7WUJ (No Gprot) | B2 | Adhesion | Adhesion | ADGRG4 | Homo sapiens | - | - | 3.3 | 2022-04-27 | 10.1038/s41586-022-04590-8 | ||
7SF8 | B2 | Adhesion | Adhesion | ADGRG1 | Homo sapiens | - | - | chim(NtGi2-G13)/β1/γ2 | 2.7 | 2022-04-27 | 10.1038/s41586-022-04575-7 | |
7SF8 (No Gprot) | B2 | Adhesion | Adhesion | ADGRG1 | Homo sapiens | - | - | 2.7 | 2022-04-27 | 10.1038/s41586-022-04575-7 | ||
7SF7 | B2 | Adhesion | Adhesion | ADGRL3 | Homo sapiens | - | - | chim(NtGi2-G13)/β1/γ2 | 2.9 | 2022-04-27 | 10.1038/s41586-022-04575-7 | |
7SF7 (No Gprot) | B2 | Adhesion | Adhesion | ADGRL3 | Homo sapiens | - | - | 2.9 | 2022-04-27 | 10.1038/s41586-022-04575-7 | ||
7WU5 | B2 | Adhesion | Adhesion | ADGRF1 | Homo sapiens | - | K6G | Gi1/β1/γ2 | 3 | 2022-04-27 | 10.1038/s41586-022-04580-w | |
7WU5 (No Gprot) | B2 | Adhesion | Adhesion | ADGRF1 | Homo sapiens | - | K6G | 3 | 2022-04-27 | 10.1038/s41586-022-04580-w | ||
7WU4 | B2 | Adhesion | Adhesion | ADGRF1 | Homo sapiens | - | K6G | Gi1/β1/γ2 | 3.4 | 2022-04-27 | 10.1038/s41586-022-04580-w | |
7WU4 (No Gprot) | B2 | Adhesion | Adhesion | ADGRF1 | Homo sapiens | - | K6G | 3.4 | 2022-04-27 | 10.1038/s41586-022-04580-w | ||
7WU2 | B2 | Adhesion | Adhesion | ADGRD1 | Homo sapiens | - | - | Gs/β1/γ1 | 2.8 | 2022-04-27 | 10.1038/s41586-022-04580-w | |
7WU2 (No Gprot) | B2 | Adhesion | Adhesion | ADGRD1 | Homo sapiens | - | - | 2.8 | 2022-04-27 | 10.1038/s41586-022-04580-w | ||
7WU3 | B2 | Adhesion | Adhesion | ADGRF1 | Homo sapiens | - | K6G | Gs/β1/γ2 | 3.1 | 2022-04-27 | 10.1038/s41586-022-04580-w | |
7WU3 (No Gprot) | B2 | Adhesion | Adhesion | ADGRF1 | Homo sapiens | - | K6G | 3.1 | 2022-04-27 | 10.1038/s41586-022-04580-w | ||
7WUQ | B2 | Adhesion | Adhesion | ADGRG2 | Mus musculus | - | - | Gs/β1/γ2 | 2.9 | 2022-04-27 | 10.1038/s41586-022-04590-8 | |
7WUQ (No Gprot) | B2 | Adhesion | Adhesion | ADGRG2 | Mus musculus | - | - | 2.9 | 2022-04-27 | 10.1038/s41586-022-04590-8 | ||
7WQ4 | A | Peptide | Galanin | GAL2 | Homo sapiens | Galanin | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.6 | 2022-04-20 | 10.1038/s41467-022-29072-3 | |
7WQ4 (No Gprot) | A | Peptide | Galanin | GAL2 | Homo sapiens | Galanin | - | 2.6 | 2022-04-20 | 10.1038/s41467-022-29072-3 | ||
7W56 | A | Peptide | Neuromedin U | NMUR1 | Homo sapiens | Neuromedin-S | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.9 | 2022-04-20 | 10.1038/s41467-022-29683-w | |
7W56 (No Gprot) | A | Peptide | Neuromedin U | NMUR1 | Homo sapiens | Neuromedin-S | - | 2.9 | 2022-04-20 | 10.1038/s41467-022-29683-w | ||
7W53 | A | Peptide | Neuromedin U | NMUR1 | Homo sapiens | Neuromedin-U-25 | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.2 | 2022-04-20 | 10.1038/s41467-022-29683-w | |
7W53 (No Gprot) | A | Peptide | Neuromedin U | NMUR1 | Homo sapiens | Neuromedin-U-25 | - | 3.2 | 2022-04-20 | 10.1038/s41467-022-29683-w | ||
7W57 | A | Peptide | Neuromedin U | NMUR2 | Homo sapiens | Neuromedin-S | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.2 | 2022-04-20 | 10.1038/s41467-022-29683-w | |
7W57 (No Gprot) | A | Peptide | Neuromedin U | NMUR2 | Homo sapiens | Neuromedin-S | - | 3.2 | 2022-04-20 | 10.1038/s41467-022-29683-w | ||
7W55 | A | Peptide | Neuromedin U | NMUR2 | Homo sapiens | Neuromedin-U-25 | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.8 | 2022-04-20 | 10.1038/s41467-022-29683-w | |
7W55 (No Gprot) | A | Peptide | Neuromedin U | NMUR2 | Homo sapiens | Neuromedin-U-25 | - | 2.8 | 2022-04-20 | 10.1038/s41467-022-29683-w | ||
7WQ3 | A | Peptide | Galanin | GAL1 | Homo sapiens | Galanin | - | Gi1/β1/γ2 | 2.7 | 2022-04-20 | 10.1038/s41467-022-29072-3 | |
7WQ3 (No Gprot) | A | Peptide | Galanin | GAL1 | Homo sapiens | Galanin | - | 2.7 | 2022-04-20 | 10.1038/s41467-022-29072-3 | ||
7SCG | A | Peptide | Opioid | μ | Mus musculus | FH210 | - | Gi1/β1/γ2 | 3 | 2022-04-20 | 10.1002/anie.202200269 | |
7SCG (No Gprot) | A | Peptide | Opioid | μ | Mus musculus | FH210 | - | 3 | 2022-04-20 | 10.1002/anie.202200269 | ||
7SBF | A | Peptide | Opioid | μ | Mus musculus | PZM21 | - | Gi1/β1/γ2 | 2.9 | 2022-04-20 | 10.1002/anie.202200269 | |
7SBF (No Gprot) | A | Peptide | Opioid | μ | Mus musculus | PZM21 | - | 2.9 | 2022-04-20 | 10.1002/anie.202200269 | ||
7EZC | A | Nucleotide | Adenosine | A2A | Homo sapiens | UKA | - | - | 3.8 | 2022-04-13 | 10.1107/S2052252522001907 | |
7TUY | A | Orphan | Orphan | GPR183 | Homo sapiens | GSK682753A | - | - | 2.98 | 2022-04-13 | 10.1016/j.str.2022.04.006 | |
7RBT | B1 | Peptide | Glucagon | GIP | Homo sapiens | Tirzepatide | PubChem 163183774 | chim(NtGi1-Gs)/β1/γ2 | 3.08 | 2022-04-13 | 10.1073/pnas.2116506119 | |
7RBT (No Gprot) | B1 | Peptide | Glucagon | GIP | Homo sapiens | Tirzepatide | PubChem 163183774 | 3.08 | 2022-04-13 | 10.1073/pnas.2116506119 | ||
7RA3 | B1 | Peptide | Glucagon | GIP | Homo sapiens | GIP | - | chim(NtGi1-Gs)/β1/γ2 | 3.24 | 2022-04-13 | 10.1073/pnas.2116506119 | |
7RA3 (No Gprot) | B1 | Peptide | Glucagon | GIP | Homo sapiens | GIP | - | 3.24 | 2022-04-13 | 10.1073/pnas.2116506119 | ||
7RGP | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Tirzepatide | - | chim(NtGi1-Gs)/β1/γ2 | 2.9 | 2022-04-13 | 10.1073/pnas.2116506119 | |
7RGP (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Tirzepatide | - | 2.9 | 2022-04-13 | 10.1073/pnas.2116506119 | ||
7RG9 | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | - | - | chim(NtGi1-Gs)/β1/γ2 | 3.2 | 2022-04-13 | 10.1073/pnas.2116506119 | |
7RG9 (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | - | - | 3.2 | 2022-04-13 | 10.1073/pnas.2116506119 | ||
7WVU | A | Peptide | Formylpeptide | FPR1-ALX | Homo sapiens | fMLF | - | Gi1/β1/γ2 | 3.3 | 2022-04-13 | 10.1038/s41467-022-29361-x | |
7WVU (No Gprot) | A | Peptide | Formylpeptide | FPR1-ALX | Homo sapiens | fMLF | - | 3.3 | 2022-04-13 | 10.1038/s41467-022-29361-x | ||
7TUZ | A | Orphan | Orphan | GPR183 | Homo sapiens | 7-α,25-dihydroxycholesterol | - | Gi1/β1/γ2 | 3.12 | 2022-04-13 | 10.1016/j.str.2022.04.006 | |
7TUZ (No Gprot) | A | Orphan | Orphan | GPR183 | Homo sapiens | 7-α,25-dihydroxycholesterol | - | 3.12 | 2022-04-13 | 10.1016/j.str.2022.04.006 | ||
7EJX | A | Orphan | Orphan | GPR88 | Homo sapiens | - | (1R;2R)-2-PCCA | Gi1/β1/γ2 | 2.4 | 2022-04-13 | 10.1038/s41467-022-30081-5 | |
7EJX (No Gprot) | A | Orphan | Orphan | GPR88 | Homo sapiens | - | (1R;2R)-2-PCCA | 2.4 | 2022-04-13 | 10.1038/s41467-022-30081-5 | ||
7WVY | A | Peptide | Formylpeptide | FPR2-ALX | Homo sapiens | Amyloid-β42 | - | Gi2/β1/γ2 | 3 | 2022-04-13 | 10.1038/s41467-022-29361-x | |
7WVY (No Gprot) | A | Peptide | Formylpeptide | FPR2-ALX | Homo sapiens | Amyloid-β42 | - | 3 | 2022-04-13 | 10.1038/s41467-022-29361-x | ||
7WVX | A | Peptide | Formylpeptide | FPR2-ALX | Homo sapiens | Humanin | - | Gi2/β1/γ2 | 2.8 | 2022-04-13 | 10.1038/s41467-022-29361-x | |
7WVX (No Gprot) | A | Peptide | Formylpeptide | FPR2-ALX | Homo sapiens | Humanin | - | 2.8 | 2022-04-13 | 10.1038/s41467-022-29361-x | ||
7WVW | A | Peptide | Formylpeptide | FPR2-ALX | Homo sapiens | fMYFINILTL | - | Gi2/β1/γ2 | 3.1 | 2022-04-13 | 10.1038/s41467-022-29361-x | |
7WVW (No Gprot) | A | Peptide | Formylpeptide | FPR2-ALX | Homo sapiens | fMYFINILTL | - | 3.1 | 2022-04-13 | 10.1038/s41467-022-29361-x | ||
7WVV | A | Peptide | Formylpeptide | FPR2-ALX | Homo sapiens | fMLFII | - | Gi2/β1/γ2 | 2.9 | 2022-04-13 | 10.1038/s41467-022-29361-x | |
7WVV (No Gprot) | A | Peptide | Formylpeptide | FPR2-ALX | Homo sapiens | fMLFII | - | 2.9 | 2022-04-13 | 10.1038/s41467-022-29361-x | ||
7EJK | A | Amine | Adrenergic | α2a | Homo sapiens | Oxymetazoline | - | Go/β1/γ2 | 3.4 | 2022-04-13 | 10.1126/sciadv.abj5347 | |
7EJK (No Gprot) | A | Amine | Adrenergic | α2a | Homo sapiens | Oxymetazoline | - | 3.4 | 2022-04-13 | 10.1126/sciadv.abj5347 | ||
7EJA | A | Amine | Adrenergic | α2a | Homo sapiens | Dexmedetomidine | - | Go/β1/γ2 | 3.6 | 2022-04-13 | 10.1126/sciadv.abj5347 | |
7EJA (No Gprot) | A | Amine | Adrenergic | α2a | Homo sapiens | Dexmedetomidine | - | 3.6 | 2022-04-13 | 10.1126/sciadv.abj5347 | ||
7EJ8 | A | Amine | Adrenergic | α2a | Homo sapiens | Brimonidine | - | Go/β1/γ2 | 3 | 2022-04-13 | 10.1126/sciadv.abj5347 | |
7EJ8 (No Gprot) | A | Amine | Adrenergic | α2a | Homo sapiens | Brimonidine | - | 3 | 2022-04-13 | 10.1126/sciadv.abj5347 | ||
7EJ0 | A | Amine | Adrenergic | α2a | Homo sapiens | L-Norepinephrine | - | Go/β1/γ2 | 3.2 | 2022-04-13 | 10.1126/sciadv.abj5347 | |
7EJ0 (No Gprot) | A | Amine | Adrenergic | α2a | Homo sapiens | L-Norepinephrine | - | 3.2 | 2022-04-13 | 10.1126/sciadv.abj5347 | ||
7V9L | B1 | Peptide | Glucagon | GHRH (SV1) | Homo sapiens | - | - | chim(NtGi1-Gs)/β1/γ2 | 2.6 | 2022-04-06 | 10.1073/pnas.2106606118 | |
7V9L (No Gprot) | B1 | Peptide | Glucagon | GHRH (SV1) | Homo sapiens | - | - | 2.6 | 2022-04-06 | 10.1073/pnas.2106606118 | ||
7T6B | A | Lipid | Lysophospholipid | S1P2 | Homo sapiens | S1P | - | chim(NtGi1L-G13)/β1/γ2 | 3.19 | 2022-04-06 | 10.1126/sciadv.abn0067 | |
7T6B (No Gprot) | A | Lipid | Lysophospholipid | S1P2 | Homo sapiens | S1P | - | 3.19 | 2022-04-06 | 10.1126/sciadv.abn0067 | ||
7VBH | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Peptide-20 | - | Gs/β1/γ2 | 3 | 2022-04-06 | 10.1038/s41467-022-28683-0 | |
7VBH (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Peptide-20 | - | 3 | 2022-04-06 | 10.1038/s41467-022-28683-0 | ||
7T6T | A | Peptide | Formylpeptide | FPR1-ALX | Homo sapiens | fMLFII | - | Gi1/β1/γ2 | 3.2 | 2022-03-30 | 10.1038/s41467-022-28586-0 | |
7T6T (No Gprot) | A | Peptide | Formylpeptide | FPR1-ALX | Homo sapiens | fMLFII | - | 3.2 | 2022-03-30 | 10.1038/s41467-022-28586-0 | ||
7T6V | A | Peptide | Formylpeptide | FPR2-ALX | Homo sapiens | fMLFII | - | Gi1/β1/γ2 | 3.1 | 2022-03-30 | 10.1038/s41467-022-28586-0 | |
7T6V (No Gprot) | A | Peptide | Formylpeptide | FPR2-ALX | Homo sapiens | fMLFII | - | 3.1 | 2022-03-30 | 10.1038/s41467-022-28586-0 | ||
7T6U | A | Peptide | Formylpeptide | FPR2-ALX | Homo sapiens | CGEN-855A | - | Gi1/β1/γ2 | 2.9 | 2022-03-30 | 10.1038/s41467-022-28586-0 | |
7T6U (No Gprot) | A | Peptide | Formylpeptide | FPR2-ALX | Homo sapiens | CGEN-855A | - | 2.9 | 2022-03-30 | 10.1038/s41467-022-28586-0 | ||
7T6S | A | Peptide | Formylpeptide | FPR2-ALX | Homo sapiens | PubChem 24776341 | - | Gi1/β1/γ2 | 3 | 2022-03-30 | 10.1038/s41467-022-28586-0 | |
7T6S (No Gprot) | A | Peptide | Formylpeptide | FPR2-ALX | Homo sapiens | PubChem 24776341 | - | 3 | 2022-03-30 | 10.1038/s41467-022-28586-0 | ||
7TYN | B1 | Peptide | Calcitonin | CT | Homo sapiens | Calcitonin-1 | - | Gs/β1/γ2 | 2.6 | 2022-03-30 | 10.1126/science.abm9609 | |
7TYN (No Gprot) | B1 | Peptide | Calcitonin | CT | Homo sapiens | Calcitonin-1 | - | 2.6 | 2022-03-30 | 10.1126/science.abm9609 | ||
7TYI | B1 | Peptide | Calcitonin | CT | Homo sapiens | Amylin | - | Gs/β1/γ2 | 3.3 | 2022-03-30 | 10.1126/science.abm9609 | |
7TYI (No Gprot) | B1 | Peptide | Calcitonin | CT | Homo sapiens | Amylin | - | 3.3 | 2022-03-30 | 10.1126/science.abm9609 | ||
7TYX | B1 | Peptide | Calcitonin | CT (AMY2) | Homo sapiens | Amylin | - | Gs/β1/γ2; RAMP2 | 2.55 | 2022-03-30 | 10.1126/science.abm9609 | |
7TYX (No Gprot) | B1 | Peptide | Calcitonin | CT (AMY2) | Homo sapiens | Amylin | - | 2.55 | 2022-03-30 | 10.1126/science.abm9609 | ||
7VLA | A | Protein | Chemokine | CCR1 | Homo sapiens | CCL15(27-92) | - | Gi1/β1/γ2 | 2.7 | 2022-03-23 | 10.1038/s41589-021-00918-z | |
7VLA (No Gprot) | A | Protein | Chemokine | CCR1 | Homo sapiens | CCL15(27-92) | - | 2.7 | 2022-03-23 | 10.1038/s41589-021-00918-z | ||
7VL9 | A | Protein | Chemokine | CCR1 | Homo sapiens | CCL15(26-92) | - | Gi1/β1/γ2 | 2.6 | 2022-03-23 | 10.1038/s41589-021-00918-z | |
7VL9 (No Gprot) | A | Protein | Chemokine | CCR1 | Homo sapiens | CCL15(26-92) | - | 2.6 | 2022-03-23 | 10.1038/s41589-021-00918-z | ||
7VL8 | A | Protein | Chemokine | CCR1 | Homo sapiens | - | - | Gi1/β1/γ2 | 2.9 | 2022-03-23 | 10.1038/s41589-021-00918-z | |
7VL8 (No Gprot) | A | Protein | Chemokine | CCR1 | Homo sapiens | - | - | 2.9 | 2022-03-23 | 10.1038/s41589-021-00918-z | ||
7TYO | B1 | Peptide | Calcitonin | CT | Homo sapiens | Calcitonin | - | Gs/β1/γ2 | 2.7 | 2022-03-23 | 10.1126/science.abm9609 | |
7TYO (No Gprot) | B1 | Peptide | Calcitonin | CT | Homo sapiens | Calcitonin | - | 2.7 | 2022-03-23 | 10.1126/science.abm9609 | ||
7TYL | B1 | Peptide | Calcitonin | CT | Homo sapiens | Amylin | - | Gs/β1/γ2 | 3.3 | 2022-03-23 | 10.1126/science.abm9609 | |
7TYL (No Gprot) | B1 | Peptide | Calcitonin | CT | Homo sapiens | Amylin | - | 3.3 | 2022-03-23 | 10.1126/science.abm9609 | ||
7TYW | B1 | Peptide | Calcitonin | CT (AMY1) | Homo sapiens | Calcitonin-1 | - | Gs/β1/γ2; RAMP1 | 3 | 2022-03-23 | 10.1126/science.abm9609 | |
7TYW (No Gprot) | B1 | Peptide | Calcitonin | CT (AMY1) | Homo sapiens | Calcitonin-1 | - | 3 | 2022-03-23 | 10.1126/science.abm9609 | ||
7TYF | B1 | Peptide | Calcitonin | CT (AMY1) | Homo sapiens | Amylin | - | Gs/β1/γ2; RAMP1 | 2.2 | 2022-03-23 | 10.1126/science.abm9609 | |
7TYF (No Gprot) | B1 | Peptide | Calcitonin | CT (AMY1) | Homo sapiens | Amylin | - | 2.2 | 2022-03-23 | 10.1126/science.abm9609 | ||
7TYY | B1 | Peptide | Calcitonin | CT (AMY2) | Homo sapiens | Calcitonin-1 | - | Gs/β1/γ2; RAMP2 | 3 | 2022-03-23 | 10.1126/science.abm9609 | |
7TYY (No Gprot) | B1 | Peptide | Calcitonin | CT (AMY2) | Homo sapiens | Calcitonin-1 | - | 3 | 2022-03-23 | 10.1126/science.abm9609 | ||
7TYH | B1 | Peptide | Calcitonin | CT (AMY2) | Homo sapiens | Calcitonin-1 | - | Gs/β1/γ2; RAMP2 | 3.3 | 2022-03-23 | 10.1126/science.abm9609 | |
7TYH (No Gprot) | B1 | Peptide | Calcitonin | CT (AMY2) | Homo sapiens | Calcitonin-1 | - | 3.3 | 2022-03-23 | 10.1126/science.abm9609 | ||
7TZF | B1 | Peptide | Calcitonin | CT (AMY3) | Homo sapiens | Amylin | - | Gs/β1/γ2; RAMP3 | 2.4 | 2022-03-23 | 10.1126/science.abm9609 | |
7TZF (No Gprot) | B1 | Peptide | Calcitonin | CT (AMY3) | Homo sapiens | Amylin | - | 2.4 | 2022-03-23 | 10.1126/science.abm9609 | ||
7WIH | C | Aminoacid | Metabotropic Glutamate | mGlu3; mGlu3 | Homo sapiens | LY2794193 | - | - | 3.68 | 2022-03-16 | 10.1038/s41422-022-00623-z | |
7WI8 | C | Aminoacid | Metabotropic Glutamate | mGlu3; mGlu3 | Homo sapiens | LY341495 | - | - | 4.17 | 2022-03-16 | 10.1038/s41422-022-00623-z | |
7WI6 | C | Aminoacid | Metabotropic Glutamate | mGlu3; mGlu3 | Homo sapiens | LY341495 | - | - | 3.71 | 2022-03-16 | 10.1038/s41422-022-00623-z | |
7QBI | D1 | Ste2-like | STE2 | STE2 | Saccharomyces cerevisiae | α-factor mating pheromone | - | - | 3.46 | 2022-03-16 | 10.1038/s41586-022-04498-3 | |
7QBC | D1 | Ste2-like | STE2 | STE2 | Saccharomyces cerevisiae | α-factor mating pheromone | - | - | 3.53 | 2022-03-16 | 10.1038/s41586-022-04498-3 | |
7QB9 | D1 | Ste2-like | STE2 | STE2 | Saccharomyces cerevisiae | - | - | - | 3.1 | 2022-03-16 | 10.1038/s41586-022-04498-3 | |
7QA8 | D1 | Ste2-like | STE2 | STE2 | Saccharomyces cerevisiae | Peptide | - | - | 2.7 | 2022-03-16 | 10.1038/s41586-022-04498-3 | |
7RYC | A | Peptide | Vasopressin and Oxytocin | OT | Homo sapiens | Oxytocin | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 2.9 | 2022-03-09 | 10.1038/s41594-022-00728-4 | |
7RYC (No Gprot) | A | Peptide | Vasopressin and Oxytocin | OT | Homo sapiens | Oxytocin | - | 2.9 | 2022-03-09 | 10.1038/s41594-022-00728-4 | ||
7VKT | A | Lipid | Leukotriene | BLT1 | Homo sapiens | LTB4 | - | Gi1/β1/γ2 | 2.9 | 2022-03-09 | 10.1038/s41467-022-28820-9 | |
7VKT (No Gprot) | A | Lipid | Leukotriene | BLT1 | Homo sapiens | LTB4 | - | 2.9 | 2022-03-09 | 10.1038/s41467-022-28820-9 | ||
7PYR | A | Nucleotide | Adenosine | A2A | Homo sapiens | PSB-2115 | - | - | 2.6 | 2022-03-02 | 10.1002/anie.202115545 | |
7PX4 | A | Nucleotide | Adenosine | A2A | Homo sapiens | PSB-2113 | - | - | 2.25 | 2022-03-02 | 10.1002/anie.202115545 | |
7VAB | B1 | Peptide | Glucagon | GIP | Homo sapiens | Non-Acylated Tirzepatide | - | chim(NtGi1-Gs)/β1/γ2 | 3.2 | 2022-03-02 | 10.1038/s41467-022-28683-0 | |
7VAB (No Gprot) | B1 | Peptide | Glucagon | GIP | Homo sapiens | Non-Acylated Tirzepatide | - | 3.2 | 2022-03-02 | 10.1038/s41467-022-28683-0 | ||
7VH0 | A | Melatonin | Melatonin | MT2 | Homo sapiens | Ramelteon | - | Gi1/β1/γ1 | 3.46 | 2022-03-02 | 10.1038/s41467-022-28111-3 | |
7VH0 (No Gprot) | A | Melatonin | Melatonin | MT2 | Homo sapiens | Ramelteon | - | 3.46 | 2022-03-02 | 10.1038/s41467-022-28111-3 | ||
7VGZ | A | Melatonin | Melatonin | MT1 | Homo sapiens | Remalteon | - | Gi1/β1/γ2 | 3.3 | 2022-03-02 | 10.1038/s41467-022-28111-3 | |
7VGZ (No Gprot) | A | Melatonin | Melatonin | MT1 | Homo sapiens | Remalteon | - | 3.3 | 2022-03-02 | 10.1038/s41467-022-28111-3 | ||
7VGY | A | Melatonin | Melatonin | MT1 | Homo sapiens | 2-Iodomelatonin | - | Gi1/β1/γ2 | 3.1 | 2022-03-02 | 10.1038/s41467-022-28111-3 | |
7VGY (No Gprot) | A | Melatonin | Melatonin | MT1 | Homo sapiens | 2-Iodomelatonin | - | 3.1 | 2022-03-02 | 10.1038/s41467-022-28111-3 | ||
7FIY | B1 | Peptide | Glucagon | GIP | Homo sapiens | Tirzepatide | - | Gs/β1/γ2 | 3.4 | 2022-03-02 | 10.1038/s41467-022-28683-0 | |
7FIY (No Gprot) | B1 | Peptide | Glucagon | GIP | Homo sapiens | Tirzepatide | - | 3.4 | 2022-03-02 | 10.1038/s41467-022-28683-0 | ||
7VBI | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Non-Acylated Tirzepatide | - | Gs/β1/γ2 | 3 | 2022-03-02 | 10.1038/s41467-022-28683-0 | |
7VBI (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Non-Acylated Tirzepatide | - | 3 | 2022-03-02 | 10.1038/s41467-022-28683-0 | ||
7FIM | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Tirzepatide | - | Gs/β1/γ2 | 3.4 | 2022-03-02 | 10.1038/s41467-022-28683-0 | |
7FIM (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Tirzepatide | - | 3.4 | 2022-03-02 | 10.1038/s41467-022-28683-0 | ||
7V35 | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | Peptide-20 | - | Gs/β1/γ2 | 3.5 | 2022-03-02 | 10.1038/s41467-022-28683-0 | |
7V35 (No Gprot) | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | Peptide-20 | - | 3.5 | 2022-03-02 | 10.1038/s41467-022-28683-0 | ||
7VGX | A | Peptide | Neuropeptide Y | Y1 | Homo sapiens | Neuropeptide-Y | - | Gi1/β1/γ2 | 3.2 | 2022-02-23 | 10.1038/s41467-022-28510-6 | |
7VGX (No Gprot) | A | Peptide | Neuropeptide Y | Y1 | Homo sapiens | Neuropeptide-Y | - | 3.2 | 2022-02-23 | 10.1038/s41467-022-28510-6 | ||
7FIN | B1 | Peptide | Glucagon | GIP | Homo sapiens | Peptide-20; GGL | - | Gs/β1/γ2 | 3.1 | 2022-02-23 | 10.1038/s41467-022-28683-0 | |
7FIN (No Gprot) | B1 | Peptide | Glucagon | GIP | Homo sapiens | Peptide-20; GGL | - | 3.1 | 2022-02-23 | 10.1038/s41467-022-28683-0 | ||
7JNI | A | Peptide | Angiotensin | AT2 | Homo sapiens | Olodanrigan | - | - | 3 | 2022-02-09 | 10.1073/pnas.2116289119 | |
7TD2 | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | LPA | - | Gi1/β1/γ2 | 3.11 | 2022-02-09 | 10.1038/s41467-022-28417-2 | |
7TD2 (No Gprot) | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | LPA | - | 3.11 | 2022-02-09 | 10.1038/s41467-022-28417-2 | ||
7TD1 | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | LPA | - | Gi1/β1/γ2 | 3.08 | 2022-02-09 | 10.1038/s41467-022-28417-2 | |
7TD1 (No Gprot) | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | LPA | - | 3.08 | 2022-02-09 | 10.1038/s41467-022-28417-2 | ||
7TD0 | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | LPA | - | Gi1/β1/γ2 | 2.83 | 2022-02-09 | 10.1038/s41467-022-28417-2 | |
7TD0 (No Gprot) | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | LPA | - | 2.83 | 2022-02-09 | 10.1038/s41467-022-28417-2 | ||
7TD4 | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | Siponimod | - | Gi1/β1/γ2 | 2.6 | 2022-02-09 | 10.1038/s41467-022-28417-2 | |
7TD4 (No Gprot) | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | Siponimod | - | 2.6 | 2022-02-09 | 10.1038/s41467-022-28417-2 | ||
7TD3 | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | S1P | - | Gi1/β1/γ2 | 3 | 2022-02-09 | 10.1038/s41467-022-28417-2 | |
7TD3 (No Gprot) | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | S1P | - | 3 | 2022-02-09 | 10.1038/s41467-022-28417-2 | ||
7WC9 | A | Amine | 5-Hydroxytryptamine | 5-HT2A | Homo sapiens | PubChem 162421364 | - | - | 2.5 | 2022-01-26 | 10.1126/science.abl8615 | |
7WC8 | A | Amine | 5-Hydroxytryptamine | 5-HT2A | Homo sapiens | Lumateperone | - | - | 2.45 | 2022-01-26 | 10.1126/science.abl8615 | |
7WC7 | A | Amine | 5-Hydroxytryptamine | 5-HT2A | Homo sapiens | Lisuride | - | - | 2.6 | 2022-01-26 | 10.1126/science.abl8615 | |
7WC6 | A | Amine | 5-Hydroxytryptamine | 5-HT2A | Homo sapiens | LSD | - | - | 2.6 | 2022-01-26 | 10.1126/science.abl8615 | |
7WC5 | A | Amine | 5-Hydroxytryptamine | 5-HT2A | Homo sapiens | Psilocin | - | - | 3.2 | 2022-01-26 | 10.1126/science.abl8615 | |
7WC4 | A | Amine | 5-Hydroxytryptamine | 5-HT2A | Homo sapiens | Serotonin | - | - | 3.2 | 2022-01-26 | 10.1126/science.abl8615 | |
7RKF | A | Other | Unclassified | US28 | Human betaherpesvirus 5 | Fractalkine | GDP | chim(NtGi1-G11)/β1/γ2 | 4 | 2022-01-26 | 10.1126/sciadv.abl5442 | |
7RKF (No Gprot) | A | Other | Unclassified | US28 | Human betaherpesvirus 5 | Fractalkine | GDP | 4 | 2022-01-26 | 10.1126/sciadv.abl5442 | ||
7RKX | A | Other | Unclassified | US27 | Human betaherpesvirus 5 | - | - | Gi1/β1/γ2 | 3.1 | 2022-01-26 | 10.1126/sciadv.abl5442 | |
7RKX (No Gprot) | A | Other | Unclassified | US27 | Human betaherpesvirus 5 | - | - | 3.1 | 2022-01-26 | 10.1126/sciadv.abl5442 | ||
7RKN | A | Other | Unclassified | US28 | Human betaherpesvirus 5 | Fractalkine | - | Gi1/β1/γ2 | 3.6 | 2022-01-26 | 10.1126/sciadv.abl5442 | |
7RKN (No Gprot) | A | Other | Unclassified | US28 | Human betaherpesvirus 5 | Fractalkine | - | 3.6 | 2022-01-26 | 10.1126/sciadv.abl5442 | ||
7RKM | A | Other | Unclassified | US28 | Human betaherpesvirus 5 | Fractalkine | - | Gi1/β1/γ2 | 3.5 | 2022-01-26 | 10.1126/sciadv.abl5442 | |
7RKM (No Gprot) | A | Other | Unclassified | US28 | Human betaherpesvirus 5 | Fractalkine | - | 3.5 | 2022-01-26 | 10.1126/sciadv.abl5442 | ||
7SIN | C | Ion | Calcium Sensing | CaS | Homo sapiens | - | NPS-2143 | - | 5.9 | 2022-01-19 | 10.1073/pnas.2115849118 | |
7SIM | C | Ion | Calcium Sensing | CaS | Homo sapiens | Ca | Ca; Ca; Cyclomethyltryptophan; PO4 | - | 2.7 | 2022-01-19 | 10.1073/pnas.2115849118 | |
7SIL | C | Ion | Calcium Sensing | CaS | Homo sapiens | Ca | Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4 | - | 2.7 | 2022-01-19 | 10.1073/pnas.2115849118 | |
7F83 | A | Peptide | Ghrelin | Ghrelin | Homo sapiens | PF-05190457 | - | - | 2.94 | 2022-01-19 | 10.1038/s41467-022-27975-9 | |
7W2Z | A | Peptide | Ghrelin | Ghrelin | Homo sapiens | Ghrelin | - | Go/β1/γ2 | 2.8 | 2022-01-19 | 10.1038/s41467-022-27975-9 | |
7W2Z (No Gprot) | A | Peptide | Ghrelin | Ghrelin | Homo sapiens | Ghrelin | - | 2.8 | 2022-01-19 | 10.1038/s41467-022-27975-9 | ||
7B6W | A | Amine | Adrenergic | α1b | Homo sapiens | Cyclazosin | - | - | 2.87 | 2022-01-12 | 10.1038/s41467-021-27911-3 | |
7LLY | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Oxyntomodulin | - | Gs/β1/γ2 | 3.3 | 2022-01-12 | 10.1038/s41467-021-27760-0 | |
7LLY (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Oxyntomodulin | - | 3.3 | 2022-01-12 | 10.1038/s41467-021-27760-0 | ||
7LLL | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Exendin-4 | - | Gs/β1/γ2 | 3.7 | 2022-01-12 | 10.1038/s41467-021-27760-0 | |
7LLL (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Exendin-4 | - | 3.7 | 2022-01-12 | 10.1038/s41467-021-27760-0 | ||
7WF7 | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | S1P | - | Gi1/β1/γ2 | 3.4 | 2022-01-05 | 10.1038/s41589-021-00930-3 | |
7WF7 (No Gprot) | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | S1P | - | 3.4 | 2022-01-05 | 10.1038/s41589-021-00930-3 | ||
7EO4 | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | BAF312 | - | Gi1/β1/γ2 | 2.86 | 2022-01-05 | 10.1038/s41589-021-00930-3 | |
7EO4 (No Gprot) | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | BAF312 | - | 2.86 | 2022-01-05 | 10.1038/s41589-021-00930-3 | ||
7EO2 | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | FTY720-P | - | Gi1/β1/γ2 | 2.89 | 2022-01-05 | 10.1038/s41589-021-00930-3 | |
7EO2 (No Gprot) | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | FTY720-P | - | 2.89 | 2022-01-05 | 10.1038/s41589-021-00930-3 | ||
7F6I | A | Peptide | Bradykinin | BK2 | Homo sapiens | Kallidin | - | Gq/β1/γ2 | 2.8 | 2022-01-05 | 10.1038/s41467-022-28399-1 | |
7F6I (No Gprot) | A | Peptide | Bradykinin | BK2 | Homo sapiens | Kallidin | - | 2.8 | 2022-01-05 | 10.1038/s41467-022-28399-1 | ||
7F6H | A | Peptide | Bradykinin | BK2 | Homo sapiens | Bradykinin | - | Gq/β1/γ2 | 2.9 | 2022-01-05 | 10.1038/s41467-022-28399-1 | |
7F6H (No Gprot) | A | Peptide | Bradykinin | BK2 | Homo sapiens | Bradykinin | - | 2.9 | 2022-01-05 | 10.1038/s41467-022-28399-1 | ||
7S3I | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | - | - | Gs/β1/γ2 | 2.51 | 2022-01-05 | 10.1038/s41589-021-00945-w | |
7S3I (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | - | - | 2.51 | 2022-01-05 | 10.1038/s41589-021-00945-w | ||
7S1M | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Ex4-D-Ala | - | Gs/β1/γ2 | 2.41 | 2022-01-05 | 10.1038/s41589-021-00945-w | |
7S1M (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Ex4-D-Ala | - | 2.41 | 2022-01-05 | 10.1038/s41589-021-00945-w | ||
7F8X | A | Peptide | Cholecystokinin | CCKA | Homo sapiens | NN9056 | - | - | 3 | 2021-12-29 | 10.1038/s41589-021-00866-8 | |
7VUJ | A | Orphan | Orphan | GPR139 | Homo sapiens | JNJ-63533054 | GDP | chim(Gs-CtGq)/β1/γ2 | 3.8 | 2021-12-29 | 10.1038/s41422-021-00591-w | |
7VUJ (No Gprot) | A | Orphan | Orphan | GPR139 | Homo sapiens | JNJ-63533054 | GDP | 3.8 | 2021-12-29 | 10.1038/s41422-021-00591-w | ||
7VUI | A | Orphan | Orphan | GPR139 | Homo sapiens | JNJ-63533054 | GTP | chim(Gs-CtGq)/β1/γ2 | 3.3 | 2021-12-29 | 10.1038/s41422-021-00591-w | |
7VUI (No Gprot) | A | Orphan | Orphan | GPR139 | Homo sapiens | JNJ-63533054 | GTP | 3.3 | 2021-12-29 | 10.1038/s41422-021-00591-w | ||
7VUH | A | Orphan | Orphan | GPR139 | Homo sapiens | JNJ-63533054 | - | chim(Gs-CtGq)/β1/γ2 | 3.22 | 2021-12-29 | 10.1038/s41422-021-00591-w | |
7VUH (No Gprot) | A | Orphan | Orphan | GPR139 | Homo sapiens | JNJ-63533054 | - | 3.22 | 2021-12-29 | 10.1038/s41422-021-00591-w | ||
7VUG | A | Orphan | Orphan | GPR139 | Homo sapiens | JNJ-63533054 | - | Gi1/β1/γ2 | 3.2 | 2021-12-29 | 10.1038/s41422-021-00591-w | |
7VUG (No Gprot) | A | Orphan | Orphan | GPR139 | Homo sapiens | JNJ-63533054 | - | 3.2 | 2021-12-29 | 10.1038/s41422-021-00591-w | ||
7VOE | A | Amine | 5-Hydroxytryptamine | 5-HT2A | Homo sapiens | Aripiprazole | - | - | 2.9 | 2021-12-22 | 10.1038/s41593-021-00971-w | |
7VOD | A | Amine | 5-Hydroxytryptamine | 5-HT2A | Homo sapiens | Cariprazine | - | - | 3.3 | 2021-12-22 | 10.1038/s41593-021-00971-w | |
7P00 | A | Peptide | Tachykinin | NK1 | Homo sapiens | Substance-P | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.71 | 2021-12-15 | 10.1126/sciadv.abk2872 | |
7P00 (No Gprot) | A | Peptide | Tachykinin | NK1 | Homo sapiens | Substance-P | - | 2.71 | 2021-12-15 | 10.1126/sciadv.abk2872 | ||
7P02 | A | Peptide | Tachykinin | NK1 | Homo sapiens | Protachykinin-1 | - | chim(NtGi1-Gs)/β1/γ2 | 2.87 | 2021-12-15 | 10.1126/sciadv.abk2872 | |
7P02 (No Gprot) | A | Peptide | Tachykinin | NK1 | Homo sapiens | Protachykinin-1 | - | 2.87 | 2021-12-15 | 10.1126/sciadv.abk2872 | ||
7NA8 | A | Peptide | Ghrelin | Ghrelin | Homo sapiens | PubChem 178024 | - | Gi1/β1/γ2 | 2.7 | 2021-12-15 | 10.1038/s41467-021-26735-5 | |
7NA8 (No Gprot) | A | Peptide | Ghrelin | Ghrelin | Homo sapiens | PubChem 178024 | - | 2.7 | 2021-12-15 | 10.1038/s41467-021-26735-5 | ||
7NA7 | A | Peptide | Ghrelin | Ghrelin | Homo sapiens | Ghrelin-27 | - | Gi1/β1/γ2 | 2.7 | 2021-12-15 | 10.1038/s41467-021-26735-5 | |
7NA7 (No Gprot) | A | Peptide | Ghrelin | Ghrelin | Homo sapiens | Ghrelin-27 | - | 2.7 | 2021-12-15 | 10.1038/s41467-021-26735-5 | ||
7SHE | C | Orphan | Orphan | GPR158 | Homo sapiens | - | PI; PE | - | 3.4 | 2021-12-01 | 10.1126/science.abl4732 | |
7EWL | C | Orphan | Orphan | GPR158 | Homo sapiens | - | - | - | 3.52 | 2021-12-01 | 10.1038/s41467-021-27147-1 | |
7VV6 | A | Orphan | Orphan | MRGPRX2 | Homo sapiens | C48/80 | - | - | 3.3 | 2021-12-01 | 10.1038/s41586-021-04077-y | |
7VV4 | A | Orphan | Orphan | MRGPRX2 | Homo sapiens | Cortistatin-14 | - | - | 2.97 | 2021-12-01 | 10.1038/s41586-021-04077-y | |
7VV0 | A | Orphan | Orphan | MRGPRX2 | Homo sapiens | PAMP-12 | - | - | 3.5 | 2021-12-01 | 10.1038/s41586-021-04077-y | |
7SHF | C | Orphan | Orphan | GPR158 | Homo sapiens | - | PI; PE | B5; RGS7 | 3.4 | 2021-12-01 | 10.1126/science.abl4732 | |
7EWR | C | Orphan | Orphan | GPR158 | Homo sapiens | - | - | B5; RGS7 | 4.7 | 2021-12-01 | 10.1038/s41467-021-27147-1 | |
7EWP | C | Orphan | Orphan | GPR158 | Homo sapiens | - | - | B5; RGS7 | 4.3 | 2021-12-01 | 10.1038/s41467-021-27147-1 | |
7VV5 | A | Orphan | Orphan | MRGPRX2 | Homo sapiens | C48/80 | - | Gi1/β1/γ2 | 2.76 | 2021-12-01 | 10.1038/s41586-021-04077-y | |
7VV5 (No Gprot) | A | Orphan | Orphan | MRGPRX2 | Homo sapiens | C48/80 | - | 2.76 | 2021-12-01 | 10.1038/s41586-021-04077-y | ||
7VV3 | A | Orphan | Orphan | MRGPRX2 | Homo sapiens | - | - | Gi1/β1/γ2 | 2.97 | 2021-12-01 | 10.1038/s41586-021-04077-y | |
7VV3 (No Gprot) | A | Orphan | Orphan | MRGPRX2 | Homo sapiens | - | - | 2.97 | 2021-12-01 | 10.1038/s41586-021-04077-y | ||
7VUZ | A | Orphan | Orphan | MRGPRX2 | Homo sapiens | - | - | Gi1/β1/γ2 | 2.89 | 2021-12-01 | 10.1038/s41586-021-04077-y | |
7VUZ (No Gprot) | A | Orphan | Orphan | MRGPRX2 | Homo sapiens | - | - | 2.89 | 2021-12-01 | 10.1038/s41586-021-04077-y | ||
7VUY | A | Orphan | Orphan | MRGPRX2 | Homo sapiens | - | - | Gi1/β1/γ2 | 2.84 | 2021-12-01 | 10.1038/s41586-021-04077-y | |
7VUY (No Gprot) | A | Orphan | Orphan | MRGPRX2 | Homo sapiens | - | - | 2.84 | 2021-12-01 | 10.1038/s41586-021-04077-y | ||
7VDM | A | Orphan | Orphan | MRGPRX2 | Homo sapiens | Substance-P | - | Gi1/β1/γ2 | 2.98 | 2021-12-01 | 10.1038/s41586-021-04077-y | |
7VDM (No Gprot) | A | Orphan | Orphan | MRGPRX2 | Homo sapiens | Substance-P | - | 2.98 | 2021-12-01 | 10.1038/s41586-021-04077-y | ||
7VDL | A | Orphan | Orphan | MRGPRX2 | Homo sapiens | Cortistatin-14 | - | Gi1/β1/γ2 | 3.22 | 2021-12-01 | 10.1038/s41586-021-04077-y | |
7VDL (No Gprot) | A | Orphan | Orphan | MRGPRX2 | Homo sapiens | Cortistatin-14 | - | 3.22 | 2021-12-01 | 10.1038/s41586-021-04077-y | ||
7VDH | A | Orphan | Orphan | MRGPRX2 | Homo sapiens | C48/80 | - | Gi1/β1/γ2 | 2.9 | 2021-12-01 | 10.1038/s41586-021-04077-y | |
7VDH (No Gprot) | A | Orphan | Orphan | MRGPRX2 | Homo sapiens | C48/80 | - | 2.9 | 2021-12-01 | 10.1038/s41586-021-04077-y | ||
7V3Z | A | Lipid | Cannabinoid | CB1 | Homo sapiens | CP55940 | - | - | 3.29 | 2021-11-24 | 10.1021/jacs.1c06847 | |
7S0G | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Isoprenaline | - | chim(Gi1-CtGs)/β1/γ2 | 3.86 | 2021-11-17 | 10.1038/s41594-021-00679-2 | |
7S0G (No Gprot) | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Isoprenaline | - | 3.86 | 2021-11-17 | 10.1038/s41594-021-00679-2 | ||
7S8N | A | Orphan | Orphan | MRGPRX2 | Homo sapiens | R-Zinc-3573 | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 2.9 | 2021-11-17 | 10.1038/s41586-021-04126-6 | |
7S8N (No Gprot) | A | Orphan | Orphan | MRGPRX2 | Homo sapiens | R-Zinc-3573 | - | 2.9 | 2021-11-17 | 10.1038/s41586-021-04126-6 | ||
7S8L | A | Orphan | Orphan | MRGPRX2 | Homo sapiens | Cortistatin-14 | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 2.45 | 2021-11-17 | 10.1038/s41586-021-04126-6 | |
7S8L (No Gprot) | A | Orphan | Orphan | MRGPRX2 | Homo sapiens | Cortistatin-14 | - | 2.45 | 2021-11-17 | 10.1038/s41586-021-04126-6 | ||
7S8P | A | Orphan | Orphan | MRGPRX4 | Homo sapiens | MS47134 | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 2.6 | 2021-11-17 | 10.1038/s41586-021-04126-6 | |
7S8P (No Gprot) | A | Orphan | Orphan | MRGPRX4 | Homo sapiens | MS47134 | - | 2.6 | 2021-11-17 | 10.1038/s41586-021-04126-6 | ||
7S0F | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Isoprenaline | - | Gi1/β1/γ2 | 2.96 | 2021-11-17 | 10.1038/s41594-021-00679-2 | |
7S0F (No Gprot) | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Isoprenaline | - | 2.96 | 2021-11-17 | 10.1038/s41594-021-00679-2 | ||
7S8O | A | Orphan | Orphan | MRGPRX2 | Homo sapiens | R-Zinc-3573 | - | Gi1/β1/γ2 | 2.58 | 2021-11-17 | 10.1038/s41586-021-04126-6 | |
7S8O (No Gprot) | A | Orphan | Orphan | MRGPRX2 | Homo sapiens | R-Zinc-3573 | - | 2.58 | 2021-11-17 | 10.1038/s41586-021-04126-6 | ||
7S8M | A | Orphan | Orphan | MRGPRX2 | Homo sapiens | Cortistatin-14 | - | Gi1/β1/γ2 | 2.54 | 2021-11-17 | 10.1038/s41586-021-04126-6 | |
7S8M (No Gprot) | A | Orphan | Orphan | MRGPRX2 | Homo sapiens | Cortistatin-14 | - | 2.54 | 2021-11-17 | 10.1038/s41586-021-04126-6 | ||
7PIV | A | Peptide | Melanocortin | MC4 | Homo sapiens | Setmelanotide | - | Gs/β1/γ2 | 2.86 | 2021-11-17 | 10.1038/s41422-021-00569-8 | |
7PIV (No Gprot) | A | Peptide | Melanocortin | MC4 | Homo sapiens | Setmelanotide | - | 2.86 | 2021-11-17 | 10.1038/s41422-021-00569-8 | ||
7PIU | A | Peptide | Melanocortin | MC4 | Homo sapiens | Setmelanotide | - | Gs/β1/γ2 | 2.58 | 2021-11-17 | 10.1038/s41422-021-00569-8 | |
7PIU (No Gprot) | A | Peptide | Melanocortin | MC4 | Homo sapiens | Setmelanotide | - | 2.58 | 2021-11-17 | 10.1038/s41422-021-00569-8 | ||
7RMI | A | Peptide | Tachykinin | NK1 | Homo sapiens | Substance-P | - | chim(Gs-CtGq)/β1/γ2 | 3.2 | 2021-11-03 | 10.1038/s41589-021-00890-8 | |
7RMI (No Gprot) | A | Peptide | Tachykinin | NK1 | Homo sapiens | Substance-P | - | 3.2 | 2021-11-03 | 10.1038/s41589-021-00890-8 | ||
7RMG | A | Peptide | Tachykinin | NK1 | Homo sapiens | Substance-P | - | chim(Gs-CtGq)/β1/γ2 | 3 | 2021-11-03 | 10.1038/s41589-021-00890-8 | |
7RMG (No Gprot) | A | Peptide | Tachykinin | NK1 | Homo sapiens | Substance-P | - | 3 | 2021-11-03 | 10.1038/s41589-021-00890-8 | ||
7F58 | A | Peptide | Melanocortin | MC4 | Homo sapiens | THIQ | - | Gs/β1/γ2 | 3.1 | 2021-11-03 | 10.1038/s41422-021-00552-3 | |
7F58 (No Gprot) | A | Peptide | Melanocortin | MC4 | Homo sapiens | THIQ | - | 3.1 | 2021-11-03 | 10.1038/s41422-021-00552-3 | ||
7F55 | A | Peptide | Melanocortin | MC4 | Homo sapiens | Bremelanotide | - | Gs/β1/γ2 | 3.1 | 2021-11-03 | 10.1038/s41422-021-00552-3 | |
7F55 (No Gprot) | A | Peptide | Melanocortin | MC4 | Homo sapiens | Bremelanotide | - | 3.1 | 2021-11-03 | 10.1038/s41422-021-00552-3 | ||
7F54 | A | Peptide | Melanocortin | MC4 | Homo sapiens | Afamelanotide | - | Gs/β1/γ2 | 3 | 2021-11-03 | 10.1038/s41422-021-00552-3 | |
7F54 (No Gprot) | A | Peptide | Melanocortin | MC4 | Homo sapiens | Afamelanotide | - | 3 | 2021-11-03 | 10.1038/s41422-021-00552-3 | ||
7F53 | A | Peptide | Melanocortin | MC4 | Homo sapiens | α-MSH | - | Gs/β1/γ2 | 3 | 2021-11-03 | 10.1038/s41422-021-00552-3 | |
7F53 (No Gprot) | A | Peptide | Melanocortin | MC4 | Homo sapiens | α-MSH | - | 3 | 2021-11-03 | 10.1038/s41422-021-00552-3 | ||
7RMH | A | Peptide | Tachykinin | NK1 | Homo sapiens | Substance-P | - | Gs/β1/γ2 | 3.1 | 2021-11-03 | 10.1038/s41589-021-00890-8 | |
7RMH (No Gprot) | A | Peptide | Tachykinin | NK1 | Homo sapiens | Substance-P | - | 3.1 | 2021-11-03 | 10.1038/s41589-021-00890-8 | ||
7V9M | B1 | Peptide | Glucagon | GHRH (SV1) | Homo sapiens | Somatoliberin | - | Gs/β1/γ2 | 3.29 | 2021-10-20 | 10.1073/pnas.2106606118 | |
7V9M (No Gprot) | B1 | Peptide | Glucagon | GHRH (SV1) | Homo sapiens | Somatoliberin | - | 3.29 | 2021-10-20 | 10.1073/pnas.2106606118 | ||
7F8Y | A | Peptide | Cholecystokinin | CCKA | Homo sapiens | Devazepide | - | - | 2.5 | 2021-10-13 | 10.1038/s41589-021-00866-8 | |
7F8U | A | Peptide | Cholecystokinin | CCKA | Homo sapiens | Lintitript | - | - | 2.8 | 2021-10-13 | 10.1038/s41589-021-00866-8 | |
7EIB | A | Peptide | Bradykinin | BK1 | Homo sapiens | Des-Arg10-Kallidin | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3 | 2021-10-13 | 10.1038/s41594-021-00645-y | |
7EIB (No Gprot) | A | Peptide | Bradykinin | BK1 | Homo sapiens | Des-Arg10-Kallidin | - | 3 | 2021-10-13 | 10.1038/s41594-021-00645-y | ||
7F2O | A | Peptide | Bradykinin | BK2 | Homo sapiens | Bradykinin | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.9 | 2021-10-13 | 10.1038/s41594-021-00645-y | |
7F2O (No Gprot) | A | Peptide | Bradykinin | BK2 | Homo sapiens | Bradykinin | - | 2.9 | 2021-10-13 | 10.1038/s41594-021-00645-y | ||
7F8W | A | Peptide | Cholecystokinin | CCKB | Homo sapiens | Gastrin-17 | - | chim(NtGsL-Gq)/β1/γ2 | 3.1 | 2021-10-13 | 10.1038/s41589-021-00866-8 | |
7F8W (No Gprot) | A | Peptide | Cholecystokinin | CCKB | Homo sapiens | Gastrin-17 | - | 3.1 | 2021-10-13 | 10.1038/s41589-021-00866-8 | ||
7F8V | A | Peptide | Cholecystokinin | CCKB | Homo sapiens | Gastrin-17 | - | Gi2/β1/γ2 | 3.3 | 2021-10-13 | 10.1038/s41589-021-00866-8 | |
7F8V (No Gprot) | A | Peptide | Cholecystokinin | CCKB | Homo sapiens | Gastrin-17 | - | 3.3 | 2021-10-13 | 10.1038/s41589-021-00866-8 | ||
6ZG9 | A | Amine | Acetylcholine (muscarinic) | M1 | Homo sapiens | GSK1034702 | - | - | 2.5 | 2021-10-06 | 10.1016/j.cell.2021.11.001 | |
6ZG4 | A | Amine | Acetylcholine (muscarinic) | M1 | Homo sapiens | HTL0009936 | - | - | 2.33 | 2021-10-06 | 10.1016/j.cell.2021.11.001 | |
6ZFZ | A | Amine | Acetylcholine (muscarinic) | M1 | Homo sapiens | 77-LH-28-1 | - | - | 2.17 | 2021-10-06 | 10.1016/j.cell.2021.11.001 | |
7RTB | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Peptide-19 | - | Gs/β1/γ2 | 2.14 | 2021-10-06 | 10.1016/j.bbrc.2021.09.016 | |
7RTB (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Peptide-19 | - | 2.14 | 2021-10-06 | 10.1016/j.bbrc.2021.09.016 | ||
7FIJ | A | Protein | Glycoprotein Hormone | LH | Homo sapiens | - | - | - | 3.8 | 2021-09-29 | 10.1038/s41586-021-03924-2 | |
7FII | A | Protein | Glycoprotein Hormone | LH | Homo sapiens | hCG | - | chim(NtGi1-Gs)/β1/γ2 | 4.3 | 2021-09-29 | 10.1038/s41586-021-03924-2 | |
7FII (No Gprot) | A | Protein | Glycoprotein Hormone | LH | Homo sapiens | hCG | - | 4.3 | 2021-09-29 | 10.1038/s41586-021-03924-2 | ||
7FIH | A | Protein | Glycoprotein Hormone | LH | Homo sapiens | hCG | Org43553 | chim(NtGi1-Gs)/β1/γ2 | 3.2 | 2021-09-29 | 10.1038/s41586-021-03924-2 | |
7FIH (No Gprot) | A | Protein | Glycoprotein Hormone | LH | Homo sapiens | hCG | Org43553 | 3.2 | 2021-09-29 | 10.1038/s41586-021-03924-2 | ||
7FIG | A | Protein | Glycoprotein Hormone | LH | Homo sapiens | hCG | - | chim(NtGi1L-Gs)/β1/γ2 | 3.9 | 2021-09-29 | 10.1038/s41586-021-03924-2 | |
7FIG (No Gprot) | A | Protein | Glycoprotein Hormone | LH | Homo sapiens | hCG | - | 3.9 | 2021-09-29 | 10.1038/s41586-021-03924-2 | ||
7EW7 | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | SEW2871 | - | Gi1/β1/γ2 | 3.27 | 2021-09-29 | 10.1038/s41422-021-00566-x | |
7EW7 (No Gprot) | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | SEW2871 | - | 3.27 | 2021-09-29 | 10.1038/s41422-021-00566-x | ||
7EW0 | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | Ozanimod | - | Gi1/β1/γ2 | 3.42 | 2021-09-29 | 10.1038/s41422-021-00566-x | |
7EW0 (No Gprot) | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | Ozanimod | - | 3.42 | 2021-09-29 | 10.1038/s41422-021-00566-x | ||
7EVZ | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | Cenerimod | - | Gi1/β1/γ2 | 3.07 | 2021-09-29 | 10.1038/s41422-021-00566-x | |
7EVZ (No Gprot) | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | Cenerimod | - | 3.07 | 2021-09-29 | 10.1038/s41422-021-00566-x | ||
7EVY | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | Siponimod | - | Gi1/β1/γ2 | 2.98 | 2021-09-29 | 10.1038/s41422-021-00566-x | |
7EVY (No Gprot) | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | Siponimod | - | 2.98 | 2021-09-29 | 10.1038/s41422-021-00566-x | ||
7EW4 | A | Lipid | Lysophospholipid | S1P3 | Homo sapiens | CYM5541 | - | Gi1/β1/γ2 | 3.2 | 2021-09-29 | 10.1038/s41422-021-00567-w | |
7EW4 (No Gprot) | A | Lipid | Lysophospholipid | S1P3 | Homo sapiens | CYM5541 | - | 3.2 | 2021-09-29 | 10.1038/s41422-021-00567-w | ||
7EW3 | A | Lipid | Lysophospholipid | S1P3 | Homo sapiens | S1P | - | Gi1/β1/γ2 | 3.1 | 2021-09-29 | 10.1038/s41422-021-00567-w | |
7EW3 (No Gprot) | A | Lipid | Lysophospholipid | S1P3 | Homo sapiens | S1P | - | 3.1 | 2021-09-29 | 10.1038/s41422-021-00567-w | ||
7EW2 | A | Lipid | Lysophospholipid | S1P3 | Homo sapiens | Fingolimod | - | Gi1/β1/γ2 | 3.1 | 2021-09-29 | 10.1038/s41422-021-00567-w | |
7EW2 (No Gprot) | A | Lipid | Lysophospholipid | S1P3 | Homo sapiens | Fingolimod | - | 3.1 | 2021-09-29 | 10.1038/s41422-021-00567-w | ||
7EW1 | A | Lipid | Lysophospholipid | S1P5 | Homo sapiens | Siponimod | - | Gi1/β1/γ2 | 3.4 | 2021-09-29 | 10.1038/s41422-021-00566-x | |
7EW1 (No Gprot) | A | Lipid | Lysophospholipid | S1P5 | Homo sapiens | Siponimod | - | 3.4 | 2021-09-29 | 10.1038/s41422-021-00566-x | ||
7E6U | C | Ion | Calcium Sensing | CaS | Homo sapiens | - | - | - | 6 | 2021-09-22 | 10.7554/eLife.68578 | |
7E6T | C | Ion | Calcium Sensing | CaS | Homo sapiens | Ca | Ca; Ca; Cyclomethyltryptophan; PO4 | - | 3 | 2021-09-22 | 10.7554/eLife.68578 | |
7DGE | C | Aminoacid | Metabotropic Glutamate | mGlu1; mGlu1 | Homo sapiens | Quisqualate | - | - | 3.65 | 2021-09-22 | 10.1007/s13238-020-00808-5 | |
7DGD | C | Aminoacid | Metabotropic Glutamate | mGlu1; mGlu1 | Homo sapiens | - | - | - | 3.96 | 2021-09-22 | 10.1007/s13238-020-00808-5 | |
7RM5 | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | Na | - | 2.79 | 2021-09-08 | 10.1073/pnas.2106041118 | |
7P2L | C | Aminoacid | Metabotropic Glutamate | mGlu5 | Homo sapiens | - | 4YI | - | 2.54 | 2021-09-08 | 10.1016/j.celrep.2021.109648 | |
7FD9 | C | Aminoacid | Metabotropic Glutamate | mGlu5; mGlu5 | Homo sapiens | LY341495 | - | - | 4 | 2021-09-08 | 10.1016/j.celrep.2021.109648 | |
7FD8 | C | Aminoacid | Metabotropic Glutamate | mGlu5; mGlu5 | Homo sapiens | Quisqualate | - | - | 3.8 | 2021-09-08 | 10.1016/j.celrep.2021.109648 | |
7F4I | A | Peptide | Melanocortin | MC1 | Homo sapiens | SHU9119 | - | chim(NtGi1-Gs)/β1/γ2 | 3.1 | 2021-09-08 | 10.1038/s41422-021-00557-y | |
7F4I (No Gprot) | A | Peptide | Melanocortin | MC1 | Homo sapiens | SHU9119 | - | 3.1 | 2021-09-08 | 10.1038/s41422-021-00557-y | ||
7F4H | A | Peptide | Melanocortin | MC1 | Homo sapiens | Afamelanotide | - | chim(NtGi1-Gs)/β1/γ2 | 2.7 | 2021-09-08 | 10.1038/s41422-021-00557-y | |
7F4H (No Gprot) | A | Peptide | Melanocortin | MC1 | Homo sapiens | Afamelanotide | - | 2.7 | 2021-09-08 | 10.1038/s41422-021-00557-y | ||
7F4F | A | Peptide | Melanocortin | MC1 | Homo sapiens | Afamelanotide | - | chim(NtGi1-Gs)/β1/γ2 | 2.9 | 2021-09-08 | 10.1038/s41422-021-00557-y | |
7F4F (No Gprot) | A | Peptide | Melanocortin | MC1 | Homo sapiens | Afamelanotide | - | 2.9 | 2021-09-08 | 10.1038/s41422-021-00557-y | ||
7F4D | A | Peptide | Melanocortin | MC1 | Homo sapiens | α-MSH | - | chim(NtGi1-Gs)/β1/γ2 | 3 | 2021-09-08 | 10.1038/s41422-021-00557-y | |
7F4D (No Gprot) | A | Peptide | Melanocortin | MC1 | Homo sapiens | α-MSH | - | 3 | 2021-09-08 | 10.1038/s41422-021-00557-y | ||
7LD4 | A | Nucleotide | Adenosine | A1 | Homo sapiens | Adenosine | - | Gi2/β1/γ2 | 3.3 | 2021-09-08 | 10.1038/s41586-021-03897-2 | |
7LD4 (No Gprot) | A | Nucleotide | Adenosine | A1 | Homo sapiens | Adenosine | - | 3.3 | 2021-09-08 | 10.1038/s41586-021-03897-2 | ||
7LD3 | A | Nucleotide | Adenosine | A1 | Homo sapiens | Adenosine | PubChem 25263603 | Gi2/β1/γ2 | 3.2 | 2021-09-08 | 10.1038/s41586-021-03897-2 | |
7LD3 (No Gprot) | A | Nucleotide | Adenosine | A1 | Homo sapiens | Adenosine | PubChem 25263603 | 3.2 | 2021-09-08 | 10.1038/s41586-021-03897-2 | ||
7M8W | A | Lipid | Prostanoid | DP2 | Homo sapiens | 15r-Methyl-Prostaglandin D2 | Na | - | 2.61 | 2021-08-25 | 10.1073/pnas.2102813118 | |
7EZK | A | Peptide | Cholecystokinin | CCKA | Homo sapiens | Cholecystokinin-8 | - | chim(NtGi1-Gs)/β1/γ2 | 3.1 | 2021-08-25 | 10.1038/s41589-021-00841-3 | |
7EZK (No Gprot) | A | Peptide | Cholecystokinin | CCKA | Homo sapiens | Cholecystokinin-8 | - | 3.1 | 2021-08-25 | 10.1038/s41589-021-00841-3 | ||
7EZM | A | Peptide | Cholecystokinin | CCKA | Homo sapiens | Cholecystokinin-8 | - | chim(NtGsL-Gq)/β1/γ2 | 2.9 | 2021-08-25 | 10.1038/s41589-021-00841-3 | |
7EZM (No Gprot) | A | Peptide | Cholecystokinin | CCKA | Homo sapiens | Cholecystokinin-8 | - | 2.9 | 2021-08-25 | 10.1038/s41589-021-00841-3 | ||
7EZH | A | Peptide | Cholecystokinin | CCKA | Homo sapiens | Cholecystokinin-8 | - | Gi1/β1/γ2 | 3.2 | 2021-08-25 | 10.1038/s41589-021-00841-3 | |
7EZH (No Gprot) | A | Peptide | Cholecystokinin | CCKA | Homo sapiens | Cholecystokinin-8 | - | 3.2 | 2021-08-25 | 10.1038/s41589-021-00841-3 | ||
7F9Z | A | Peptide | Ghrelin | Ghrelin | Homo sapiens | GHRP-6 | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.2 | 2021-08-18 | 10.1038/s41467-021-25364-2 | |
7F9Z (No Gprot) | A | Peptide | Ghrelin | Ghrelin | Homo sapiens | GHRP-6 | - | 3.2 | 2021-08-18 | 10.1038/s41467-021-25364-2 | ||
7F9Y | A | Peptide | Ghrelin | Ghrelin | Homo sapiens | Ghrelin-28 | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 2.9 | 2021-08-18 | 10.1038/s41467-021-25364-2 | |
7F9Y (No Gprot) | A | Peptide | Ghrelin | Ghrelin | Homo sapiens | Ghrelin-28 | - | 2.9 | 2021-08-18 | 10.1038/s41467-021-25364-2 | ||
7DB6 | A | Melatonin | Melatonin | MT1 | Homo sapiens | Ramelteon | - | Gi1/β1/γ2 | 3.3 | 2021-08-18 | 10.1038/s41594-021-00634-1 | |
7DB6 (No Gprot) | A | Melatonin | Melatonin | MT1 | Homo sapiens | Ramelteon | - | 3.3 | 2021-08-18 | 10.1038/s41594-021-00634-1 | ||
7F16 | B1 | Peptide | Parathyroid Hormone | PTH2 | Homo sapiens | TIP39 | - | Gs/β1/γ2 | 2.8 | 2021-08-18 | 10.1073/pnas.2101279118 | |
7F16 (No Gprot) | B1 | Peptide | Parathyroid Hormone | PTH2 | Homo sapiens | TIP39 | - | 2.8 | 2021-08-18 | 10.1073/pnas.2101279118 | ||
7EVM | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | - | PubChem 156022738 | Gs/β1/γ2 | 2.5 | 2021-08-11 | 10.1038/s41467-021-24058-z | |
7EVM (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | - | PubChem 156022738 | 2.5 | 2021-08-11 | 10.1038/s41467-021-24058-z | ||
7DUR | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | - | PubChem 156022738 | Gs/β1/γ2 | 3.3 | 2021-08-11 | 10.1038/s41467-021-24058-z | |
7DUR (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | - | PubChem 156022738 | 3.3 | 2021-08-11 | 10.1038/s41467-021-24058-z | ||
7EXD | A | Amine | 5-Hydroxytryptamine | 5-HT1F | Homo sapiens | Lasmiditan | - | Gi1/β1/γ2 | 3.4 | 2021-08-04 | 10.1038/s41422-021-00527-4 | |
7EXD (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT1F | Homo sapiens | Lasmiditan | - | 3.4 | 2021-08-04 | 10.1038/s41422-021-00527-4 | ||
7DH5 | A | Amine | Adrenergic | β3 | Canis lupus familiaris | Mirabegron | - | Gs/β1/γ2 | 3.16 | 2021-08-04 | 10.1016/j.molcel.2021.06.024 | |
7DH5 (No Gprot) | A | Amine | Adrenergic | β3 | Canis lupus familiaris | Mirabegron | - | 3.16 | 2021-08-04 | 10.1016/j.molcel.2021.06.024 | ||
7EVW | F | Protein | Frizzled | FZD7 | Homo sapiens | - | - | Gs/β1/γ2 | 3.22 | 2021-08-04 | 10.1038/s41422-021-00525-6 | |
7EVW (No Gprot) | F | Protein | Frizzled | FZD7 | Homo sapiens | - | - | 3.22 | 2021-08-04 | 10.1038/s41422-021-00525-6 | ||
7DTY | B1 | Peptide | Glucagon | GIP | Homo sapiens | GIP | - | Gs/β1/γ2 | 2.98 | 2021-08-04 | 10.7554/eLife.68719 | |
7DTY (No Gprot) | B1 | Peptide | Glucagon | GIP | Homo sapiens | GIP | - | 2.98 | 2021-08-04 | 10.7554/eLife.68719 | ||
7KI1 | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Taspoglutide | - | Gs/β1/γ2 | 2.5 | 2021-08-04 | 10.1016/j.celrep.2021.109374 | |
7KI1 (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Taspoglutide | - | 2.5 | 2021-08-04 | 10.1016/j.celrep.2021.109374 | ||
7KI0 | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Semaglutide | - | Gs/β1/γ2 | 2.5 | 2021-08-04 | 10.1016/j.celrep.2021.109374 | |
7KI0 (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Semaglutide | - | 2.5 | 2021-08-04 | 10.1016/j.celrep.2021.109374 | ||
7DW9 | A | Peptide | Vasopressin and Oxytocin | V2 | Homo sapiens | AVP | - | chim(NtGi1-Gs)/β1/γ2 | 2.6 | 2021-07-21 | 10.1038/s41422-021-00480-2 | |
7DW9 (No Gprot) | A | Peptide | Vasopressin and Oxytocin | V2 | Homo sapiens | AVP | - | 2.6 | 2021-07-21 | 10.1038/s41422-021-00480-2 | ||
7F1T | A | Protein | Chemokine | CCR5 | Homo sapiens | MIP-1a | - | - | 2.6 | 2021-07-14 | 10.1038/s41467-021-24438-5 | |
7F1S | A | Protein | Chemokine | CCR5 | Homo sapiens | - | - | Gi1/β1/γ2 | 2.8 | 2021-07-14 | 10.1038/s41467-021-24438-5 | |
7F1S (No Gprot) | A | Protein | Chemokine | CCR5 | Homo sapiens | - | - | 2.8 | 2021-07-14 | 10.1038/s41467-021-24438-5 | ||
7F1R | A | Protein | Chemokine | CCR5 | Homo sapiens | - | - | Gi1/β1/γ2 | 3 | 2021-07-14 | 10.1038/s41467-021-24438-5 | |
7F1R (No Gprot) | A | Protein | Chemokine | CCR5 | Homo sapiens | - | - | 3 | 2021-07-14 | 10.1038/s41467-021-24438-5 | ||
7F1Q | A | Protein | Chemokine | CCR5 | Homo sapiens | MIP-1a | - | Gi1/β1/γ2 | 2.9 | 2021-07-14 | 10.1038/s41467-021-24438-5 | |
7F1Q (No Gprot) | A | Protein | Chemokine | CCR5 | Homo sapiens | MIP-1a | - | 2.9 | 2021-07-14 | 10.1038/s41467-021-24438-5 | ||
7DUQ | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | GLP-1 | PubChem 156022738 | Gs/β1/γ2 | 2.5 | 2021-07-14 | 10.1038/s41467-021-24058-z | |
7DUQ (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | GLP-1 | PubChem 156022738 | 2.5 | 2021-07-14 | 10.1038/s41467-021-24058-z | ||
7MTR | C | Aminoacid | Metabotropic Glutamate | mGlu2; mGlu2 | Homo sapiens | Glutamate | ADX55164 | - | 3.3 | 2021-07-07 | 10.1038/s41586-021-03680-3 | |
7MTQ | C | Aminoacid | Metabotropic Glutamate | mGlu2; mGlu2 | Homo sapiens | LY341495 | - | - | 3.65 | 2021-07-07 | 10.1038/s41586-021-03680-3 | |
7JHJ | A | Other | Unclassified | BILF1 | Human gammaherpesvirus 4 | - | - | Gi1/β1/γ2 | 3.2 | 2021-07-07 | 10.1016/j.immuni.2021.06.001 | |
7JHJ (No Gprot) | A | Other | Unclassified | BILF1 | Human gammaherpesvirus 4 | - | - | 3.2 | 2021-07-07 | 10.1016/j.immuni.2021.06.001 | ||
7MTS | C | Aminoacid | Metabotropic Glutamate | mGlu2; mGlu2 | Homo sapiens | Glutamate | ADX55164 | Gi1/β1/γ2 | 3.2 | 2021-07-07 | 10.1038/s41586-021-03680-3 | |
7MTS (No Gprot) | C | Aminoacid | Metabotropic Glutamate | mGlu2; mGlu2 | Homo sapiens | Glutamate | ADX55164 | 3.2 | 2021-07-07 | 10.1038/s41586-021-03680-3 | ||
7MTB | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | GRK1 | 4 | 2021-07-07 | 10.1038/s41586-021-03721-x | |
7MTB (No Gprot) | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | 4 | 2021-07-07 | 10.1038/s41586-021-03721-x | ||
7MTA | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | GRK1 | 4.1 | 2021-07-07 | 10.1038/s41586-021-03721-x | |
7MTA (No Gprot) | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | 4.1 | 2021-07-07 | 10.1038/s41586-021-03721-x | ||
7MT9 | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | GRK1 | 7 | 2021-07-07 | 10.1038/s41586-021-03721-x | |
7MT9 (No Gprot) | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | 7 | 2021-07-07 | 10.1038/s41586-021-03721-x | ||
7MT8 | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | GRK1 | 5.8 | 2021-07-07 | 10.1038/s41586-021-03721-x | |
7MT8 (No Gprot) | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | 5.8 | 2021-07-07 | 10.1038/s41586-021-03721-x | ||
7E14 | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Orforglipron | PubChem 156022738 | Gs/β1/γ2 | 2.9 | 2021-07-07 | 10.1038/s41467-021-24058-z | |
7E14 (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Orforglipron | PubChem 156022738 | 2.9 | 2021-07-07 | 10.1038/s41467-021-24058-z | ||
7M3J | C | Ion | Calcium Sensing | CaS | Homo sapiens | - | NPS-2143; PO4 | - | 4.1 | 2021-06-30 | 10.1038/s41586-021-03691-0 | |
7M3G | C | Ion | Calcium Sensing | CaS | Homo sapiens | - | Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4 | - | 2.5 | 2021-06-30 | 10.1038/s41586-021-03691-0 | |
7M3F | C | Ion | Calcium Sensing | CaS | Homo sapiens | - | Ca; Ca; Tryptophan; Cinacalcet; PO4 | - | 2.8 | 2021-06-30 | 10.1038/s41586-021-03691-0 | |
7M3E | C | Ion | Calcium Sensing | CaS | Homo sapiens | - | Ca; Ca; Tryptophan; NPS-2143 | - | 3.2 | 2021-06-30 | 10.1038/s41586-021-03691-0 | |
7O7F | A | Protein | Chemokine | CCR5 | Homo sapiens | 6P4-CCL5 | - | Gi1/β1/γ1 | 3.15 | 2021-06-30 | 10.1126/sciadv.abg8685 | |
7O7F (No Gprot) | A | Protein | Chemokine | CCR5 | Homo sapiens | 6P4-CCL5 | - | 3.15 | 2021-06-30 | 10.1126/sciadv.abg8685 | ||
7EPF | C | Aminoacid | Metabotropic Glutamate | mGlu2; mGlu2 | Homo sapiens | - | NAM597 | - | 2.7 | 2021-06-23 | 10.1038/s41586-021-03641-w | |
7EPE | C | Aminoacid | Metabotropic Glutamate | mGlu2; mGlu2 | Homo sapiens | - | NAM563 | - | 2.5 | 2021-06-23 | 10.1038/s41586-021-03641-w | |
7EPB | C | Aminoacid | Metabotropic Glutamate | mGlu2; mGlu2 | Homo sapiens | Eglumetad | - | - | 3.1 | 2021-06-23 | 10.1038/s41586-021-03641-w | |
7EPA | C | Aminoacid | Metabotropic Glutamate | mGlu2; mGlu2 | Homo sapiens | - | - | - | 3.6 | 2021-06-23 | 10.1038/s41586-021-03641-w | |
7EPD | C | Aminoacid | Metabotropic Glutamate | mGlu2, mGlu7 | Homo sapiens | - | - | - | 3.9 | 2021-06-23 | 10.1038/s41586-021-03641-w | |
7EPC | C | Aminoacid | Metabotropic Glutamate | mGlu7; mGlu7 | Homo sapiens | - | - | - | 4 | 2021-06-23 | 10.1038/s41586-021-03641-w | |
7E9G | C | Aminoacid | Metabotropic Glutamate | mGlu2; mGlu2 | Homo sapiens | Eglumetad | JNJ-40411813 | Gi1/β1/γ2 | 3.5 | 2021-06-23 | 10.1038/s41586-021-03495-2 | |
7E9G (No Gprot) | C | Aminoacid | Metabotropic Glutamate | mGlu2; mGlu2 | Homo sapiens | Eglumetad | JNJ-40411813 | 3.5 | 2021-06-23 | 10.1038/s41586-021-03495-2 | ||
7E9H | C | Aminoacid | Metabotropic Glutamate | mGlu4; mGlu4 | Homo sapiens | Phosphoserine | - | Gi3/β1/γ2 | 4 | 2021-06-23 | 10.1038/s41586-021-03495-2 | |
7E9H (No Gprot) | C | Aminoacid | Metabotropic Glutamate | mGlu4; mGlu4 | Homo sapiens | Phosphoserine | - | 4 | 2021-06-23 | 10.1038/s41586-021-03495-2 | ||
7DD7 | C | Ion | Calcium Sensing | CaS | Gallus gallus | Ca | Ca; Ca; Tryptophan; Evocalcet | - | 3.2 | 2021-06-16 | 10.1126/sciadv.abg1483 | |
7DD6 | C | Ion | Calcium Sensing | CaS | Gallus gallus | Ca | Ca; Ca; Tryptophan | - | 3.2 | 2021-06-16 | 10.1126/sciadv.abg1483 | |
7DD5 | C | Ion | Calcium Sensing | CaS | Gallus gallus | Ca | Ca; Ca; Tryptophan; NPS-2143 | - | 3.2 | 2021-06-16 | 10.1126/sciadv.abg1483 | |
7C4S | A | Lipid | Lysophospholipid | S1P3 | Homo sapiens | S1P | - | - | 3.2 | 2021-06-09 | 10.1126/sciadv.abf5325 | |
7BB7 | A | Peptide | Vasopressin and Oxytocin | V2 | Homo sapiens | AVP | - | Gs/β1/γ2 | 4.4 | 2021-06-02 | 10.1126/sciadv.abg5628 | |
7BB7 (No Gprot) | A | Peptide | Vasopressin and Oxytocin | V2 | Homo sapiens | AVP | - | 4.4 | 2021-06-02 | 10.1126/sciadv.abg5628 | ||
7BB6 | A | Peptide | Vasopressin and Oxytocin | V2 | Homo sapiens | AVP | - | Gs/β1/γ2 | 4.2 | 2021-06-02 | 10.1126/sciadv.abg5628 | |
7BB6 (No Gprot) | A | Peptide | Vasopressin and Oxytocin | V2 | Homo sapiens | AVP | - | 4.2 | 2021-06-02 | 10.1126/sciadv.abg5628 | ||
7KH0 | A | Peptide | Vasopressin and Oxytocin | V2 | Homo sapiens | AVP | - | chim(NtGi1-Gs)/β1/γ2 | 2.8 | 2021-05-26 | 10.1038/s41422-021-00483-z | |
7KH0 (No Gprot) | A | Peptide | Vasopressin and Oxytocin | V2 | Homo sapiens | AVP | - | 2.8 | 2021-05-26 | 10.1038/s41422-021-00483-z | ||
7MBY | A | Peptide | Cholecystokinin | CCKA | Homo sapiens | Cholecystokinin-8 | - | chim(NtGi1L-Gs-CtGq)/β1/γ2 | 2.44 | 2021-05-26 | 10.1371/journal.pbio.3001295 | |
7MBY (No Gprot) | A | Peptide | Cholecystokinin | CCKA | Homo sapiens | Cholecystokinin-8 | - | 2.44 | 2021-05-26 | 10.1371/journal.pbio.3001295 | ||
7MBX | A | Peptide | Cholecystokinin | CCKA | Homo sapiens | Cholecystokinin-8 | - | Gs/β1/γ1 | 1.95 | 2021-05-26 | 10.1371/journal.pbio.3001295 | |
7MBX (No Gprot) | A | Peptide | Cholecystokinin | CCKA | Homo sapiens | Cholecystokinin-8 | - | 1.95 | 2021-05-26 | 10.1371/journal.pbio.3001295 | ||
7EB2 | C | Aminoacid | GABAB | GABAB2; GABAB1 | Homo sapiens | Baclofen | rac-BHFF | Gi1/β1/γ2 | 3.5 | 2021-05-05 | 10.1038/s41586-021-03507-1 | |
7EB2 (No Gprot) | C | Aminoacid | GABAB | GABAB2; GABAB1 | Homo sapiens | Baclofen | rac-BHFF | 3.5 | 2021-05-05 | 10.1038/s41586-021-03507-1 | ||
7CX4 | A | Lipid | Prostanoid | EP2 | Homo sapiens | Evatanepag | - | Gs/β1/γ2 | 2.9 | 2021-05-05 | 10.1126/sciadv.abf1268 | |
7CX4 (No Gprot) | A | Lipid | Prostanoid | EP2 | Homo sapiens | Evatanepag | - | 2.9 | 2021-05-05 | 10.1126/sciadv.abf1268 | ||
7CX3 | A | Lipid | Prostanoid | EP2 | Homo sapiens | Taprenepag | - | Gs/β1/γ2 | 2.8 | 2021-05-05 | 10.1126/sciadv.abf1268 | |
7CX3 (No Gprot) | A | Lipid | Prostanoid | EP2 | Homo sapiens | Taprenepag | - | 2.8 | 2021-05-05 | 10.1126/sciadv.abf1268 | ||
7CX2 | A | Lipid | Prostanoid | EP2 | Homo sapiens | PGE2 | - | Gs/β1/γ2 | 2.8 | 2021-05-05 | 10.1126/sciadv.abf1268 | |
7CX2 (No Gprot) | A | Lipid | Prostanoid | EP2 | Homo sapiens | PGE2 | - | 2.8 | 2021-05-05 | 10.1126/sciadv.abf1268 | ||
7AUE | A | Peptide | Melanocortin | MC4 | Homo sapiens | Setmelanotide | - | chim(NtGi1L-Gs)/β1/γ2 | 2.97 | 2021-04-28 | 10.1126/science.abf7958 | |
7AUE (No Gprot) | A | Peptide | Melanocortin | MC4 | Homo sapiens | Setmelanotide | - | 2.97 | 2021-04-28 | 10.1126/science.abf7958 | ||
7E32 | A | Amine | 5-Hydroxytryptamine | 5-HT1D | Homo sapiens | Serotonin | - | Gi1/β1/γ2 | 2.9 | 2021-04-21 | 10.1038/s41586-021-03376-8 | |
7E32 (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT1D | Homo sapiens | Serotonin | - | 2.9 | 2021-04-21 | 10.1038/s41586-021-03376-8 | ||
7E2Z | A | Amine | 5-Hydroxytryptamine | 5-HT1A | Homo sapiens | Aripiprazole | - | Gi1/β1/γ2 | 3.1 | 2021-04-14 | 10.1038/s41586-021-03376-8 | |
7E2Z (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT1A | Homo sapiens | Aripiprazole | - | 3.1 | 2021-04-14 | 10.1038/s41586-021-03376-8 | ||
7E2Y | A | Amine | 5-Hydroxytryptamine | 5-HT1A | Homo sapiens | Serotonin | - | Gi1/β1/γ2 | 3 | 2021-04-14 | 10.1038/s41586-021-03376-8 | |
7E2Y (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT1A | Homo sapiens | Serotonin | - | 3 | 2021-04-14 | 10.1038/s41586-021-03376-8 | ||
7E2X | A | Amine | 5-Hydroxytryptamine | 5-HT1A | Homo sapiens | - | - | Gi1/β1/γ2 | 3 | 2021-04-14 | 10.1038/s41586-021-03376-8 | |
7E2X (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT1A | Homo sapiens | - | - | 3 | 2021-04-14 | 10.1038/s41586-021-03376-8 | ||
7E33 | A | Amine | 5-Hydroxytryptamine | 5-HT1E | Homo sapiens | BRL-54443 | - | Gi1/β1/γ2 | 2.9 | 2021-04-14 | 10.1038/s41586-021-03376-8 | |
7E33 (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT1E | Homo sapiens | BRL-54443 | - | 2.9 | 2021-04-14 | 10.1038/s41586-021-03376-8 | ||
7JOZ | A | Amine | Dopamine | D1 | Homo sapiens | VFP | - | Gs/β1/γ2 | 3.8 | 2021-04-14 | 10.1038/s41467-021-23519-9 | |
7JOZ (No Gprot) | A | Amine | Dopamine | D1 | Homo sapiens | VFP | - | 3.8 | 2021-04-14 | 10.1038/s41467-021-23519-9 | ||
7ARO | A | Nucleotide | Adenosine | A2A | Homo sapiens | LUF5833 | Na | - | 3.12 | 2021-04-07 | 10.1021/acs.jmedchem.0c01856 | |
7DFL | A | Amine | Histamine | H1 | Homo sapiens | Histamine | - | chim(NtGi1L-Gq)/β1/γ2 | 3.3 | 2021-03-31 | 10.1038/s41467-021-22427-2 | |
7DFL (No Gprot) | A | Amine | Histamine | H1 | Homo sapiens | Histamine | - | 3.3 | 2021-03-31 | 10.1038/s41467-021-22427-2 | ||
7DTW | C | Ion | Calcium Sensing | CaS | Homo sapiens | - | - | - | 4.5 | 2021-03-10 | 10.1038/s41422-021-00474-0 | |
7DTV | C | Ion | Calcium Sensing | CaS | Homo sapiens | Ca | Ca; Tryptophan | - | 3.5 | 2021-03-10 | 10.1038/s41422-021-00474-0 | |
7DTU | C | Ion | Calcium Sensing | CaS | Homo sapiens | - | Tryptophan | - | 4.4 | 2021-03-10 | 10.1038/s41422-021-00474-0 | |
7DTT | C | Ion | Calcium Sensing | CaS | Homo sapiens | Ca | Ca | - | 3.8 | 2021-03-10 | 10.1038/s41422-021-00474-0 | |
7CMV | A | Amine | Dopamine | D3 | Homo sapiens | PD128907 | - | Gi1/β1/γ2 | 2.7 | 2021-03-10 | 10.1016/j.molcel.2021.01.003 | |
7CMV (No Gprot) | A | Amine | Dopamine | D3 | Homo sapiens | PD128907 | - | 2.7 | 2021-03-10 | 10.1016/j.molcel.2021.01.003 | ||
7CMU | A | Amine | Dopamine | D3 | Homo sapiens | Pramipexole | - | Gi1/β1/γ2 | 3 | 2021-03-10 | 10.1016/j.molcel.2021.01.003 | |
7CMU (No Gprot) | A | Amine | Dopamine | D3 | Homo sapiens | Pramipexole | - | 3 | 2021-03-10 | 10.1016/j.molcel.2021.01.003 | ||
7LJD | A | Amine | Dopamine | D1 | Homo sapiens | Dopamine | Mevidalen | Gs/β1/γ1 | 3.2 | 2021-03-03 | 10.1038/s41422-021-00482-0 | |
7LJD (No Gprot) | A | Amine | Dopamine | D1 | Homo sapiens | Dopamine | Mevidalen | 3.2 | 2021-03-03 | 10.1038/s41422-021-00482-0 | ||
7LJC | A | Amine | Dopamine | D1 | Homo sapiens | SKF-81297 | Mevidalen | Gs/β1/γ2 | 3 | 2021-03-03 | 10.1038/s41422-021-00482-0 | |
7LJC (No Gprot) | A | Amine | Dopamine | D1 | Homo sapiens | SKF-81297 | Mevidalen | 3 | 2021-03-03 | 10.1038/s41422-021-00482-0 | ||
7CRH | A | Amine | Dopamine | D1 | Homo sapiens | SKF83959 | - | Gs/β1/γ2 | 3.3 | 2021-03-03 | 10.1016/j.cell.2021.01.028 | |
7CRH (No Gprot) | A | Amine | Dopamine | D1 | Homo sapiens | SKF83959 | - | 3.3 | 2021-03-03 | 10.1016/j.cell.2021.01.028 | ||
7CKZ | A | Amine | Dopamine | D1 | Homo sapiens | Dopamine | Mevidalen | Gs/β1/γ2 | 3.1 | 2021-03-03 | 10.1016/j.cell.2021.01.028 | |
7CKZ (No Gprot) | A | Amine | Dopamine | D1 | Homo sapiens | Dopamine | Mevidalen | 3.1 | 2021-03-03 | 10.1016/j.cell.2021.01.028 | ||
7CKY | A | Amine | Dopamine | D1 | Homo sapiens | PW0464 | - | Gs/β1/γ2 | 3.2 | 2021-03-03 | 10.1016/j.cell.2021.01.028 | |
7CKY (No Gprot) | A | Amine | Dopamine | D1 | Homo sapiens | PW0464 | - | 3.2 | 2021-03-03 | 10.1016/j.cell.2021.01.028 | ||
7CKX | A | Amine | Dopamine | D1 | Homo sapiens | A77636 | - | Gs/β1/γ2 | 3.54 | 2021-03-03 | 10.1016/j.cell.2021.01.028 | |
7CKX (No Gprot) | A | Amine | Dopamine | D1 | Homo sapiens | A77636 | - | 3.54 | 2021-03-03 | 10.1016/j.cell.2021.01.028 | ||
7CKW | A | Amine | Dopamine | D1 | Homo sapiens | Fenoldopam | - | Gs/β1/γ2 | 3.22 | 2021-03-03 | 10.1016/j.cell.2021.01.028 | |
7CKW (No Gprot) | A | Amine | Dopamine | D1 | Homo sapiens | Fenoldopam | - | 3.22 | 2021-03-03 | 10.1016/j.cell.2021.01.028 | ||
7JVR | A | Amine | Dopamine | D2 | Homo sapiens | Bromoergocryptine | - | Gi1/β1/γ2 | 2.8 | 2021-02-24 | 10.1016/j.cell.2021.01.027 | |
7JVR (No Gprot) | A | Amine | Dopamine | D2 | Homo sapiens | Bromoergocryptine | - | 2.8 | 2021-02-24 | 10.1016/j.cell.2021.01.027 | ||
7JVQ | A | Amine | Dopamine | D1 | Homo sapiens | Apomorphine | - | Gs/β1/γ2 | 3 | 2021-02-24 | 10.1016/j.cell.2021.01.027 | |
7JVQ (No Gprot) | A | Amine | Dopamine | D1 | Homo sapiens | Apomorphine | - | 3 | 2021-02-24 | 10.1016/j.cell.2021.01.027 | ||
7JVP | A | Amine | Dopamine | D1 | Homo sapiens | SKF83959 | - | Gs/β1/γ2 | 2.9 | 2021-02-24 | 10.1016/j.cell.2021.01.027 | |
7JVP (No Gprot) | A | Amine | Dopamine | D1 | Homo sapiens | SKF83959 | - | 2.9 | 2021-02-24 | 10.1016/j.cell.2021.01.027 | ||
7JV5 | A | Amine | Dopamine | D1 | Homo sapiens | SKF81297 | - | Gs/β1/γ2 | 3 | 2021-02-24 | 10.1016/j.cell.2021.01.027 | |
7JV5 (No Gprot) | A | Amine | Dopamine | D1 | Homo sapiens | SKF81297 | - | 3 | 2021-02-24 | 10.1016/j.cell.2021.01.027 | ||
7KNU | B1 | Peptide | Calcitonin | CT Like | Homo sapiens | Calcitonin gene-related peptide-1 | - | RAMP1 | 3.49 | 2021-02-24 | 10.1126/science.abf7258 | |
7KNT | B1 | Peptide | Calcitonin | CT Like | Homo sapiens | - | - | RAMP1 | 3.15 | 2021-02-24 | 10.1126/science.abf7258 | |
7K15 | A | Lipid | Leukotriene | BLT1 | Homo sapiens | MKD046 | Na | - | 2.88 | 2021-02-17 | 10.1038/s41467-021-23149-1 | |
6ZIN | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | SR48692 | - | - | 2.64 | 2021-02-10 | 10.1126/sciadv.abe5504 | |
6ZA8 | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | RTI-3a | - | - | 2.72 | 2021-02-10 | 10.1126/sciadv.abe5504 | |
6Z8N | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | SRI-9829 | - | - | 2.8 | 2021-02-10 | 10.1126/sciadv.abe5504 | |
6Z66 | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | - | - | - | 3.19 | 2021-02-10 | 10.1126/sciadv.abe5504 | |
6Z4V | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | NTS8-13 | - | - | 2.6 | 2021-02-10 | 10.1126/sciadv.abe5504 | |
6Z4S | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | SR48692 | - | - | 2.71 | 2021-02-10 | 10.1126/sciadv.abe5504 | |
6Z4Q | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | SR142948A | - | - | 2.92 | 2021-02-10 | 10.1126/sciadv.abe5504 | |
6YVR | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | NTS8-13 | - | - | 2.46 | 2021-02-10 | 10.1126/sciadv.abe5504 | |
7L1V | A | Peptide | Orexin | OX2 | Homo sapiens | PubChem 155491009 | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3 | 2021-02-10 | 10.1038/s41467-021-21087-6 | |
7L1V (No Gprot) | A | Peptide | Orexin | OX2 | Homo sapiens | PubChem 155491009 | - | 3 | 2021-02-10 | 10.1038/s41467-021-21087-6 | ||
7L1U | A | Peptide | Orexin | OX2 | Homo sapiens | Orexin | - | chim(NtGi1-Gs-CtGq)/β1/γ2 | 3.2 | 2021-02-10 | 10.1038/s41467-021-21087-6 | |
7L1U (No Gprot) | A | Peptide | Orexin | OX2 | Homo sapiens | Orexin | - | 3.2 | 2021-02-10 | 10.1038/s41467-021-21087-6 | ||
7D77 | B2 | Adhesion | Adhesion | ADGRG3 | Homo sapiens | Hydrocortisone | - | Go/β1/γ2 | 2.9 | 2021-02-03 | 10.1038/s41586-020-03083-w | |
7D77 (No Gprot) | B2 | Adhesion | Adhesion | ADGRG3 | Homo sapiens | Hydrocortisone | - | 2.9 | 2021-02-03 | 10.1038/s41586-020-03083-w | ||
7D76 | B2 | Adhesion | Adhesion | ADGRG3 | Homo sapiens | Beclomethasone | - | Go/β1/γ2 | 3.1 | 2021-02-03 | 10.1038/s41586-020-03083-w | |
7D76 (No Gprot) | B2 | Adhesion | Adhesion | ADGRG3 | Homo sapiens | Beclomethasone | - | 3.1 | 2021-02-03 | 10.1038/s41586-020-03083-w | ||
7DDZ | A | Peptide | Neuropeptide Y | Y2 | Homo sapiens | JNJ-31020028 | - | - | 2.8 | 2021-01-27 | 10.1038/s41467-021-21030-9 | |
7LCK | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Danuglipron | - | - | 3.24 | 2021-01-20 | 10.1016/j.str.2021.04.008 | |
7LCJ | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Danuglipron | - | - | 2.82 | 2021-01-20 | 10.1016/j.str.2021.04.008 | |
7LCI | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Danuglipron | - | Gs/β1/γ2 | 2.9 | 2021-01-20 | 10.1016/j.str.2021.04.008 | |
7LCI (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Danuglipron | - | 2.9 | 2021-01-20 | 10.1016/j.str.2021.04.008 | ||
7L0S | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | Neurotensin | - | Gi1/β1/γ1 | 4.5 | 2021-01-06 | 10.1038/s41594-020-00554-6 | |
7L0S (No Gprot) | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | Neurotensin | - | 4.5 | 2021-01-06 | 10.1038/s41594-020-00554-6 | ||
7L0R | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | Neurotensin | - | Gi1/β1/γ1 | 4.2 | 2021-01-06 | 10.1038/s41594-020-00554-6 | |
7L0R (No Gprot) | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | Neurotensin | - | 4.2 | 2021-01-06 | 10.1038/s41594-020-00554-6 | ||
7L0Q | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | Neurotensin | - | Gi1/β1/γ1 | 4.3 | 2021-01-06 | 10.1038/s41594-020-00554-6 | |
7L0Q (No Gprot) | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | Neurotensin | - | 4.3 | 2021-01-06 | 10.1038/s41594-020-00554-6 | ||
7L0P | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | Neurotensin | - | Gi1/β1/γ1 | 4.1 | 2021-01-06 | 10.1038/s41594-020-00554-6 | |
7L0P (No Gprot) | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | Neurotensin | - | 4.1 | 2021-01-06 | 10.1038/s41594-020-00554-6 | ||
7DFP | A | Amine | Dopamine | D2 | Homo sapiens | Spiperone | - | - | 3.1 | 2020-12-30 | 10.1038/s41467-020-20221-0 | |
7DHR | A | Amine | Adrenergic | β2 | Homo sapiens | Isoprenaline | - | Gs/β1/γ2 | 3.8 | 2020-12-16 | 10.1093/nsr/nwaa284 | |
7DHR (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Isoprenaline | - | 3.8 | 2020-12-16 | 10.1093/nsr/nwaa284 | ||
7DHI | A | Amine | Adrenergic | β2 | Homo sapiens | Salbutamol | - | Gs/β1/γ2 | 3.26 | 2020-12-16 | 10.1093/nsr/nwaa284 | |
7DHI (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Salbutamol | - | 3.26 | 2020-12-16 | 10.1093/nsr/nwaa284 | ||
7D68 | B1 | Peptide | Glucagon | GLP-2 | Homo sapiens | GLP-2 | - | Gs/β1/γ2 | 3 | 2020-12-16 | 10.1038/s41422-020-00442-0 | |
7D68 (No Gprot) | B1 | Peptide | Glucagon | GLP-2 | Homo sapiens | GLP-2 | - | 3 | 2020-12-16 | 10.1038/s41422-020-00442-0 | ||
7AD3 | D1 | Ste2-like | STE2 | STE2 | Saccharomyces cerevisiae | α-factor mating pheromone | - | Gi1/STE4/γ2 | 3.3 | 2020-12-09 | 10.1038/s41586-020-2994-1 | |
7AD3 (No Gprot) | D1 | Ste2-like | STE2 | STE2 | Saccharomyces cerevisiae | α-factor mating pheromone | - | 3.3 | 2020-12-09 | 10.1038/s41586-020-2994-1 | ||
7BVQ | A | Amine | Adrenergic | β1 | Homo sapiens | S-Carazolol | - | - | 2.5 | 2020-12-02 | 10.1038/s41422-020-00424-2 | |
7BU7 | A | Amine | Adrenergic | β1 | Homo sapiens | BI167107 | - | - | 2.6 | 2020-12-02 | 10.1038/s41422-020-00424-2 | |
7BU6 | A | Amine | Adrenergic | β1 | Homo sapiens | L-Norepinephrine | - | - | 2.7 | 2020-12-02 | 10.1038/s41422-020-00424-2 | |
7BTS | A | Amine | Adrenergic | β1 | Homo sapiens | L-Epinephrine | - | - | 3.13 | 2020-12-02 | 10.1038/s41422-020-00424-2 | |
6LPL | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | Na | - | 2 | 2020-11-25 | 10.1038/s41598-020-76277-x | |
6LPK | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | Na | - | 1.8 | 2020-11-25 | 10.1038/s41598-020-76277-x | |
6LPJ | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | Na | - | 1.8 | 2020-11-25 | 10.1038/s41598-020-76277-x | |
6WQA | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | Na | - | 2 | 2020-11-18 | 10.1107/S2052252520012701 | |
6XOX | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Orforglipron | - | chim(NtGi1-Gs)/β1/γ2 | 3.1 | 2020-11-18 | 10.1073/pnas.2014879117 | |
6XOX (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Orforglipron | - | 3.1 | 2020-11-18 | 10.1073/pnas.2014879117 | ||
7D7M | A | Lipid | Prostanoid | EP4 | Homo sapiens | Dinoprostone | - | Gs/β1/γ1 | 3.3 | 2020-11-18 | 10.1016/j.str.2020.11.007 | |
7D7M (No Gprot) | A | Lipid | Prostanoid | EP4 | Homo sapiens | Dinoprostone | - | 3.3 | 2020-11-18 | 10.1016/j.str.2020.11.007 | ||
7CZ5 | B1 | Peptide | Glucagon | GHRH | Homo sapiens | Somatoliberin | - | Gs/β1/γ2 | 2.6 | 2020-11-18 | 10.1038/s41467-020-18945-0 | |
7CZ5 (No Gprot) | B1 | Peptide | Glucagon | GHRH | Homo sapiens | Somatoliberin | - | 2.6 | 2020-11-18 | 10.1038/s41467-020-18945-0 | ||
7CUM | C | Aminoacid | GABAB | GABAB1, GABAB2 | Homo sapiens | CGP54626 | Phospholipid | - | 3.52 | 2020-11-11 | 10.1016/j.jmb.2020.09.023 | |
7CA5 | C | Aminoacid | GABAB | GABAB1, GABAB2 | Homo sapiens | - | - | - | 7.6 | 2020-11-11 | 10.1016/j.jmb.2020.09.023 | |
7CA3 | C | Aminoacid | GABAB | GABAB1, GABAB2 | Homo sapiens | - | rac-BHFF | - | 4.5 | 2020-11-11 | 10.1016/j.jmb.2020.09.023 | |
7D3S | B1 | Peptide | Glucagon | Secretin | Homo sapiens | Secretin | - | Gs/β1/γ2 | 2.9 | 2020-11-04 | 10.1016/j.bbrc.2020.08.042 | |
7D3S (No Gprot) | B1 | Peptide | Glucagon | Secretin | Homo sapiens | Secretin | - | 2.9 | 2020-11-04 | 10.1016/j.bbrc.2020.08.042 | ||
7BR3 | A | Peptide | Gonadotrophin Releasing Hormone | GnRH1 | Homo sapiens | Elagolix | - | - | 2.79 | 2020-10-07 | 10.1038/s41467-020-19109-w | |
6XBM | F | Protein | Frizzled | SMO | Homo sapiens | - | 25(S)-Epoxycholesterol | Gi1/β1/γ2 | 3.14 | 2020-09-30 | 10.1038/s41589-020-0646-2 | |
6XBM (No Gprot) | F | Protein | Frizzled | SMO | Homo sapiens | - | 25(S)-Epoxycholesterol | 3.14 | 2020-09-30 | 10.1038/s41589-020-0646-2 | ||
6XBL | F | Protein | Frizzled | SMO | Homo sapiens | SAG | Cholesterol | Gi1/β1/γ2 | 3.96 | 2020-09-30 | 10.1038/s41589-020-0646-2 | |
6XBL (No Gprot) | F | Protein | Frizzled | SMO | Homo sapiens | SAG | Cholesterol | 3.96 | 2020-09-30 | 10.1038/s41589-020-0646-2 | ||
6XBK | F | Protein | Frizzled | SMO | Homo sapiens | - | Cholesterol | Gi1/β1/γ2 | 3.24 | 2020-09-30 | 10.1038/s41589-020-0646-2 | |
6XBK (No Gprot) | F | Protein | Frizzled | SMO | Homo sapiens | - | Cholesterol | 3.24 | 2020-09-30 | 10.1038/s41589-020-0646-2 | ||
6XBJ | F | Protein | Frizzled | SMO | Homo sapiens | - | Cholesterol | Gi1/β1/γ2 | 3.88 | 2020-09-30 | 10.1038/s41589-020-0646-2 | |
6XBJ (No Gprot) | F | Protein | Frizzled | SMO | Homo sapiens | - | Cholesterol | 3.88 | 2020-09-30 | 10.1038/s41589-020-0646-2 | ||
6WH4 | A | Amine | 5-Hydroxytryptamine | 5-HT2A | Homo sapiens | Methiothepin | - | - | 3.4 | 2020-09-23 | 10.1016/j.cell.2020.08.024 | |
6WH4 (Multimeric) | A | Amine | 5-Hydroxytryptamine | 5-HT2A | Homo sapiens | Methiothepin | - | 3.4 | 2020-09-23 | 10.1016/j.cell.2020.08.024 | ||
6WGT | A | Amine | 5-Hydroxytryptamine | 5-HT2A | Homo sapiens | LSD | - | - | 3.4 | 2020-09-23 | 10.1016/j.cell.2020.08.024 | |
6WGT (Multimeric) | A | Amine | 5-Hydroxytryptamine | 5-HT2A | Homo sapiens | LSD | - | 3.4 | 2020-09-23 | 10.1016/j.cell.2020.08.024 | ||
6WHA | A | Amine | 5-Hydroxytryptamine | 5-HT2A | Homo sapiens | DB13948 | - | chim(NtGi2L-Gs-CtGq)/β1/γ2 | 3.36 | 2020-09-23 | 10.1016/j.cell.2020.08.024 | |
6WHA (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT2A | Homo sapiens | DB13948 | - | 3.36 | 2020-09-23 | 10.1016/j.cell.2020.08.024 | ||
6ZDV | A | Nucleotide | Adenosine | A2A | Homo sapiens | Chromone 5d | Na | - | 2.13 | 2020-09-16 | 10.1002/anie.202003788 | |
6ZDR | A | Nucleotide | Adenosine | A2A | Homo sapiens | HMS1413f12 | Na | - | 1.92 | 2020-09-16 | 10.1002/anie.202003788 | |
6Z10 | A | Alicarboxylic acid | Succinate | Succinate | Rattus norvegicus | PubChem 154585554 | - | - | 2.27 | 2020-09-16 | 10.1021/acs.jmedchem.0c01020 | |
6X1A | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Danuglipron | - | Gs/β1/γ2 | 2.5 | 2020-09-09 | 10.1016/j.molcel.2020.09.020 | |
6X1A (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Danuglipron | - | 2.5 | 2020-09-09 | 10.1016/j.molcel.2020.09.020 | ||
6X19 | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | CHU-128 | - | Gs/β1/γ2 | 2.1 | 2020-09-09 | 10.1016/j.molcel.2020.09.020 | |
6X19 (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | CHU-128 | - | 2.1 | 2020-09-09 | 10.1016/j.molcel.2020.09.020 | ||
6X18 | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | GLP-1 | - | Gs/β1/γ2 | 2.1 | 2020-09-09 | 10.1016/j.molcel.2020.09.020 | |
6X18 (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | GLP-1 | - | 2.1 | 2020-09-09 | 10.1016/j.molcel.2020.09.020 | ||
7CFN | A | Steroid | Bile Acid | GPBA | Homo sapiens | INT-777 | - | Gs/β1/γ2 | 3 | 2020-09-09 | 10.1038/s41586-020-2569-1 | |
7CFN (No Gprot) | A | Steroid | Bile Acid | GPBA | Homo sapiens | INT-777 | - | 3 | 2020-09-09 | 10.1038/s41586-020-2569-1 | ||
7CFM | A | Steroid | Bile Acid | GPBA | Homo sapiens | P395 | - | Gs/β1/γ2 | 3 | 2020-09-09 | 10.1038/s41586-020-2569-1 | |
7CFM (No Gprot) | A | Steroid | Bile Acid | GPBA | Homo sapiens | P395 | - | 3 | 2020-09-09 | 10.1038/s41586-020-2569-1 | ||
6LFL | A | Protein | Chemokine | CXCR2 | Homo sapiens | - | PubChem 153466996 | - | 3.2 | 2020-09-02 | 10.1038/s41586-020-2492-5 | |
7BW0 | A | Steroid | Bile Acid | GPBA | Homo sapiens | - | - | chim(NtGi1-Gs)/β1/γ2 | 3.9 | 2020-09-02 | 10.1038/s41392-020-00262-z | |
7BW0 (No Gprot) | A | Steroid | Bile Acid | GPBA | Homo sapiens | - | - | 3.9 | 2020-09-02 | 10.1038/s41392-020-00262-z | ||
6LFO | A | Protein | Chemokine | CXCR2 | Homo sapiens | Interleukin-8 | - | Gi1/β1/γ2 | 3.4 | 2020-09-02 | 10.1038/s41586-020-2492-5 | |
6LFO (No Gprot) | A | Protein | Chemokine | CXCR2 | Homo sapiens | Interleukin-8 | - | 3.4 | 2020-09-02 | 10.1038/s41586-020-2492-5 | ||
6LFM | A | Protein | Chemokine | CXCR2 | Homo sapiens | Interleukin-8 | - | Gi1/β1/γ2 | 3.5 | 2020-09-02 | 10.1038/s41586-020-2492-5 | |
6LFM (No Gprot) | A | Protein | Chemokine | CXCR2 | Homo sapiens | Interleukin-8 | - | 3.5 | 2020-09-02 | 10.1038/s41586-020-2492-5 | ||
7JJO | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Isoprenaline | - | Gs/β1/γ2 | 2.6 | 2020-09-02 | 10.1016/j.molcel.2020.08.001 | |
7JJO (No Gprot) | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Isoprenaline | - | 2.6 | 2020-09-02 | 10.1016/j.molcel.2020.08.001 | ||
6VN7 | B1 | Peptide | VIP and PACAP | VPAC1 | Homo sapiens | PACAP | - | Gs/β1/γ2 | 3.2 | 2020-09-02 | 10.1038/s41467-020-17933-8 | |
6VN7 (No Gprot) | B1 | Peptide | VIP and PACAP | VPAC1 | Homo sapiens | PACAP | - | 3.2 | 2020-09-02 | 10.1038/s41467-020-17933-8 | ||
7C2E | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | PubChem 149050799 | - | Gs/β1/γ2 | 4.2 | 2020-08-26 | 10.1038/s41422-020-0384-8 | |
7C2E (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | PubChem 149050799 | - | 4.2 | 2020-08-26 | 10.1038/s41422-020-0384-8 | ||
6WW2 | F | Protein | Frizzled | FZD5 | Homo sapiens | - | - | - | 3.7 | 2020-08-19 | 10.7554/eLife.58464 | |
6KO5 | A | Peptide | Ghrelin | Ghrelin | Homo sapiens | PubChem 57400002 | - | - | 3.3 | 2020-08-12 | 10.1038/s41467-020-17554-1 | |
6WPW | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | Glucagon derivative ZP3780 | - | Gs/β1/γ2 | 3.1 | 2020-08-12 | 10.1126/science.aba3373 | |
6WPW (No Gprot) | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | Glucagon derivative ZP3780 | - | 3.1 | 2020-08-12 | 10.1126/science.aba3373 | ||
6WZG | B1 | Peptide | Glucagon | Secretin | Homo sapiens | Secretin | - | Gs/β1/γ2 | 2.3 | 2020-08-12 | 10.1038/s41467-020-17791-4 | |
6WZG (No Gprot) | B1 | Peptide | Glucagon | Secretin | Homo sapiens | Secretin | - | 2.3 | 2020-08-12 | 10.1038/s41467-020-17791-4 | ||
6WI9 | B1 | Peptide | Glucagon | Secretin | Homo sapiens | Secretin | - | Gs/β1/γ2 | 4.3 | 2020-08-12 | 10.1038/s41467-020-17791-4 | |
6WI9 (No Gprot) | B1 | Peptide | Glucagon | Secretin | Homo sapiens | Secretin | - | 4.3 | 2020-08-12 | 10.1038/s41467-020-17791-4 | ||
6TPK | A | Peptide | Vasopressin and Oxytocin | OT | Homo sapiens | Retosiban | - | - | 3.2 | 2020-08-05 | 10.1126/sciadv.abb5419 | |
7BZ2 | A | Amine | Adrenergic | β2 | Homo sapiens | Arformoterol | - | Gs/β1/γ2 | 3.82 | 2020-08-05 | 10.1038/s41421-020-0176-9 | |
7BZ2 (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | Arformoterol | - | 3.82 | 2020-08-05 | 10.1038/s41421-020-0176-9 | ||
7C61 | A | Amine | 5-Hydroxytryptamine | 5-HT1B | Homo sapiens | Ergotamine | - | - | 3 | 2020-07-29 | 10.1038/s41598-020-68355-x | |
7C6A | A | Peptide | Angiotensin | AT2 | Homo sapiens | (Sar1,Ile8)-Angiotensin II | - | - | 3.4 | 2020-07-29 | 10.1038/s41598-020-68355-x | |
6VCB | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | GLP-1 | LSN3160440 | Gs/β1/γ2 | 3.3 | 2020-07-22 | 10.1038/s41589-020-0589-7 | |
6VCB (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | GLP-1 | LSN3160440 | 3.3 | 2020-07-22 | 10.1038/s41589-020-0589-7 | ||
6S0Q | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | - | - | 2.65 | 2020-07-15 | 10.1107/S2052252520011379 | |
6S0L | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | - | - | 2.65 | 2020-07-15 | 10.1107/S2052252520011379 | |
6V9S | A | Peptide | Orexin | OX1 | Homo sapiens | GTPL11403 | - | - | 3.5 | 2020-07-15 | 10.1073/pnas.2002704117 | |
6WJC | A | Amine | Acetylcholine (muscarinic) | M1 | Homo sapiens | Atropine | Muscarinic toxin 7 | - | 2.55 | 2020-07-08 | 10.1126/science.aax2517 | |
6W2Y | C | Aminoacid | GABAB | GABAB1; GABAB1 | Homo sapiens | PubChem 5311042 | PubChem 23727970 | - | 3.2 | 2020-07-01 | 10.1038/s41586-020-2469-4 | |
7C7S | C | Aminoacid | GABAB | GABAB1, GABAB2 | Homo sapiens | CGP54626 | - | - | 2.9 | 2020-07-01 | 10.1038/s41422-020-0350-5 | |
7C7Q | C | Aminoacid | GABAB | GABAB1, GABAB2 | Homo sapiens | Baclofen | PubChem 7023848 | - | 3 | 2020-07-01 | 10.1038/s41422-020-0350-5 | |
6WIV | C | Aminoacid | GABAB | GABAB1, GABAB2 | Homo sapiens | - | PubChem 52923113; PubChem 52924645 | - | 3.3 | 2020-07-01 | 10.1038/s41586-020-2452-0 | |
6W2X | C | Aminoacid | GABAB | GABAB1, GABAB2 | Homo sapiens | PubChem 5311042 | PubChem 23727970 | - | 3.6 | 2020-07-01 | 10.1038/s41586-020-2469-4 | |
6PH7 | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | Nerol | Gt(CT) | 2.9 | 2020-07-01 | To be published | |
6PH7 (No Gprot) | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | Nerol | 2.9 | 2020-07-01 | To be published | ||
6PGS | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | Geraniol | Gt(CT) | 2.9 | 2020-07-01 | To be published | |
6PGS (No Gprot) | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | Geraniol | 2.9 | 2020-07-01 | To be published | ||
6WWZ | A | Protein | Chemokine | CCR6 | Homo sapiens | CCL20 | - | Go/β1/γ2 | 3.34 | 2020-06-24 | 10.1038/s41467-020-16820-6 | |
6WWZ (No Gprot) | A | Protein | Chemokine | CCR6 | Homo sapiens | CCL20 | - | 3.34 | 2020-06-24 | 10.1038/s41467-020-16820-6 | ||
6PEL | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | Citronellol | Gt(CT) | 3.19 | 2020-06-24 | To be published | |
6PEL (No Gprot) | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | Citronellol | 3.19 | 2020-06-24 | To be published | ||
6TKO | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Arformoterol | - | Arrestin2 | 3.3 | 2020-06-17 | 10.1038/s41586-020-2419-1 | |
6VMS | A | Amine | Dopamine | D2 | Homo sapiens | Bromoergocryptine | - | Gi1/β1/γ2 | 3.8 | 2020-06-17 | 10.1038/s41586-020-2379-5 | |
6VMS (No Gprot) | A | Amine | Dopamine | D2 | Homo sapiens | Bromoergocryptine | - | 3.8 | 2020-06-17 | 10.1038/s41586-020-2379-5 | ||
6VJM | C | Aminoacid | GABAB | GABAB1, GABAB2 | Homo sapiens | - | - | - | 3.97 | 2020-06-10 | 10.1038/s41586-020-2408-4 | |
6UOA | C | Aminoacid | GABAB | GABAB1, GABAB2 | Homo sapiens | - | - | - | 6.3 | 2020-06-10 | 10.1038/s41586-020-2408-4 | |
6UO9 | C | Aminoacid | GABAB | GABAB1, GABAB2 | Homo sapiens | SKF97541 | - | - | 4.8 | 2020-06-10 | 10.1038/s41586-020-2408-4 | |
6UO8 | C | Aminoacid | GABAB | GABAB1, GABAB2 | Homo sapiens | SKF97541 | GS39783 | - | 3.63 | 2020-06-10 | 10.1038/s41586-020-2408-4 | |
6WHC | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | Glu16 analog of GCG | - | Gs/β1/γ2 | 3.4 | 2020-05-27 | 10.1074/jbc.RA120.013793 | |
6WHC (No Gprot) | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | Glu16 analog of GCG | - | 3.4 | 2020-05-27 | 10.1074/jbc.RA120.013793 | ||
6W25 | A | Peptide | Melanocortin | MC4 | Homo sapiens | SHU9119 | Ca | - | 2.75 | 2020-04-29 | 10.1126/science.aaz8995 | |
6K42 | A | Amine | Adrenergic | α2b | Homo sapiens | Dexmedetomidine | - | Gi1/β1/γ2 | 4.1 | 2020-04-15 | 10.1038/s41589-020-0492-2 | |
6K42 (No Gprot) | A | Amine | Adrenergic | α2b | Homo sapiens | Dexmedetomidine | - | 4.1 | 2020-04-15 | 10.1038/s41589-020-0492-2 | ||
6K41 | A | Amine | Adrenergic | α2b | Homo sapiens | Dexmedetomidine | - | Go/β1/γ2 | 2.9 | 2020-04-15 | 10.1038/s41589-020-0492-2 | |
6K41 (No Gprot) | A | Amine | Adrenergic | α2b | Homo sapiens | Dexmedetomidine | - | 2.9 | 2020-04-15 | 10.1038/s41589-020-0492-2 | ||
6LML | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | Glucagon | - | Gi1/β1/γ1 | 3.9 | 2020-04-01 | 10.1126/science.aaz5346 | |
6LML (No Gprot) | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | Glucagon | - | 3.9 | 2020-04-01 | 10.1126/science.aaz5346 | ||
6LMK | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | Glucagon | - | Gs/β1/γ2 | 3.7 | 2020-04-01 | 10.1126/science.aaz5346 | |
6LMK (No Gprot) | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | Glucagon | - | 3.7 | 2020-04-01 | 10.1126/science.aaz5346 | ||
6UVA | B1 | Peptide | Calcitonin | CT Like (AM2) | Homo sapiens | Adrenomedullin-2 | - | Gs/β1/γ2; RAMP3 | 2.3 | 2020-04-01 | 10.1021/acsptsci.9b00080 | |
6UVA (No Gprot) | B1 | Peptide | Calcitonin | CT Like (AM2) | Homo sapiens | Adrenomedullin-2 | - | 2.3 | 2020-04-01 | 10.1021/acsptsci.9b00080 | ||
6UUS | B1 | Peptide | Calcitonin | CT Like (AM2) | Homo sapiens | Adrenomedullin | - | Gs/β1/γ2; RAMP3 | 2.4 | 2020-04-01 | 10.1021/acsptsci.9b00080 | |
6UUS (No Gprot) | B1 | Peptide | Calcitonin | CT Like (AM2) | Homo sapiens | Adrenomedullin | - | 2.4 | 2020-04-01 | 10.1021/acsptsci.9b00080 | ||
6OBA | A | Amine | Adrenergic | β2 | Homo sapiens | S-Alprenolol | GTPL11074 | - | 3.1 | 2020-03-25 | 10.1038/s41589-020-0549-2 | |
6LW5 | A | Peptide | Formylpeptide | FPR2-ALX | Homo sapiens | WKYMVm | - | - | 2.8 | 2020-03-25 | 10.1038/s41467-020-15009-1 | |
6UUN | B1 | Peptide | Calcitonin | CT Like (AM1) | Homo sapiens | Adrenomedullin | - | Gs/β1/γ2; RAMP2 | 3 | 2020-03-25 | 10.1021/acsptsci.9b00080 | |
6UUN (No Gprot) | B1 | Peptide | Calcitonin | CT Like (AM1) | Homo sapiens | Adrenomedullin | - | 3 | 2020-03-25 | 10.1021/acsptsci.9b00080 | ||
6LN2 | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | - | PubChem 68178630 | - | 3.2 | 2020-03-18 | 10.1038/s41467-020-14934-5 | |
6VI4 | A | Peptide | Opioid | κ | Homo sapiens | JDTic | - | - | 3.3 | 2020-03-18 | 10.1038/s41467-020-14889-7 | |
6KP6 | A | Amine | Acetylcholine (muscarinic) | M4 | Homo sapiens | - | - | - | 3 | 2020-03-11 | 10.1107/S2052252520000597 | |
6LPB | B1 | Peptide | VIP and PACAP | PAC1 | Homo sapiens | PACAP | - | Gs/β1/γ1 | 3.9 | 2020-03-11 | 10.1038/s41594-020-0386-8 | |
6LPB (No Gprot) | B1 | Peptide | VIP and PACAP | PAC1 | Homo sapiens | PACAP | - | 3.9 | 2020-03-11 | 10.1038/s41594-020-0386-8 | ||
6M1I | B1 | Peptide | VIP and PACAP | PAC1 | Homo sapiens | PACAP | - | Gs/β1/γ2 | 3.5 | 2020-03-11 | 10.1038/s41422-020-0280-2 | |
6M1I (No Gprot) | B1 | Peptide | VIP and PACAP | PAC1 | Homo sapiens | PACAP | - | 3.5 | 2020-03-11 | 10.1038/s41422-020-0280-2 | ||
6M1H | B1 | Peptide | VIP and PACAP | PAC1 | Homo sapiens | Maxadilan | - | Gs/β1/γ2 | 3.6 | 2020-03-11 | 10.1038/s41422-020-0280-2 | |
6M1H (No Gprot) | B1 | Peptide | VIP and PACAP | PAC1 | Homo sapiens | Maxadilan | - | 3.6 | 2020-03-11 | 10.1038/s41422-020-0280-2 | ||
6LUQ | A | Amine | Dopamine | D2 | Homo sapiens | Haloperidol | - | - | 3.1 | 2020-03-04 | 10.1038/s41467-020-14884-y | |
6LI2 | A | Orphan | Orphan | GPR52 | Homo sapiens | - | - | - | 2.8 | 2020-02-26 | 10.1038/s41586-020-2019-0 | |
6LI1 | A | Orphan | Orphan | GPR52 | Homo sapiens | - | - | - | 2.9 | 2020-02-26 | 10.1038/s41586-020-2019-0 | |
6LI0 | A | Orphan | Orphan | GPR52 | Homo sapiens | - | C17 | - | 2.2 | 2020-02-26 | 10.1038/s41586-020-2019-0 | |
6U1N | A | Amine | Acetylcholine (muscarinic) | M2 | Homo sapiens | - | LY2119620 | Arrestin2 | 4 | 2020-02-26 | 10.1038/s41586-020-1954-0 | |
6UP7 | A | Peptide | Neurotensin | NTS1 | Homo sapiens | Neurotensin | - | Arrestin2 | 4.2 | 2020-02-26 | 10.1038/s41586-020-1953-1 | |
6OMM | A | Peptide | Formylpeptide | FPR2-ALX | Homo sapiens | WKYMVX | - | Gi1/β1/γ2 | 3.17 | 2020-02-26 | 10.1038/s41467-020-14728-9 | |
6OMM (No Gprot) | A | Peptide | Formylpeptide | FPR2-ALX | Homo sapiens | WKYMVX | - | 3.17 | 2020-02-26 | 10.1038/s41467-020-14728-9 | ||
6LI3 | A | Orphan | Orphan | GPR52 | Homo sapiens | - | - | Gs/β1/γ2 | 3.32 | 2020-02-26 | 10.1038/s41586-020-2019-0 | |
6LI3 (No Gprot) | A | Orphan | Orphan | GPR52 | Homo sapiens | - | - | 3.32 | 2020-02-26 | 10.1038/s41586-020-2019-0 | ||
6OS2 | A | Peptide | Angiotensin | AT1 | Homo sapiens | TRV026 | - | - | 2.7 | 2020-02-19 | 10.1126/science.aay9813 | |
6OS1 | A | Peptide | Angiotensin | AT1 | Homo sapiens | TRV026 | - | - | 2.79 | 2020-02-19 | 10.1126/science.aay9813 | |
6OS0 | A | Peptide | Angiotensin | AT1 | Homo sapiens | Angiotensinogen | - | - | 2.9 | 2020-02-19 | 10.1126/science.aay9813 | |
6KPC | A | Lipid | Cannabinoid | CB2 | Homo sapiens | PubChem 145915889 | - | - | 3.2 | 2020-02-12 | 10.1016/j.cell.2020.01.008 | |
6LRY | A | Peptide | Endothelin | ETB | Homo sapiens | Sarafotoxin-B | - | - | 3 | 2020-02-12 | 10.1016/j.bbrc.2019.12.091 | |
6PB0 | B1 | Peptide | Corticotropin Releasing Factor | CRF1 | Homo sapiens | Urocortin | - | chim(NtGi1-Gs)/β1/γ2 | 3 | 2020-02-12 | 10.1016/j.molcel.2020.01.013 | |
6PB0 (No Gprot) | B1 | Peptide | Corticotropin Releasing Factor | CRF1 | Homo sapiens | Urocortin | - | 3 | 2020-02-12 | 10.1016/j.molcel.2020.01.013 | ||
6PB1 | B1 | Peptide | Corticotropin Releasing Factor | CRF2 | Homo sapiens | Urocortin | - | chim(NtGi1-Gs)/β1/γ2 | 2.8 | 2020-02-12 | 10.1016/j.molcel.2020.01.013 | |
6PB1 (No Gprot) | B1 | Peptide | Corticotropin Releasing Factor | CRF2 | Homo sapiens | Urocortin | - | 2.8 | 2020-02-12 | 10.1016/j.molcel.2020.01.013 | ||
6KPG | A | Lipid | Cannabinoid | CB1 | Homo sapiens | AM841 | - | Gi1/β1/γ2 | 3 | 2020-02-12 | 10.1016/j.cell.2020.01.008 | |
6KPG (No Gprot) | A | Lipid | Cannabinoid | CB1 | Homo sapiens | AM841 | - | 3 | 2020-02-12 | 10.1016/j.cell.2020.01.008 | ||
6PT0 | A | Lipid | Cannabinoid | CB2 | Homo sapiens | WIN 55212-2 | - | Gi1/β1/γ2 | 3.2 | 2020-02-12 | 10.1016/j.cell.2020.01.007 | |
6PT0 (No Gprot) | A | Lipid | Cannabinoid | CB2 | Homo sapiens | WIN 55212-2 | - | 3.2 | 2020-02-12 | 10.1016/j.cell.2020.01.007 | ||
6KPF | A | Lipid | Cannabinoid | CB2 | Homo sapiens | PubChem 145915889 | - | Gi1/β1/γ2 | 2.9 | 2020-02-12 | 10.1016/j.cell.2020.01.008 | |
6KPF (No Gprot) | A | Lipid | Cannabinoid | CB2 | Homo sapiens | PubChem 145915889 | - | 2.9 | 2020-02-12 | 10.1016/j.cell.2020.01.008 | ||
6NWE | A | Sensory | Opsins | Rhodopsin | Bos taurus | Octyl-β-D-Glucopyranoside | - | Gt(CT) | 2.71 | 2020-02-12 | To be published | |
6NWE (No Gprot) | A | Sensory | Opsins | Rhodopsin | Bos taurus | Octyl-β-D-Glucopyranoside | - | 2.71 | 2020-02-12 | To be published | ||
6P9X | B1 | Peptide | Corticotropin Releasing Factor | CRF1 | Homo sapiens | Corticoliberin | - | Gs/β1/γ2 | 2.91 | 2020-02-05 | 10.1016/j.molcel.2020.01.012 | |
6P9X (No Gprot) | B1 | Peptide | Corticotropin Releasing Factor | CRF1 | Homo sapiens | Corticoliberin | - | 2.91 | 2020-02-05 | 10.1016/j.molcel.2020.01.012 | ||
6P9Y | B1 | Peptide | VIP and PACAP | PAC1 | Homo sapiens | PACAP | - | Gs/β1/γ2 | 3.01 | 2020-02-05 | 10.1016/j.molcel.2020.01.012 | |
6P9Y (No Gprot) | B1 | Peptide | VIP and PACAP | PAC1 | Homo sapiens | PACAP | - | 3.01 | 2020-02-05 | 10.1016/j.molcel.2020.01.012 | ||
6KNM | A | Peptide | Apelin | Apelin | Homo sapiens | JN241-9 | - | - | 3.2 | 2020-01-29 | 10.1126/sciadv.aax7379 | |
6JOD | A | Peptide | Angiotensin | AT2 | Homo sapiens | Angiotensin II | - | - | 3.2 | 2020-01-15 | 10.1016/j.str.2019.12.003 | |
6TOT | A | Peptide | Orexin | OX1 | Homo sapiens | Lemborexant | - | - | 2.22 | 2020-01-15 | 10.1021/acs.jmedchem.9b01787 | |
6TOS | A | Peptide | Orexin | OX1 | Homo sapiens | GSK1059865 | Na | - | 2.13 | 2020-01-15 | 10.1021/acs.jmedchem.9b01787 | |
6ORV | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | - | TT-OAD2 | Gs/β1/γ2 | 3 | 2020-01-08 | 10.1038/s41586-019-1902-z | |
6ORV (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | - | TT-OAD2 | 3 | 2020-01-08 | 10.1038/s41586-019-1902-z | ||
6TQ9 | A | Peptide | Orexin | OX1 | Homo sapiens | SB-408124 | - | - | 2.65 | 2020-01-01 | 10.1021/acs.jmedchem.9b01787 | |
6TQ7 | A | Peptide | Orexin | OX1 | Homo sapiens | SB-334867 | - | - | 2.66 | 2020-01-01 | 10.1021/acs.jmedchem.9b01787 | |
6TQ6 | A | Peptide | Orexin | OX1 | Homo sapiens | PubChem 145714283 | - | - | 2.55 | 2020-01-01 | 10.1021/acs.jmedchem.9b01787 | |
6TQ4 | A | Peptide | Orexin | OX1 | Homo sapiens | PubChem 16046844 | Na | - | 2.3 | 2020-01-01 | 10.1021/acs.jmedchem.9b01787 | |
6TP6 | A | Peptide | Orexin | OX1 | Homo sapiens | Filorexant | - | - | 2.34 | 2020-01-01 | 10.1021/acs.jmedchem.9b01787 | |
6TP4 | A | Peptide | Orexin | OX1 | Homo sapiens | ACT-462206 | - | - | 3.01 | 2020-01-01 | 10.1021/acs.jmedchem.9b01787 | |
6TP3 | A | Peptide | Orexin | OX1 | Homo sapiens | Nemorexant | - | - | 3.04 | 2020-01-01 | 10.1021/acs.jmedchem.9b01787 | |
6TOD | A | Peptide | Orexin | OX1 | Homo sapiens | EMPA | Na | - | 2.11 | 2020-01-01 | 10.1021/acs.jmedchem.9b01787 | |
6TO7 | A | Peptide | Orexin | OX1 | Homo sapiens | Suvorexant | Na | - | 2.26 | 2020-01-01 | 10.1021/acs.jmedchem.9b01787 | |
6TPN | A | Peptide | Orexin | OX2 | Homo sapiens | HTL6641 | - | - | 2.61 | 2020-01-01 | 10.1021/acs.jmedchem.9b01787 | |
6TPJ | A | Peptide | Orexin | OX2 | Homo sapiens | Suvorexant | - | - | 2.74 | 2020-01-01 | 10.1021/acs.jmedchem.9b01787 | |
6TPG | A | Peptide | Orexin | OX2 | Homo sapiens | EMPA | - | - | 2.74 | 2020-01-01 | 10.1021/acs.jmedchem.9b01787 | |
6RZ9 | A | Lipid | Leukotriene | CysLT2 | Homo sapiens | ONO-2770372 | - | - | 2.73 | 2019-12-11 | 10.1038/s41467-019-13348-2 | |
6RZ8 | A | Lipid | Leukotriene | CysLT2 | Homo sapiens | ONO-2080365 | - | - | 2.7 | 2019-12-11 | 10.1038/s41467-019-13348-2 | |
6RZ7 | A | Lipid | Leukotriene | CysLT2 | Homo sapiens | ONO-2570366 | - | - | 2.43 | 2019-12-11 | 10.1038/s41467-019-13348-2 | |
6RZ6 | A | Lipid | Leukotriene | CysLT2 | Homo sapiens | ONO-2570366 | - | - | 2.43 | 2019-12-11 | 10.1038/s41467-019-13348-2 | |
6PT3 | A | Peptide | Opioid | δ | Homo sapiens | DPI-287 | - | - | 3.3 | 2019-12-11 | 10.1126/sciadv.aax9115 | |
6PT2 | A | Peptide | Opioid | δ | Homo sapiens | KGCHM07 | - | - | 2.8 | 2019-12-11 | 10.1126/sciadv.aax9115 | |
6OL9 | A | Amine | Acetylcholine (muscarinic) | M5 | Homo sapiens | Tiotropium | - | - | 2.54 | 2019-12-11 | 10.1073/pnas.1914446116 | |
6KUY | A | Amine | Adrenergic | α2a | Homo sapiens | PubChem 145704643 | - | - | 3.2 | 2019-12-04 | 10.1038/nature06325 | |
6KUX | A | Amine | Adrenergic | α2a | Homo sapiens | RS-79948 | - | - | 2.7 | 2019-12-04 | 10.1038/nature06325 | |
6KUW | A | Amine | Adrenergic | α2c | Homo sapiens | PubChem 57213234 | - | - | 2.8 | 2019-12-04 | 10.1038/nature06325 | |
6KUW (Multimeric) | A | Amine | Adrenergic | α2c | Homo sapiens | PubChem 57213234 | - | 2.8 | 2019-12-04 | 10.1038/nature06325 | ||
6IQL | A | Amine | Dopamine | D4 | Mus musculus | L745870 | - | - | 3.5 | 2019-12-04 | 10.7554/eLife.48822 | |
6PWC | A | Peptide | Neurotensin | NTS1 | Homo sapiens | Neurotensin | - | Arrestin2 | 4.9 | 2019-12-04 | 10.1038/s41422-019-0256-2 | |
6NI3 | A | Amine | Adrenergic | β2 | Homo sapiens | BI167107 | - | Gs/β1/γ2 | 3.8 | 2019-11-20 | 10.1038/s41594-019-0330-y | |
6NI3 (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | BI167107 | - | 3.8 | 2019-11-20 | 10.1038/s41594-019-0330-y | ||
6PS7 | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | Na | - | 1.85 | 2019-11-13 | 10.1107/S2052252519013137 | |
6PS6 | A | Amine | Adrenergic | β2 | Homo sapiens | Timolol | - | - | 2.7 | 2019-11-13 | 10.1107/S2052252519013137 | |
6PS5 | A | Amine | Adrenergic | β2 | Homo sapiens | S-Propranolol | - | - | 2.9 | 2019-11-13 | 10.1107/S2052252519013137 | |
6PS4 | A | Amine | Adrenergic | β2 | Homo sapiens | ICI118-551 | - | - | 2.6 | 2019-11-13 | 10.1107/S2052252519013137 | |
6PS3 | A | Amine | Adrenergic | β2 | Homo sapiens | S-Carvedilol | - | - | 2.5 | 2019-11-13 | 10.1107/S2052252519013137 | |
6PS2 | A | Amine | Adrenergic | β2 | Homo sapiens | S-Alprenolol | - | - | 2.4 | 2019-11-13 | 10.1107/S2052252519013137 | |
6PS1 | A | Amine | Adrenergic | β2 | Homo sapiens | Timolol | - | - | 3.2 | 2019-11-13 | 10.1107/S2052252519013137 | |
6PS0 | A | Amine | Adrenergic | β2 | Homo sapiens | S-Carazolol | - | - | 3.4 | 2019-11-13 | 10.1107/S2052252519013137 | |
6PRZ | A | Amine | Adrenergic | β2 | Homo sapiens | S-Alprenolol | - | - | 2.8 | 2019-11-13 | 10.1107/S2052252519013137 | |
6KK7 | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | - | PubChem 68178630 | - | 3.1 | 2019-11-13 | 10.1107/S2052252519013496 | |
6KK1 | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | - | PubChem 68178630 | - | 2.8 | 2019-11-13 | 10.1107/S2052252519013496 | |
6KJV | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | - | PubChem 68178630 | - | 2.8 | 2019-11-13 | 10.1107/S2052252519013496 | |
6PS8 | A | Melatonin | Melatonin | MT1 | Homo sapiens | 2-Phenylmelatonin | - | - | 3.3 | 2019-11-13 | 10.1107/S2052252519013137 | |
6JZH | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | Na | - | 2.25 | 2019-10-30 | 10.1107/S1600576719012846 | |
6RZ5 | A | Lipid | Leukotriene | CysLT1 | Homo sapiens | Zafirlukast | Na | - | 2.53 | 2019-10-30 | 10.1126/sciadv.aax2518 | |
6RZ4 | A | Lipid | Leukotriene | CysLT1 | Homo sapiens | Pranlukast | Na | - | 2.7 | 2019-10-30 | 10.1126/sciadv.aax2518 | |
6KQI | A | Lipid | Cannabinoid | CB1 | Homo sapiens | CP55940 | Org27569 | - | 3.25 | 2019-10-23 | 10.1038/s41589-019-0387-2 | |
6QZH | A | Protein | Chemokine | CCR7 | Homo sapiens | - | HY-133073; Na | - | 2.1 | 2019-09-04 | 10.1016/j.cell.2019.07.028 | |
6OFJ | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | - | - | 4.5 | 2019-08-21 | 10.1074/jbc.RA119.010089 | |
6OFJ (Multimeric) | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | - | 4.5 | 2019-08-21 | 10.1074/jbc.RA119.010089 | ||
6RNK | A | Alicarboxylic acid | Succinate | Succinate | Rattus norvegicus | NF-56-EJ40 | - | - | 1.94 | 2019-08-14 | 10.1038/s41586-019-1663-8 | |
6IBB | A | Alicarboxylic acid | Succinate | Succinate | Rattus norvegicus | - | - | - | 2.12 | 2019-08-14 | 10.1038/s41586-019-1663-8 | |
6OYA | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | Gt/β1/γ1 | 3.3 | 2019-07-24 | 10.1016/j.molcel.2019.06.007 | |
6OYA (No Gprot) | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | 3.3 | 2019-07-24 | 10.1016/j.molcel.2019.06.007 | ||
6OY9 | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | Gt/β1/γ1 | 3.9 | 2019-07-24 | 10.1016/j.molcel.2019.06.007 | |
6OY9 (No Gprot) | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | 3.9 | 2019-07-24 | 10.1016/j.molcel.2019.06.007 | ||
6K1Q | A | Peptide | Endothelin | ETB | Homo sapiens | IRL2500 | - | - | 2.7 | 2019-07-17 | 10.1038/s42003-019-0482-7 | |
6QNO | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | Gi1/β1/γ1 | 4.38 | 2019-07-10 | 10.7554/eLife.46041 | |
6QNO (No Gprot) | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | 4.38 | 2019-07-10 | 10.7554/eLife.46041 | ||
6OSA | A | Peptide | Neurotensin | NTS1 | Homo sapiens | JMV449 | - | Gi1/β1/γ2 | 3 | 2019-07-10 | 10.1038/s41586-019-1337-6 | |
6OSA (No Gprot) | A | Peptide | Neurotensin | NTS1 | Homo sapiens | JMV449 | - | 3 | 2019-07-10 | 10.1038/s41586-019-1337-6 | ||
6OS9 | A | Peptide | Neurotensin | NTS1 | Homo sapiens | JMV449 | - | Gi1/β1/γ2 | 3 | 2019-07-10 | 10.1038/s41586-019-1337-6 | |
6OS9 (No Gprot) | A | Peptide | Neurotensin | NTS1 | Homo sapiens | JMV449 | - | 3 | 2019-07-10 | 10.1038/s41586-019-1337-6 | ||
6I9K | A | Sensory | Opsins | Rhodopsin | Hasarius adansoni | 9-cis-Retinal | - | - | 2.15 | 2019-07-03 | 10.1073/pnas.1902192116 | |
6O3C | F | Protein | Frizzled | SMO | Mus musculus | SAG21k | Cholesterol | - | 2.8 | 2019-07-03 | 10.1038/s41586-019-1355-4 | |
6GT3 | A | Nucleotide | Adenosine | A2A | Homo sapiens | Imaradenant | Na | - | 2 | 2019-06-26 | 10.1136/jitc-2019-000417 | |
6N48 | A | Amine | Adrenergic | β2 | Homo sapiens | BI167107 | PubChem 138454256 | - | 3.2 | 2019-06-26 | 10.1126/science.aaw8981 | |
6OT0 | F | Protein | Frizzled | SMO | Homo sapiens | - | 25(S)-Epoxycholesterol | Gi1/β1/γ2 | 3.84 | 2019-06-12 | 10.1038/s41586-019-1286-0 | |
6OT0 (No Gprot) | F | Protein | Frizzled | SMO | Homo sapiens | - | 25(S)-Epoxycholesterol | 3.84 | 2019-06-12 | 10.1038/s41586-019-1286-0 | ||
6E67 | A | Amine | Adrenergic | β2 | Homo sapiens | BI167107 | - | Gs (fused) | 3.7 | 2019-06-05 | 10.1016/j.cell.2019.04.021 | |
6E67 (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | BI167107 | - | 3.7 | 2019-06-05 | 10.1016/j.cell.2019.04.021 | ||
6OIK | A | Amine | Acetylcholine (muscarinic) | M2 | Homo sapiens | Iperoxo | LY2119620 | chim(NtGi1-Go)/β1/γ2 | 3.6 | 2019-05-08 | 10.1126/science.aaw5188 | |
6OIK (No Gprot) | A | Amine | Acetylcholine (muscarinic) | M2 | Homo sapiens | Iperoxo | LY2119620 | 3.6 | 2019-05-08 | 10.1126/science.aaw5188 | ||
6OIJ | A | Amine | Acetylcholine (muscarinic) | M1 | Homo sapiens | Iperoxo | - | chim(NtGi1L-G11)/β1/γ2 | 3.3 | 2019-05-08 | 10.1126/science.aaw5188 | |
6OIJ (No Gprot) | A | Amine | Acetylcholine (muscarinic) | M1 | Homo sapiens | Iperoxo | - | 3.3 | 2019-05-08 | 10.1126/science.aaw5188 | ||
6MH8 | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | - | - | 4.2 | 2019-04-24 | 10.1107/S205225251900263X | |
6ME5 | A | Melatonin | Melatonin | MT1 | Homo sapiens | Agomelatine | - | - | 3.2 | 2019-04-24 | 10.1038/s41586-019-1141-3 | |
6ME4 | A | Melatonin | Melatonin | MT1 | Homo sapiens | 2-Iodomelatonin | - | - | 3.2 | 2019-04-24 | 10.1038/s41586-019-1141-3 | |
6ME3 | A | Melatonin | Melatonin | MT1 | Homo sapiens | 2-Phenylmelatonin | - | - | 2.9 | 2019-04-24 | 10.1038/s41586-019-1141-3 | |
6ME2 | A | Melatonin | Melatonin | MT1 | Homo sapiens | Ramelteon | - | - | 2.8 | 2019-04-24 | 10.1038/s41586-019-1141-3 | |
6ME9 | A | Melatonin | Melatonin | MT2 | Homo sapiens | Ramelteon | - | - | 3.3 | 2019-04-24 | 10.1038/s41586-019-1144-0 | |
6ME8 | A | Melatonin | Melatonin | MT2 | Homo sapiens | 2-Phenylmelatonin | - | - | 3.1 | 2019-04-24 | 10.1038/s41586-019-1144-0 | |
6ME7 | A | Melatonin | Melatonin | MT2 | Homo sapiens | 2-Phenylmelatonin | - | - | 3.2 | 2019-04-24 | 10.1038/s41586-019-1144-0 | |
6ME6 | A | Melatonin | Melatonin | MT2 | Homo sapiens | 2-Phenylmelatonin | - | - | 2.8 | 2019-04-24 | 10.1038/s41586-019-1144-0 | |
6NBI | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | Long-Acting PTH Analog | - | Gs/β1/γ2 | 4 | 2019-04-17 | 10.1126/science.aav7942 | |
6NBI (No Gprot) | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | Long-Acting PTH Analog | - | 4 | 2019-04-17 | 10.1126/science.aav7942 | ||
6NBH | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | Long-Acting PTH Analog | - | Gs/β1/γ2 | 3.5 | 2019-04-17 | 10.1126/science.aav7942 | |
6NBH (No Gprot) | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | Long-Acting PTH Analog | - | 3.5 | 2019-04-17 | 10.1126/science.aav7942 | ||
6NBF | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | Long-Acting PTH Analog | - | Gs/β1/γ2 | 3 | 2019-04-17 | 10.1126/science.aav7942 | |
6NBF (No Gprot) | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | Long-Acting PTH Analog | - | 3 | 2019-04-17 | 10.1126/science.aav7942 | ||
6J21 | A | Peptide | Tachykinin | NK1 | Homo sapiens | Aprepitant | - | - | 3.2 | 2019-03-06 | 10.1038/s41467-019-08568-5 | |
6J20 | A | Peptide | Tachykinin | NK1 | Homo sapiens | Aprepitant | - | - | 2.7 | 2019-03-06 | 10.1038/s41467-019-08568-5 | |
6A94 | A | Amine | 5-Hydroxytryptamine | 5-HT2A | Homo sapiens | Zotepine | - | - | 2.9 | 2019-02-13 | 10.1038/s41594-018-0180-z | |
6A93 | A | Amine | 5-Hydroxytryptamine | 5-HT2A | Homo sapiens | Risperidone | - | - | 3 | 2019-02-13 | 10.1038/s41594-018-0180-z | |
6DO1 | A | Peptide | Angiotensin | AT1 | Homo sapiens | Angiotensin-like peptide S1I8 | - | - | 2.9 | 2019-01-30 | 10.1016/j.cell.2018.12.006 | |
5ZTY | A | Lipid | Cannabinoid | CB2 | Homo sapiens | AM10257 | - | - | 2.8 | 2019-01-30 | 10.1016/j.cell.2018.12.011 | |
6N4B | A | Lipid | Cannabinoid | CB1 | Homo sapiens | MDMB-Fubinaca | - | Gi1/β1/γ2 | 3 | 2019-01-30 | 10.1016/j.cell.2018.11.040 | |
6N4B (No Gprot) | A | Lipid | Cannabinoid | CB1 | Homo sapiens | MDMB-Fubinaca | - | 3 | 2019-01-30 | 10.1016/j.cell.2018.11.040 | ||
6N52 | C | Aminoacid | Metabotropic Glutamate | mGlu5; mGlu5 | Homo sapiens | - | - | - | 4 | 2019-01-23 | 10.1038/s41586-019-0881-4 | |
6N51 | C | Aminoacid | Metabotropic Glutamate | mGlu5; mGlu5 | Homo sapiens | Quisqualate | - | - | 4 | 2019-01-23 | 10.1038/s41586-019-0881-4 | |
6NIY | B1 | Peptide | Calcitonin | CT | Homo sapiens | Adrenomedullin | - | Gs/β1/γ2 | 3.34 | 2019-01-23 | 10.1021/acsptsci.8b00056 | |
6NIY (No Gprot) | B1 | Peptide | Calcitonin | CT | Homo sapiens | Adrenomedullin | - | 3.34 | 2019-01-23 | 10.1021/acsptsci.8b00056 | ||
6HLP | A | Peptide | Tachykinin | NK1 | Homo sapiens | Netupitant | - | - | 2.2 | 2019-01-16 | 10.1038/s41467-018-07939-8 | |
6HLO | A | Peptide | Tachykinin | NK1 | Homo sapiens | Aprepitant | - | - | 2.4 | 2019-01-16 | 10.1038/s41467-018-07939-8 | |
6HLL | A | Peptide | Tachykinin | NK1 | Homo sapiens | CP99994 | - | - | 3.27 | 2019-01-16 | 10.1038/s41467-018-07939-8 | |
6IBL | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Arformoterol | - | - | 2.7 | 2019-01-09 | 10.1038/s41586-020-2419-1 | |
6GPX | A | Protein | Chemokine | CCR2 | Homo sapiens | MK0812 | - | - | 2.7 | 2019-01-02 | 10.1016/j.str.2018.10.027 | |
6GPS | A | Protein | Chemokine | CCR2 | Homo sapiens | MK0812 | - | - | 3.3 | 2019-01-02 | 10.1016/j.str.2018.10.027 | |
6IIV | A | Lipid | Prostanoid | TP | Homo sapiens | Daltroban | - | - | 3 | 2018-12-19 | 10.1038/s41589-018-0170-9 | |
6IIU | A | Lipid | Prostanoid | TP | Homo sapiens | Ramatroban | - | - | 2.5 | 2018-12-19 | 10.1038/s41589-018-0170-9 | |
6MET | A | Protein | Chemokine | CCR5 | Homo sapiens | Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4 | - | - | 4.5 | 2018-12-12 | 10.1038/s41586-018-0804-9 | |
6MEO | A | Protein | Chemokine | CCR5 | Homo sapiens | Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4 | - | - | 3.9 | 2018-12-12 | 10.1038/s41586-018-0804-9 | |
6E59 | A | Peptide | Tachykinin | NK1 | Homo sapiens | L-760735 | - | - | 3.4 | 2018-12-12 | 10.1073/pnas.1812717115 | |
6M9T | A | Lipid | Prostanoid | EP3 | Homo sapiens | Misoprostol-FA | - | - | 2.5 | 2018-12-05 | 10.1038/s41589-018-0160-y | |
6AK3 | A | Lipid | Prostanoid | EP3 | Homo sapiens | Dinoprostone IPGE2 | - | - | 2.9 | 2018-12-05 | 10.1038/s41589-018-0171-8 | |
6AK3 (Multimeric) | A | Lipid | Prostanoid | EP3 | Homo sapiens | Dinoprostone IPGE2 | - | 2.9 | 2018-12-05 | 10.1038/s41589-018-0171-8 | ||
5YWY | A | Lipid | Prostanoid | EP4 | Homo sapiens | ONO-AE3-208 | - | - | 3.2 | 2018-12-05 | 10.1038/s41589-018-0131-3 | |
5YHL | A | Lipid | Prostanoid | EP4 | Homo sapiens | PubChem 135121352 | - | - | 4.2 | 2018-12-05 | 10.1038/s41589-018-0131-3 | |
5ZHP | A | Amine | Acetylcholine (muscarinic) | M3 | Rattus norvegicus | PubChem 134828589 | - | - | 3.1 | 2018-11-28 | 10.1073/pnas.1813988115 | |
6IGL | A | Peptide | Endothelin | ETB | Homo sapiens | IRL1620 | - | - | 2.7 | 2018-11-21 | 10.1038/s41467-018-07094-0 | |
6IGK | A | Peptide | Endothelin | ETB | Homo sapiens | Endothelin-3 | - | - | 2 | 2018-11-21 | 10.1038/s41467-018-07094-0 | |
5ZKC | A | Amine | Acetylcholine (muscarinic) | M2 | Homo sapiens | N-Methyl-Scopolamine | - | - | 2.3 | 2018-11-21 | 10.1038/s41589-018-0152-y | |
5ZKB | A | Amine | Acetylcholine (muscarinic) | M2 | Homo sapiens | AF-DX 384 | - | - | 2.95 | 2018-11-21 | 10.1038/s41589-018-0152-y | |
5ZK8 | A | Amine | Acetylcholine (muscarinic) | M2 | Homo sapiens | N-Methyl-Scopolamine | - | - | 3 | 2018-11-21 | 10.1038/s41589-018-0152-y | |
5ZK3 | A | Amine | Acetylcholine (muscarinic) | M2 | Homo sapiens | 3-quinuclidinyl-benzilate | - | - | 2.6 | 2018-11-21 | 10.1038/s41589-018-0152-y | |
5YC8 | A | Amine | Acetylcholine (muscarinic) | M2 | Homo sapiens | N-Methyl-Scopolamine | - | - | 2.5 | 2018-11-21 | 10.1038/s41589-018-0152-y | |
6FJ3 | B1 | Peptide | Parathyroid Hormone | PTH1 | Homo sapiens | PTH | - | - | 2.5 | 2018-11-21 | 10.1038/s41594-018-0151-4 | |
6MXT | A | Amine | Adrenergic | β2 | Homo sapiens | Salmeterol | - | - | 2.96 | 2018-11-14 | 10.1038/s41589-018-0145-x | |
6AKY | A | Protein | Chemokine | CCR5 | Homo sapiens | - | Maraviroc | - | 2.8 | 2018-10-24 | 10.1021/acs.jmedchem.8b01077 | |
6AKX | A | Protein | Chemokine | CCR5 | Homo sapiens | - | A4R | - | 2.8 | 2018-10-24 | 10.1021/acs.jmedchem.8b01077 | |
6H7O | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Cyanopindolol | - | - | 2.8 | 2018-10-17 | 10.1126/science.aau5595 | |
6H7N | A | Amine | Adrenergic | β1 | Meleagris gallopavo | S-Xamoterol | - | - | 2.5 | 2018-10-17 | 10.1101/436212 | |
6H7M | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Salbutamol | - | - | 2.76 | 2018-10-17 | 10.1126/science.aau5595 | |
6H7L | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Dobutamine | - | - | 2.7 | 2018-10-17 | 10.1126/science.aau5595 | |
6H7J | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Isoprenaline | - | - | 2.8 | 2018-10-17 | 10.1126/science.aau5595 | |
6D27 | A | Lipid | Prostanoid | DP2 | Homo sapiens | CAY10471 | - | - | 2.74 | 2018-10-03 | 10.1016/j.molcel.2018.08.009 | |
6D26 | A | Lipid | Prostanoid | DP2 | Homo sapiens | Fevipiprant | - | - | 2.8 | 2018-10-03 | 10.1016/j.molcel.2018.08.009 | |
6FUF | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | Go | 3.12 | 2018-10-03 | 10.1126/sciadv.aat7052 | |
6FUF (No Gprot) | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | 3.12 | 2018-10-03 | 10.1126/sciadv.aat7052 | ||
6E3Y | B1 | Peptide | Calcitonin | CT Like | Homo sapiens | Calcitonin gene-related peptide-1 | - | Gs/β1/γ2; RAMP1 | 3.3 | 2018-09-19 | 10.1038/s41586-018-0535-y | |
6E3Y (No Gprot) | B1 | Peptide | Calcitonin | CT Like | Homo sapiens | Calcitonin gene-related peptide-1 | - | 3.3 | 2018-09-19 | 10.1038/s41586-018-0535-y | ||
6DS0 | A | Amine | 5-Hydroxytryptamine | 5-HT2B | Homo sapiens | Ly266097 | - | - | 3.19 | 2018-08-29 | 10.1038/s41594-018-0116-7 | |
6DRZ | A | Amine | 5-Hydroxytryptamine | 5-HT2B | Homo sapiens | Methysergide | - | - | 3.1 | 2018-08-29 | 10.1038/s41594-018-0116-7 | |
6DRY | A | Amine | 5-Hydroxytryptamine | 5-HT2B | Homo sapiens | Methylergonovine | - | - | 2.92 | 2018-08-29 | 10.1038/s41594-018-0116-7 | |
6DRX | A | Amine | 5-Hydroxytryptamine | 5-HT2B | Homo sapiens | Lisuride | - | - | 3.1 | 2018-08-29 | 10.1038/s41594-018-0116-7 | |
6BD4 | F | Protein | Frizzled | FZD4 | Homo sapiens | - | - | - | 2.4 | 2018-08-22 | 10.1038/s41586-018-0447-x | |
5XJM | A | Peptide | Angiotensin | AT2 | Homo sapiens | (Sar1,Ile8)-Angiotensin II | - | - | 3.2 | 2018-07-11 | 10.1038/s41594-018-0079-8 | |
5ZKQ | A | Lipid | Platelet Activating Factor | PAF | Homo sapiens | ABT-491 | - | - | 2.9 | 2018-06-20 | 10.1038/s41594-018-0068-y | |
5ZKP | A | Lipid | Platelet Activating Factor | PAF | Homo sapiens | Foropafant (SR27417) | - | - | 2.81 | 2018-06-20 | 10.1038/s41594-018-0068-y | |
6CMO | A | Sensory | Opsins | Rhodopsin | Homo sapiens | - | - | Gi1/β1/γ2 | 4.5 | 2018-06-20 | 10.1038/s41586-018-0215-y | |
6CMO (No Gprot) | A | Sensory | Opsins | Rhodopsin | Homo sapiens | - | - | 4.5 | 2018-06-20 | 10.1038/s41586-018-0215-y | ||
6D9H | A | Nucleotide | Adenosine | A1 | Homo sapiens | Adenosine | - | Gi2/β1/γ2 | 3.6 | 2018-06-20 | 10.1038/s41586-018-0236-6 | |
6D9H (No Gprot) | A | Nucleotide | Adenosine | A1 | Homo sapiens | Adenosine | - | 3.6 | 2018-06-20 | 10.1038/s41586-018-0236-6 | ||
6G79 | A | Amine | 5-Hydroxytryptamine | 5-HT1B | Homo sapiens | Donitriptan | - | Go/β1/γ2 | 3.78 | 2018-06-20 | 10.1038/s41586-018-0241-9 | |
6G79 (No Gprot) | A | Amine | 5-Hydroxytryptamine | 5-HT1B | Homo sapiens | Donitriptan | - | 3.78 | 2018-06-20 | 10.1038/s41586-018-0241-9 | ||
5WB2 | A | Other | Unclassified | US28 | Human cytomegalovirus (strain towne) | CX3CL1.35 | - | - | 3.5 | 2018-06-13 | 10.7554/eLife.35850 | |
5WB1 | A | Other | Unclassified | US28 | Human cytomegalovirus (strain towne) | - | - | - | 3.51 | 2018-06-13 | 10.7554/eLife.35850 | |
6DDF | A | Peptide | Opioid | μ | Mus musculus | Damgo | - | Gi1/β1/γ2 | 3.5 | 2018-06-13 | 10.1038/s41586-018-0219-7 | |
6DDF (No Gprot) | A | Peptide | Opioid | μ | Mus musculus | Damgo | - | 3.5 | 2018-06-13 | 10.1038/s41586-018-0219-7 | ||
6DDE | A | Peptide | Opioid | μ | Mus musculus | Damgo | - | Gi1/β1/γ2 | 3.5 | 2018-06-13 | 10.1038/s41586-018-0219-7 | |
6DDE (No Gprot) | A | Peptide | Opioid | μ | Mus musculus | Damgo | - | 3.5 | 2018-06-13 | 10.1038/s41586-018-0219-7 | ||
6C1R | A | Peptide | Complement Peptide | C5a1 | Homo sapiens | PMX53 | Avacopan; Na | - | 2.2 | 2018-05-30 | 10.1038/s41594-018-0067-z | |
6C1Q | A | Peptide | Complement Peptide | C5a1 | Homo sapiens | PMX53 | NDT9513727 | - | 2.9 | 2018-05-30 | 10.1038/s41594-018-0067-z | |
6D35 | F | Protein | Frizzled | SMO | Xenopus laevis | - | Cholesterol | - | 3.9 | 2018-05-23 | 10.1016/j.cell.2018.04.029 | |
6D32 | F | Protein | Frizzled | SMO | Xenopus laevis | Cyclopamine | Cyclopamine | - | 3.75 | 2018-05-23 | 10.1016/j.cell.2018.04.029 | |
6GDG | A | Nucleotide | Adenosine | A2A | Homo sapiens | NECA | - | Gs/β1/γ1 | 4.11 | 2018-05-16 | 10.7554/eLife.35946 | |
6GDG (No Gprot) | A | Nucleotide | Adenosine | A2A | Homo sapiens | NECA | - | 4.11 | 2018-05-16 | 10.7554/eLife.35946 | ||
5KW2 | A | Lipid | Free Fatty Acid | FFA1 | Homo sapiens | - | PubChem 133053953 | - | 2.76 | 2018-05-02 | 10.1038/s41467-017-01240-w | |
5ZBQ | A | Peptide | Neuropeptide Y | Y1 | Homo sapiens | UR-MK-299 | - | - | 2.7 | 2018-04-25 | 10.1038/s41586-018-0046-x | |
5ZBH | A | Peptide | Neuropeptide Y | Y1 | Homo sapiens | BMS-193885 | - | - | 3 | 2018-04-25 | 10.1038/s41586-018-0046-x | |
6FKD | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | PubChem 137349183 | - | 2.49 | 2018-04-04 | 10.1073/pnas.1718084115 | |
6FKC | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | PubChem 132473039 | - | 2.46 | 2018-04-04 | 10.1073/pnas.1718084115 | |
6FKB | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | PubChem 132473038 | - | 3.03 | 2018-04-04 | 10.1073/pnas.1718084115 | |
6FKA | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | PubChem 132473037 | - | 2.7 | 2018-04-04 | 10.1073/pnas.1718084115 | |
6FK9 | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | PubChem 132473036 | - | 2.63 | 2018-04-04 | 10.1073/pnas.1718084115 | |
6FK8 | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | PubChem 132473035 | - | 2.87 | 2018-04-04 | 10.1073/pnas.1718084115 | |
6FK7 | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | PubChem 132473034 | - | 2.62 | 2018-04-04 | 10.1073/pnas.1718084115 | |
6FK6 | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | PubChem 132473033 | - | 2.36 | 2018-04-04 | 10.1073/pnas.1718084115 | |
6CM4 | A | Amine | Dopamine | D2 | Homo sapiens | Risperidone | - | - | 2.87 | 2018-03-14 | 10.1038/nature25758 | |
6FFI | C | Aminoacid | Metabotropic Glutamate | mGlu5 | Homo sapiens | - | MMPEP | - | 2.2 | 2018-03-07 | 10.1021/acs.jmedchem.7b01722 | |
6FFH | C | Aminoacid | Metabotropic Glutamate | mGlu5 | Homo sapiens | - | Fenobam | - | 2.65 | 2018-03-07 | 10.1021/acs.jmedchem.7b01722 | |
5WF6 | A | Nucleotide | Adenosine | A2A | Homo sapiens | UK-432097 | - | - | 2.9 | 2018-02-21 | 10.1016/j.str.2017.12.013 | |
5WF5 | A | Nucleotide | Adenosine | A2A | Homo sapiens | UK-432097 | - | - | 2.6 | 2018-02-21 | 10.1016/j.str.2017.12.013 | |
6B3J | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Exendin-P5 | - | Gs/β1/γ2 | 3.3 | 2018-02-21 | 10.1038/nature25773 | |
6B3J (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | Exendin-P5 | - | 3.3 | 2018-02-21 | 10.1038/nature25773 | ||
6BQH | A | Amine | 5-Hydroxytryptamine | 5-HT2C | Homo sapiens | Ritanserin | - | - | 2.7 | 2018-02-14 | 10.1016/j.cell.2018.01.001 | |
6BQG | A | Amine | 5-Hydroxytryptamine | 5-HT2C | Homo sapiens | Ergotamine | - | - | 3 | 2018-02-14 | 10.1016/j.cell.2018.01.001 | |
5V54 | A | Amine | 5-Hydroxytryptamine | 5-HT1B | Homo sapiens | Methiothepin | - | - | 3.9 | 2018-02-07 | 10.1038/s41421-018-0009-2 | |
5OM4 | A | Nucleotide | Adenosine | A2A | Homo sapiens | PubChem 135566609 | Na | - | 2 | 2018-01-17 | 10.1038/s41598-017-18570-w | |
5OM1 | A | Nucleotide | Adenosine | A2A | Homo sapiens | PubChem 135566609 | Na | - | 2.1 | 2018-01-17 | 10.1038/s41598-017-18570-w | |
5OLZ | A | Nucleotide | Adenosine | A2A | Homo sapiens | PubChem 135566609 | Na | - | 1.9 | 2018-01-17 | 10.1038/s41598-017-18570-w | |
5OLV | A | Nucleotide | Adenosine | A2A | Homo sapiens | LUAA41063 | Na | - | 2 | 2018-01-17 | 10.1038/s41598-017-18570-w | |
5OLO | A | Nucleotide | Adenosine | A2A | Homo sapiens | Tozadenant | Na | - | 3.1 | 2018-01-17 | 10.1038/s41598-017-18570-w | |
5OLH | A | Nucleotide | Adenosine | A2A | Homo sapiens | Vipadenant | Na | - | 2.6 | 2018-01-17 | 10.1038/s41598-017-18570-w | |
5OLG | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | Na | - | 1.87 | 2018-01-17 | 10.1038/s41598-017-18570-w | |
5YQZ | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | Glucagon analogue | - | - | 3 | 2018-01-17 | 10.1038/nature25153 | |
6B73 | A | Peptide | Opioid | κ | Homo sapiens | MP1104 | - | - | 3.1 | 2018-01-17 | 10.1016/j.cell.2017.12.011 | |
6AQF | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | - | - | 2.51 | 2018-01-10 | 10.1016/j.cell.2017.12.004 | |
5O9H | A | Peptide | Complement Peptide | C5a1 | Homo sapiens | - | NDT9513727 | - | 2.7 | 2018-01-10 | 10.1038/nature25025 | |
5O9H (Multimeric) | A | Peptide | Complement Peptide | C5a1 | Homo sapiens | - | NDT9513727 | 2.7 | 2018-01-10 | 10.1038/nature25025 | ||
5X33 | A | Lipid | Leukotriene | BLT1 | Cavia porcellus | BIIL260 | - | - | 3.7 | 2018-01-03 | 10.1038/nchembio.2547 | |
5VRA | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | Na | - | 2.35 | 2017-12-13 | 10.1038/nprot.2017.135 | |
5WS3 | A | Peptide | Orexin | OX2 | Homo sapiens | EMPA | - | - | 2.3 | 2017-12-13 | 10.1016/j.str.2017.11.005 | |
5WKT | A | Sensory | Opsins | Rhodopsin | Bos taurus | Octyl-β-D-Glucopyranoside | - | Gt(CT) | 3.2 | 2017-12-13 | 10.1038/nprot.2017.135 | |
5WKT (No Gprot) | A | Sensory | Opsins | Rhodopsin | Bos taurus | Octyl-β-D-Glucopyranoside | - | 3.2 | 2017-12-13 | 10.1038/nprot.2017.135 | ||
5WQC | A | Peptide | Orexin | OX2 | Homo sapiens | EMPA | - | - | 1.96 | 2017-11-29 | 10.1016/j.str.2017.11.005 | |
5WIV | A | Amine | Dopamine | D4 | Homo sapiens | Nemonapride | Na | - | 2.14 | 2017-10-18 | 10.1126/science.aan5468 | |
5WIU | A | Amine | Dopamine | D4 | Homo sapiens | Nemonapride | - | - | 1.96 | 2017-10-18 | 10.1126/science.aan5468 | |
5NM4 | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | Na | - | 1.7 | 2017-09-27 | 10.1038/s41467-017-00630-4 | |
5NM2 | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | Na | - | 1.95 | 2017-09-27 | 10.1038/s41467-017-00630-4 | |
5NLX | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | Na | - | 2.14 | 2017-09-27 | 10.1038/s41467-017-00630-4 | |
5X7D | A | Amine | Adrenergic | β2 | Homo sapiens | S-Carazolol | PubChem 129318963 | - | 2.7 | 2017-08-16 | 10.1038/nature23652 | |
5XPR | A | Peptide | Endothelin | ETB | Homo sapiens | Bosentan | - | - | 3.6 | 2017-08-16 | 10.1038/nsmb.3450 | |
5X93 | A | Peptide | Endothelin | ETB | Homo sapiens | K-8794 | - | - | 2.2 | 2017-08-16 | 10.1038/nsmb.3450 | |
5XSZ | A | Lipid | Lysophospholipid | LPA6 | Danio rerio | Glyceryl-mono-oleate | - | - | 3.2 | 2017-08-16 | 10.1038/nature23448 | |
5W0P | A | Sensory | Opsins | Rhodopsin | Homo sapiens | - | - | Arrestin1 | 3.01 | 2017-08-09 | 10.1016/j.cell.2017.07.002 | |
5TUD | A | Amine | 5-Hydroxytryptamine | 5-HT2B | Homo sapiens | Ergotamine | - | - | 3 | 2017-07-26 | 10.1073/pnas.1700891114 | |
5N2S | A | Nucleotide | Adenosine | A1 | Homo sapiens | PSB36 | - | - | 3.3 | 2017-07-26 | 10.1016/j.str.2017.06.012 | |
5N2R | A | Nucleotide | Adenosine | A2A | Homo sapiens | PSB-36 | Na | - | 2.8 | 2017-07-26 | 10.1016/j.str.2017.06.012 | |
5MZP | A | Nucleotide | Adenosine | A2A | Homo sapiens | Caffeine | Na | - | 2.1 | 2017-07-26 | 10.1016/j.str.2017.06.012 | |
5MZJ | A | Nucleotide | Adenosine | A2A | Homo sapiens | Theophylline | Na | - | 2 | 2017-07-26 | 10.1016/j.str.2017.06.012 | |
5XRA | A | Lipid | Cannabinoid | CB1 | Homo sapiens | AM11542 | - | - | 2.8 | 2017-07-12 | 10.1038/nature23272 | |
5XR8 | A | Lipid | Cannabinoid | CB1 | Homo sapiens | AM841 | - | - | 2.95 | 2017-07-12 | 10.1038/nature23272 | |
5UIW | A | Protein | Chemokine | CCR5 | Homo sapiens | 5P7-CCL5 | - | - | 2.2 | 2017-06-28 | 10.1016/j.immuni.2017.05.002 | |
5NX2 | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | GLP-1 (Truncated) | - | - | 3.7 | 2017-06-14 | 10.1038/nature22800 | |
5TZY | A | Lipid | Free Fatty Acid | FFA1 | Homo sapiens | - | MK8666; PubChem 127053597 | - | 3.22 | 2017-06-07 | 10.1038/nsmb.3417 | |
5TZR | A | Lipid | Free Fatty Acid | FFA1 | Homo sapiens | - | MK8666 | - | 2.2 | 2017-06-07 | 10.1038/nsmb.3417 | |
5JTB | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | - | - | 2.8 | 2017-05-31 | 10.1126/sciadv.1602952 | |
5VBL | A | Peptide | Apelin | Apelin | Homo sapiens | Apelin mimetic peptide agonist | - | - | 2.6 | 2017-05-31 | 10.1016/j.str.2017.04.008 | |
5UVI | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | - | - | 3.2 | 2017-05-24 | 10.1107/S205225251700570X | |
5VEW | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | - | PF-06372222 | - | 2.7 | 2017-05-24 | 10.1038/nature22378 | |
5XF1 | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | - | NNC0640 | - | 3.19 | 2017-05-24 | 10.1038/nature22363 | |
5XEZ | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | - | NNC0640 | - | 3 | 2017-05-24 | 10.1038/nature22363 | |
5V57 | F | Protein | Frizzled | SMO | Homo sapiens | TC114 | - | - | 3 | 2017-05-24 | 10.1038/ncomms15383 | |
5V56 | F | Protein | Frizzled | SMO | Homo sapiens | TC114 | - | - | 2.9 | 2017-05-24 | 10.1038/ncomms15383 | |
5VAI | B1 | Peptide | Glucagon | GLP-1 | Oryctolagus cuniculus | GLP-1 | - | Gs/β1/γ2 | 4.1 | 2017-05-24 | 10.1038/nature22394 | |
5VAI (No Gprot) | B1 | Peptide | Glucagon | GLP-1 | Oryctolagus cuniculus | GLP-1 | - | 4.1 | 2017-05-24 | 10.1038/nature22394 | ||
5VEX | B1 | Peptide | Glucagon | GLP-1 | Homo sapiens | - | NNC0640 | - | 3 | 2017-05-17 | 10.1038/nature22378 | |
5NJ6 | A | Peptide | Proteinase Activated | PAR2 | Homo sapiens | - | - | - | 4 | 2017-05-03 | 10.1038/nature22309 | |
5NDZ | A | Peptide | Proteinase Activated | PAR2 | Homo sapiens | - | AZ3451; Na | - | 3.6 | 2017-05-03 | 10.1038/nature22309 | |
5NDD | A | Peptide | Proteinase Activated | PAR2 | Homo sapiens | - | AZ8838; Na | - | 2.8 | 2017-05-03 | 10.1038/nature22309 | |
5UZ7 | B1 | Peptide | Calcitonin | CT | Homo sapiens | - | - | Gs/β1/γ2 | 4.1 | 2017-05-03 | 10.1038/nature22327 | |
5UZ7 (No Gprot) | B1 | Peptide | Calcitonin | CT | Homo sapiens | - | - | 4.1 | 2017-05-03 | 10.1038/nature22327 | ||
5UNH | A | Peptide | Angiotensin | AT2 | Homo sapiens | PubChem 126456406 | - | - | 2.9 | 2017-04-05 | 10.1038/nature22035 | |
5UNG | A | Peptide | Angiotensin | AT2 | Homo sapiens | PubChem 15780052 | - | - | 2.8 | 2017-04-05 | 10.1038/nature22035 | |
5UNF | A | Peptide | Angiotensin | AT2 | Homo sapiens | PubChem 15780052 | - | - | 2.8 | 2017-04-05 | 10.1038/nature22035 | |
5TE5 | A | Sensory | Opsins | Rhodopsin | Bos taurus | 20-Methanoretinal | - | - | 4.01 | 2017-03-15 | 10.1073/pnas.1617446114 | |
5TE3 | A | Sensory | Opsins | Rhodopsin | Bos taurus | Octyl-β-D-Glucopyranoside | - | - | 2.7 | 2017-03-15 | 10.1073/pnas.1617446114 | |
5UEN | A | Nucleotide | Adenosine | A1 | Homo sapiens | DU172 | - | - | 3.2 | 2017-03-01 | 10.1016/j.cell.2017.01.042 | |
5UIG | A | Nucleotide | Adenosine | A2A | Homo sapiens | Cmpd-1 | - | - | 3.5 | 2017-02-08 | 10.1073/pnas.1621423114 | |
5TVN | A | Amine | 5-Hydroxytryptamine | 5-HT2B | Homo sapiens | LSD | - | - | 2.9 | 2017-02-01 | 10.1016/j.cell.2016.12.033 | |
5T04 | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | Neurotensin | - | - | 3.3 | 2016-12-21 | 10.1038/srep38564 | |
5T1A | A | Protein | Chemokine | CCR2 | Homo sapiens | - | PubChem 68764898; PubChem 12093170 | - | 2.81 | 2016-12-14 | 10.1038/nature20605 | |
5U09 | A | Lipid | Cannabinoid | CB1 | Homo sapiens | Taranabant | - | - | 2.6 | 2016-12-07 | 10.1038/nature20613 | |
5LWE | A | Protein | Chemokine | CCR9 | Homo sapiens | - | Vercirnon | - | 2.8 | 2016-12-07 | 10.1038/nature20606 | |
5TGZ | A | Lipid | Cannabinoid | CB1 | Homo sapiens | AM6538 | - | - | 2.8 | 2016-11-02 | 10.1016/j.cell.2016.10.004 | |
5K2D | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | Na | - | 1.9 | 2016-09-21 | 10.1126/sciadv.1600292 | |
5K2C | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | Na | - | 1.9 | 2016-09-21 | 10.1126/sciadv.1600292 | |
5K2B | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | Na | - | 2.5 | 2016-09-21 | 10.1126/sciadv.1600292 | |
5K2A | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | Na | - | 2.5 | 2016-09-21 | 10.1126/sciadv.1600292 | |
5GLI | A | Peptide | Endothelin | ETB | Homo sapiens | - | - | - | 2.5 | 2016-09-07 | 10.1038/nature19319 | |
5GLH | A | Peptide | Endothelin | ETB | Homo sapiens | Endothelin-1 | - | - | 2.8 | 2016-09-07 | 10.1038/nature19319 | |
5D6L | A | Amine | Adrenergic | β2 | Homo sapiens | S-Carazolol | - | - | 3.2 | 2016-08-17 | 10.1038/nprot.2017.057 | |
5DYS | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | - | 2.3 | 2016-08-10 | 10.15252/embr.201642671 | |
5EN0 | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | Gt(CT) | 2.81 | 2016-08-10 | 10.15252/embr.201642671 | |
5EN0 (No Gprot) | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | 2.81 | 2016-08-10 | 10.15252/embr.201642671 | ||
5G53 | A | Nucleotide | Adenosine | A2A | Homo sapiens | NECA | - | Gs | 3.4 | 2016-08-03 | 10.1038/nature18966 | |
5G53 (No Gprot) | A | Nucleotide | Adenosine | A2A | Homo sapiens | NECA | - | 3.4 | 2016-08-03 | 10.1038/nature18966 | ||
5L7I | F | Protein | Frizzled | SMO | Homo sapiens | Vismodegib | - | - | 3.3 | 2016-07-20 | 10.1038/nature18934 | |
5L7D | F | Protein | Frizzled | SMO | Homo sapiens | - | Cholesterol | - | 3.2 | 2016-07-20 | 10.1038/nature18934 | |
5JQH | A | Amine | Adrenergic | β2 | Homo sapiens | S-Carazolol | - | - | 3.2 | 2016-07-13 | 10.1038/nature18636 | |
5IUB | A | Nucleotide | Adenosine | A2A | Homo sapiens | Q27456344 | Na | - | 2.1 | 2016-06-29 | 10.1021/acs.jmedchem.6b00653 | |
5IUA | A | Nucleotide | Adenosine | A2A | Homo sapiens | Q27456348 | Na | - | 2.2 | 2016-06-29 | 10.1021/acs.jmedchem.6b00653 | |
5IU8 | A | Nucleotide | Adenosine | A2A | Homo sapiens | Q27456347 | Na | - | 2 | 2016-06-29 | 10.1021/acs.jmedchem.6b00653 | |
5IU7 | A | Nucleotide | Adenosine | A2A | Homo sapiens | Q27456346 | Na | - | 1.9 | 2016-06-29 | 10.1021/acs.jmedchem.6b00653 | |
5IU4 | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | Na | - | 1.72 | 2016-06-29 | 10.1021/acs.jmedchem.6b00653 | |
4Z9G | B1 | Peptide | Corticotropin Releasing Factor | CRF1 | Homo sapiens | - | CP-376395 | - | 3.18 | 2016-06-29 | 10.2174/1874467210666170110114727 | |
5EE7 | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | - | MK0893 | - | 2.5 | 2016-04-20 | 10.1038/nature17414 | |
5DGY | A | Sensory | Opsins | Rhodopsin | Homo sapiens | - | - | Arrestin1 | 7.7 | 2016-03-23 | 10.1038/sdata.2016.21 | |
5DSG | A | Amine | Acetylcholine (muscarinic) | M4 | Homo sapiens | Tiotropium | - | - | 2.6 | 2016-03-16 | 10.1038/nature17188 | |
5CXV | A | Amine | Acetylcholine (muscarinic) | M1 | Homo sapiens | Tiotropium | - | - | 2.7 | 2016-03-09 | 10.1038/nature17188 | |
4ZJC | A | Peptide | Orexin | OX1 | Homo sapiens | SB-674042 | - | - | 2.83 | 2016-03-09 | 10.1038/nsmb.3183 | |
4ZJ8 | A | Peptide | Orexin | OX1 | Homo sapiens | Suvorexant | - | - | 2.75 | 2016-03-09 | 10.1038/nsmb.3183 | |
5D5B | A | Amine | Adrenergic | β2 | Homo sapiens | S-Carazolol | - | - | 3.8 | 2016-01-13 | 10.1107/S2059798315021683 | |
5D5A | A | Amine | Adrenergic | β2 | Homo sapiens | S-Carazolol | - | - | 2.48 | 2016-01-13 | 10.1107/S2059798315021683 | |
5F8U | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Cyanopindolol | - | - | 3.35 | 2015-12-23 | 10.1038/nsmb.3130 | |
4X1H | A | Sensory | Opsins | Rhodopsin | Bos taurus | Nonyl-β-D-Glucopyranoside | - | Gt(CT) | 2.29 | 2015-11-04 | 10.1016/j.str.2015.09.015 | |
4X1H (No Gprot) | A | Sensory | Opsins | Rhodopsin | Bos taurus | Nonyl-β-D-Glucopyranoside | - | 2.29 | 2015-11-04 | 10.1016/j.str.2015.09.015 | ||
5DHH | A | Peptide | Opioid | NOP | Homo sapiens | SB-612111 | - | - | 3 | 2015-10-21 | 10.1016/j.str.2015.07.024 | |
5DHG | A | Peptide | Opioid | NOP | Homo sapiens | C-35 | - | - | 3 | 2015-10-21 | 10.1016/j.str.2015.07.024 | |
4ZUD | A | Peptide | Angiotensin | AT1 | Homo sapiens | Olmesartan | - | - | 2.8 | 2015-10-07 | 10.1074/jbc.M115.689000 | |
5A8E | A | Amine | Adrenergic | β1 | Meleagris gallopavo | 7-Methylcyanopindolol | Na | - | 2.4 | 2015-09-30 | 10.1124/mol.115.101030 | |
5CGD | C | Aminoacid | Metabotropic Glutamate | mGlu5 | Homo sapiens | - | HTL14242 | - | 2.6 | 2015-08-12 | 10.1021/acs.jmedchem.5b00892 | |
5CGC | C | Aminoacid | Metabotropic Glutamate | mGlu5 | Homo sapiens | - | HTL14242 | - | 3.1 | 2015-08-12 | 10.1021/acs.jmedchem.5b00892 | |
5C1M | A | Peptide | Opioid | μ | Mus musculus | BU72 | - | - | 2.07 | 2015-08-05 | 10.1038/nature14886 | |
4XES | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | Neurotensin | - | - | 2.6 | 2015-07-29 | 10.1038/ncomms8895 | |
4XEE | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | Neurotensin | - | - | 2.9 | 2015-07-29 | 10.1038/ncomms8895 | |
4ZWJ | A | Sensory | Opsins | Rhodopsin | Homo sapiens | - | - | Arrestin1 | 3.3 | 2015-07-29 | 10.1038/nature14656 | |
4WW3 | A | Sensory | Opsins | Rhodopsin | Todarodes pacificus | All-trans-Retinal | - | - | 2.8 | 2015-06-17 | 10.1371/journal.pone.0126970 | |
4Z36 | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | ONO-3080573 | - | - | 2.9 | 2015-06-03 | 10.1016/j.cell.2015.06.002 | |
4Z35 | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | ONO-9910539 | - | - | 2.9 | 2015-06-03 | 10.1016/j.cell.2015.06.002 | |
4Z34 | A | Lipid | Lysophospholipid | LPA1 | Homo sapiens | ONO-9780307 | - | - | 3 | 2015-06-03 | 10.1016/j.cell.2015.06.002 | |
4YAY | A | Peptide | Angiotensin | AT1 | Homo sapiens | ZD-7155 | - | - | 2.9 | 2015-04-22 | 10.1016/j.cell.2015.04.011 | |
4UHR | A | Nucleotide | Adenosine | A2A | Homo sapiens | CGS21680 | - | - | 2.6 | 2015-04-08 | 10.1124/mol.114.097360 | |
4UG2 | A | Nucleotide | Adenosine | A2A | Homo sapiens | CGS21680 | - | - | 2.6 | 2015-04-08 | 10.1124/mol.114.097360 | |
4XNW | A | Nucleotide | P2Y | P2Y1 | Homo sapiens | MRS2500 | - | - | 2.7 | 2015-04-01 | 10.1038/nature14287 | |
4XNV | A | Nucleotide | P2Y | P2Y1 | Homo sapiens | - | BPTU | - | 2.2 | 2015-04-01 | 10.1038/nature14287 | |
4XT3 | A | Other | Unclassified | US28 | Human cytomegalovirus (strain ad169) | Fractalkine | - | - | 3.8 | 2015-03-04 | 10.1126/science.aaa5026 | |
4XT1 | A | Other | Unclassified | US28 | Human cytomegalovirus (strain ad169) | Fractalkine | - | - | 2.89 | 2015-03-04 | 10.1126/science.aaa5026 | |
4RWS | A | Protein | Chemokine | CXCR4 | Homo sapiens | vMIP-II | - | - | 3.1 | 2015-02-11 | 10.1126/science.1261064 | |
4RWD | A | Peptide | Opioid | δ | Homo sapiens | DIPP-NH2 | Na | - | 2.7 | 2015-01-14 | 10.1038/nsmb.2965 | |
4RWA | A | Peptide | Opioid | δ | Homo sapiens | DIPP-NH2 | - | - | 3.28 | 2015-01-14 | 10.1038/nsmb.2965 | |
4S0V | A | Peptide | Orexin | OX2 | Homo sapiens | Suvorexant | - | - | 2.5 | 2015-01-14 | 10.1038/nature14035 | |
4U16 | A | Amine | Acetylcholine (muscarinic) | M3 | Rattus norvegicus | N-Methyl-Scopolamine | - | - | 3.7 | 2014-11-26 | 10.1016/j.str.2014.08.022 | |
4U15 | A | Amine | Acetylcholine (muscarinic) | M3 | Rattus norvegicus | Tiotropium | - | - | 2.8 | 2014-11-26 | 10.1016/j.str.2014.08.022 | |
4U14 | A | Amine | Acetylcholine (muscarinic) | M3 | Rattus norvegicus | Tiotropium | - | - | 3.57 | 2014-11-26 | 10.1016/j.str.2014.08.022 | |
4PXF | A | Sensory | Opsins | Rhodopsin | Bos taurus | Octyl-β-D-Glucopyranoside | - | Arrestin1 Finger Loop | 2.75 | 2014-09-17 | 10.1038/ncomms5801 | |
4QKX | A | Amine | Adrenergic | β2 | Homo sapiens | 35V | - | - | 3.3 | 2014-07-23 | 10.1073/pnas.1410415111 | |
4QIN | F | Protein | Frizzled | SMO | Homo sapiens | SAG1.5 | - | - | 2.6 | 2014-07-23 | 10.1038/ncomms5355 | |
4QIM | F | Protein | Frizzled | SMO | Homo sapiens | ANTA XV | - | - | 2.61 | 2014-07-23 | 10.1038/ncomms5355 | |
4PHU | A | Lipid | Free Fatty Acid | FFA1 | Homo sapiens | - | Fasiglifam | - | 2.33 | 2014-07-16 | 10.1038/nature13494 | |
4OO9 | C | Aminoacid | Metabotropic Glutamate | mGlu5 | Homo sapiens | - | Mavoglurant | - | 2.6 | 2014-07-02 | 10.1038/nature13396 | |
4PY0 | A | Nucleotide | P2Y | P2Y12 | Homo sapiens | 2MeSATP | - | - | 3.1 | 2014-04-30 | 10.1038/nature13288 | |
4PXZ | A | Nucleotide | P2Y | P2Y12 | Homo sapiens | 2MeSADP | - | - | 2.5 | 2014-04-30 | 10.1038/nature13288 | |
4BVN | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Cyanopindolol | Na | - | 2.1 | 2014-04-02 | 10.1371/journal.pone.0092727 | |
4NTJ | A | Nucleotide | P2Y | P2Y12 | Homo sapiens | AZD1283 | - | - | 2.62 | 2014-03-26 | 10.1038/nature13083 | |
4OR2 | C | Aminoacid | Metabotropic Glutamate | mGlu1; mGlu1 | Homo sapiens | - | FITM | - | 2.8 | 2014-03-19 | 10.1126/science.1249489 | |
4O9R | F | Protein | Frizzled | SMO | Homo sapiens | Cyclopamine | - | - | 3.2 | 2014-03-05 | 10.1038/ncomms4309 | |
4BWB | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | Neurotensin | - | - | 3.57 | 2014-01-29 | 10.1073/pnas.1317903111 | |
4BV0 | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | Neurotensin | - | - | 3.1 | 2014-01-29 | 10.1073/pnas.1317903111 | |
4BUO | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | Neurotensin | - | - | 2.75 | 2014-01-29 | 10.1073/pnas.1317903111 | |
3ZEV | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | Neurotensin | - | - | 3 | 2014-01-29 | 10.1073/pnas.1317903111 | |
4N4W | F | Protein | Frizzled | SMO | Homo sapiens | - | SANT-1 | - | 2.8 | 2014-01-22 | 10.1038/ncomms5355 | |
4N6H | A | Peptide | Opioid | δ | Homo sapiens | Naltrindole | Na | - | 1.8 | 2013-12-25 | 10.1038/nature12944 | |
4NC3 | A | Amine | 5-Hydroxytryptamine | 5-HT2B | Homo sapiens | Ergotamine | - | - | 2.8 | 2013-12-18 | 10.1126/science.1244142 | |
4MQT | A | Amine | Acetylcholine (muscarinic) | M2 | Homo sapiens | Iperoxo | LY2119620 | - | 3.7 | 2013-11-27 | 10.1038/nature12735 | |
4MQS | A | Amine | Acetylcholine (muscarinic) | M2 | Homo sapiens | Iperoxo | - | - | 3.5 | 2013-11-27 | 10.1038/nature12735 | |
4J4Q | A | Sensory | Opsins | Rhodopsin | Bos taurus | Octyl β-D-Glucopyranoside | - | Gt(CT) | 2.65 | 2013-10-30 | 10.1002/anie.201302374 | |
4J4Q (No Gprot) | A | Sensory | Opsins | Rhodopsin | Bos taurus | Octyl β-D-Glucopyranoside | - | 2.65 | 2013-10-30 | 10.1002/anie.201302374 | ||
4LDO | A | Amine | Adrenergic | β2 | Homo sapiens | L-Epinephrine | - | - | 3.2 | 2013-09-25 | 10.1038/nature12572 | |
4LDL | A | Amine | Adrenergic | β2 | Homo sapiens | Hydroxybenzylisoproterenol | - | - | 3.1 | 2013-09-25 | 10.1038/nature12572 | |
4LDE | A | Amine | Adrenergic | β2 | Homo sapiens | BI167107 | - | - | 2.79 | 2013-09-25 | 10.1038/nature12572 | |
4MBS | A | Protein | Chemokine | CCR5 | Homo sapiens | - | Maraviroc | - | 2.71 | 2013-09-11 | 10.1126/science.1241475 | |
4L6R | B1 | Peptide | Glucagon | Glucagon | Homo sapiens | - | - | - | 3.3 | 2013-07-24 | 10.1038/nature12393 | |
4K5Y | B1 | Peptide | Corticotropin Releasing Factor | CRF1 | Homo sapiens | - | CP-376395 | - | 2.98 | 2013-07-17 | 10.1038/nature12357 | |
4BEY | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | - | Gt(CT) | 2.9 | 2013-05-08 | 10.1038/embor.2013.44 | |
4BEY (No Gprot) | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | - | 2.9 | 2013-05-08 | 10.1038/embor.2013.44 | ||
4BEZ | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | - | - | 3.3 | 2013-04-24 | 10.1038/embor.2013.44 | |
4JKV | F | Protein | Frizzled | SMO | Homo sapiens | Taladegib | - | - | 2.45 | 2013-04-24 | 10.1038/nature12167 | |
4JKV (Multimeric) | F | Protein | Frizzled | SMO | Homo sapiens | Taladegib | - | 2.45 | 2013-04-24 | 10.1038/nature12167 | ||
3ZPR | A | Amine | Adrenergic | β1 | Meleagris gallopavo | 4-methyl-2-(piperazin-1-yl) | Na | - | 2.7 | 2013-04-03 | 10.1021/jm400140q | |
3ZPQ | A | Amine | Adrenergic | β1 | Meleagris gallopavo | 4-(piperazin-1- yl)-1H-indole | Na | - | 2.8 | 2013-04-03 | 10.1021/jm400140q | |
4IAR | A | Amine | 5-Hydroxytryptamine | 5-HT1B | Homo sapiens | Ergotamine | - | - | 2.7 | 2013-03-13 | 10.1126/science.1232807 | |
4IAQ | A | Amine | 5-Hydroxytryptamine | 5-HT1B | Homo sapiens | Dihydroergotamine | - | - | 2.8 | 2013-03-13 | 10.1126/science.1232807 | |
4IB4 | A | Amine | 5-Hydroxytryptamine | 5-HT2B | Homo sapiens | Ergotamine | - | - | 2.7 | 2013-03-13 | 10.1126/science.1232808 | |
4GPO | A | Amine | Adrenergic | β1 | Meleagris gallopavo | - | - | - | 3.5 | 2013-02-27 | 10.1038/nsmb.2504 | |
4GPO (Multimeric) | A | Amine | Adrenergic | β1 | Meleagris gallopavo | - | - | 3.5 | 2013-02-27 | 10.1038/nsmb.2504 | ||
3VW7 | A | Peptide | Proteinase Activated | PAR1 | Homo sapiens | - | Vorapaxar; Na | - | 2.2 | 2012-12-12 | 10.1038/nature11701 | |
4GBR | A | Amine | Adrenergic | β2 | Homo sapiens | S-Carazolol | - | - | 3.99 | 2012-10-24 | 10.1371/journal.pone.0046039 | |
4GRV | A | Peptide | Neurotensin | NTS1 | Rattus norvegicus | Neurotensin-(8-13) | - | - | 2.8 | 2012-10-17 | 10.1038/nature11558 | |
4EIY | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | Na | - | 1.8 | 2012-07-25 | 10.1126/science.1219218 | |
4AMJ | A | Amine | Adrenergic | β1 | Meleagris gallopavo | S-Carvedilol | - | - | 2.3 | 2012-05-23 | 10.1016/j.str.2012.03.014 | |
4AMI | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Bucindolol | - | - | 3.2 | 2012-05-23 | 10.1016/j.str.2012.03.014 | |
4EJ4 | A | Peptide | Opioid | δ | Mus musculus | Naltrindole | - | - | 3.4 | 2012-05-16 | 10.1038/nature11111 | |
4EA3 | A | Peptide | Opioid | NOP | Homo sapiens | PubChem 10296561 | - | - | 3.01 | 2012-04-25 | 10.1038/nature11085 | |
3UZC | A | Nucleotide | Adenosine | A2A | Homo sapiens | 4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol | - | - | 3.34 | 2012-03-21 | 10.1021/jm201376w | |
3UZA | A | Nucleotide | Adenosine | A2A | Homo sapiens | GTPL9236 | - | - | 3.27 | 2012-03-21 | 10.1021/jm201376w | |
4DJH | A | Peptide | Opioid | κ | Homo sapiens | JDTic | - | - | 2.9 | 2012-03-21 | 10.1038/nature10939 | |
4DJH (Multimeric) | A | Peptide | Opioid | κ | Homo sapiens | JDTic | - | 2.9 | 2012-03-21 | 10.1038/nature10939 | ||
4DKL | A | Peptide | Opioid | μ | Mus musculus | β-Funaltrexamine | - | - | 2.8 | 2012-03-21 | 10.1038/nature10954 | |
4DAJ | A | Amine | Acetylcholine (muscarinic) | M3 | Rattus norvegicus | Tiotropium | - | - | 3.4 | 2012-02-22 | 10.1038/nature10867 | |
3V2Y | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | PubChem 51892645 | - | - | 2.8 | 2012-02-15 | 10.1126/science.1215904 | |
3V2W | A | Lipid | Lysophospholipid | S1P1 | Homo sapiens | PubChem 51892645 | - | - | 3.35 | 2012-02-15 | 10.1126/science.1215904 | |
3VGA | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | Antibody | - | 3.1 | 2012-02-01 | 10.1038/nature10750 | |
3VG9 | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | Antibody | - | 2.7 | 2012-02-01 | 10.1038/nature10750 | |
3UON | A | Amine | Acetylcholine (muscarinic) | M2 | Homo sapiens | 3-quinuclidinyl-benzilate | - | - | 3 | 2012-02-01 | 10.1038/nature10753 | |
4A4M | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | Gt(CT) | 3.3 | 2012-01-25 | 10.1073/pnas.1114089108 | |
4A4M (No Gprot) | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | 3.3 | 2012-01-25 | 10.1073/pnas.1114089108 | ||
3RFM | A | Nucleotide | Adenosine | A2A | Homo sapiens | Caffeine | - | - | 3.6 | 2011-09-07 | 10.1016/j.str.2011.06.014 | |
3REY | A | Nucleotide | Adenosine | A2A | Homo sapiens | XAC | - | - | 3.31 | 2011-09-07 | 10.1016/j.str.2011.06.014 | |
3PWH | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | - | - | 3.3 | 2011-09-07 | 10.1016/j.str.2011.06.014 | |
3AYN | A | Sensory | Opsins | Rhodopsin | Todarodes pacificus | 9-cis-Retinal | - | - | 2.7 | 2011-08-17 | 10.1016/j.jmb.2011.08.044 | |
3AYM | A | Sensory | Opsins | Rhodopsin | Todarodes pacificus | All-trans-Retinal | - | - | 2.8 | 2011-08-17 | 10.1016/j.jmb.2011.08.044 | |
3SN6 | A | Amine | Adrenergic | β2 | Homo sapiens | BI167107 | - | Gs/β1/γ2 | 3.2 | 2011-07-20 | 10.1038/nature10361 | |
3SN6 (No Gprot) | A | Amine | Adrenergic | β2 | Homo sapiens | BI167107 | - | 3.2 | 2011-07-20 | 10.1038/nature10361 | ||
3RZE | A | Amine | Histamine | H1 | Homo sapiens | Cidoxepin | - | - | 3.1 | 2011-06-15 | 10.1038/nature10236 | |
2YCY | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Cyanopindolol | - | - | 3.15 | 2011-06-08 | 10.1073/pnas.1100185108 | |
2YCZ | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Iodocyanopindolol | - | - | 3.65 | 2011-06-01 | 10.1073/pnas.1100185108 | |
2YCX | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Cyanopindolol | - | - | 3.25 | 2011-06-01 | 10.1073/pnas.1100185108 | |
2YCW | A | Amine | Adrenergic | β1 | Meleagris gallopavo | S-Carazolol | - | - | 3 | 2011-06-01 | 10.1073/pnas.1100185108 | |
2YDV | A | Nucleotide | Adenosine | A2A | Homo sapiens | NECA | - | - | 2.6 | 2011-05-18 | 10.1038/nature10136 | |
2YDO | A | Nucleotide | Adenosine | A2A | Homo sapiens | Adenosine | - | - | 3 | 2011-05-18 | 10.1038/nature10136 | |
2Y01 | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Dobutamine | - | - | 2.6 | 2011-03-30 | 10.1038/nature09746 | |
2X72 | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | Gt(CT) | 3 | 2011-03-16 | 10.1038/nature09795 | |
2X72 (No Gprot) | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | 3 | 2011-03-16 | 10.1038/nature09795 | ||
3QAK | A | Nucleotide | Adenosine | A2A | Homo sapiens | UK-432097 | - | - | 2.71 | 2011-03-09 | 10.1126/science.1202793 | |
3PXO | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | - | 3 | 2011-03-09 | 10.1038/nature09789 | |
3PQR | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | Gt(CT) | 2.85 | 2011-03-09 | 10.1038/nature09789 | |
3PQR (No Gprot) | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | 2.85 | 2011-03-09 | 10.1038/nature09789 | ||
3P0G | A | Amine | Adrenergic | β2 | Homo sapiens | BI167107 | - | - | 3.5 | 2011-01-19 | 10.1038/nature09648 | |
3OAX | A | Sensory | Opsins | Rhodopsin | Bos taurus | 11-cis-Retinal | - | - | 2.6 | 2011-01-19 | 10.1016/j.bpj.2010.08.003 | |
2Y04 | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Salbutamol | - | - | 3.05 | 2011-01-12 | 10.1038/nature09746 | |
2Y03 | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Isoprenaline | - | - | 2.85 | 2011-01-12 | 10.1038/nature09746 | |
2Y02 | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Carmoterol | - | - | 2.6 | 2011-01-12 | 10.1038/nature09746 | |
2Y00 | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Dobutamine | - | - | 2.5 | 2011-01-12 | 10.1038/nature09746 | |
3PDS | A | Amine | Adrenergic | β2 | Homo sapiens | Hydroxybenzylisoproterenol | - | - | 3.5 | 2011-01-12 | 10.1038/nature09665 | |
3PBL | A | Amine | Dopamine | D3 | Homo sapiens | Eticlopride | - | - | 2.89 | 2010-11-03 | 10.1126/science.1197410 | |
3OE9 | A | Protein | Chemokine | CXCR4 | Homo sapiens | IT1t | - | - | 3.1 | 2010-10-27 | 10.1126/science.1194396 | |
3OE9 (Multimeric) | A | Protein | Chemokine | CXCR4 | Homo sapiens | IT1t | - | 3.1 | 2010-10-27 | 10.1126/science.1194396 | ||
3OE8 | A | Protein | Chemokine | CXCR4 | Homo sapiens | IT1t | - | - | 3.1 | 2010-10-27 | 10.1126/science.1194396 | |
3OE8 (Multimeric) | A | Protein | Chemokine | CXCR4 | Homo sapiens | IT1t | - | 3.1 | 2010-10-27 | 10.1126/science.1194396 | ||
3OE6 | A | Protein | Chemokine | CXCR4 | Homo sapiens | IT1t | - | - | 3.2 | 2010-10-27 | 10.1126/science.1194396 | |
3OE0 | A | Protein | Chemokine | CXCR4 | Homo sapiens | CVX15 | - | - | 2.9 | 2010-10-27 | 10.1126/science.1194396 | |
3ODU | A | Protein | Chemokine | CXCR4 | Homo sapiens | IT1t | - | - | 2.5 | 2010-10-27 | 10.1126/science.1194396 | |
3ODU (Multimeric) | A | Protein | Chemokine | CXCR4 | Homo sapiens | IT1t | - | 2.5 | 2010-10-27 | 10.1126/science.1194396 | ||
3NYA | A | Amine | Adrenergic | β2 | Homo sapiens | S-Alprenolol | - | - | 3.16 | 2010-08-11 | 10.1021/ja105108q | |
3NY9 | A | Amine | Adrenergic | β2 | Homo sapiens | ICI118-551 | - | - | 2.84 | 2010-08-11 | 10.1021/ja105108q | |
3NY8 | A | Amine | Adrenergic | β2 | Homo sapiens | ICI118-551 | - | - | 2.84 | 2010-08-11 | 10.1021/ja105108q | |
3KJ6 | A | Amine | Adrenergic | β2 | Homo sapiens | - | - | - | 3.4 | 2010-02-16 | 10.1038/nature08650 | |
3EML | A | Nucleotide | Adenosine | A2A | Homo sapiens | ZM-241385 | - | - | 2.6 | 2008-10-14 | 10.1126/science.1164772 | |
3DQB | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | - | Gt(CT) | 3.2 | 2008-09-23 | 10.1038/nature07330 | |
3DQB (No Gprot) | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | - | 3.2 | 2008-09-23 | 10.1038/nature07330 | ||
3C9M | A | Sensory | Opsins | Rhodopsin | Bos taurus | 11-cis-Retinal | - | - | 3.4 | 2008-08-05 | 10.1107/S0907444908017162 | |
3C9L | A | Sensory | Opsins | Rhodopsin | Bos taurus | 11-cis-Retinal | - | - | 2.65 | 2008-08-05 | 10.1107/S0907444908017162 | |
2VT4 | A | Amine | Adrenergic | β1 | Meleagris gallopavo | Cyanopindolol | - | - | 2.7 | 2008-06-24 | 10.1038/nature07101 | |
3CAP | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | - | - | 2.9 | 2008-06-24 | 10.1038/nature07063 | |
3CAP (Multimeric) | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | - | 2.9 | 2008-06-24 | 10.1038/nature07063 | ||
3D4S | A | Amine | Adrenergic | β2 | Homo sapiens | Timolol | - | - | 2.8 | 2008-06-17 | 10.1016/j.str.2008.05.001 | |
2Z73 | A | Sensory | Opsins | Rhodopsin | Todarodes pacificus | 11-cis-Retinal | - | - | 2.5 | 2008-05-13 | 10.1038/nature06925 | |
2ZIY | A | Sensory | Opsins | Rhodopsin | Todarodes pacificus | 11-cis-Retinal | - | - | 3.7 | 2008-05-06 | 10.1074/jbc.C800040200 | |
2R4S | A | Amine | Adrenergic | β2 | Homo sapiens | - | - | - | 3.4 | 2007-11-06 | 10.1038/nature06325 | |
2R4R | A | Amine | Adrenergic | β2 | Homo sapiens | - | - | - | 3.4 | 2007-11-06 | 10.1038/nature06325 | |
2RH1 | A | Amine | Adrenergic | β2 | Homo sapiens | S-Carazolol | - | - | 2.4 | 2007-10-30 | 10.1126/science.1150577 | |
2PED | A | Sensory | Opsins | Rhodopsin | Bos taurus | 9-cis-Retinal | - | - | 2.95 | 2007-10-30 | 10.1529/biophysj.107.108225 | |
2J4Y | A | Sensory | Opsins | Rhodopsin | Bos taurus | 11-cis-Retinal | - | - | 3.4 | 2007-09-25 | 10.1016/j.jmb.2007.03.007 | |
2I37 | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | - | - | 4.15 | 2006-10-17 | 10.1073/pnas.0608022103 | |
2I36 | A | Sensory | Opsins | Rhodopsin | Bos taurus | - | - | - | 4.1 | 2006-10-17 | 10.1073/pnas.0608022103 | |
2I35 | A | Sensory | Opsins | Rhodopsin | Bos taurus | 11-cis-Retinal | - | - | 3.8 | 2006-10-17 | 10.1073/pnas.0608022103 | |
2G87 | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | - | 2.6 | 2006-09-02 | 10.1002/anie.200600595 | |
2HPY | A | Sensory | Opsins | Rhodopsin | Bos taurus | All-trans-Retinal | - | - | 2.8 | 2006-08-22 | 10.1073/pnas.0601765103 | |
1U19 | A | Sensory | Opsins | Rhodopsin | Bos taurus | 11-cis-Retinal | - | - | 2.2 | 2004-10-12 | 10.1016/j.jmb.2004.07.044 | |
1GZM | A | Sensory | Opsins | Rhodopsin | Bos taurus | 11-cis-Retinal | - | - | 2.65 | 2003-11-20 | 10.1016/j.jmb.2004.08.090 | |
1L9H | A | Sensory | Opsins | Rhodopsin | Bos taurus | 11-cis-Retinal | - | - | 2.6 | 2002-05-15 | 10.1073/pnas.082666399 | |
1HZX | A | Sensory | Opsins | Rhodopsin | Bos taurus | 11-cis-Retinal | - | - | 2.8 | 2001-07-04 | 10.1021/bi0155091 | |
1F88 | A | Sensory | Opsins | Rhodopsin | Bos taurus | 11-cis-Retinal | - | - | 2.8 | 2000-08-04 | 10.1126/science.289.5480.739 |