psnGPCRdb

Receptors → Single PSN

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Show: Click this button to access the corresponding database entry page.

PDB: PDB code of the receptor used to compute the network and a direct link to the corresponding entry in the Protein Data Bank.

Class: Receptor Class.

SubFamily: Receptor Sub Family.

Type: Receptor Type.

Subtype: Receptor SubType.

Species: Organism.

Orthosteric Ligand: Name of the orthosteric ligand, if present.

Other Ligand(s): Name of other allosteric ligands, if present.

Protein Partners: G Protein, Arrestin or Kinase coupled to a given receptor.

Resolution: Structure resolution.

Date: Deposition date.

DOI: DOI and link of the corresponding paper.


ShowPDBClassSubFamilyTypeSubTypeSpeciesOrthosteric LigandOther Ligand(s)Protein PartnersResolutionDateDOI
7E2XAAmine5-Hydroxytryptamine5-HT1AHomo sapiens--Gi1/β1/γ232021-04-14doi.org/10.1038/s41586-021-03376-8
7E2X (No Gprot) AAmine5-Hydroxytryptamine5-HT1AHomo sapiens--32021-04-14doi.org/10.1038/s41586-021-03376-8
7E2YAAmine5-Hydroxytryptamine5-HT1AHomo sapiensSerotonin-Gi1/β1/γ232021-04-14doi.org/10.1038/s41586-021-03376-8
7E2Y (No Gprot) AAmine5-Hydroxytryptamine5-HT1AHomo sapiensSerotonin-32021-04-14doi.org/10.1038/s41586-021-03376-8
7E2ZAAmine5-Hydroxytryptamine5-HT1AHomo sapiensAripiprazole-Gi1/β1/γ23.12021-04-14doi.org/10.1038/s41586-021-03376-8
7E2Z (No Gprot) AAmine5-Hydroxytryptamine5-HT1AHomo sapiensAripiprazole-3.12021-04-14doi.org/10.1038/s41586-021-03376-8
8W8BAAmine5-Hydroxytryptamine5-HT1AHomo sapiensSEP-363856-Gi1/β1/γ232023-11-22doi.org/10.1038/s41586-023-06775-1
8W8B (No Gprot) AAmine5-Hydroxytryptamine5-HT1AHomo sapiensSEP-363856-32023-11-22doi.org/10.1038/s41586-023-06775-1
8JSPAAmine5-Hydroxytryptamine5-HT1AHomo sapiensUlotaront-Gi1/β1/γ23.652023-11-15doi.org/10.1038/s41586-023-06804-z
8JSP (No Gprot) AAmine5-Hydroxytryptamine5-HT1AHomo sapiensUlotaront-3.652023-11-15doi.org/10.1038/s41586-023-06804-z
8FY8AAmine5-Hydroxytryptamine5-HT1AHomo sapiens5-MeO-DMT-Gi1/β1/γ12.792024-05-15doi.org/10.1038/s41586-024-07403-2
8FY8 (No Gprot) AAmine5-Hydroxytryptamine5-HT1AHomo sapiens5-MeO-DMT-2.792024-05-15doi.org/10.1038/s41586-024-07403-2
8FYEAAmine5-Hydroxytryptamine5-HT1AHomo sapiens4-F,5-MeO-PyrT-Gi1/β1/γ12.852024-05-15doi.org/10.1038/s41586-024-07403-2
8FYE (No Gprot) AAmine5-Hydroxytryptamine5-HT1AHomo sapiens4-F,5-MeO-PyrT-2.852024-05-15doi.org/10.1038/s41586-024-07403-2
8FYLAAmine5-Hydroxytryptamine5-HT1AHomo sapiensVilazodone-Gi1/β1/γ12.942024-05-15doi.org/10.1038/s41586-024-07403-2
8FYL (No Gprot) AAmine5-Hydroxytryptamine5-HT1AHomo sapiensVilazodone-2.942024-05-15doi.org/10.1038/s41586-024-07403-2
8FYTAAmine5-Hydroxytryptamine5-HT1AHomo sapiensLSD-Gi1/β1/γ12.642024-05-15doi.org/10.1038/s41586-024-07403-2
8FYT (No Gprot) AAmine5-Hydroxytryptamine5-HT1AHomo sapiensLSD-2.642024-05-15doi.org/10.1038/s41586-024-07403-2
8FYXAAmine5-Hydroxytryptamine5-HT1AHomo sapiensBuspirone-Gi1/β1/γ12.722024-05-15doi.org/10.1038/s41586-024-07403-2
8FYX (No Gprot) AAmine5-Hydroxytryptamine5-HT1AHomo sapiensBuspirone-2.722024-05-15doi.org/10.1038/s41586-024-07403-2
8JT6AAmine5-Hydroxytryptamine5-HT1AHomo sapiens(R)-IHCH-7179-Gi1/β1/γ232024-02-28doi.org/10.1016/j.cell.2024.02.034
8JT6 (No Gprot) AAmine5-Hydroxytryptamine5-HT1AHomo sapiens(R)-IHCH-7179-32024-02-28doi.org/10.1016/j.cell.2024.02.034
8PJKAAmine5-Hydroxytryptamine5-HT1AHomo sapiensST171-Gi1/β1/γ12.42024-05-29doi.org/10.1126/sciadv.adv9267
8PJK (No Gprot) AAmine5-Hydroxytryptamine5-HT1AHomo sapiensST171-2.42024-05-29doi.org/10.1126/sciadv.adv9267
8PKMAAmine5-Hydroxytryptamine5-HT1AHomo sapiensBefiradol-Gi1/β1/γ12.92024-05-29doi.org/10.1126/sciadv.adv9267
8PKM (No Gprot) AAmine5-Hydroxytryptamine5-HT1AHomo sapiensBefiradol-2.92024-05-29doi.org/10.1126/sciadv.adv9267
9GL2AAmine5-Hydroxytryptamine5-HT1AHomo sapiensBefiradol-Gs/β1/γ23.22025-07-02doi.org/10.1126/sciadv.adv9267
9GL2 (No Gprot) AAmine5-Hydroxytryptamine5-HT1AHomo sapiensBefiradol-3.22025-07-02doi.org/10.1126/sciadv.adv9267
5V54AAmine5-Hydroxytryptamine5-HT1BHomo sapiensMethiothepin--3.92018-02-07doi.org/10.1038/s41421-018-0009-2
6G79AAmine5-Hydroxytryptamine5-HT1BHomo sapiensDonitriptan-Go/β1/γ23.782018-06-20doi.org/10.1038/s41586-018-0241-9
6G79 (No Gprot) AAmine5-Hydroxytryptamine5-HT1BHomo sapiensDonitriptan-3.782018-06-20doi.org/10.1038/s41586-018-0241-9
7C61AAmine5-Hydroxytryptamine5-HT1BHomo sapiensErgotamine--32020-07-29doi.org/10.1038/s41598-020-68355-x
4IAQAAmine5-Hydroxytryptamine5-HT1BHomo sapiensDihydroergotamine--2.82013-03-13doi.org/10.1126/science.1232807
4IARAAmine5-Hydroxytryptamine5-HT1BHomo sapiensErgotamine--2.72013-03-13doi.org/10.1126/science.1232807
7E32AAmine5-Hydroxytryptamine5-HT1DHomo sapiensSerotonin-Gi1/β1/γ22.92021-04-21doi.org/10.1038/s41586-021-03376-8
7E32 (No Gprot) AAmine5-Hydroxytryptamine5-HT1DHomo sapiensSerotonin-2.92021-04-21doi.org/10.1038/s41586-021-03376-8
7E33AAmine5-Hydroxytryptamine5-HT1EHomo sapiensBRL-54443-Gi1/β1/γ22.92021-04-14doi.org/10.1038/s41586-021-03376-8
7E33 (No Gprot) AAmine5-Hydroxytryptamine5-HT1EHomo sapiensBRL-54443-2.92021-04-14doi.org/10.1038/s41586-021-03376-8
8UGYAAmine5-Hydroxytryptamine5-HT1EHomo sapiensMianserin-Gi1/β1/γ13.312024-05-01doi.org/10.1126/sciadv.adk4855
8UGY (No Gprot) AAmine5-Hydroxytryptamine5-HT1EHomo sapiensMianserin-3.312024-05-01doi.org/10.1126/sciadv.adk4855
8UH3AAmine5-Hydroxytryptamine5-HT1EHomo sapiensSetiptiline-Gi1/β1/γ13.312024-05-01doi.org/10.1126/sciadv.adk4855
8UH3 (No Gprot) AAmine5-Hydroxytryptamine5-HT1EHomo sapiensSetiptiline-3.312024-05-01doi.org/10.1126/sciadv.adk4855
7EXDAAmine5-Hydroxytryptamine5-HT1FHomo sapiensLasmiditan-Gi1/β1/γ23.42021-08-04doi.org/10.1038/s41422-021-00527-4
7EXD (No Gprot) AAmine5-Hydroxytryptamine5-HT1FHomo sapiensLasmiditan-3.42021-08-04doi.org/10.1038/s41422-021-00527-4
6WGTAAmine5-Hydroxytryptamine5-HT2AHomo sapiensLSD--3.42020-09-23doi.org/10.1016/j.cell.2020.08.024
6WH4AAmine5-Hydroxytryptamine5-HT2AHomo sapiensMethiothepin--3.42020-09-23doi.org/10.1016/j.cell.2020.08.024
6WHAAAmine5-Hydroxytryptamine5-HT2AHomo sapiensDB13948-chim(NtGi2L-Gs-CtGq)/β1/γ23.362020-09-23doi.org/10.1016/j.cell.2020.08.024
6WHA (No Gprot) AAmine5-Hydroxytryptamine5-HT2AHomo sapiensDB13948-3.362020-09-23doi.org/10.1016/j.cell.2020.08.024
8ZMGAAmine5-Hydroxytryptamine5-HT2AHomo sapiensPimavanserin--3.42024-08-28doi.org/10.1021/acs.jmedchem.4c01244
7RANAAmine5-Hydroxytryptamine5-HT2AHomo sapiensPubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ23.452022-07-06doi.org/10.1038/s41586-022-05258-z
7RAN (No Gprot) AAmine5-Hydroxytryptamine5-HT2AHomo sapiensPubChem 164575847-3.452022-07-06doi.org/10.1038/s41586-022-05258-z
7VODAAmine5-Hydroxytryptamine5-HT2AHomo sapiensCariprazine--3.32021-12-22doi.org/10.1038/s41593-021-00971-w
7VOEAAmine5-Hydroxytryptamine5-HT2AHomo sapiensAripiprazole--2.92021-12-22doi.org/10.1038/s41593-021-00971-w
6A93AAmine5-Hydroxytryptamine5-HT2AHomo sapiensRisperidone--32019-02-13doi.org/10.1038/s41594-018-0180-z
6A94AAmine5-Hydroxytryptamine5-HT2AHomo sapiensZotepine--2.92019-02-13doi.org/10.1038/s41594-018-0180-z
7WC4AAmine5-Hydroxytryptamine5-HT2AHomo sapiensSerotonin--3.22022-01-26doi.org/10.1126/science.abl8615
7WC5AAmine5-Hydroxytryptamine5-HT2AHomo sapiensPsilocin--3.22022-01-26doi.org/10.1126/science.abl8615
7WC6AAmine5-Hydroxytryptamine5-HT2AHomo sapiensLSD--2.62022-01-26doi.org/10.1126/science.abl8615
7WC7AAmine5-Hydroxytryptamine5-HT2AHomo sapiensLisuride--2.62022-01-26doi.org/10.1126/science.abl8615
7WC8AAmine5-Hydroxytryptamine5-HT2AHomo sapiensLumateperone--2.452022-01-26doi.org/10.1126/science.abl8615
7WC9AAmine5-Hydroxytryptamine5-HT2AHomo sapiensPubChem 162421364--2.52022-01-26doi.org/10.1126/science.abl8615
8UWLAAmine5-Hydroxytryptamine5-HT2AHomo sapiensLisuride-chim(NtGi2-Gs-CtGq)/β1/γ22.82024-05-29doi.org/10.1126/science.adn6354
8UWL (No Gprot) AAmine5-Hydroxytryptamine5-HT2AHomo sapiensLisuride-2.82024-05-29doi.org/10.1126/science.adn6354
8V6UAAmine5-Hydroxytryptamine5-HT2AHomo sapiensPubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ232024-05-29doi.org/10.1126/science.adn6354
8V6U (No Gprot) AAmine5-Hydroxytryptamine5-HT2AHomo sapiensPubChem 171392456-32024-05-29doi.org/10.1126/science.adn6354
8JT8AAmine5-Hydroxytryptamine5-HT2AHomo sapiens(R)-IHCH-7179--2.72024-02-28doi.org/10.1016/j.cell.2024.02.034
9ARXAAmine5-Hydroxytryptamine5-HT2AHomo sapiensSerotonin--3.242025-04-02doi.org/10.1038/s41467-025-57956-7
9ARYAAmine5-Hydroxytryptamine5-HT2AHomo sapiensSerotonin-chim(NtGi1-Gs-CtGq)/β1/γ23.272025-04-02doi.org/10.1038/s41467-025-57956-7
9ARY (No Gprot) AAmine5-Hydroxytryptamine5-HT2AHomo sapiensSerotonin-3.272025-04-02doi.org/10.1038/s41467-025-57956-7
9ARZAAmine5-Hydroxytryptamine5-HT2AHomo sapiens2-bromo-LSD--3.372025-04-02doi.org/10.1038/s41467-025-57956-7
9AS0AAmine5-Hydroxytryptamine5-HT2AHomo sapiens2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ23.382025-04-02doi.org/10.1038/s41467-025-57956-7
9AS0 (No Gprot) AAmine5-Hydroxytryptamine5-HT2AHomo sapiens2-bromo-LSD-3.382025-04-02doi.org/10.1038/s41467-025-57956-7
9AS1AAmine5-Hydroxytryptamine5-HT2AHomo sapiensDMT--3.382025-04-02doi.org/10.1038/s41467-025-57956-7
9AS2AAmine5-Hydroxytryptamine5-HT2AHomo sapiensDMT-chim(NtGi1-Gs-CtGq)/β1/γ23.212025-04-02doi.org/10.1038/s41467-025-57956-7
9AS2 (No Gprot) AAmine5-Hydroxytryptamine5-HT2AHomo sapiensDMT-3.212025-04-02doi.org/10.1038/s41467-025-57956-7
9AS3AAmine5-Hydroxytryptamine5-HT2AHomo sapiensLSD--3.182025-04-02doi.org/10.1038/s41467-025-57956-7
9AS4AAmine5-Hydroxytryptamine5-HT2AHomo sapiensLSD-chim(NtGi1-Gs-CtGq)/β1/γ23.062025-04-02doi.org/10.1038/s41467-025-57956-7
9AS4 (No Gprot) AAmine5-Hydroxytryptamine5-HT2AHomo sapiensLSD-3.062025-04-02doi.org/10.1038/s41467-025-57956-7
9AS5AAmine5-Hydroxytryptamine5-HT2AHomo sapiensMescaline--3.342025-04-02doi.org/10.1038/s41467-025-57956-7
9AS6AAmine5-Hydroxytryptamine5-HT2AHomo sapiensMescaline-chim(NtGi1-Gs-CtGq)/β1/γ23.072025-04-02doi.org/10.1038/s41467-025-57956-7
9AS6 (No Gprot) AAmine5-Hydroxytryptamine5-HT2AHomo sapiensMescaline-3.072025-04-02doi.org/10.1038/s41467-025-57956-7
9AS7AAmine5-Hydroxytryptamine5-HT2AHomo sapiensPsilocin--2.722025-04-02doi.org/10.1038/s41467-025-57956-7
9AS9AAmine5-Hydroxytryptamine5-HT2AHomo sapiensRS130-180--3.472025-04-02doi.org/10.1038/s41467-025-57956-7
9ASAAAmine5-Hydroxytryptamine5-HT2AHomo sapiensRS130-180-chim(NtGi1-Gs-CtGq)/β1/γ23.122025-04-02doi.org/10.1038/s41467-025-57956-7
9ASA (No Gprot) AAmine5-Hydroxytryptamine5-HT2AHomo sapiensRS130-180-3.122025-04-02doi.org/10.1038/s41467-025-57956-7
5TVNAAmine5-Hydroxytryptamine5-HT2BHomo sapiensLSD--2.92017-02-01doi.org/10.1016/j.cell.2016.12.033
7SRQAAmine5-Hydroxytryptamine5-HT2BHomo sapiensLSD--2.72022-09-21doi.org/10.1016/j.neuron.2022.08.006
7SRRAAmine5-Hydroxytryptamine5-HT2BHomo sapiensLSD-chim(NtGi2L-Gs-CtGq)/β1/γ22.92022-09-21doi.org/10.1016/j.neuron.2022.08.006
7SRR (No Gprot) AAmine5-Hydroxytryptamine5-HT2BHomo sapiensLSD-2.92022-09-21doi.org/10.1016/j.neuron.2022.08.006
7SRSAAmine5-Hydroxytryptamine5-HT2BHomo sapiensLSD-Arrestin23.32022-09-21doi.org/10.1016/j.neuron.2022.08.006
6DRXAAmine5-Hydroxytryptamine5-HT2BHomo sapiensLisuride--3.12018-08-29doi.org/10.1038/s41594-018-0116-7
6DRYAAmine5-Hydroxytryptamine5-HT2BHomo sapiensMethylergonovine--2.922018-08-29doi.org/10.1038/s41594-018-0116-7
6DRZAAmine5-Hydroxytryptamine5-HT2BHomo sapiensMethysergide--3.12018-08-29doi.org/10.1038/s41594-018-0116-7
6DS0AAmine5-Hydroxytryptamine5-HT2BHomo sapiensLy266097--3.192018-08-29doi.org/10.1038/s41594-018-0116-7
5TUDAAmine5-Hydroxytryptamine5-HT2BHomo sapiensErgotamine--32017-07-26doi.org/10.1073/pnas.1700891114
4IB4AAmine5-Hydroxytryptamine5-HT2BHomo sapiensErgotamine--2.72013-03-13doi.org/10.1126/science.1232808
4NC3AAmine5-Hydroxytryptamine5-HT2BHomo sapiensErgotamine--2.82013-12-18doi.org/10.1126/science.1244142
6BQGAAmine5-Hydroxytryptamine5-HT2CHomo sapiensErgotamine--32018-02-14doi.org/10.1016/j.cell.2018.01.001
6BQHAAmine5-Hydroxytryptamine5-HT2CHomo sapiensRitanserin--2.72018-02-14doi.org/10.1016/j.cell.2018.01.001
8DPFAAmine5-Hydroxytryptamine5-HT2CHomo sapiensLorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ22.842022-08-24doi.org/10.1016/j.celrep.2022.111211
8DPF (No Gprot) AAmine5-Hydroxytryptamine5-HT2CHomo sapiensLorcaserin-2.842022-08-24doi.org/10.1016/j.celrep.2022.111211
8DPGAAmine5-Hydroxytryptamine5-HT2CHomo sapiensPsilocin-chim(NtGi2L-Gs-CtGq)/β1/γ23.62022-08-24doi.org/10.1016/j.celrep.2022.111211
8DPG (No Gprot) AAmine5-Hydroxytryptamine5-HT2CHomo sapiensPsilocin-3.62022-08-24doi.org/10.1016/j.celrep.2022.111211
8DPHAAmine5-Hydroxytryptamine5-HT2CHomo sapiensLorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ23.22022-08-24doi.org/10.1016/j.celrep.2022.111211
8DPH (No Gprot) AAmine5-Hydroxytryptamine5-HT2CHomo sapiensLorcaserin-3.22022-08-24doi.org/10.1016/j.celrep.2022.111211
8DPIAAmine5-Hydroxytryptamine5-HT2CHomo sapiensLorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ23.42022-08-24doi.org/10.1016/j.celrep.2022.111211
8DPI (No Gprot) AAmine5-Hydroxytryptamine5-HT2CHomo sapiensLorcaserin-3.42022-08-24doi.org/10.1016/j.celrep.2022.111211
8ZMFAAmine5-Hydroxytryptamine5-HT2CHomo sapiensA1L10--3.62024-08-28doi.org/10.1021/acs.jmedchem.4c01244
7XT8AAmine5-Hydroxytryptamine5-HT4Homo sapiensSerotonin-Gs/β1/γ23.12022-07-27doi.org/10.1016/j.molcel.2022.05.031
7XT8 (No Gprot) AAmine5-Hydroxytryptamine5-HT4Homo sapiensSerotonin-3.12022-07-27doi.org/10.1016/j.molcel.2022.05.031
7XT9AAmine5-Hydroxytryptamine5-HT4Homo sapiensSerotonin-Gs/β1/γ23.22022-07-27doi.org/10.1016/j.molcel.2022.05.031
7XT9 (No Gprot) AAmine5-Hydroxytryptamine5-HT4Homo sapiensSerotonin-3.22022-07-27doi.org/10.1016/j.molcel.2022.05.031
7XTAAAmine5-Hydroxytryptamine5-HT4Homo sapiensSerotonin-Gi1/β1/γ23.22022-07-27doi.org/10.1016/j.molcel.2022.05.031
7XTA (No Gprot) AAmine5-Hydroxytryptamine5-HT4Homo sapiensSerotonin-3.22022-07-27doi.org/10.1016/j.molcel.2022.05.031
7X5HAAmine5-Hydroxytryptamine5-HT5AHomo sapiens5-CT-Gi1/β1/γ23.12022-09-14doi.org/10.1038/s41421-022-00412-3
7X5H (No Gprot) AAmine5-Hydroxytryptamine5-HT5AHomo sapiens5-CT-3.12022-09-14doi.org/10.1038/s41421-022-00412-3
7UM4AAmine5-Hydroxytryptamine5-HT5AHomo sapiensAS2674723--2.82022-07-20doi.org/10.1038/s41594-022-00796-6
7UM5AAmine5-Hydroxytryptamine5-HT5AHomo sapiens5-CT-chim(NtGi1-Go)/β1/γ22.732022-07-20doi.org/10.1038/s41594-022-00796-6
7UM5 (No Gprot) AAmine5-Hydroxytryptamine5-HT5AHomo sapiens5-CT-2.732022-07-20doi.org/10.1038/s41594-022-00796-6
7UM6AAmine5-Hydroxytryptamine5-HT5AHomo sapiensLisuride-chim(NtGi1-Go)/β1/γ22.792022-07-20doi.org/10.1038/s41594-022-00796-6
7UM6 (No Gprot) AAmine5-Hydroxytryptamine5-HT5AHomo sapiensLisuride-2.792022-07-20doi.org/10.1038/s41594-022-00796-6
7UM7AAmine5-Hydroxytryptamine5-HT5AHomo sapiensMethylergometrine-chim(NtGi1-Go)/β1/γ22.752022-07-20doi.org/10.1038/s41594-022-00796-6
7UM7 (No Gprot) AAmine5-Hydroxytryptamine5-HT5AHomo sapiensMethylergometrine-2.752022-07-20doi.org/10.1038/s41594-022-00796-6
8JLZAAmine5-Hydroxytryptamine5-HT6Homo sapiensST1936-Gs/β1/γ23.092023-06-28doi.org/10.1016/j.bbrc.2023.05.126
8JLZ (No Gprot) AAmine5-Hydroxytryptamine5-HT6Homo sapiensST1936-3.092023-06-28doi.org/10.1016/j.bbrc.2023.05.126
7XTBAAmine5-Hydroxytryptamine5-HT6Homo sapiensSerotonin-Gs/β1/γ23.32022-07-27doi.org/10.1016/j.molcel.2022.05.031
7XTB (No Gprot) AAmine5-Hydroxytryptamine5-HT6Homo sapiensSerotonin-3.32022-07-27doi.org/10.1016/j.molcel.2022.05.031
7YS6AAmine5-Hydroxytryptamine5-HT6Homo sapiensSerotonin-chim(NtGi1-Gs)/β1/γ232023-03-29doi.org/10.1073/pnas.2209917120
7YS6 (No Gprot) AAmine5-Hydroxytryptamine5-HT6Homo sapiensSerotonin-32023-03-29doi.org/10.1073/pnas.2209917120
7XTCAAmine5-Hydroxytryptamine5-HT7Homo sapiens5-CT-Gs/β1/γ23.22022-07-27doi.org/10.1016/j.molcel.2022.05.031
7XTC (No Gprot) AAmine5-Hydroxytryptamine5-HT7Homo sapiens5-CT-3.22022-07-27doi.org/10.1016/j.molcel.2022.05.031
8FX5AAmineAcetylcholine (muscarinic)M4Homo sapiensXanomelineXanomelineGi1/β1/γ22.452023-09-13doi.org/10.1038/s41467-023-41199-5
8FX5 (No Gprot) AAmineAcetylcholine (muscarinic)M4Homo sapiensXanomelineXanomeline2.452023-09-13doi.org/10.1038/s41467-023-41199-5
7TRQAAmineAcetylcholine (muscarinic)M4Homo sapiensIperoxoVU0467154Gi1/β1/γ22.52023-05-17doi.org/10.2139/ssrn.4034884
7TRQ (No Gprot) AAmineAcetylcholine (muscarinic)M4Homo sapiensIperoxoVU04671542.52023-05-17doi.org/10.2139/ssrn.4034884
7V6AAAmineAcetylcholine (muscarinic)M4Homo sapiens-PubChem 9864275Gi1/β1/γ23.62022-05-11doi.org/10.1038/s41467-022-30595-y
7V6A (No Gprot) AAmineAcetylcholine (muscarinic)M4Homo sapiens-PubChem 98642753.62022-05-11doi.org/10.1038/s41467-022-30595-y
6WJCAAmineAcetylcholine (muscarinic)M1Homo sapiensAtropineMuscarinic toxin 7-2.552020-07-08doi.org/10.1126/science.aax2517
4MQTAAmineAcetylcholine (muscarinic)M2Homo sapiensIperoxoLY2119620-3.72013-11-27doi.org/10.1038/nature12735
7T94AAmineAcetylcholine (muscarinic)M2Homo sapiensAcetylcholineLY2119620chim(NtGi1-Go)/β1/γ23.162023-01-25doi.org/10.1038/s41467-022-35726-z
7T94 (No Gprot) AAmineAcetylcholine (muscarinic)M2Homo sapiensAcetylcholineLY21196203.162023-01-25doi.org/10.1038/s41467-022-35726-z
6U1NAAmineAcetylcholine (muscarinic)M2Homo sapiens-LY2119620Arrestin242020-02-26doi.org/10.1038/s41586-020-1954-0
6OIKAAmineAcetylcholine (muscarinic)M2Homo sapiensIperoxoLY2119620chim(NtGi1-Go)/β1/γ23.62019-05-08doi.org/10.1126/science.aaw5188
6OIK (No Gprot) AAmineAcetylcholine (muscarinic)M2Homo sapiensIperoxoLY21196203.62019-05-08doi.org/10.1126/science.aaw5188
7T96AAmineAcetylcholine (muscarinic)M2Homo sapiensAcetylcholineLY2119620Go/β1/γ23.222023-01-25doi.org/10.1038/s41467-022-35726-z
7T96 (No Gprot) AAmineAcetylcholine (muscarinic)M2Homo sapiensAcetylcholineLY21196203.222023-01-25doi.org/10.1038/s41467-022-35726-z
7V68AAmineAcetylcholine (muscarinic)M4Homo sapiensIperoxoLY2119620Gi1/β1/γ23.42022-05-11doi.org/10.1038/s41467-022-30595-y
7V68 (No Gprot) AAmineAcetylcholine (muscarinic)M4Homo sapiensIperoxoLY21196203.42022-05-11doi.org/10.1038/s41467-022-30595-y
7TRPAAmineAcetylcholine (muscarinic)M4Homo sapiensIperoxoLY2033298Gi1/β1/γ22.42023-05-17doi.org/10.2139/ssrn.4034884
7TRP (No Gprot) AAmineAcetylcholine (muscarinic)M4Homo sapiensIperoxoLY20332982.42023-05-17doi.org/10.2139/ssrn.4034884
6ZFZAAmineAcetylcholine (muscarinic)M1Homo sapiens77-LH-28-1--2.172021-10-06doi.org/10.1016/j.cell.2021.11.001
6ZG4AAmineAcetylcholine (muscarinic)M1Homo sapiensHTL0009936--2.332021-10-06doi.org/10.1016/j.cell.2021.11.001
6ZG9AAmineAcetylcholine (muscarinic)M1Homo sapiensGSK1034702--2.52021-10-06doi.org/10.1016/j.cell.2021.11.001
5CXVAAmineAcetylcholine (muscarinic)M1Homo sapiensTiotropium--2.72016-03-09doi.org/10.1038/nature17188
6OIJAAmineAcetylcholine (muscarinic)M1Homo sapiensIperoxo-chim(NtGi1L-G11)/β1/γ23.32019-05-08doi.org/10.1126/science.aaw5188
6OIJ (No Gprot) AAmineAcetylcholine (muscarinic)M1Homo sapiensIperoxo-3.32019-05-08doi.org/10.1126/science.aaw5188
9JEAAAmineAcetylcholine (muscarinic)M1Homo sapiensAtropine--3.42025-07-09To be published
3UONAAmineAcetylcholine (muscarinic)M2Homo sapiens3-quinuclidinyl-benzilate--32012-02-01doi.org/10.1038/nature10753
4MQSAAmineAcetylcholine (muscarinic)M2Homo sapiensIperoxo--3.52013-11-27doi.org/10.1038/nature12735
7T8XAAmineAcetylcholine (muscarinic)M2Homo sapiensAcetylcholine-chim(NtGi1-Go)/β1/γ23.212023-01-25doi.org/10.1038/s41467-022-35726-z
7T8X (No Gprot) AAmineAcetylcholine (muscarinic)M2Homo sapiensAcetylcholine-3.212023-01-25doi.org/10.1038/s41467-022-35726-z
7T90AAmineAcetylcholine (muscarinic)M2Homo sapiensAcetylcholine-chim(NtGi1-Go)/β1/γ23.322023-01-25doi.org/10.1038/s41467-022-35726-z
7T90 (No Gprot) AAmineAcetylcholine (muscarinic)M2Homo sapiensAcetylcholine-3.322023-01-25doi.org/10.1038/s41467-022-35726-z
5YC8AAmineAcetylcholine (muscarinic)M2Homo sapiensN-Methyl-Scopolamine--2.52018-11-21doi.org/10.1038/s41589-018-0152-y
5ZK3AAmineAcetylcholine (muscarinic)M2Homo sapiens3-quinuclidinyl-benzilate--2.62018-11-21doi.org/10.1038/s41589-018-0152-y
5ZK8AAmineAcetylcholine (muscarinic)M2Homo sapiensN-Methyl-Scopolamine--32018-11-21doi.org/10.1038/s41589-018-0152-y
5ZKBAAmineAcetylcholine (muscarinic)M2Homo sapiensAF-DX 384--2.952018-11-21doi.org/10.1038/s41589-018-0152-y
5ZKCAAmineAcetylcholine (muscarinic)M2Homo sapiensN-Methyl-Scopolamine--2.32018-11-21doi.org/10.1038/s41589-018-0152-y
4U14AAmineAcetylcholine (muscarinic)M3Rattus norvegicusTiotropium--3.572014-11-26doi.org/10.1016/j.str.2014.08.022
4U15AAmineAcetylcholine (muscarinic)M3Rattus norvegicusTiotropium--2.82014-11-26doi.org/10.1016/j.str.2014.08.022
4U16AAmineAcetylcholine (muscarinic)M3Rattus norvegicusN-Methyl-Scopolamine--3.72014-11-26doi.org/10.1016/j.str.2014.08.022
4DAJAAmineAcetylcholine (muscarinic)M3Rattus norvegicusTiotropium--3.42012-02-22doi.org/10.1038/nature10867
8E9WAAmineAcetylcholine (muscarinic)M3Homo sapiens2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ22.692022-11-30doi.org/10.1038/s41586-022-05489-0
8E9W (No Gprot) AAmineAcetylcholine (muscarinic)M3Homo sapiens2-Deoxycytidine-2.692022-11-30doi.org/10.1038/s41586-022-05489-0
8E9YAAmineAcetylcholine (muscarinic)M3Homo sapiensClozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ22.792022-11-30doi.org/10.1038/s41586-022-05489-0
8E9Y (No Gprot) AAmineAcetylcholine (muscarinic)M3Homo sapiensClozapine-N-oxide-2.792022-11-30doi.org/10.1038/s41586-022-05489-0
8E9ZAAmineAcetylcholine (muscarinic)M3Homo sapiensIperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ22.692022-11-30doi.org/10.1038/s41586-022-05489-0
8E9Z (No Gprot) AAmineAcetylcholine (muscarinic)M3Homo sapiensIperoxo-2.692022-11-30doi.org/10.1038/s41586-022-05489-0
8EA0AAmineAcetylcholine (muscarinic)M3Homo sapiensIperoxo--2.562022-11-30doi.org/10.1038/s41586-022-05489-0
5ZHPAAmineAcetylcholine (muscarinic)M3Rattus norvegicusPubChem 134828589--3.12018-11-28doi.org/10.1073/pnas.1813988115
5DSGAAmineAcetylcholine (muscarinic)M4Homo sapiensTiotropium--2.62016-03-16doi.org/10.1038/nature17188
7V69AAmineAcetylcholine (muscarinic)M4Homo sapiens--Gi1/β1/γ23.42022-05-11doi.org/10.1038/s41467-022-30595-y
7V69 (No Gprot) AAmineAcetylcholine (muscarinic)M4Homo sapiens--3.42022-05-11doi.org/10.1038/s41467-022-30595-y
8E9XAAmineAcetylcholine (muscarinic)M4Homo sapiens2-Deoxycytidine-chim(NtGi1-Go)/β1/γ22.72022-11-30doi.org/10.1038/s41586-022-05489-0
8E9X (No Gprot) AAmineAcetylcholine (muscarinic)M4Homo sapiens2-Deoxycytidine-2.72022-11-30doi.org/10.1038/s41586-022-05489-0
6KP6AAmineAcetylcholine (muscarinic)M4Homo sapiens---32020-03-11doi.org/10.1107/S2052252520000597
7TRKAAmineAcetylcholine (muscarinic)M4Homo sapiensIperoxo-Gi1/β1/γ22.82023-05-17doi.org/10.2139/ssrn.4034884
7TRK (No Gprot) AAmineAcetylcholine (muscarinic)M4Homo sapiensIperoxo-2.82023-05-17doi.org/10.2139/ssrn.4034884
7TRSAAmineAcetylcholine (muscarinic)M4Homo sapiensAcetylcholine-Gi1/β1/γ22.82023-05-17doi.org/10.2139/ssrn.4034884
7TRS (No Gprot) AAmineAcetylcholine (muscarinic)M4Homo sapiensAcetylcholine-2.82023-05-17doi.org/10.2139/ssrn.4034884
6OL9AAmineAcetylcholine (muscarinic)M5Homo sapiensTiotropium--2.542019-12-11doi.org/10.1073/pnas.1914446116
6ZDRANucleotideAdenosineA2AHomo sapiensHMS1413f12Na-1.922020-09-16doi.org/10.1002/anie.202003788
6ZDVANucleotideAdenosineA2AHomo sapiensChromone 5dNa-2.132020-09-16doi.org/10.1002/anie.202003788
8JWZANucleotideAdenosineA2AHomo sapiensAB928Na-2.372023-08-16doi.org/10.1007/s11427-023-2459-8
5MZJANucleotideAdenosineA2AHomo sapiensTheophyllineNa-22017-07-26doi.org/10.1016/j.str.2017.06.012
5MZPANucleotideAdenosineA2AHomo sapiensCaffeineNa-2.12017-07-26doi.org/10.1016/j.str.2017.06.012
5N2RANucleotideAdenosineA2AHomo sapiensPSB-36Na-2.82017-07-26doi.org/10.1016/j.str.2017.06.012
7AROANucleotideAdenosineA2AHomo sapiensLUF5833Na-3.122021-04-07doi.org/10.1021/acs.jmedchem.0c01856
8CU7ANucleotideAdenosineA2AHomo sapiensLJ-4517Na-2.052022-08-31doi.org/10.1021/acs.jmedchem.2c00462
5IU4ANucleotideAdenosineA2AHomo sapiensZM-241385Na-1.722016-06-29doi.org/10.1021/acs.jmedchem.6b00653
5IU7ANucleotideAdenosineA2AHomo sapiensQ27456346Na-1.92016-06-29doi.org/10.1021/acs.jmedchem.6b00653
5IU8ANucleotideAdenosineA2AHomo sapiensQ27456347Na-22016-06-29doi.org/10.1021/acs.jmedchem.6b00653
5IUAANucleotideAdenosineA2AHomo sapiensQ27456348Na-2.22016-06-29doi.org/10.1021/acs.jmedchem.6b00653
5IUBANucleotideAdenosineA2AHomo sapiensQ27456344Na-2.12016-06-29doi.org/10.1021/acs.jmedchem.6b00653
5VRAANucleotideAdenosineA2AHomo sapiensZM-241385Na-2.352017-12-13doi.org/10.1038/nprot.2017.135
5NLXANucleotideAdenosineA2AHomo sapiensZM-241385Na-2.142017-09-27doi.org/10.1038/s41467-017-00630-4
5NM2ANucleotideAdenosineA2AHomo sapiensZM-241385Na-1.952017-09-27doi.org/10.1038/s41467-017-00630-4
5NM4ANucleotideAdenosineA2AHomo sapiensZM-241385Na-1.72017-09-27doi.org/10.1038/s41467-017-00630-4
8FYNANucleotideAdenosineA2AHomo sapiensZM-241385Na-22023-03-08doi.org/10.1038/s41467-023-36733-4
8RW0ANucleotideAdenosineA2AHomo sapiensIstradefyllineNa-1.942025-01-08doi.org/10.1038/s41467-024-55109-w
5OLGANucleotideAdenosineA2AHomo sapiensZM-241385Na-1.872018-01-17doi.org/10.1038/s41598-017-18570-w
5OLHANucleotideAdenosineA2AHomo sapiensVipadenantNa-2.62018-01-17doi.org/10.1038/s41598-017-18570-w
5OLOANucleotideAdenosineA2AHomo sapiensTozadenantNa-3.12018-01-17doi.org/10.1038/s41598-017-18570-w
5OLVANucleotideAdenosineA2AHomo sapiensLUAA41063Na-22018-01-17doi.org/10.1038/s41598-017-18570-w
5OLZANucleotideAdenosineA2AHomo sapiensPubChem 135566609Na-1.92018-01-17doi.org/10.1038/s41598-017-18570-w
5OM1ANucleotideAdenosineA2AHomo sapiensPubChem 135566609Na-2.12018-01-17doi.org/10.1038/s41598-017-18570-w
5OM4ANucleotideAdenosineA2AHomo sapiensPubChem 135566609Na-22018-01-17doi.org/10.1038/s41598-017-18570-w
6LPJANucleotideAdenosineA2AHomo sapiensZM-241385Na-1.82020-11-25doi.org/10.1038/s41598-020-76277-x
6LPKANucleotideAdenosineA2AHomo sapiensZM-241385Na-1.82020-11-25doi.org/10.1038/s41598-020-76277-x
6LPLANucleotideAdenosineA2AHomo sapiensZM-241385Na-22020-11-25doi.org/10.1038/s41598-020-76277-x
8CICANucleotideAdenosineA2AHomo sapiensEtrumadenantNa-2.12023-05-31doi.org/10.1038/s42004-023-00894-6
7RM5ANucleotideAdenosineA2AHomo sapiensZM-241385Na-2.792021-09-08doi.org/10.1073/pnas.2106041118
6JZHANucleotideAdenosineA2AHomo sapiensZM-241385Na-2.252019-10-30doi.org/10.1107/S1600576719012846
8A2OANucleotideAdenosineA2AHomo sapiensTheophyllineNa-3.452023-08-30doi.org/10.1107/S1600576723006428
8A2PANucleotideAdenosineA2AHomo sapiensLUAA47070Na-3.52023-08-30doi.org/10.1107/S1600576723006428
6PS7ANucleotideAdenosineA2AHomo sapiensZM-241385Na-1.852019-11-13doi.org/10.1107/S2052252519013137
6WQAANucleotideAdenosineA2AHomo sapiensZM-241385Na-22020-11-18doi.org/10.1107/S2052252520012701
8GNEANucleotideAdenosineA2AHomo sapiensKW-6356Na-2.32023-03-22doi.org/10.1124/molpharm.122.000633
5K2AANucleotideAdenosineA2AHomo sapiensZM-241385Na-2.52016-09-21doi.org/10.1126/sciadv.1600292
5K2BANucleotideAdenosineA2AHomo sapiensZM-241385Na-2.52016-09-21doi.org/10.1126/sciadv.1600292
5K2CANucleotideAdenosineA2AHomo sapiensZM-241385Na-1.92016-09-21doi.org/10.1126/sciadv.1600292
5K2DANucleotideAdenosineA2AHomo sapiensZM-241385Na-1.92016-09-21doi.org/10.1126/sciadv.1600292
4EIYANucleotideAdenosineA2AHomo sapiensZM-241385Na-1.82012-07-25doi.org/10.1126/science.1219218
6GT3ANucleotideAdenosineA2AHomo sapiensImaradenantNa-22019-06-26doi.org/10.1136/jitc-2019-000417
8RQQANucleotideAdenosineA2AHomo sapiensZM-241385Na-2.372024-04-03doi.org/10.1021/acs.cgd.4c00087
8RVWANucleotideAdenosineA2AHomo sapiensStilSwitch3Na-2.652025-01-08doi.org/10.1038/s41467-024-55109-w
8RW4ANucleotideAdenosineA2AHomo sapiensAzoSwitch2Na-2.22025-01-08doi.org/10.1038/s41467-024-55109-w
8RW7ANucleotideAdenosineA2AHomo sapiensStilSwitch1Na-2.252025-01-08doi.org/10.1038/s41467-024-55109-w
8RWCANucleotideAdenosineA2AHomo sapiensStilSwitch2Na-2.312025-01-08doi.org/10.1038/s41467-024-55109-w
8RWDANucleotideAdenosineA2AHomo sapiensStilSwitch3Na-2.052025-01-08doi.org/10.1038/s41467-024-55109-w
8RWEANucleotideAdenosineA2AHomo sapiensStilSwitch4Na-2.22025-01-08doi.org/10.1038/s41467-024-55109-w
8RWHANucleotideAdenosineA2AHomo sapiensStilSwitch2Na-2.452025-01-08doi.org/10.1038/s41467-024-55109-w
8RWIANucleotideAdenosineA2AHomo sapiensStilSwitch2Na-2.82025-01-08doi.org/10.1038/s41467-024-55109-w
8RWXANucleotideAdenosineA2AHomo sapiensStilSwitch3Na-3.052025-01-08doi.org/10.1038/s41467-024-55109-w
9FUPANucleotideAdenosineA2AHomo sapiensIstradefyllineNa-2.52025-01-22doi.org/10.1038/s42004-024-01404-y
9H2XANucleotideAdenosineA2AHomo sapiensA1IR1Na-1.752025-06-18To be published
9H37ANucleotideAdenosineA2AHomo sapiensA1IR0Na-1.712025-06-18To be published
7LD3ANucleotideAdenosineA1Homo sapiensAdenosineMIPS521Gi2/β1/γ23.22021-09-08doi.org/10.1038/s41586-021-03897-2
7LD3 (No Gprot) ANucleotideAdenosineA1Homo sapiensAdenosineMIPS5213.22021-09-08doi.org/10.1038/s41586-021-03897-2
3VG9ANucleotideAdenosineA2AHomo sapiensZM-241385Antibody-2.72012-02-01doi.org/10.1038/nature10750
3VGAANucleotideAdenosineA2AHomo sapiensZM-241385Antibody-3.12012-02-01doi.org/10.1038/nature10750
5UENANucleotideAdenosineA1Homo sapiensDU172--3.22017-03-01doi.org/10.1016/j.cell.2017.01.042
5N2SANucleotideAdenosineA1Homo sapiensPSB36--3.32017-07-26doi.org/10.1016/j.str.2017.06.012
6D9HANucleotideAdenosineA1Homo sapiensAdenosine-Gi2/β1/γ23.62018-06-20doi.org/10.1038/s41586-018-0236-6
6D9H (No Gprot) ANucleotideAdenosineA1Homo sapiensAdenosine-3.62018-06-20doi.org/10.1038/s41586-018-0236-6
7LD4ANucleotideAdenosineA1Homo sapiensAdenosine-Gi2/β1/γ23.32021-09-08doi.org/10.1038/s41586-021-03897-2
7LD4 (No Gprot) ANucleotideAdenosineA1Homo sapiensAdenosine-3.32021-09-08doi.org/10.1038/s41586-021-03897-2
7PX4ANucleotideAdenosineA2AHomo sapiensPSB-2113--2.252022-03-02doi.org/10.1002/anie.202115545
7PYRANucleotideAdenosineA2AHomo sapiensPSB-2115--2.62022-03-02doi.org/10.1002/anie.202115545
8JWYANucleotideAdenosineA2AHomo sapiens2-118--2.332023-08-16doi.org/10.1007/s11427-023-2459-8
6AQFANucleotideAdenosineA2AHomo sapiensZM-241385--2.512018-01-10doi.org/10.1016/j.cell.2017.12.004
8DU3ANucleotideAdenosineA2AHomo sapiensPubChem 105526064--2.52022-08-10doi.org/10.1016/j.ejmech.2022.114620
3PWHANucleotideAdenosineA2AHomo sapiensZM-241385--3.32011-09-07doi.org/10.1016/j.str.2011.06.014
3REYANucleotideAdenosineA2AHomo sapiensXAC--3.312011-09-07doi.org/10.1016/j.str.2011.06.014
3RFMANucleotideAdenosineA2AHomo sapiensCaffeine--3.62011-09-07doi.org/10.1016/j.str.2011.06.014
5WF5ANucleotideAdenosineA2AHomo sapiensUK-432097--2.62018-02-21doi.org/10.1016/j.str.2017.12.013
5WF6ANucleotideAdenosineA2AHomo sapiensUK-432097--2.92018-02-21doi.org/10.1016/j.str.2017.12.013
8CU6ANucleotideAdenosineA2AHomo sapiensLJ-4517--2.82022-08-31doi.org/10.1021/acs.jmedchem.2c00462
3UZAANucleotideAdenosineA2AHomo sapiensGTPL9236--3.272012-03-21doi.org/10.1021/jm201376w
3UZCANucleotideAdenosineA2AHomo sapiens4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol--3.342012-03-21doi.org/10.1021/jm201376w
2YDOANucleotideAdenosineA2AHomo sapiensAdenosine--32011-05-18doi.org/10.1038/nature10136
2YDVANucleotideAdenosineA2AHomo sapiensNECA--2.62011-05-18doi.org/10.1038/nature10136
5G53ANucleotideAdenosineA2AHomo sapiensNECA-Gs3.42016-08-03doi.org/10.1038/nature18966
5G53 (No Gprot) ANucleotideAdenosineA2AHomo sapiensNECA-3.42016-08-03doi.org/10.1038/nature18966
7T32ANucleotideAdenosineA2AHomo sapiensZM-241385--3.42022-08-10doi.org/10.1038/s41467-022-32125-2
8C9WANucleotideAdenosineA2AHomo sapiensEtrumadenant--2.112023-07-12doi.org/10.1038/s42004-023-00894-6
8PWNANucleotideAdenosineA2AHomo sapiensTheophylline--2.752023-10-25doi.org/10.1038/s42004-023-01014-0
5UIGANucleotideAdenosineA2AHomo sapiensCmpd-1--3.52017-02-08doi.org/10.1073/pnas.1621423114
5UVIANucleotideAdenosineA2AHomo sapiensZM-241385--3.22017-05-24doi.org/10.1107/S205225251700570X
6MH8ANucleotideAdenosineA2AHomo sapiensZM-241385--4.22019-04-24doi.org/10.1107/S205225251900263X
6S0LANucleotideAdenosineA2AHomo sapiensZM-241385--2.652020-07-15doi.org/10.1107/S2052252520011379
6S0QANucleotideAdenosineA2AHomo sapiensZM-241385--2.652020-07-15doi.org/10.1107/S2052252520011379
7EZCANucleotideAdenosineA2AHomo sapiensUKA--3.82022-04-13doi.org/10.1107/S2052252522001907
4UG2ANucleotideAdenosineA2AHomo sapiensCGS21680--2.62015-04-08doi.org/10.1124/mol.114.097360
4UHRANucleotideAdenosineA2AHomo sapiensCGS21680--2.62015-04-08doi.org/10.1124/mol.114.097360
8GNGANucleotideAdenosineA2AHomo sapiensIstradefylline--3.22023-03-22doi.org/10.1124/molpharm.122.000633
5JTBANucleotideAdenosineA2AHomo sapiensZM-241385--2.82017-05-31doi.org/10.1126/sciadv.1602952
3EMLANucleotideAdenosineA2AHomo sapiensZM-241385--2.62008-10-14doi.org/10.1126/science.1164772
3QAKANucleotideAdenosineA2AHomo sapiensUK-432097--2.712011-03-09doi.org/10.1126/science.1202793
6GDGANucleotideAdenosineA2AHomo sapiensNECA-Gs/β1/γ14.112018-05-16doi.org/10.7554/eLife.35946
6GDG (No Gprot) ANucleotideAdenosineA2AHomo sapiensNECA-4.112018-05-16doi.org/10.7554/eLife.35946
8WDTANucleotideAdenosineA2AHomo sapiensphotoNECA--3.342024-01-17doi.org/10.1016/j.bbrc.2023.149393
8RLNANucleotideAdenosineA2AHomo sapiensLUF5834--2.432024-06-19doi.org/10.1021/acsptsci.4c00051
9EE8ANucleotideAdenosineA2AHomo sapiensAdenosine-Gs/β1/γ22.632025-04-09doi.org/10.1038/s41467-025-56434-4
9EE8 (No Gprot) ANucleotideAdenosineA2AHomo sapiensAdenosine-2.632025-04-09doi.org/10.1038/s41467-025-56434-4
9EE9ANucleotideAdenosineA2AHomo sapiensAdenosine-Gs/β1/γ23.162025-04-09doi.org/10.1038/s41467-025-56434-4
9EE9 (No Gprot) ANucleotideAdenosineA2AHomo sapiensAdenosine-3.162025-04-09doi.org/10.1038/s41467-025-56434-4
9EEAANucleotideAdenosineA2AHomo sapiensAdenosine-Gs/β1/γ23.362025-04-09doi.org/10.1038/s41467-025-56434-4
9EEA (No Gprot) ANucleotideAdenosineA2AHomo sapiensAdenosine-3.362025-04-09doi.org/10.1038/s41467-025-56434-4
8UGWANucleotideAdenosineA2AHomo sapiensPubChem 3086599--3.92024-12-18doi.org/10.1038/s41557-024-01719-2
8HDOANucleotideAdenosineA2BHomo sapiensBAY 60-6583-Gs/β1/γ22.872023-01-18doi.org/10.1038/s41421-022-00503-1
8HDO (No Gprot) ANucleotideAdenosineA2BHomo sapiensBAY 60-6583-2.872023-01-18doi.org/10.1038/s41421-022-00503-1
8HDPANucleotideAdenosineA2BHomo sapiensAdenosine-Gs/β1/γ23.22023-01-18doi.org/10.1038/s41421-022-00503-1
8HDP (No Gprot) ANucleotideAdenosineA2BHomo sapiensAdenosine-3.22023-01-18doi.org/10.1038/s41421-022-00503-1
7XY6ANucleotideAdenosineA2BHomo sapiensBAY 60-6583-chim(NtGi1-Gs)/β1/γ22.992023-05-03doi.org/10.1126/sciadv.add3709
7XY6 (No Gprot) ANucleotideAdenosineA2BHomo sapiensBAY 60-6583-2.992023-05-03doi.org/10.1126/sciadv.add3709
7XY7ANucleotideAdenosineA2BHomo sapiensNECA-chim(NtGi1-Gs)/β1/γ23.262023-05-03doi.org/10.1126/sciadv.add3709
7XY7 (No Gprot) ANucleotideAdenosineA2BHomo sapiensNECA-3.262023-05-03doi.org/10.1126/sciadv.add3709
8X16ANucleotideAdenosineA3AHomo sapiensPiclidenoson-Gi1/β1/γ23.292024-04-24doi.org/10.1038/s41467-024-47207-6
8X16 (No Gprot) ANucleotideAdenosineA3AHomo sapiensPiclidenoson-3.292024-04-24doi.org/10.1038/s41467-024-47207-6
8X17ANucleotideAdenosineA3AHomo sapiensNamodenoson-Gi1/β1/γ23.192024-04-24doi.org/10.1038/s41467-024-47207-6
8X17 (No Gprot) ANucleotideAdenosineA3AHomo sapiensNamodenoson-3.192024-04-24doi.org/10.1038/s41467-024-47207-6
8YH0ANucleotideAdenosineA3AHomo sapiensNECA-Gi1/β1/γ22.862024-11-06doi.org/10.1038/s41467-024-53473-1
8YH0 (No Gprot) ANucleotideAdenosineA3AHomo sapiensNECA-2.862024-11-06doi.org/10.1038/s41467-024-53473-1
8YH2ANucleotideAdenosineA3AHomo sapiensAdenosine-Gi1/β1/γ23.272024-11-06doi.org/10.1038/s41467-024-53473-1
8YH2 (No Gprot) ANucleotideAdenosineA3AHomo sapiensAdenosine-3.272024-11-06doi.org/10.1038/s41467-024-53473-1
8YH3ANucleotideAdenosineA3AHomo sapiensN-methyladenosine-Gi1/β1/γ23.42024-11-06doi.org/10.1038/s41467-024-53473-1
8YH3 (No Gprot) ANucleotideAdenosineA3AHomo sapiensN-methyladenosine-3.42024-11-06doi.org/10.1038/s41467-024-53473-1
8YH5ANucleotideAdenosineA3AHomo sapiensRiboprine-Gi1/β1/γ23.662024-11-06doi.org/10.1038/s41467-024-53473-1
8YH5 (No Gprot) ANucleotideAdenosineA3AHomo sapiensRiboprine-3.662024-11-06doi.org/10.1038/s41467-024-53473-1
8YH6ANucleotideAdenosineA3AHomo sapiensNamodenoson-Gi1/β1/γ23.622024-11-06doi.org/10.1038/s41467-024-53473-1
8YH6 (No Gprot) ANucleotideAdenosineA3AHomo sapiensNamodenoson-3.622024-11-06doi.org/10.1038/s41467-024-53473-1
8G2YB2AdhesionAdhesionADGRF1Homo sapiens-LPCchim(Gs-CtGq)/β1/γ23.442023-05-10doi.org/10.1038/s41467-023-38083-7
8G2Y (No Gprot) B2AdhesionAdhesionADGRF1Homo sapiens-LPC3.442023-05-10doi.org/10.1038/s41467-023-38083-7
7WU3B2AdhesionAdhesionADGRF1Homo sapiens-K6GGs/β1/γ23.12022-04-27doi.org/10.1038/s41586-022-04580-w
7WU3 (No Gprot) B2AdhesionAdhesionADGRF1Homo sapiens-K6G3.12022-04-27doi.org/10.1038/s41586-022-04580-w
7WU4B2AdhesionAdhesionADGRF1Homo sapiens-K6GGi1/β1/γ23.42022-04-27doi.org/10.1038/s41586-022-04580-w
7WU4 (No Gprot) B2AdhesionAdhesionADGRF1Homo sapiens-K6G3.42022-04-27doi.org/10.1038/s41586-022-04580-w
7WU5B2AdhesionAdhesionADGRF1Homo sapiens-K6GGi1/β1/γ232022-04-27doi.org/10.1038/s41586-022-04580-w
7WU5 (No Gprot) B2AdhesionAdhesionADGRF1Homo sapiens-K6G32022-04-27doi.org/10.1038/s41586-022-04580-w
7WU2B2AdhesionAdhesionADGRD1Homo sapiens--Gs/β1/γ12.82022-04-27doi.org/10.1038/s41586-022-04580-w
7WU2 (No Gprot) B2AdhesionAdhesionADGRD1Homo sapiens--2.82022-04-27doi.org/10.1038/s41586-022-04580-w
7EPTB2AdhesionAdhesionADGRD1Homo sapiens--Gs/β1/γ232022-05-11doi.org/10.1038/s41586-022-04619-y
7EPT (No Gprot) B2AdhesionAdhesionADGRD1Homo sapiens--32022-05-11doi.org/10.1038/s41586-022-04619-y
8X9SB2AdhesionAdhesionADGRD1Homo sapiens5α-DHT-chim(NtGi1-Gs)/β1/γ23.492025-02-12doi.org/10.1016/j.cell.2025.01.006
8X9S (No Gprot) B2AdhesionAdhesionADGRD1Homo sapiens5α-DHT-3.492025-02-12doi.org/10.1016/j.cell.2025.01.006
8X9TB2AdhesionAdhesionADGRD1Homo sapiensAP503-chim(NtGi1-Gs)/β1/γ22.752025-02-12doi.org/10.1016/j.cell.2025.01.006
8X9T (No Gprot) B2AdhesionAdhesionADGRD1Homo sapiensAP503-2.752025-02-12doi.org/10.1016/j.cell.2025.01.006
8X9UB2AdhesionAdhesionADGRD1Homo sapiensMetenolone-chim(NtGi1-Gs)/β1/γ22.882025-02-12doi.org/10.1016/j.cell.2025.01.006
8X9U (No Gprot) B2AdhesionAdhesionADGRD1Homo sapiensMetenolone-2.882025-02-12doi.org/10.1016/j.cell.2025.01.006
9IV1B2AdhesionAdhesionADGRD1Homo sapiens5α-DHT-chim(NtGi1-Gs)/β1/γ22.982025-02-12doi.org/10.1016/j.cell.2025.01.006
9IV1 (No Gprot) B2AdhesionAdhesionADGRD1Homo sapiens5α-DHT-2.982025-02-12doi.org/10.1016/j.cell.2025.01.006
9IV2B2AdhesionAdhesionADGRD1Homo sapiens5α-DHT-chim(NtGi1-Gs)/β1/γ23.532025-02-12doi.org/10.1016/j.cell.2025.01.006
9IV2 (No Gprot) B2AdhesionAdhesionADGRD1Homo sapiens5α-DHT-3.532025-02-12doi.org/10.1016/j.cell.2025.01.006
7YDHB2AdhesionAdhesionADGRE5Homo sapiens--chim(NtGi2-G13)/β1/γ23.12023-07-12doi.org/10.1016/j.chembiol.2023.08.003
7YDH (No Gprot) B2AdhesionAdhesionADGRE5Homo sapiens--3.12023-07-12doi.org/10.1016/j.chembiol.2023.08.003
7YDMB2AdhesionAdhesionADGRE5Homo sapiens--chim(NtGi1-Gs-CtGq)/β1/γ22.892023-07-12doi.org/10.1016/j.chembiol.2023.08.003
7YDM (No Gprot) B2AdhesionAdhesionADGRE5Homo sapiens--2.892023-07-12doi.org/10.1016/j.chembiol.2023.08.003
7YDPB2AdhesionAdhesionADGRE5Homo sapiens--chim(NtGi1-Gs)/β1/γ23.12023-07-12doi.org/10.1016/j.chembiol.2023.08.003
7YDP (No Gprot) B2AdhesionAdhesionADGRE5Homo sapiens--3.12023-07-12doi.org/10.1016/j.chembiol.2023.08.003
8IKLB2AdhesionAdhesionADGRE5Homo sapiens--chim(NtGi1L-G13)/β1/γ22.332024-01-24doi.org/10.1016/j.molcel.2023.12.020
8IKL (No Gprot) B2AdhesionAdhesionADGRE5Homo sapiens--2.332024-01-24doi.org/10.1016/j.molcel.2023.12.020
8IKJB2AdhesionAdhesionADGRE5Homo sapiens---3.22024-02-14doi.org/10.1016/j.molcel.2023.12.020
7YDJB2AdhesionAdhesionADGRE5Homo sapiens--chim(NtGi1-G12)/β1/γ23.032023-07-12To be published
7YDJ (No Gprot) B2AdhesionAdhesionADGRE5Homo sapiens--3.032023-07-12To be published
7WXUB2AdhesionAdhesionADGRF1Homo sapiens--chim(NtGi1-Gs-CtGq)/β1/γ22.852022-09-28doi.org/10.1038/s41467-022-33173-4
7WXU (No Gprot) B2AdhesionAdhesionADGRF1Homo sapiens--2.852022-09-28doi.org/10.1038/s41467-022-33173-4
7WXWB2AdhesionAdhesionADGRF1Homo sapiens--chim(NtGi1-Gs)/β1/γ22.842022-09-28doi.org/10.1038/s41467-022-33173-4
7WXW (No Gprot) B2AdhesionAdhesionADGRF1Homo sapiens--2.842022-09-28doi.org/10.1038/s41467-022-33173-4
7WY0B2AdhesionAdhesionADGRF1Homo sapiens--chim(NtGi1L-G13)/β1/γ22.832022-09-28doi.org/10.1038/s41467-022-33173-4
7WY0 (No Gprot) B2AdhesionAdhesionADGRF1Homo sapiens--2.832022-09-28doi.org/10.1038/s41467-022-33173-4
7WZ7B2AdhesionAdhesionADGRF1Homo sapiens--chim(NtGi1-G12)/β1/γ22.832022-09-28doi.org/10.1038/s41467-022-33173-4
7WZ7 (No Gprot) B2AdhesionAdhesionADGRF1Homo sapiens--2.832022-09-28doi.org/10.1038/s41467-022-33173-4
7X2VB2AdhesionAdhesionADGRF1Homo sapiens--Gi1/β1/γ23.092022-09-28doi.org/10.1038/s41467-022-33173-4
7X2V (No Gprot) B2AdhesionAdhesionADGRF1Homo sapiens--3.092022-09-28doi.org/10.1038/s41467-022-33173-4
7SF8B2AdhesionAdhesionADGRG1Homo sapiens--chim(NtGi2-G13)/β1/γ22.72022-04-27doi.org/10.1038/s41586-022-04575-7
7SF8 (No Gprot) B2AdhesionAdhesionADGRG1Homo sapiens--2.72022-04-27doi.org/10.1038/s41586-022-04575-7
7WUIB2AdhesionAdhesionADGRG2Mus musculusIP15-chim(NtGi1-Gs)/β1/γ23.12022-04-27doi.org/10.1038/s41586-022-04590-8
7WUI (No Gprot) B2AdhesionAdhesionADGRG2Mus musculusIP15-3.12022-04-27doi.org/10.1038/s41586-022-04590-8
7WUQB2AdhesionAdhesionADGRG2Mus musculus--Gs/β1/γ22.92022-04-27doi.org/10.1038/s41586-022-04590-8
7WUQ (No Gprot) B2AdhesionAdhesionADGRG2Mus musculus--2.92022-04-27doi.org/10.1038/s41586-022-04590-8
7XKDB2AdhesionAdhesionADGRG2Mus musculusβ-Hydroxyandrosterone-Gs/β1/γ22.42022-08-10doi.org/10.1038/s41589-022-01084-6
7XKD (No Gprot) B2AdhesionAdhesionADGRG2Mus musculusβ-Hydroxyandrosterone-2.42022-08-10doi.org/10.1038/s41589-022-01084-6
7XKEB2AdhesionAdhesionADGRG2Mus musculusβ-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ22.92022-08-10doi.org/10.1038/s41589-022-01084-6
7XKE (No Gprot) B2AdhesionAdhesionADGRG2Mus musculusβ-Hydroxyandrosterone-2.92022-08-10doi.org/10.1038/s41589-022-01084-6
7XKFB2AdhesionAdhesionADGRG2Mus musculusβ-Hydroxyandrosterone-Gs/β1/γ22.42022-08-10doi.org/10.1038/s41589-022-01084-6
7XKF (No Gprot) B2AdhesionAdhesionADGRG2Mus musculusβ-Hydroxyandrosterone-2.42022-08-10doi.org/10.1038/s41589-022-01084-6
7YP7B2AdhesionAdhesionADGRG2Mus musculus--Gs/β1/γ23.12022-08-24doi.org/10.1038/s41589-022-01084-6
7YP7 (No Gprot) B2AdhesionAdhesionADGRG2Mus musculus--3.12022-08-24doi.org/10.1038/s41589-022-01084-6
7D76B2AdhesionAdhesionADGRG3Homo sapiensBeclomethasone-Go/β1/γ23.12021-02-03doi.org/10.1038/s41586-020-03083-w
7D76 (No Gprot) B2AdhesionAdhesionADGRG3Homo sapiensBeclomethasone-3.12021-02-03doi.org/10.1038/s41586-020-03083-w
7D77B2AdhesionAdhesionADGRG3Homo sapiensHydrocortisone-Go/β1/γ22.92021-02-03doi.org/10.1038/s41586-020-03083-w
7D77 (No Gprot) B2AdhesionAdhesionADGRG3Homo sapiensHydrocortisone-2.92021-02-03doi.org/10.1038/s41586-020-03083-w
7WUJB2AdhesionAdhesionADGRG4Homo sapiens--chim(NtGi1-Gs)/β1/γ23.32022-04-27doi.org/10.1038/s41586-022-04590-8
7WUJ (No Gprot) B2AdhesionAdhesionADGRG4Homo sapiens--3.32022-04-27doi.org/10.1038/s41586-022-04590-8
7EQ1B2AdhesionAdhesionADGRG5Homo sapiens--chim(NtGi1-Gs)/β1/γ23.32022-05-11doi.org/10.1038/s41586-022-04619-y
7EQ1 (No Gprot) B2AdhesionAdhesionADGRG5Homo sapiens--3.32022-05-11doi.org/10.1038/s41586-022-04619-y
7WY5B2AdhesionAdhesionADGRL3Mus musculus--chim(NtGi1-Gs-CtGq)/β1/γ22.832022-10-26doi.org/10.1016/j.molcel.2022.10.009
7WY5 (No Gprot) B2AdhesionAdhesionADGRL3Mus musculus--2.832022-10-26doi.org/10.1016/j.molcel.2022.10.009
7WY8B2AdhesionAdhesionADGRL3Mus musculus--chim(NtGi1-Gs)/β1/γ22.832022-10-26doi.org/10.1016/j.molcel.2022.10.009
7WY8 (No Gprot) B2AdhesionAdhesionADGRL3Mus musculus--2.832022-10-26doi.org/10.1016/j.molcel.2022.10.009
7WYBB2AdhesionAdhesionADGRL3Mus musculus--Gi1/β1/γ22.972022-10-26doi.org/10.1016/j.molcel.2022.10.009
7WYB (No Gprot) B2AdhesionAdhesionADGRL3Mus musculus--2.972022-10-26doi.org/10.1016/j.molcel.2022.10.009
7X10B2AdhesionAdhesionADGRL3Mus musculus--chim(NtGi1-G12)/β1/γ22.932022-10-26doi.org/10.1016/j.molcel.2022.10.009
7X10 (No Gprot) B2AdhesionAdhesionADGRL3Mus musculus--2.932022-10-26doi.org/10.1016/j.molcel.2022.10.009
7SF7B2AdhesionAdhesionADGRL3Homo sapiens--chim(NtGi2-G13)/β1/γ22.92022-04-27doi.org/10.1038/s41586-022-04575-7
7SF7 (No Gprot) B2AdhesionAdhesionADGRL3Homo sapiens--2.92022-04-27doi.org/10.1038/s41586-022-04575-7
8JMTB2AdhesionAdhesionADGRL3Homo sapiens---3.32023-09-06doi.org/10.1038/s41589-023-01389-0
9M4QAAmineAdrenegicAlpha1AHomo sapiensDoxazosin--2.992025-07-02doi.org/10.1016/j.jbc.2025.110348
9M4TAAmineAdrenegicAlpha1AHomo sapiensSilodosin--3.192025-07-02doi.org/10.1016/j.jbc.2025.110348
6N48AAmineAdrenergicβ2Homo sapiensBI167107PubChem 138454256-3.22019-06-26doi.org/10.1126/science.aaw8981
3ZPQAAmineAdrenergicβ1Meleagris gallopavo4-(piperazin-1- yl)-1H-indoleNa-2.82013-04-03doi.org/10.1021/jm400140q
3ZPRAAmineAdrenergicβ1Meleagris gallopavo4-methyl-2-(piperazin-1-yl)Na-2.72013-04-03doi.org/10.1021/jm400140q
5A8EAAmineAdrenergicβ1Meleagris gallopavo7-MethylcyanopindololNa-2.42015-09-30doi.org/10.1124/mol.115.101030
4BVNAAmineAdrenergicβ1Meleagris gallopavoCyanopindololNa-2.12014-04-02doi.org/10.1371/journal.pone.0092727
7XK9AAmineAdrenergicβ2Homo sapiensConstrained IsoproterenolNa-3.42023-04-26doi.org/10.1038/s41467-023-37808-y
6OBAAAmineAdrenergicβ2Homo sapiensS-AlprenololGTPL11074-3.12020-03-25doi.org/10.1038/s41589-020-0549-2
8UO1AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP; MgGs/β1/γ23.62024-03-06doi.org/10.1038/s41586-024-07153-1
8UO1 (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP; Mg3.62024-03-06doi.org/10.1038/s41586-024-07153-1
8UO3AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP; MgGs/β1/γ23.52024-03-06doi.org/10.1038/s41586-024-07153-1
8UO3 (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP; Mg3.52024-03-06doi.org/10.1038/s41586-024-07153-1
8UO4AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP; MgGs/β1/γ242024-03-06doi.org/10.1038/s41586-024-07153-1
8UO4 (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP; Mg42024-03-06doi.org/10.1038/s41586-024-07153-1
8GFVAAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.12024-03-06doi.org/10.1038/s41586-024-07153-1
8GFV (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.12024-03-06doi.org/10.1038/s41586-024-07153-1
8GFWAAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ232024-03-06doi.org/10.1038/s41586-024-07153-1
8GFW (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP32024-03-06doi.org/10.1038/s41586-024-07153-1
8GFXAAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ232024-03-06doi.org/10.1038/s41586-024-07153-1
8GFX (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP32024-03-06doi.org/10.1038/s41586-024-07153-1
8GFYAAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ232024-03-06doi.org/10.1038/s41586-024-07153-1
8GFY (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP32024-03-06doi.org/10.1038/s41586-024-07153-1
8GFZAAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ232024-03-06doi.org/10.1038/s41586-024-07153-1
8GFZ (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP32024-03-06doi.org/10.1038/s41586-024-07153-1
8GG0AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ22.92024-03-06doi.org/10.1038/s41586-024-07153-1
8GG0 (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP2.92024-03-06doi.org/10.1038/s41586-024-07153-1
8GG1AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ232024-03-06doi.org/10.1038/s41586-024-07153-1
8GG1 (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP32024-03-06doi.org/10.1038/s41586-024-07153-1
8GG2AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ232024-03-06doi.org/10.1038/s41586-024-07153-1
8GG2 (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP32024-03-06doi.org/10.1038/s41586-024-07153-1
8GG3AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.12024-03-06doi.org/10.1038/s41586-024-07153-1
8GG3 (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.12024-03-06doi.org/10.1038/s41586-024-07153-1
8GG4AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.22024-03-06doi.org/10.1038/s41586-024-07153-1
8GG4 (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.22024-03-06doi.org/10.1038/s41586-024-07153-1
8GG5AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.22024-03-06doi.org/10.1038/s41586-024-07153-1
8GG5 (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.22024-03-06doi.org/10.1038/s41586-024-07153-1
8GG6AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.32024-03-06doi.org/10.1038/s41586-024-07153-1
8GG6 (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.32024-03-06doi.org/10.1038/s41586-024-07153-1
8GG7AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.32024-03-06doi.org/10.1038/s41586-024-07153-1
8GG7 (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.32024-03-06doi.org/10.1038/s41586-024-07153-1
8GG8AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.32024-03-06doi.org/10.1038/s41586-024-07153-1
8GG8 (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.32024-03-06doi.org/10.1038/s41586-024-07153-1
8GG9AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.42024-03-06doi.org/10.1038/s41586-024-07153-1
8GG9 (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.42024-03-06doi.org/10.1038/s41586-024-07153-1
8GGAAAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.52024-03-06doi.org/10.1038/s41586-024-07153-1
8GGA (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.52024-03-06doi.org/10.1038/s41586-024-07153-1
8GGBAAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.52024-03-06doi.org/10.1038/s41586-024-07153-1
8GGB (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.52024-03-06doi.org/10.1038/s41586-024-07153-1
8GGCAAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.42024-03-06doi.org/10.1038/s41586-024-07153-1
8GGC (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.42024-03-06doi.org/10.1038/s41586-024-07153-1
8GGEAAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.52024-03-06doi.org/10.1038/s41586-024-07153-1
8GGE (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.52024-03-06doi.org/10.1038/s41586-024-07153-1
8GGFAAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.62024-03-06doi.org/10.1038/s41586-024-07153-1
8GGF (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.62024-03-06doi.org/10.1038/s41586-024-07153-1
8UNLAAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.32024-03-06doi.org/10.1038/s41586-024-07153-1
8UNL (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.32024-03-06doi.org/10.1038/s41586-024-07153-1
8UNMAAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.42024-03-06doi.org/10.1038/s41586-024-07153-1
8UNM (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.42024-03-06doi.org/10.1038/s41586-024-07153-1
8UNNAAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.42024-03-06doi.org/10.1038/s41586-024-07153-1
8UNN (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.42024-03-06doi.org/10.1038/s41586-024-07153-1
8UNOAAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.32024-03-06doi.org/10.1038/s41586-024-07153-1
8UNO (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.32024-03-06doi.org/10.1038/s41586-024-07153-1
8UNPAAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.32024-03-06doi.org/10.1038/s41586-024-07153-1
8UNP (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.32024-03-06doi.org/10.1038/s41586-024-07153-1
8UNQAAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.32024-03-06doi.org/10.1038/s41586-024-07153-1
8UNQ (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.32024-03-06doi.org/10.1038/s41586-024-07153-1
8UNRAAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.42024-03-06doi.org/10.1038/s41586-024-07153-1
8UNR (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.42024-03-06doi.org/10.1038/s41586-024-07153-1
8UNSAAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.42024-03-06doi.org/10.1038/s41586-024-07153-1
8UNS (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.42024-03-06doi.org/10.1038/s41586-024-07153-1
8UNTAAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.42024-03-06doi.org/10.1038/s41586-024-07153-1
8UNT (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.42024-03-06doi.org/10.1038/s41586-024-07153-1
8UNUAAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.52024-03-06doi.org/10.1038/s41586-024-07153-1
8UNU (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.52024-03-06doi.org/10.1038/s41586-024-07153-1
8UNVAAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.32024-03-06doi.org/10.1038/s41586-024-07153-1
8UNV (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.32024-03-06doi.org/10.1038/s41586-024-07153-1
8UNWAAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.42024-03-06doi.org/10.1038/s41586-024-07153-1
8UNW (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.42024-03-06doi.org/10.1038/s41586-024-07153-1
8UNXAAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.62024-03-06doi.org/10.1038/s41586-024-07153-1
8UNX (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.62024-03-06doi.org/10.1038/s41586-024-07153-1
8UNYAAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.62024-03-06doi.org/10.1038/s41586-024-07153-1
8UNY (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.62024-03-06doi.org/10.1038/s41586-024-07153-1
8UNZAAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.82024-03-06doi.org/10.1038/s41586-024-07153-1
8UNZ (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.82024-03-06doi.org/10.1038/s41586-024-07153-1
8UO0AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.52024-03-06doi.org/10.1038/s41586-024-07153-1
8UO0 (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.52024-03-06doi.org/10.1038/s41586-024-07153-1
8UO2AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTPGs/β1/γ23.62024-03-06doi.org/10.1038/s41586-024-07153-1
8UO2 (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained EpinephrineGTP3.62024-03-06doi.org/10.1038/s41586-024-07153-1
5X7DAAmineAdrenergicβ2Homo sapiensS-CarazololCmpd-15-2.72017-08-16doi.org/10.1038/nature23652
7YM8AAmineAdrenergicAlpha1AHomo sapiensOxymetazoline-chim(Gs-CtGq)2.922023-07-05doi.org/10.1038/s41467-023-39310-x
7YM8 (No Gprot) AAmineAdrenergicAlpha1AHomo sapiensOxymetazoline-2.922023-07-05doi.org/10.1038/s41467-023-39310-x
7YMHAAmineAdrenergicAlpha1AHomo sapiensNorepinephrine-chim(Gs-CtGq)3.522023-07-05doi.org/10.1038/s41467-023-39310-x
7YMH (No Gprot) AAmineAdrenergicAlpha1AHomo sapiensNorepinephrine-3.522023-07-05doi.org/10.1038/s41467-023-39310-x
7YMJAAmineAdrenergicAlpha1AHomo sapiensTamsulosin--3.352023-07-05doi.org/10.1038/s41467-023-39310-x
8THKAAmineAdrenergicAlpha1AHomo sapiensA61603-chim(NtGi2L-Gs-CtGq)/β1/γ22.62023-08-16doi.org/10.1038/s41467-023-40524-2
8THK (No Gprot) AAmineAdrenergicAlpha1AHomo sapiensA61603-2.62023-08-16doi.org/10.1038/s41467-023-40524-2
8THLAAmineAdrenergicAlpha1AHomo sapiensEpinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ23.12023-08-16doi.org/10.1038/s41467-023-40524-2
8THL (No Gprot) AAmineAdrenergicAlpha1AHomo sapiensEpinephrine-3.12023-08-16doi.org/10.1038/s41467-023-40524-2
8HN1AAmineAdrenergicAlpha1AHomo sapiensToxin AdTx1--2.92023-12-20To be published
7B6WAAmineAdrenergicα1bHomo sapiensCyclazosin--2.872022-01-12doi.org/10.1038/s41467-021-27911-3
6KUXAAmineAdrenergicα2aHomo sapiensRS-79948--2.72019-12-04doi.org/10.1038/nature06325
6KUYAAmineAdrenergicα2aHomo sapiensPubChem 145704643--3.22019-12-04doi.org/10.1038/nature06325
7EJ0AAmineAdrenergicα2aHomo sapiensL-Norepinephrine-Go/β1/γ23.22022-04-13doi.org/10.1126/sciadv.abj5347
7EJ0 (No Gprot) AAmineAdrenergicα2aHomo sapiensL-Norepinephrine-3.22022-04-13doi.org/10.1126/sciadv.abj5347
7EJ8AAmineAdrenergicα2aHomo sapiensBrimonidine-Go/β1/γ232022-04-13doi.org/10.1126/sciadv.abj5347
7EJ8 (No Gprot) AAmineAdrenergicα2aHomo sapiensBrimonidine-32022-04-13doi.org/10.1126/sciadv.abj5347
7EJAAAmineAdrenergicα2aHomo sapiensDexmedetomidine-Go/β1/γ23.62022-04-13doi.org/10.1126/sciadv.abj5347
7EJA (No Gprot) AAmineAdrenergicα2aHomo sapiensDexmedetomidine-3.62022-04-13doi.org/10.1126/sciadv.abj5347
7EJKAAmineAdrenergicα2aHomo sapiensOxymetazoline-Go/β1/γ23.42022-04-13doi.org/10.1126/sciadv.abj5347
7EJK (No Gprot) AAmineAdrenergicα2aHomo sapiensOxymetazoline-3.42022-04-13doi.org/10.1126/sciadv.abj5347
7W6PAAmineAdrenergicα2aHomo sapiensN-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ23.472022-09-28doi.org/10.1126/science.abn7065
7W6P (No Gprot) AAmineAdrenergicα2aHomo sapiensN-pyridin-4-ylisoquinolin-4-amine-3.472022-09-28doi.org/10.1126/science.abn7065
7W7EAAmineAdrenergicα2aHomo sapiensPubChem 164946676-Go/β1/γ23.42022-09-28doi.org/10.1126/science.abn7065
7W7E (No Gprot) AAmineAdrenergicα2aHomo sapiensPubChem 164946676-3.42022-09-28doi.org/10.1126/science.abn7065
9CBLAAmineAdrenergicα2aHomo sapiensEpinephrine-Gi1/β1/γ22.82024-09-11doi.org/10.1038/s12276-024-01296-x
9CBL (No Gprot) AAmineAdrenergicα2aHomo sapiensEpinephrine-2.82024-09-11doi.org/10.1038/s12276-024-01296-x
9CBMAAmineAdrenergicα2aHomo sapiensDexmedetomidine-Gi1/β1/γ23.22024-09-11doi.org/10.1038/s12276-024-01296-x
9CBM (No Gprot) AAmineAdrenergicα2aHomo sapiensDexmedetomidine-3.22024-09-11doi.org/10.1038/s12276-024-01296-x
6K41AAmineAdrenergicα2bHomo sapiensDexmedetomidine-Go/β1/γ22.92020-04-15doi.org/10.1038/s41589-020-0492-2
6K41 (No Gprot) AAmineAdrenergicα2bHomo sapiensDexmedetomidine-2.92020-04-15doi.org/10.1038/s41589-020-0492-2
6K42AAmineAdrenergicα2bHomo sapiensDexmedetomidine-Gi1/β1/γ24.12020-04-15doi.org/10.1038/s41589-020-0492-2
6K42 (No Gprot) AAmineAdrenergicα2bHomo sapiensDexmedetomidine-4.12020-04-15doi.org/10.1038/s41589-020-0492-2
6KUWAAmineAdrenergicα2cHomo sapiensPubChem 57213234--2.82019-12-04doi.org/10.1038/nature06325
7JJOAAmineAdrenergicβ1Meleagris gallopavoIsoprenaline-Gs/β1/γ22.62020-09-02doi.org/10.1016/j.molcel.2020.08.001
7JJO (No Gprot) AAmineAdrenergicβ1Meleagris gallopavoIsoprenaline-2.62020-09-02doi.org/10.1016/j.molcel.2020.08.001
4AMIAAmineAdrenergicβ1Meleagris gallopavoBucindolol--3.22012-05-23doi.org/10.1016/j.str.2012.03.014
4AMJAAmineAdrenergicβ1Meleagris gallopavoS-Carvedilol--2.32012-05-23doi.org/10.1016/j.str.2012.03.014
2VT4AAmineAdrenergicβ1Meleagris gallopavoCyanopindolol--2.72008-06-24doi.org/10.1038/nature07101
2Y00AAmineAdrenergicβ1Meleagris gallopavoDobutamine--2.52011-01-12doi.org/10.1038/nature09746
2Y02AAmineAdrenergicβ1Meleagris gallopavoCarmoterol--2.62011-01-12doi.org/10.1038/nature09746
2Y03AAmineAdrenergicβ1Meleagris gallopavoIsoprenaline--2.852011-01-12doi.org/10.1038/nature09746
2Y04AAmineAdrenergicβ1Meleagris gallopavoSalbutamol--3.052011-01-12doi.org/10.1038/nature09746
2Y01AAmineAdrenergicβ1Meleagris gallopavoDobutamine--2.62011-03-30doi.org/10.1038/nature09746
4GPOAAmineAdrenergicβ1Meleagris gallopavo---3.52013-02-27doi.org/10.1038/nsmb.2504
5F8UAAmineAdrenergicβ1Meleagris gallopavoCyanopindolol--3.352015-12-23doi.org/10.1038/nsmb.3130
7BTSAAmineAdrenergicβ1Homo sapiensL-Epinephrine--3.132020-12-02doi.org/10.1038/s41422-020-00424-2
7BU6AAmineAdrenergicβ1Homo sapiensL-Norepinephrine--2.72020-12-02doi.org/10.1038/s41422-020-00424-2
7BU7AAmineAdrenergicβ1Homo sapiensBI167107--2.62020-12-02doi.org/10.1038/s41422-020-00424-2
7BVQAAmineAdrenergicβ1Homo sapiensS-Carazolol--2.52020-12-02doi.org/10.1038/s41422-020-00424-2
8DCRAAmineAdrenergicβ1Meleagris gallopavoDobutamine-Gs/β1/γ22.62022-07-27doi.org/10.1038/s41467-022-31823-1
8DCR (No Gprot) AAmineAdrenergicβ1Meleagris gallopavoDobutamine-2.62022-07-27doi.org/10.1038/s41467-022-31823-1
8DCSAAmineAdrenergicβ1Meleagris gallopavoCyanopindolol-Gs/β1/γ22.52022-07-27doi.org/10.1038/s41467-022-31823-1
8DCS (No Gprot) AAmineAdrenergicβ1Meleagris gallopavoCyanopindolol-2.52022-07-27doi.org/10.1038/s41467-022-31823-1
6IBLAAmineAdrenergicβ1Meleagris gallopavoArformoterol--2.72019-01-09doi.org/10.1038/s41586-020-2419-1
6TKOAAmineAdrenergicβ1Meleagris gallopavoArformoterol-Arrestin23.32020-06-17doi.org/10.1038/s41586-020-2419-1
7S0FAAmineAdrenergicβ1Meleagris gallopavoIsoprenaline-Gi1/β1/γ22.962021-11-17doi.org/10.1038/s41594-021-00679-2
7S0F (No Gprot) AAmineAdrenergicβ1Meleagris gallopavoIsoprenaline-2.962021-11-17doi.org/10.1038/s41594-021-00679-2
7S0GAAmineAdrenergicβ1Meleagris gallopavoIsoprenaline-chim(Gi1-CtGs)/β1/γ23.862021-11-17doi.org/10.1038/s41594-021-00679-2
7S0G (No Gprot) AAmineAdrenergicβ1Meleagris gallopavoIsoprenaline-3.862021-11-17doi.org/10.1038/s41594-021-00679-2
2YCWAAmineAdrenergicβ1Meleagris gallopavoS-Carazolol--32011-06-01doi.org/10.1073/pnas.1100185108
2YCXAAmineAdrenergicβ1Meleagris gallopavoCyanopindolol--3.252011-06-01doi.org/10.1073/pnas.1100185108
2YCZAAmineAdrenergicβ1Meleagris gallopavoIodocyanopindolol--3.652011-06-01doi.org/10.1073/pnas.1100185108
2YCYAAmineAdrenergicβ1Meleagris gallopavoCyanopindolol--3.152011-06-08doi.org/10.1073/pnas.1100185108
6H7NAAmineAdrenergicβ1Meleagris gallopavoS-Xamoterol--2.52018-10-17doi.org/10.1101/436212
6H7JAAmineAdrenergicβ1Meleagris gallopavoIsoprenaline--2.82018-10-17doi.org/10.1126/science.aau5595
6H7LAAmineAdrenergicβ1Meleagris gallopavoDobutamine--2.72018-10-17doi.org/10.1126/science.aau5595
6H7MAAmineAdrenergicβ1Meleagris gallopavoSalbutamol--2.762018-10-17doi.org/10.1126/science.aau5595
6H7OAAmineAdrenergicβ1Meleagris gallopavoCyanopindolol--2.82018-10-17doi.org/10.1126/science.aau5595
8S2TAAmineAdrenergicβ1Homo sapiensIsoprenaline-chim(NtGi1-Gs)/β1/γ23.32025-05-21To be published
8S2T (No Gprot) AAmineAdrenergicβ1Homo sapiensIsoprenaline-3.32025-05-21To be published
6E67AAmineAdrenergicβ2Homo sapiensBI167107-Gs(CT)3.72019-06-05doi.org/10.1016/j.cell.2019.04.021
6E67 (No Gprot) AAmineAdrenergicβ2Homo sapiensBI167107-3.72019-06-05doi.org/10.1016/j.cell.2019.04.021
3D4SAAmineAdrenergicβ2Homo sapiensTimolol--2.82008-06-17doi.org/10.1016/j.str.2008.05.001
3NY8AAmineAdrenergicβ2Homo sapiensICI118-551--2.842010-08-11doi.org/10.1021/ja105108q
3NY9AAmineAdrenergicβ2Homo sapiensICI118-551--2.842010-08-11doi.org/10.1021/ja105108q
3NYAAAmineAdrenergicβ2Homo sapiensS-Alprenolol--3.162010-08-11doi.org/10.1021/ja105108q
2R4RAAmineAdrenergicβ2Homo sapiens---3.42007-11-06doi.org/10.1038/nature06325
2R4SAAmineAdrenergicβ2Homo sapiens---3.42007-11-06doi.org/10.1038/nature06325
3KJ6AAmineAdrenergicβ2Homo sapiens---3.42010-02-16doi.org/10.1038/nature08650
3P0GAAmineAdrenergicβ2Homo sapiensBI167107--3.52011-01-19doi.org/10.1038/nature09648
3PDSAAmineAdrenergicβ2Homo sapiensHydroxybenzylisoproterenol--3.52011-01-12doi.org/10.1038/nature09665
3SN6AAmineAdrenergicβ2Homo sapiensBI167107-Gs/β1/γ23.22011-07-20doi.org/10.1038/nature10361
3SN6 (No Gprot) AAmineAdrenergicβ2Homo sapiensBI167107-3.22011-07-20doi.org/10.1038/nature10361
4LDEAAmineAdrenergicβ2Homo sapiensBI167107--2.792013-09-25doi.org/10.1038/nature12572
4LDLAAmineAdrenergicβ2Homo sapiensHydroxybenzylisoproterenol--3.12013-09-25doi.org/10.1038/nature12572
4LDOAAmineAdrenergicβ2Homo sapiensL-Epinephrine--3.22013-09-25doi.org/10.1038/nature12572
5JQHAAmineAdrenergicβ2Homo sapiensS-Carazolol--3.22016-07-13doi.org/10.1038/nature18636
5D6LAAmineAdrenergicβ2Homo sapiensS-Carazolol--3.22016-08-17doi.org/10.1038/nprot.2017.057
7BZ2AAmineAdrenergicβ2Homo sapiensArformoterol-Gs/β1/γ23.822020-08-05doi.org/10.1038/s41421-020-0176-9
7BZ2 (No Gprot) AAmineAdrenergicβ2Homo sapiensArformoterol-3.822020-08-05doi.org/10.1038/s41421-020-0176-9
7XKAAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine--3.12023-04-26doi.org/10.1038/s41467-023-37808-y
8GDZAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-Gs/β1/γ23.52024-03-06doi.org/10.1038/s41586-024-07153-1
8GDZ (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-3.52024-03-06doi.org/10.1038/s41586-024-07153-1
8GE1AAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-Gs/β1/γ23.42024-03-06doi.org/10.1038/s41586-024-07153-1
8GE1 (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-3.42024-03-06doi.org/10.1038/s41586-024-07153-1
8GE3AAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-Gs/β1/γ23.32024-03-06doi.org/10.1038/s41586-024-07153-1
8GE3 (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-3.32024-03-06doi.org/10.1038/s41586-024-07153-1
8GE4AAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-Gs/β1/γ23.32024-03-06doi.org/10.1038/s41586-024-07153-1
8GE4 (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-3.32024-03-06doi.org/10.1038/s41586-024-07153-1
8GE6AAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-Gs/β1/γ23.42024-03-06doi.org/10.1038/s41586-024-07153-1
8GE6 (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-3.42024-03-06doi.org/10.1038/s41586-024-07153-1
8GE7AAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-Gs/β1/γ23.42024-03-06doi.org/10.1038/s41586-024-07153-1
8GE7 (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-3.42024-03-06doi.org/10.1038/s41586-024-07153-1
8GE8AAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-Gs/β1/γ23.42024-03-06doi.org/10.1038/s41586-024-07153-1
8GE8 (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-3.42024-03-06doi.org/10.1038/s41586-024-07153-1
8GE9AAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-Gs/β1/γ23.52024-03-06doi.org/10.1038/s41586-024-07153-1
8GE9 (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-3.52024-03-06doi.org/10.1038/s41586-024-07153-1
8GEAAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-Gs/β1/γ23.52024-03-06doi.org/10.1038/s41586-024-07153-1
8GEA (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-3.52024-03-06doi.org/10.1038/s41586-024-07153-1
8GEBAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-Gs/β1/γ23.62024-03-06doi.org/10.1038/s41586-024-07153-1
8GEB (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-3.62024-03-06doi.org/10.1038/s41586-024-07153-1
8GECAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-Gs/β1/γ23.52024-03-06doi.org/10.1038/s41586-024-07153-1
8GEC (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-3.52024-03-06doi.org/10.1038/s41586-024-07153-1
8GEDAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-Gs/β1/γ23.52024-03-06doi.org/10.1038/s41586-024-07153-1
8GED (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-3.52024-03-06doi.org/10.1038/s41586-024-07153-1
8GEEAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-Gs/β1/γ23.72024-03-06doi.org/10.1038/s41586-024-07153-1
8GEE (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-3.72024-03-06doi.org/10.1038/s41586-024-07153-1
8GEFAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-Gs/β1/γ23.82024-03-06doi.org/10.1038/s41586-024-07153-1
8GEF (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-3.82024-03-06doi.org/10.1038/s41586-024-07153-1
8GEGAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-Gs/β1/γ23.82024-03-06doi.org/10.1038/s41586-024-07153-1
8GEG (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-3.82024-03-06doi.org/10.1038/s41586-024-07153-1
8GEHAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-Gs/β1/γ242024-03-06doi.org/10.1038/s41586-024-07153-1
8GEH (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-42024-03-06doi.org/10.1038/s41586-024-07153-1
8GEIAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-Gs/β1/γ24.12024-03-06doi.org/10.1038/s41586-024-07153-1
8GEI (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-4.12024-03-06doi.org/10.1038/s41586-024-07153-1
8GEJAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-Gs/β1/γ24.22024-03-06doi.org/10.1038/s41586-024-07153-1
8GEJ (No Gprot) AAmineAdrenergicβ2Homo sapiensConstrained Epinephrine-4.22024-03-06doi.org/10.1038/s41586-024-07153-1
8GGIAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine--3.52024-03-06doi.org/10.1038/s41586-024-07153-1
8GGJAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine--3.52024-03-06doi.org/10.1038/s41586-024-07153-1
8GGKAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine--3.32024-03-06doi.org/10.1038/s41586-024-07153-1
8GGLAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine--3.22024-03-06doi.org/10.1038/s41586-024-07153-1
8GGMAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine--3.22024-03-06doi.org/10.1038/s41586-024-07153-1
8GGNAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine--3.32024-03-06doi.org/10.1038/s41586-024-07153-1
8GGOAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine--3.22024-03-06doi.org/10.1038/s41586-024-07153-1
8GGPAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine--3.22024-03-06doi.org/10.1038/s41586-024-07153-1
8GGQAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine--3.42024-03-06doi.org/10.1038/s41586-024-07153-1
8GGRAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine--3.42024-03-06doi.org/10.1038/s41586-024-07153-1
8GGSAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine--3.52024-03-06doi.org/10.1038/s41586-024-07153-1
8GGTAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine--3.52024-03-06doi.org/10.1038/s41586-024-07153-1
8GGUAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine--3.42024-03-06doi.org/10.1038/s41586-024-07153-1
8GGVAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine--3.52024-03-06doi.org/10.1038/s41586-024-07153-1
8GGWAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine--3.62024-03-06doi.org/10.1038/s41586-024-07153-1
8GGXAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine--3.62024-03-06doi.org/10.1038/s41586-024-07153-1
8GGYAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine--3.92024-03-06doi.org/10.1038/s41586-024-07153-1
8GGZAAmineAdrenergicβ2Homo sapiensConstrained Epinephrine--3.92024-03-06doi.org/10.1038/s41586-024-07153-1
8GH0AAmineAdrenergicβ2Homo sapiensConstrained Epinephrine--42024-03-06doi.org/10.1038/s41586-024-07153-1
8GH1AAmineAdrenergicβ2Homo sapiensConstrained Epinephrine--4.12024-03-06doi.org/10.1038/s41586-024-07153-1
6MXTAAmineAdrenergicβ2Homo sapiensSalmeterol--2.962018-11-14doi.org/10.1038/s41589-018-0145-x
8JJ8AAmineAdrenergicβ2Homo sapiensFormoterol--3.22023-09-06doi.org/10.1038/s41589-023-01389-0
8JJLAAmineAdrenergicβ2Homo sapiensOlodaterol--3.22023-09-06doi.org/10.1038/s41589-023-01389-0
8JJOAAmineAdrenergicβ2Homo sapiensAlprenolol--3.42023-09-06doi.org/10.1038/s41589-023-01389-0
6NI3AAmineAdrenergicβ2Homo sapiensBI167107-Gs/β1/γ23.82019-11-20doi.org/10.1038/s41594-019-0330-y
6NI3 (No Gprot) AAmineAdrenergicβ2Homo sapiensBI167107-3.82019-11-20doi.org/10.1038/s41594-019-0330-y
4QKXAAmineAdrenergicβ2Homo sapiens35V--3.32014-07-23doi.org/10.1073/pnas.1410415111
9CHUAAmineAdrenergicβ2Homo sapiensNoradrenaline--3.492024-11-13doi.org/10.1073/pnas.2414544121
9CHVAAmineAdrenergicβ2Homo sapiens---3.952024-11-13doi.org/10.1073/pnas.2414544121
9CHXAAmineAdrenergicβ2Homo sapiensS-Carazolol--3.52024-11-13doi.org/10.1073/pnas.2414544121
7DHIAAmineAdrenergicβ2Homo sapiensSalbutamol-Gs/β1/γ23.262020-12-16doi.org/10.1093/nsr/nwaa284
7DHI (No Gprot) AAmineAdrenergicβ2Homo sapiensSalbutamol-3.262020-12-16doi.org/10.1093/nsr/nwaa284
7DHRAAmineAdrenergicβ2Homo sapiensIsoprenaline-Gs/β1/γ23.82020-12-16doi.org/10.1093/nsr/nwaa284
7DHR (No Gprot) AAmineAdrenergicβ2Homo sapiensIsoprenaline-3.82020-12-16doi.org/10.1093/nsr/nwaa284
6PRZAAmineAdrenergicβ2Homo sapiensS-Alprenolol--2.82019-11-13doi.org/10.1107/S2052252519013137
6PS0AAmineAdrenergicβ2Homo sapiensS-Carazolol--3.42019-11-13doi.org/10.1107/S2052252519013137
6PS1AAmineAdrenergicβ2Homo sapiensTimolol--3.22019-11-13doi.org/10.1107/S2052252519013137
6PS2AAmineAdrenergicβ2Homo sapiensS-Alprenolol--2.42019-11-13doi.org/10.1107/S2052252519013137
6PS3AAmineAdrenergicβ2Homo sapiensS-Carvedilol--2.52019-11-13doi.org/10.1107/S2052252519013137
6PS4AAmineAdrenergicβ2Homo sapiensICI118-551--2.62019-11-13doi.org/10.1107/S2052252519013137
6PS5AAmineAdrenergicβ2Homo sapiensS-Propranolol--2.92019-11-13doi.org/10.1107/S2052252519013137
6PS6AAmineAdrenergicβ2Homo sapiensTimolol--2.72019-11-13doi.org/10.1107/S2052252519013137
5D5AAAmineAdrenergicβ2Homo sapiensS-Carazolol--2.482016-01-13doi.org/10.1107/S2059798315021683
5D5BAAmineAdrenergicβ2Homo sapiensS-Carazolol--3.82016-01-13doi.org/10.1107/S2059798315021683
2RH1AAmineAdrenergicβ2Homo sapiensS-Carazolol--2.42007-10-30doi.org/10.1126/science.1150577
4GBRAAmineAdrenergicβ2Homo sapiensS-Carazolol--3.992012-10-24doi.org/10.1371/journal.pone.0046039
8W1VAAmineAdrenergicβ2Homo sapiensPubChem 171716265--32024-07-17doi.org/10.1021/acs.jmedchem.4c00578
9BUYAAmineAdrenergicβ2Homo sapiensLM189-Gi1/β1/γ22.92025-05-28doi.org/10.1126/sciadv.adq3971
9BUY (No Gprot) AAmineAdrenergicβ2Homo sapiensLM189-2.92025-05-28doi.org/10.1126/sciadv.adq3971
7XJIAAmineAdrenergicβ3Canis lupus familiarisSolabegron-Gs/β1/γ23.92022-05-04doi.org/10.1016/j.bbrc.2022.04.065
7XJI (No Gprot) AAmineAdrenergicβ3Canis lupus familiarisSolabegron-3.92022-05-04doi.org/10.1016/j.bbrc.2022.04.065
7DH5AAmineAdrenergicβ3Canis lupus familiarisMirabegron-Gs/β1/γ23.162021-08-04doi.org/10.1016/j.molcel.2021.06.024
7DH5 (No Gprot) AAmineAdrenergicβ3Canis lupus familiarisMirabegron-3.162021-08-04doi.org/10.1016/j.molcel.2021.06.024
7XJHAAmineAdrenergicβ3Canis lupus familiarisIsoproterenol-Gs/β1/γ23.32022-05-04doi.org/10.1016/j.molcel.2021.06.024
7XJH (No Gprot) AAmineAdrenergicβ3Canis lupus familiarisIsoproterenol-3.32022-05-04doi.org/10.1016/j.molcel.2021.06.024
9IJDAAmineAdrenergicβ3Homo sapiensCarazolol-chim(NtGi1-Gs)/β1/γ22.762024-08-21doi.org/10.1002/cplu.202400288
9IJD (No Gprot) AAmineAdrenergicβ3Homo sapiensCarazolol-2.762024-08-21doi.org/10.1002/cplu.202400288
9IJEAAmineAdrenergicβ3Homo sapiensEpinephrine-chim(NtGi1-Gs)/β1/γ22.342024-08-21doi.org/10.1002/cplu.202400288
9IJE (No Gprot) AAmineAdrenergicβ3Homo sapiensEpinephrine-2.342024-08-21doi.org/10.1002/cplu.202400288
9EAHAPeptideAngiotensinAT1Homo sapiensOlmesartanNanobody AT209-3.12025-03-05doi.org/10.1073/pnas.2423931122
9EAIAPeptideAngiotensinAT1Homo sapiensLosartanNanobody AT209-3.12025-03-05doi.org/10.1073/pnas.2423931122
9EAJAPeptideAngiotensinAT1Homo sapiens-Nanobody AT209-3.22025-03-05doi.org/10.1073/pnas.2423931122
8TH4APeptideAngiotensinAT1Homo sapiensLosartanAT118-L Nanobody-3.32024-05-22doi.org/10.1038/s41589-024-01620-6
8TH3APeptideAngiotensinAT1Homo sapiens-AT118-H Nanobody-32024-05-22doi.org/10.1038/s41589-024-01620-6
4YAYAPeptideAngiotensinAT1Homo sapiensZD-7155--2.92015-04-22doi.org/10.1016/j.cell.2015.04.011
6DO1APeptideAngiotensinAT1Homo sapiensAngiotensin-like peptide S1I8--2.92019-01-30doi.org/10.1016/j.cell.2018.12.006
4ZUDAPeptideAngiotensinAT1Homo sapiensOlmesartan--2.82015-10-07doi.org/10.1074/jbc.M115.689000
6OS0APeptideAngiotensinAT1Homo sapiensAngiotensinogen--2.92020-02-19doi.org/10.1126/science.aay9813
6OS1APeptideAngiotensinAT1Homo sapiensTRV026--2.792020-02-19doi.org/10.1126/science.aay9813
6OS2APeptideAngiotensinAT1Homo sapiensTRV026--2.72020-02-19doi.org/10.1126/science.aay9813
7F6GAPeptideAngiotensinAT1Homo sapiensSAR1-AngII-Gq/β1/γ22.92023-03-29doi.org/10.15252/embj.2022112940
7F6G (No Gprot) APeptideAngiotensinAT1Homo sapiensSAR1-AngII-2.92023-03-29doi.org/10.15252/embj.2022112940
6JODAPeptideAngiotensinAT2Homo sapiensAngiotensin II--3.22020-01-15doi.org/10.1016/j.str.2019.12.003
5UNFAPeptideAngiotensinAT2Homo sapiensPubChem 15780052--2.82017-04-05doi.org/10.1038/nature22035
5UNGAPeptideAngiotensinAT2Homo sapiensPubChem 15780052--2.82017-04-05doi.org/10.1038/nature22035
5UNHAPeptideAngiotensinAT2Homo sapiensPubChem 126456406--2.92017-04-05doi.org/10.1038/nature22035
5XJMAPeptideAngiotensinAT2Homo sapiens(Sar1,Ile8)-Angiotensin II--3.22018-07-11doi.org/10.1038/s41594-018-0079-8
7C6AAPeptideAngiotensinAT2Homo sapiens(Sar1,Ile8)-Angiotensin II--3.42020-07-29doi.org/10.1038/s41598-020-68355-x
7JNIAPeptideAngiotensinAT2Homo sapiensOlodanrigan--32022-02-09doi.org/10.1073/pnas.2116289119
8XZFAPeptideApelinApelinHomo sapiensWN561-Gi1/β1/γ232024-03-20doi.org/10.1016/j.cell.2024.02.004
8XZF (No Gprot) APeptideApelinApelinHomo sapiensWN561-32024-03-20doi.org/10.1016/j.cell.2024.02.004
8XZGAPeptideApelinApelinHomo sapiensApelin-13-Gi1/β1/γ23.22024-03-20doi.org/10.1016/j.cell.2024.02.004
8XZG (No Gprot) APeptideApelinApelinHomo sapiensApelin-13-3.22024-03-20doi.org/10.1016/j.cell.2024.02.004
8XZHAPeptideApelinApelinHomo sapiensMM07-Gi1/β1/γ22.062024-03-20doi.org/10.1016/j.cell.2024.02.004
8XZH (No Gprot) APeptideApelinApelinHomo sapiensMM07-2.062024-03-20doi.org/10.1016/j.cell.2024.02.004
8XZJAPeptideApelinApelinHomo sapiensWN353-Gi1/β1/γ232024-03-20doi.org/10.1016/j.cell.2024.02.004
8XZJ (No Gprot) APeptideApelinApelinHomo sapiensWN353-32024-03-20doi.org/10.1016/j.cell.2024.02.004
5VBLAPeptideApelinApelinHomo sapiensApelin mimetic peptide agonist--2.62017-05-31doi.org/10.1016/j.str.2017.04.008
8Z74APeptideApelinApelinHomo sapiensAgonistic antibody--3.012025-01-22doi.org/10.1038/s41467-024-55555-6
8Z7JAPeptideApelinApelinHomo sapiensAgonistic antibody-Gi1/β1/γ23.122025-01-22doi.org/10.1038/s41467-024-55555-6
8Z7J (No Gprot) APeptideApelinApelinHomo sapiensAgonistic antibody-3.122025-01-22doi.org/10.1038/s41467-024-55555-6
7SUSAPeptideApelinApelinHomo sapiensPubChem 122701908--2.72022-07-27doi.org/10.1038/s41594-022-00797-5
7W0LAPeptideApelinApelinHomo sapiensPubChem 122701908-Gi1/β1/γ23.572022-07-27doi.org/10.1038/s41594-022-00797-5
7W0L (No Gprot) APeptideApelinApelinHomo sapiensPubChem 122701908-3.572022-07-27doi.org/10.1038/s41594-022-00797-5
7W0MAPeptideApelinApelinHomo sapiensPubChem 122701908-Gi1/β1/γ23.712022-07-27doi.org/10.1038/s41594-022-00797-5
7W0M (No Gprot) APeptideApelinApelinHomo sapiensPubChem 122701908-3.712022-07-27doi.org/10.1038/s41594-022-00797-5
7W0NAPeptideApelinApelinHomo sapiensElabela-Gi1/β1/γ24.212022-07-27doi.org/10.1038/s41594-022-00797-5
7W0N (No Gprot) APeptideApelinApelinHomo sapiensElabela-4.212022-07-27doi.org/10.1038/s41594-022-00797-5
7W0OAPeptideApelinApelinHomo sapiensElabela-Gi1/β1/γ23.782022-07-27doi.org/10.1038/s41594-022-00797-5
7W0O (No Gprot) APeptideApelinApelinHomo sapiensElabela-3.782022-07-27doi.org/10.1038/s41594-022-00797-5
7W0PAPeptideApelinApelinHomo sapiensElabela-Gi1/β1/γ23.162022-07-27doi.org/10.1038/s41594-022-00797-5
7W0P (No Gprot) APeptideApelinApelinHomo sapiensElabela-3.162022-07-27doi.org/10.1038/s41594-022-00797-5
6KNMAPeptideApelinApelinHomo sapiensJN241-9--3.22020-01-29doi.org/10.1126/sciadv.aax7379
8XZIAPeptideApelinApelinHomo sapiensCMF-019-Gi1/β1/γ22.72024-03-20doi.org/10.1016/j.cell.2024.02.004
8XZI (No Gprot) APeptideApelinApelinHomo sapiensCMF-019-2.72024-03-20doi.org/10.1016/j.cell.2024.02.004
8S4DAPeptideApelinApelinHomo sapiensCMF-019--2.582024-12-04doi.org/10.1038/s41467-024-55381-w
8XQEAPeptideApelinApelinHomo sapiensApelin-13-Gi1/β1/γ23.482025-01-22doi.org/10.1038/s41467-024-55555-6
8XQE (No Gprot) APeptideApelinApelinHomo sapiensApelin-13-3.482025-01-22doi.org/10.1038/s41467-024-55555-6
8XQFAPeptideApelinApelinHomo sapiensApelin-13-Gi1/β1/γ23.132025-01-22doi.org/10.1038/s41467-024-55555-6
8XQF (No Gprot) APeptideApelinApelinHomo sapiensApelin-13-3.132025-01-22doi.org/10.1038/s41467-024-55555-6
8XQIAPeptideApelinApelinHomo sapiens---3.252025-01-22doi.org/10.1038/s41467-024-55555-6
8XQJAPeptideApelinApelinHomo sapiensJN241--2.952025-01-22doi.org/10.1038/s41467-024-55555-6
9JH3APeptideApelinApelinHomo sapiensCMF-019-Gi1/β1/γ22.932025-04-23doi.org/10.1073/pnas.2423432122
9JH3 (No Gprot) APeptideApelinApelinHomo sapiensCMF-019-2.932025-04-23doi.org/10.1073/pnas.2423432122
7BW0ASteroidBile AcidGPBAHomo sapiens--chim(NtGi1-Gs)/β1/γ23.92020-09-02doi.org/10.1038/s41392-020-00262-z
7BW0 (No Gprot) ASteroidBile AcidGPBAHomo sapiens--3.92020-09-02doi.org/10.1038/s41392-020-00262-z
7CFMASteroidBile AcidGPBAHomo sapiensP395-Gs/β1/γ232020-09-09doi.org/10.1038/s41586-020-2569-1
7CFM (No Gprot) ASteroidBile AcidGPBAHomo sapiensP395-32020-09-09doi.org/10.1038/s41586-020-2569-1
7CFNASteroidBile AcidGPBAHomo sapiensINT-777-Gs/β1/γ232020-09-09doi.org/10.1038/s41586-020-2569-1
7CFN (No Gprot) ASteroidBile AcidGPBAHomo sapiensINT-777-32020-09-09doi.org/10.1038/s41586-020-2569-1
7XTQASteroidBile AcidGPBAHomo sapiensR399-Gs/β1/γ23.22022-07-06doi.org/10.1073/pnas.2117054119
7XTQ (No Gprot) ASteroidBile AcidGPBAHomo sapiensR399-3.22022-07-06doi.org/10.1073/pnas.2117054119
9GYOASteroidBile acidGPBAHomo sapiensP395-chim(NtGi1-Gs)/β1/γ22.52024-10-09To be published
9GYO (No Gprot) ASteroidBile acidGPBAHomo sapiensP395-2.52024-10-09To be published
8H0PAPeptideBombesinBB1Homo sapiensNMB30-chim(NtGi1-Gs-CtGq)/β1/γ23.152023-08-09doi.org/10.1038/s41422-022-00743-6
8H0P (No Gprot) APeptideBombesinBB1Homo sapiensNMB30-3.152023-08-09doi.org/10.1038/s41422-022-00743-6
9JF4APeptideBombesinBB1Homo sapiensPD168368--3.62025-07-09To be published
8H0QAPeptideBombesinBB2Homo sapiensGastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ23.32023-08-09doi.org/10.1038/s41422-022-00743-6
8H0Q (No Gprot) APeptideBombesinBB2Homo sapiensGastrin Releasing Peptide-3.32023-08-09doi.org/10.1038/s41422-022-00743-6
7W3ZAPeptideBombesinBB2Homo sapiensGastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ232023-02-22doi.org/10.1073/pnas.2216230120
7W3Z (No Gprot) APeptideBombesinBB2Homo sapiensGastrin Releasing Peptide-32023-02-22doi.org/10.1073/pnas.2216230120
7W40APeptideBombesinBB2Homo sapiensBombesin-chim(NtGi1L-Gq)/β1/γ232023-02-22doi.org/10.1073/pnas.2216230120
7W40 (No Gprot) APeptideBombesinBB2Homo sapiensBombesin-32023-02-22doi.org/10.1073/pnas.2216230120
7W41APeptideBombesinBB2Homo sapiensPD176252--2.952023-02-22doi.org/10.1073/pnas.2216230120
8Y52APeptideBombesinBB3Homo sapiensBA1-chim(NtGi1-Gs-CtGq)/β1/γ22.92024-09-11doi.org/10.1016/j.celrep.2024.114511
8Y52 (No Gprot) APeptideBombesinBB3Homo sapiensBA1-2.92024-09-11doi.org/10.1016/j.celrep.2024.114511
8Y53APeptideBombesinBB3Homo sapiensMK5046-chim(NtGi1-Gs-CtGq)/β1/γ22.932024-09-11doi.org/10.1016/j.celrep.2024.114511
8Y53 (No Gprot) APeptideBombesinBB3Homo sapiensMK5046-2.932024-09-11doi.org/10.1016/j.celrep.2024.114511
8Y51APeptideBombesinBB3Homo sapiens--chim(NtGi1-Gs-CtGq)/β1/γ23.32025-02-12To be published
8Y51 (No Gprot) APeptideBombesinBB3Homo sapiens--3.32025-02-12To be published
7EIBAPeptideBradykininBK1Homo sapiensDes-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ232021-10-13doi.org/10.1038/s41594-021-00645-y
7EIB (No Gprot) APeptideBradykininBK1Homo sapiensDes-Arg10-Kallidin-32021-10-13doi.org/10.1038/s41594-021-00645-y
7F6HAPeptideBradykininBK2Homo sapiensBradykinin-Gq/β1/γ22.92022-01-05doi.org/10.1038/s41467-022-28399-1
7F6H (No Gprot) APeptideBradykininBK2Homo sapiensBradykinin-2.92022-01-05doi.org/10.1038/s41467-022-28399-1
7F6IAPeptideBradykininBK2Homo sapiensKallidin-Gq/β1/γ22.82022-01-05doi.org/10.1038/s41467-022-28399-1
7F6I (No Gprot) APeptideBradykininBK2Homo sapiensKallidin-2.82022-01-05doi.org/10.1038/s41467-022-28399-1
7F2OAPeptideBradykininBK2Homo sapiensBradykinin-chim(NtGi1-Gs-CtGq)/β1/γ22.92021-10-13doi.org/10.1038/s41594-021-00645-y
7F2O (No Gprot) APeptideBradykininBK2Homo sapiensBradykinin-2.92021-10-13doi.org/10.1038/s41594-021-00645-y
6NIYB1PeptideCalcitoninCTHomo sapiensAdrenomedullin-Gs/β1/γ23.342019-01-23doi.org/10.1021/acsptsci.8b00056
6NIY (No Gprot) B1PeptideCalcitoninCTHomo sapiensAdrenomedullin-3.342019-01-23doi.org/10.1021/acsptsci.8b00056
5UZ7B1PeptideCalcitoninCTHomo sapiens--Gs/β1/γ24.12017-05-03doi.org/10.1038/nature22327
5UZ7 (No Gprot) B1PeptideCalcitoninCTHomo sapiens--4.12017-05-03doi.org/10.1038/nature22327
8F0JB1PeptideCalcitoninCTHomo sapiensPramlintide Analogue San45-Gs/β1/γ222023-08-02doi.org/10.1038/s41589-023-01393-4
8F0J (No Gprot) B1PeptideCalcitoninCTHomo sapiensPramlintide Analogue San45-22023-08-02doi.org/10.1038/s41589-023-01393-4
7TYLB1PeptideCalcitoninCTHomo sapiensAmylin-Gs/β1/γ23.32022-03-23doi.org/10.1126/science.abm9609
7TYL (No Gprot) B1PeptideCalcitoninCTHomo sapiensAmylin-3.32022-03-23doi.org/10.1126/science.abm9609
7TYOB1PeptideCalcitoninCTHomo sapiensCalcitonin-Gs/β1/γ22.72022-03-23doi.org/10.1126/science.abm9609
7TYO (No Gprot) B1PeptideCalcitoninCTHomo sapiensCalcitonin-2.72022-03-23doi.org/10.1126/science.abm9609
7TYIB1PeptideCalcitoninCTHomo sapiensAmylin-Gs/β1/γ23.32022-03-30doi.org/10.1126/science.abm9609
7TYI (No Gprot) B1PeptideCalcitoninCTHomo sapiensAmylin-3.32022-03-30doi.org/10.1126/science.abm9609
7TYNB1PeptideCalcitoninCTHomo sapiensCalcitonin-1-Gs/β1/γ22.62022-03-30doi.org/10.1126/science.abm9609
7TYN (No Gprot) B1PeptideCalcitoninCTHomo sapiensCalcitonin-1-2.62022-03-30doi.org/10.1126/science.abm9609
9BUBB1PeptideCalcitoninCTHomo sapiensCagrilintide-Gs/β1/γ22.32025-04-23doi.org/10.1038/s41467-025-58680-y
9BUB (No Gprot) B1PeptideCalcitoninCTHomo sapiensCagrilintide-2.32025-04-23doi.org/10.1038/s41467-025-58680-y
9BLBB1PeptideCalcitoninCTHomo sapiensCagrilintide backbone (non-acylated)-Gs/β1/γ23.22025-04-16To be published
9BLB (No Gprot) B1PeptideCalcitoninCTHomo sapiensCagrilintide backbone (non-acylated)-3.22025-04-16To be published
9BLCB1PeptideCalcitoninCTHomo sapiensCagrilintide backbone (non-acylated)-Gs/β1/γ23.32025-04-16To be published
9BLC (No Gprot) B1PeptideCalcitoninCTHomo sapiensCagrilintide backbone (non-acylated)-3.32025-04-16To be published
9BUEB1PeptideCalcitoninCTHomo sapiensCagrilintide-Gs/β1/γ23.62025-04-16To be published
9BUE (No Gprot) B1PeptideCalcitoninCTHomo sapiensCagrilintide-3.62025-04-16To be published
9BUCB1PeptideCalcitoninCTHomo sapiensCagrilintide-Gs/β1/γ23.42025-04-23To be published
9BUC (No Gprot) B1PeptideCalcitoninCTHomo sapiensCagrilintide-3.42025-04-23To be published
9BUDB1PeptideCalcitoninCTHomo sapiensCagrilintide-Gs/β1/γ22.52025-04-23To be published
9BUD (No Gprot) B1PeptideCalcitoninCTHomo sapiensCagrilintide-2.52025-04-23To be published
9AUCB1PeptideCalcitoninCT (AMY1)Homo sapiensCalcitonin gene-related peptide-1-Gs/β1/γ2; RAMP12.42024-04-24doi.org/10.1021/acs.biochem.4c00114
9AUC (No Gprot) B1PeptideCalcitoninCT (AMY1)Homo sapiensCalcitonin gene-related peptide-1-2.42024-04-24doi.org/10.1021/acs.biochem.4c00114
7TYFB1PeptideCalcitoninCT (AMY1)Homo sapiensAmylin-Gs/β1/γ2; RAMP12.22022-03-23doi.org/10.1126/science.abm9609
7TYF (No Gprot) B1PeptideCalcitoninCT (AMY1)Homo sapiensAmylin-2.22022-03-23doi.org/10.1126/science.abm9609
7TYWB1PeptideCalcitoninCT (AMY1)Homo sapiensCalcitonin-1-Gs/β1/γ2; RAMP132022-03-23doi.org/10.1126/science.abm9609
7TYW (No Gprot) B1PeptideCalcitoninCT (AMY1)Homo sapiensCalcitonin-1-32022-03-23doi.org/10.1126/science.abm9609
9BLWB1PeptideCalcitoninCT (AMY1)Homo sapiensCagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP13.22025-04-16To be published
9BLW (No Gprot) B1PeptideCalcitoninCT (AMY1)Homo sapiensCagrilintide backbone (non-acylated)-3.22025-04-16To be published
9BP3B1PeptideCalcitoninCT (AMY1)Homo sapiensCagrilintide-Gs/β1/γ2; RAMP12.22025-04-23To be published
9BP3 (No Gprot) B1PeptideCalcitoninCT (AMY1)Homo sapiensCagrilintide-2.22025-04-23To be published
7TYHB1PeptideCalcitoninCT (AMY2)Homo sapiensCalcitonin-1-Gs/β1/γ2; RAMP23.32022-03-23doi.org/10.1126/science.abm9609
7TYH (No Gprot) B1PeptideCalcitoninCT (AMY2)Homo sapiensCalcitonin-1-3.32022-03-23doi.org/10.1126/science.abm9609
7TYYB1PeptideCalcitoninCT (AMY2)Homo sapiensCalcitonin-1-Gs/β1/γ2; RAMP232022-03-23doi.org/10.1126/science.abm9609
7TYY (No Gprot) B1PeptideCalcitoninCT (AMY2)Homo sapiensCalcitonin-1-32022-03-23doi.org/10.1126/science.abm9609
7TYXB1PeptideCalcitoninCT (AMY2)Homo sapiensAmylin-Gs/β1/γ2; RAMP22.552022-03-30doi.org/10.1126/science.abm9609
7TYX (No Gprot) B1PeptideCalcitoninCT (AMY2)Homo sapiensAmylin-2.552022-03-30doi.org/10.1126/science.abm9609
9BQ3B1PeptideCalcitoninCT (AMY2)Homo sapiensCagrilintide-Gs/β1/γ2; RAMP22.82025-04-23To be published
9BQ3 (No Gprot) B1PeptideCalcitoninCT (AMY2)Homo sapiensCagrilintide-2.82025-04-23To be published
8F0KB1PeptideCalcitoninCT (AMY3)Homo sapiensPramlintide Analogue San385-Gs/β1/γ2; RAMP31.92023-08-02doi.org/10.1038/s41589-023-01393-4
8F0K (No Gprot) B1PeptideCalcitoninCT (AMY3)Homo sapiensPramlintide Analogue San385-1.92023-08-02doi.org/10.1038/s41589-023-01393-4
8F2AB1PeptideCalcitoninCT (AMY3)Homo sapiensPramlintide Analogue San385-Gs/β1/γ2; RAMP32.22023-08-02doi.org/10.1038/s41589-023-01393-4
8F2A (No Gprot) B1PeptideCalcitoninCT (AMY3)Homo sapiensPramlintide Analogue San385-2.22023-08-02doi.org/10.1038/s41589-023-01393-4
8F2BB1PeptideCalcitoninCT (AMY3)Homo sapiensPramlintide Analogue San45-Gs/β1/γ2; RAMP322023-08-02doi.org/10.1038/s41589-023-01393-4
8F2B (No Gprot) B1PeptideCalcitoninCT (AMY3)Homo sapiensPramlintide Analogue San45-22023-08-02doi.org/10.1038/s41589-023-01393-4
7TZFB1PeptideCalcitoninCT (AMY3)Homo sapiensAmylin-Gs/β1/γ2; RAMP32.42022-03-23doi.org/10.1126/science.abm9609
7TZF (No Gprot) B1PeptideCalcitoninCT (AMY3)Homo sapiensAmylin-2.42022-03-23doi.org/10.1126/science.abm9609
9BTWB1PeptideCalcitoninCT (AMY3)Homo sapiensCagrilintide-Gs/β1/γ2; RAMP332025-04-16To be published
9BTW (No Gprot) B1PeptideCalcitoninCT (AMY3)Homo sapiensCagrilintide-32025-04-16To be published
6E3YB1PeptideCalcitoninCT LikeHomo sapiensCalcitonin gene-related peptide-1-Gs/β1/γ2; RAMP13.32018-09-19doi.org/10.1038/s41586-018-0535-y
6E3Y (No Gprot) B1PeptideCalcitoninCT LikeHomo sapiensCalcitonin gene-related peptide-1-3.32018-09-19doi.org/10.1038/s41586-018-0535-y
7KNTB1PeptideCalcitoninCT LikeHomo sapiens--RAMP13.152021-02-24doi.org/10.1126/science.abf7258
7KNUB1PeptideCalcitoninCT LikeHomo sapiensCalcitonin gene-related peptide-1-RAMP13.492021-02-24doi.org/10.1126/science.abf7258
6UUNB1PeptideCalcitoninCT Like (AM1)Homo sapiensAdrenomedullin-Gs/β1/γ2; RAMP232020-03-25doi.org/10.1021/acsptsci.9b00080
6UUN (No Gprot) B1PeptideCalcitoninCT Like (AM1)Homo sapiensAdrenomedullin-32020-03-25doi.org/10.1021/acsptsci.9b00080
6UUSB1PeptideCalcitoninCT Like (AM2)Homo sapiensAdrenomedullin-Gs/β1/γ2; RAMP32.42020-04-01doi.org/10.1021/acsptsci.9b00080
6UUS (No Gprot) B1PeptideCalcitoninCT Like (AM2)Homo sapiensAdrenomedullin-2.42020-04-01doi.org/10.1021/acsptsci.9b00080
6UVAB1PeptideCalcitoninCT Like (AM2)Homo sapiensAdrenomedullin-2-Gs/β1/γ2; RAMP32.32020-04-01doi.org/10.1021/acsptsci.9b00080
6UVA (No Gprot) B1PeptideCalcitoninCT Like (AM2)Homo sapiensAdrenomedullin-2-2.32020-04-01doi.org/10.1021/acsptsci.9b00080
8WPGCIonCalcium SensingCaSHomo sapiens-Tryptophan; Cinacalcet; PO4; Ca-2.72023-11-22doi.org/10.1038/s41422-023-00892-2
8WPUCIonCalcium SensingCaSHomo sapiens-Tryptophan; Cinacalcet; PO4; Cachim(NtGi2L-Gs-CtGq)/β1/γ23.12023-11-22doi.org/10.1038/s41422-023-00892-2
8WPU (No Gprot) CIonCalcium SensingCaSHomo sapiens-Tryptophan; Cinacalcet; PO4; Ca3.12023-11-22doi.org/10.1038/s41422-023-00892-2
7DTUCIonCalcium SensingCaSHomo sapiens-Tryptophan-4.42021-03-10doi.org/10.1038/s41422-021-00474-0
7M3JCIonCalcium SensingCaSHomo sapiens-NPS-2143; PO4-4.12021-06-30doi.org/10.1038/s41586-021-03691-0
7SINCIonCalcium SensingCaSHomo sapiens-NPS-2143-5.92022-01-19doi.org/10.1073/pnas.2115849118
9C1PCIonCalcium SensingCaSHomo sapiensCaCa; Tryptophan; '6218; PO4-2.82024-10-02doi.org/10.1126/science.ado1868
7DTVCIonCalcium SensingCaSHomo sapiensCaCa; Tryptophan-3.52021-03-10doi.org/10.1038/s41422-021-00474-0
7M3ECIonCalcium SensingCaSHomo sapiens-Ca; Ca; Tryptophan; NPS-2143-3.22021-06-30doi.org/10.1038/s41586-021-03691-0
7DD5CIonCalcium SensingCaSGallus gallusCaCa; Ca; Tryptophan; NPS-2143-3.22021-06-16doi.org/10.1126/sciadv.abg1483
7M3GCIonCalcium SensingCaSHomo sapiens-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4-2.52021-06-30doi.org/10.1038/s41586-021-03691-0
7DD7CIonCalcium SensingCaSGallus gallusCaCa; Ca; Tryptophan; Evocalcet-3.22021-06-16doi.org/10.1126/sciadv.abg1483
8SZFCIonCalcium SensingCaSHomo sapiens-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-2.82024-02-07doi.org/10.1038/s41586-024-07055-2
8SZGCIonCalcium SensingCaSHomo sapiens-Ca; Ca; Tryptophan; Cinacalcet; PO4; Sperminechim(NtGi1-Gq)/β1/γ23.62024-02-07doi.org/10.1038/s41586-024-07055-2
8SZG (No Gprot) CIonCalcium SensingCaSHomo sapiens-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine3.62024-02-07doi.org/10.1038/s41586-024-07055-2
8SZHCIonCalcium SensingCaSHomo sapiens-Ca; Ca; Tryptophan; Cinacalcet; PO4; SpermineGi1/β1/γ23.12024-02-07doi.org/10.1038/s41586-024-07055-2
8SZH (No Gprot) CIonCalcium SensingCaSHomo sapiens-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine3.12024-02-07doi.org/10.1038/s41586-024-07055-2
7M3FCIonCalcium SensingCaSHomo sapiens-Ca; Ca; Tryptophan; Cinacalcet; PO4-2.82021-06-30doi.org/10.1038/s41586-021-03691-0
8SZICIonCalcium SensingCaSHomo sapiens-Ca; Ca; Tryptophan; Cinacalcet; PO4Gi3/β1/γ23.52024-02-07doi.org/10.1038/s41586-024-07055-2
8SZI (No Gprot) CIonCalcium SensingCaSHomo sapiens-Ca; Ca; Tryptophan; Cinacalcet; PO43.52024-02-07doi.org/10.1038/s41586-024-07055-2
9C2FCIonCalcium SensingCaSHomo sapiensCaCa; Ca; Tryptophan; '54149; PO4-2.82024-10-02doi.org/10.1126/science.ado1868
7DD6CIonCalcium SensingCaSGallus gallusCaCa; Ca; Tryptophan-3.22021-06-16doi.org/10.1126/sciadv.abg1483
7SIMCIonCalcium SensingCaSHomo sapiensCaCa; Ca; Cyclomethyltryptophan; PO4-2.72022-01-19doi.org/10.1073/pnas.2115849118
7E6TCIonCalcium SensingCaSHomo sapiensCaCa; Ca; Cyclomethyltryptophan; PO4-32021-09-22doi.org/10.7554/eLife.68578
9ASBCIonCalcium SensingCaSHomo sapiensCaCa; Ca; Cyclomethyltryptophan; 9IG; PO4chim(NtGi1-Gs-CtGq)/β1/γ23.42024-04-17doi.org/10.1038/s41586-024-07331-1
9ASB (No Gprot) CIonCalcium SensingCaSHomo sapiensCaCa; Ca; Cyclomethyltryptophan; 9IG; PO43.42024-04-17doi.org/10.1038/s41586-024-07331-1
9AVGCIonCalcium SensingCaSHomo sapiensCaCa; Ca; Cyclomethyltryptophan; 9IG; PO4chim(NtGi1-Gs)/β1/γ23.62024-04-17doi.org/10.1038/s41586-024-07331-1
9AVG (No Gprot) CIonCalcium SensingCaSHomo sapiensCaCa; Ca; Cyclomethyltryptophan; 9IG; PO43.62024-04-17doi.org/10.1038/s41586-024-07331-1
9AVLCIonCalcium SensingCaSHomo sapiensCaCa; Ca; Cyclomethyltryptophan; 9IG; PO4Gi3/β2/γ23.82024-04-17doi.org/10.1038/s41586-024-07331-1
9AVL (No Gprot) CIonCalcium SensingCaSHomo sapiensCaCa; Ca; Cyclomethyltryptophan; 9IG; PO43.82024-04-17doi.org/10.1038/s41586-024-07331-1
9AXFCIonCalcium SensingCaSHomo sapiensCaCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4chim(NtGi1-Gs-CtGq)/β1/γ23.52024-04-17doi.org/10.1038/s41586-024-07331-1
9AXF (No Gprot) CIonCalcium SensingCaSHomo sapiensCaCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO43.52024-04-17doi.org/10.1038/s41586-024-07331-1
9AYFCIonCalcium SensingCaSHomo sapiensCaCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4Gi1/β1/γ23.62024-04-17doi.org/10.1038/s41586-024-07331-1
9AYF (No Gprot) CIonCalcium SensingCaSHomo sapiensCaCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO43.62024-04-17doi.org/10.1038/s41586-024-07331-1
7SILCIonCalcium SensingCaSHomo sapiensCaCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-2.72022-01-19doi.org/10.1073/pnas.2115849118
7DTTCIonCalcium SensingCaSHomo sapiensCaCa-3.82021-03-10doi.org/10.1038/s41422-021-00474-0
7DTWCIonCalcium SensingCaSHomo sapiens---4.52021-03-10doi.org/10.1038/s41422-021-00474-0
7E6UCIonCalcium SensingCaSHomo sapiens---62021-09-22doi.org/10.7554/eLife.68578
7FEEALipidCannabinoidCB1Homo sapiensCP55940ZCZ011-2.72022-06-15doi.org/10.1038/s41589-022-01038-y
7WV9ALipidCannabinoidCB1Homo sapiensCP55940ZCZ011Gi2/β1/γ23.362022-06-15doi.org/10.1038/s41589-022-01038-y
7WV9 (No Gprot) ALipidCannabinoidCB1Homo sapiensCP55940ZCZ0113.362022-06-15doi.org/10.1038/s41589-022-01038-y
8IKHALipidCannabinoidCB1Homo sapiens-Q2LGi1/β1/γ13.32024-06-05doi.org/10.1073/pnas.2321532121
8IKH (No Gprot) ALipidCannabinoidCB1Homo sapiens-Q2L3.32024-06-05doi.org/10.1073/pnas.2321532121
8IKGALipidCannabinoidCB1Homo sapiens-Q2BGi1/β1/γ13.42024-06-05doi.org/10.1073/pnas.2321532121
8IKG (No Gprot) ALipidCannabinoidCB1Homo sapiens-Q2B3.42024-06-05doi.org/10.1073/pnas.2321532121
6KQIALipidCannabinoidCB1Homo sapiensCP55940Org27569-3.252019-10-23doi.org/10.1038/s41589-019-0387-2
8K8JALipidCannabinoidCB1Homo sapiensFenofibrate-chim(Gs-CtGq)/β1/γ22.882024-02-14doi.org/10.1002/advs.202306311
8K8J (No Gprot) ALipidCannabinoidCB1Homo sapiensFenofibrate-2.882024-02-14doi.org/10.1002/advs.202306311
5TGZALipidCannabinoidCB1Homo sapiensAM6538--2.82016-11-02doi.org/10.1016/j.cell.2016.10.004
6N4BALipidCannabinoidCB1Homo sapiensMDMB-Fubinaca-Gi1/β1/γ232019-01-30doi.org/10.1016/j.cell.2018.11.040
6N4B (No Gprot) ALipidCannabinoidCB1Homo sapiensMDMB-Fubinaca-32019-01-30doi.org/10.1016/j.cell.2018.11.040
6KPGALipidCannabinoidCB1Homo sapiensAM841-Gi1/β1/γ232020-02-12doi.org/10.1016/j.cell.2020.01.008
6KPG (No Gprot) ALipidCannabinoidCB1Homo sapiensAM841-32020-02-12doi.org/10.1016/j.cell.2020.01.008
7V3ZALipidCannabinoidCB1Homo sapiensCP55940--3.292021-11-24doi.org/10.1021/jacs.1c06847
5U09ALipidCannabinoidCB1Homo sapiensTaranabant--2.62016-12-07doi.org/10.1038/nature20613
5XR8ALipidCannabinoidCB1Homo sapiensAM841--2.952017-07-12doi.org/10.1038/nature23272
5XRAALipidCannabinoidCB1Homo sapiensAM11542--2.82017-07-12doi.org/10.1038/nature23272
8GHVALipidCannabinoidCB1Homo sapiensAMG315-Gi1/β1/γ22.82023-05-24doi.org/10.1038/s41467-023-37864-4
8GHV (No Gprot) ALipidCannabinoidCB1Homo sapiensAMG315-2.82023-05-24doi.org/10.1038/s41467-023-37864-4
9B9ZALipidCannabinoidCB1Homo sapiensA1AKO--3.32024-11-20doi.org/10.1038/s41467-024-54206-0
9BA0ALipidCannabinoidCB1Homo sapiensA1AKN--3.132024-11-20doi.org/10.1038/s41467-024-54206-0
9B9YALipidCannabinoidCB1Homo sapiens7DY--3.52024-11-20doi.org/10.1038/s41467-024-54206-0
9B54ALipidCannabinoidCB1Homo sapiensA1AIW-Gi1/β1/γ22.862025-03-05doi.org/10.1038/s41586-025-08618-7
9B54 (No Gprot) ALipidCannabinoidCB1Homo sapiensA1AIW-2.862025-03-05doi.org/10.1038/s41586-025-08618-7
9B65ALipidCannabinoidCB1Homo sapiensKCA-Gi1/β1/γ23.032025-03-05doi.org/10.1038/s41586-025-08618-7
9B65 (No Gprot) ALipidCannabinoidCB1Homo sapiensKCA-3.032025-03-05doi.org/10.1038/s41586-025-08618-7
8WRZALipidCannabinoidCB1Homo sapiensPubChem 102336704-Arrestin23.62024-02-28doi.org/10.1093/procel/pwad055
9ERXALipidCannabinoidCB1Homo sapiensD9-THC analog-Gi1/β1/γ22.92024-06-26doi.org/10.21203/rs.3.rs-4277209/v1
9ERX (No Gprot) ALipidCannabinoidCB1Homo sapiensD9-THC analog-2.92024-06-26doi.org/10.21203/rs.3.rs-4277209/v1
8WU1ALipidCannabinoidCB1Homo sapiensPubChem 119025665-Arrestin23.22024-03-20doi.org/10.1016/j.cell.2023.11.017
9DGIALipidCannabinoidCB1Homo sapiensZ8526711350--3.352025-04-30doi.org/10.1038/s41467-025-57136-7
9EGOALipidCannabinoidCB1Homo sapiensYVF-Gi1/β1/γ23.22025-04-30doi.org/10.1038/s41467-025-57136-7
9EGO (No Gprot) ALipidCannabinoidCB1Homo sapiensYVF-3.22025-04-30doi.org/10.1038/s41467-025-57136-7
8GAGALipidCannabinoidCB1Homo sapiensPubChem 170838490-Gi1/β1/γ23.32024-02-28To be published
8GAG (No Gprot) ALipidCannabinoidCB1Homo sapiensPubChem 170838490-3.32024-02-28To be published
5ZTYALipidCannabinoidCB2Homo sapiensAM10257--2.82019-01-30doi.org/10.1016/j.cell.2018.12.011
6PT0ALipidCannabinoidCB2Homo sapiensWIN 55212-2-Gi1/β1/γ23.22020-02-12doi.org/10.1016/j.cell.2020.01.007
6PT0 (No Gprot) ALipidCannabinoidCB2Homo sapiensWIN 55212-2-3.22020-02-12doi.org/10.1016/j.cell.2020.01.007
6KPCALipidCannabinoidCB2Homo sapiensPubChem 145915889--3.22020-02-12doi.org/10.1016/j.cell.2020.01.008
6KPFALipidCannabinoidCB2Homo sapiensPubChem 145915889-Gi1/β1/γ22.92020-02-12doi.org/10.1016/j.cell.2020.01.008
6KPF (No Gprot) ALipidCannabinoidCB2Homo sapiensPubChem 145915889-2.92020-02-12doi.org/10.1016/j.cell.2020.01.008
8GUQALipidCannabinoidCB2Homo sapiensOlorinab-Gi1/β1/γ23.082023-05-10doi.org/10.1038/s41467-023-37112-9
8GUQ (No Gprot) ALipidCannabinoidCB2Homo sapiensOlorinab-3.082023-05-10doi.org/10.1038/s41467-023-37112-9
8GURALipidCannabinoidCB2Homo sapiensCP55,940-Gi1/β1/γ22.842023-05-10doi.org/10.1038/s41467-023-37112-9
8GUR (No Gprot) ALipidCannabinoidCB2Homo sapiensCP55,940-2.842023-05-10doi.org/10.1038/s41467-023-37112-9
8GUSALipidCannabinoidCB2Homo sapiensHU-308-Gi1/β1/γ22.972023-05-10doi.org/10.1038/s41467-023-37112-9
8GUS (No Gprot) ALipidCannabinoidCB2Homo sapiensHU-308-2.972023-05-10doi.org/10.1038/s41467-023-37112-9
8GUTALipidCannabinoidCB2Homo sapiensLEI-102-Gi1/β1/γ22.982023-05-10doi.org/10.1038/s41467-023-37112-9
8GUT (No Gprot) ALipidCannabinoidCB2Homo sapiensLEI-102-2.982023-05-10doi.org/10.1038/s41467-023-37112-9
8X3LALipidCannabinoidCB2Homo sapiensXWD-Gi1/β1/γ23.132024-11-20doi.org/10.1073/pnas.2401091121
8X3L (No Gprot) ALipidCannabinoidCB2Homo sapiensXWD-3.132024-11-20doi.org/10.1073/pnas.2401091121
7YKDAProteinChemerinCML1Homo sapiensChemerin-9-Gi1/β1/γ22.812023-04-19doi.org/10.1073/pnas.2214324120
7YKD (No Gprot) AProteinChemerinCML1Homo sapiensChemerin-9-2.812023-04-19doi.org/10.1073/pnas.2214324120
8SG1AProteinChemerinCML1Homo sapiensChemerin-9-Gi1/β1/γ22.942023-11-01doi.org/10.1371/journal.pbio.3002188
8SG1 (No Gprot) AProteinChemerinCML1Homo sapiensChemerin-9-2.942023-11-01doi.org/10.1371/journal.pbio.3002188
8ZJGAProteinChemerinCML1Homo sapiensChemerin-Gi1/β1/γ23.182025-01-22doi.org/10.1038/s42003-024-07228-9
8ZJG (No Gprot) AProteinChemerinCML1Homo sapiensChemerin-3.182025-01-22doi.org/10.1038/s42003-024-07228-9
9L3WAProteinChemerinCML1Homo sapiensRetinoic acid receptor responder protein 2-Gi1/β1/γ23.52025-03-12doi.org/10.1093/procel/pwae073
9L3W (No Gprot) AProteinChemerinCML1Homo sapiensRetinoic acid receptor responder protein 2-3.52025-03-12doi.org/10.1093/procel/pwae073
9L3ZAProteinChemerinCML1Homo sapiensLRH7-C2--3.92025-03-12doi.org/10.1093/procel/pwae073
9L3YAProteinChemerinCML2Homo sapiensRetinoic acid receptor responder protein 2-Gi1/β1/γ23.62025-03-12doi.org/10.1093/procel/pwae073
9L3Y (No Gprot) AProteinChemerinCML2Homo sapiensRetinoic acid receptor responder protein 2-3.62025-03-12doi.org/10.1093/procel/pwae073
8JJPAProteinChemerinCML2Homo sapiensChemerin-Gi1/β1/γ22.92024-08-21doi.org/10.1371/journal.pbio.3002838
8JJP (No Gprot) AProteinChemerinCML2Homo sapiensChemerin-2.92024-08-21doi.org/10.1371/journal.pbio.3002838
8XGMAProteinChemerinCML2Homo sapiensChemerin-Gi1/β1/γ23.292024-08-21doi.org/10.1371/journal.pbio.3002838
8XGM (No Gprot) AProteinChemerinCML2Homo sapiensChemerin-3.292024-08-21doi.org/10.1371/journal.pbio.3002838
5LWEAProteinChemokineCCR9Homo sapiens-Vercirnon-2.82016-12-07doi.org/10.1038/nature20606
6LFLAProteinChemokineCXCR2Homo sapiens-PubChem 153466996-3.22020-09-02doi.org/10.1038/s41586-020-2492-5
5T1AAProteinChemokineCCR2Homo sapiensBMS-681PubChem 12093170-2.812016-12-14doi.org/10.1038/nature20605
6AKYAProteinChemokineCCR5Homo sapiens-Maraviroc-2.82018-10-24doi.org/10.1021/acs.jmedchem.8b01077
4MBSAProteinChemokineCCR5Homo sapiens-Maraviroc-2.712013-09-11doi.org/10.1126/science.1241475
6QZHAProteinChemokineCCR7Homo sapiens-Cmp2105; Na-2.12019-09-04doi.org/10.1016/j.cell.2019.07.028
7SK7AProteinChemokineACKR3Homo sapiensCXCL12CCX662-3.32022-07-27doi.org/10.1126/sciadv.abn8063
7SK8AProteinChemokineACKR3Homo sapiensCXCL12CCX662-3.32022-07-27doi.org/10.1126/sciadv.abn8063
7SK9AProteinChemokineACKR3Homo sapiens-CCX662-3.72022-07-27doi.org/10.1126/sciadv.abn8063
6AKXAProteinChemokineCCR5Homo sapiens-A4R-2.82018-10-24doi.org/10.1021/acs.jmedchem.8b01077
8JPSAProteinChemokineACKR1Homo sapiensCCL7--3.652024-07-31doi.org/10.1016/j.cell.2024.07.005
7SK3AProteinChemokineACKR3Homo sapiensCXCL12--3.82022-07-27doi.org/10.1126/sciadv.abn8063
7SK4AProteinChemokineACKR3Homo sapiensCXCL12_LRHQ--3.32022-07-27doi.org/10.1126/sciadv.abn8063
7SK5AProteinChemokineACKR3Homo sapiensCXCL12--42022-07-27doi.org/10.1126/sciadv.abn8063
7SK6AProteinChemokineACKR3Homo sapiensCXCL12_LRHQ--42022-07-27doi.org/10.1126/sciadv.abn8063
9E82AProteinChemokineACKR3Homo sapiensSDF-1-β-Arrestin23.42025-04-02To be published
7VL8AProteinChemokineCCR1Homo sapiens--Gi1/β1/γ22.92022-03-23doi.org/10.1038/s41589-021-00918-z
7VL8 (No Gprot) AProteinChemokineCCR1Homo sapiens--2.92022-03-23doi.org/10.1038/s41589-021-00918-z
7VL9AProteinChemokineCCR1Homo sapiensCCL15(26-92)-Gi1/β1/γ22.62022-03-23doi.org/10.1038/s41589-021-00918-z
7VL9 (No Gprot) AProteinChemokineCCR1Homo sapiensCCL15(26-92)-2.62022-03-23doi.org/10.1038/s41589-021-00918-z
7VLAAProteinChemokineCCR1Homo sapiensCCL15(27-92)-Gi1/β1/γ22.72022-03-23doi.org/10.1038/s41589-021-00918-z
7VLA (No Gprot) AProteinChemokineCCR1Homo sapiensCCL15(27-92)-2.72022-03-23doi.org/10.1038/s41589-021-00918-z
6GPSAProteinChemokineCCR2Homo sapiensMK0812--3.32019-01-02doi.org/10.1016/j.str.2018.10.027
6GPXAProteinChemokineCCR2Homo sapiensMK0812--2.72019-01-02doi.org/10.1016/j.str.2018.10.027
7XA3AProteinChemokineCCR2Homo sapiensCCL2-Gi1/β1/γ22.92022-08-24doi.org/10.1038/s41421-022-00403-4
7XA3 (No Gprot) AProteinChemokineCCR2Homo sapiensCCL2-2.92022-08-24doi.org/10.1038/s41421-022-00403-4
7X9YAProteinChemokineCCR3Homo sapiens--Gi1/β1/γ23.12022-08-24doi.org/10.1038/s41421-022-00403-4
7X9Y (No Gprot) AProteinChemokineCCR3Homo sapiens--3.12022-08-24doi.org/10.1038/s41421-022-00403-4
5UIWAProteinChemokineCCR5Homo sapiens5P7-CCL5--2.22017-06-28doi.org/10.1016/j.immuni.2017.05.002
7F1QAProteinChemokineCCR5Homo sapiensMIP-1a-Gi1/β1/γ22.92021-07-14doi.org/10.1038/s41467-021-24438-5
7F1Q (No Gprot) AProteinChemokineCCR5Homo sapiensMIP-1a-2.92021-07-14doi.org/10.1038/s41467-021-24438-5
7F1RAProteinChemokineCCR5Homo sapiens--Gi1/β1/γ232021-07-14doi.org/10.1038/s41467-021-24438-5
7F1R (No Gprot) AProteinChemokineCCR5Homo sapiens--32021-07-14doi.org/10.1038/s41467-021-24438-5
7F1SAProteinChemokineCCR5Homo sapiens--Gi1/β1/γ22.82021-07-14doi.org/10.1038/s41467-021-24438-5
7F1S (No Gprot) AProteinChemokineCCR5Homo sapiens--2.82021-07-14doi.org/10.1038/s41467-021-24438-5
7F1TAProteinChemokineCCR5Homo sapiensMIP-1a--2.62021-07-14doi.org/10.1038/s41467-021-24438-5
6MEOAProteinChemokineCCR5Homo sapiensEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4--3.92018-12-12doi.org/10.1038/s41586-018-0804-9
6METAProteinChemokineCCR5Homo sapiensEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4--4.52018-12-12doi.org/10.1038/s41586-018-0804-9
7O7FAProteinChemokineCCR5Homo sapiens6P4-CCL5-Gi1/β1/γ13.152021-06-30doi.org/10.1126/sciadv.abg8685
7O7F (No Gprot) AProteinChemokineCCR5Homo sapiens6P4-CCL5-3.152021-06-30doi.org/10.1126/sciadv.abg8685
6WWZAProteinChemokineCCR6Homo sapiensCCL20-Go/β1/γ23.342020-06-24doi.org/10.1038/s41467-020-16820-6
6WWZ (No Gprot) AProteinChemokineCCR6Homo sapiensCCL20-3.342020-06-24doi.org/10.1038/s41467-020-16820-6
8TLMAProteinChemokineCCR8Homo sapiensAnti-murine CCR8 antibody--3.92023-12-20doi.org/10.1038/s41467-023-43601-8
8U1UAProteinChemokineCCR8Homo sapiensCCL1-Gi1/β1/γ23.12023-12-20doi.org/10.1038/s41467-023-43601-8
8U1U (No Gprot) AProteinChemokineCCR8Homo sapiensCCL1-3.12023-12-20doi.org/10.1038/s41467-023-43601-8
8KFXAProteinChemokineCCR8Homo sapiensLMD-009-Gi1/β1/γ22.962024-02-07doi.org/10.1126/sciadv.adj7500
8KFX (No Gprot) AProteinChemokineCCR8Homo sapiensLMD-009-2.962024-02-07doi.org/10.1126/sciadv.adj7500
8KFYAProteinChemokineCCR8Homo sapiensZK-756326-Gi1/β1/γ23.062024-02-07doi.org/10.1126/sciadv.adj7500
8KFY (No Gprot) AProteinChemokineCCR8Homo sapiensZK-756326-3.062024-02-07doi.org/10.1126/sciadv.adj7500
8KFZAProteinChemokineCCR8Homo sapiens--Gi1/β1/γ23.32024-02-07doi.org/10.1126/sciadv.adj7500
8KFZ (No Gprot) AProteinChemokineCCR8Homo sapiens--3.32024-02-07doi.org/10.1126/sciadv.adj7500
8XMLAProteinChemokineCCR8Homo sapiens--Gi1/β1/γ22.582025-01-01To be published
8XML (No Gprot) AProteinChemokineCCR8Homo sapiens--2.582025-01-01To be published
7XBWAProteinChemokineCX3CR1Homo sapiens--Gi1/β1/γ22.82022-07-13doi.org/10.1126/sciadv.abn8048
7XBW (No Gprot) AProteinChemokineCX3CR1Homo sapiens--2.82022-07-13doi.org/10.1126/sciadv.abn8048
7XBXAProteinChemokineCX3CR1Homo sapiensCX3CL1-Gi1/β1/γ23.42022-07-13doi.org/10.1126/sciadv.abn8048
7XBX (No Gprot) AProteinChemokineCX3CR1Homo sapiensCX3CL1-3.42022-07-13doi.org/10.1126/sciadv.abn8048
8IC0AProteinChemokineCXCR1Homo sapiensInterleukin-8-Gi1/β1/γ23.412023-07-19doi.org/10.1038/s41467-023-39799-2
8IC0 (No Gprot) AProteinChemokineCXCR1Homo sapiensInterleukin-8-3.412023-07-19doi.org/10.1038/s41467-023-39799-2
6LFMAProteinChemokineCXCR2Homo sapiensInterleukin-8-Gi1/β1/γ23.52020-09-02doi.org/10.1038/s41586-020-2492-5
6LFM (No Gprot) AProteinChemokineCXCR2Homo sapiensInterleukin-8-3.52020-09-02doi.org/10.1038/s41586-020-2492-5
6LFOAProteinChemokineCXCR2Homo sapiensInterleukin-8-Gi1/β1/γ23.42020-09-02doi.org/10.1038/s41586-020-2492-5
6LFO (No Gprot) AProteinChemokineCXCR2Homo sapiensInterleukin-8-3.42020-09-02doi.org/10.1038/s41586-020-2492-5
8XVUAProteinChemokineCXCR2Homo sapiensCXCL2--3.092025-01-15doi.org/10.1016/j.molcel.2025.01.024
8XWAAProteinChemokineCXCR2Homo sapiensCXCL1--3.482025-01-15doi.org/10.1016/j.molcel.2025.01.024
8XWFAProteinChemokineCXCR2Homo sapiensCXCL3--3.652025-01-15doi.org/10.1016/j.molcel.2025.01.024
8XWMAProteinChemokineCXCR2Homo sapiensCXCL6--3.712025-01-15doi.org/10.1016/j.molcel.2025.01.024
8XWNAProteinChemokineCXCR2Homo sapiensCXCL8--3.292025-01-15doi.org/10.1016/j.molcel.2025.01.024
8XWSAProteinChemokineCXCR2Homo sapiensCXCL5--3.062025-01-15doi.org/10.1016/j.molcel.2025.01.024
8XWVAProteinChemokineCXCR2Homo sapiensCXCL1-Go/β1/γ23.072025-01-15doi.org/10.1016/j.molcel.2025.01.024
8XWV (No Gprot) AProteinChemokineCXCR2Homo sapiensCXCL1-3.072025-01-15doi.org/10.1016/j.molcel.2025.01.024
8XX3AProteinChemokineCXCR2Homo sapiensCXCL3-Go/β1/γ23.382025-01-15doi.org/10.1016/j.molcel.2025.01.024
8XX3 (No Gprot) AProteinChemokineCXCR2Homo sapiensCXCL3-3.382025-01-15doi.org/10.1016/j.molcel.2025.01.024
8XX6AProteinChemokineCXCR2Homo sapiensCXCL8-Go/β1/γ22.992025-01-15doi.org/10.1016/j.molcel.2025.01.024
8XX6 (No Gprot) AProteinChemokineCXCR2Homo sapiensCXCL8-2.992025-01-15doi.org/10.1016/j.molcel.2025.01.024
8XX7AProteinChemokineCXCR2Homo sapiensCXCL5-Go/β1/γ23.322025-01-15doi.org/10.1016/j.molcel.2025.01.024
8XX7 (No Gprot) AProteinChemokineCXCR2Homo sapiensCXCL5-3.322025-01-15doi.org/10.1016/j.molcel.2025.01.024
8XXHAProteinChemokineCXCR2Homo sapiensCXCL2-Go/β1/γ22.82025-01-15doi.org/10.1016/j.molcel.2025.01.024
8XXH (No Gprot) AProteinChemokineCXCR2Homo sapiensCXCL2-2.82025-01-15doi.org/10.1016/j.molcel.2025.01.024
8XXRAProteinChemokineCXCR2Homo sapiens--Go/β1/γ23.172025-01-15doi.org/10.1016/j.molcel.2025.01.024
8XXR (No Gprot) AProteinChemokineCXCR2Homo sapiens--3.172025-01-15doi.org/10.1016/j.molcel.2025.01.024
8XXXAProteinChemokineCXCR2Homo sapiensCXCL6-Go/β1/γ23.172025-01-15doi.org/10.1016/j.molcel.2025.01.024
8XXX (No Gprot) AProteinChemokineCXCR2Homo sapiensCXCL6-3.172025-01-15doi.org/10.1016/j.molcel.2025.01.024
8HNKAProteinChemokineCXCR3Homo sapiensCXCL11-Gi1/β1/γ23.012023-11-29doi.org/10.1038/s41594-023-01175-5
8HNK (No Gprot) AProteinChemokineCXCR3Homo sapiensCXCL11-3.012023-11-29doi.org/10.1038/s41594-023-01175-5
8HNLAProteinChemokineCXCR3Homo sapiensPS372424-Gi1/β1/γ22.982023-11-29doi.org/10.1038/s41594-023-01175-5
8HNL (No Gprot) AProteinChemokineCXCR3Homo sapiensPS372424-2.982023-11-29doi.org/10.1038/s41594-023-01175-5
8HNMAProteinChemokineCXCR3Homo sapiensVUF11222-Gi1/β1/γ22.942023-11-29doi.org/10.1038/s41594-023-01175-5
8HNM (No Gprot) AProteinChemokineCXCR3Homo sapiensVUF11222-2.942023-11-29doi.org/10.1038/s41594-023-01175-5
8HNNAProteinChemokineCXCR3Homo sapiensSCH546738--3.62023-11-29doi.org/10.1038/s41594-023-01175-5
8K2WAProteinChemokineCXCR3Homo sapiensAMG487--32023-11-29doi.org/10.1038/s41594-023-01175-5
8K2XAProteinChemokineCXCR3Homo sapiensCXCL10-Gi1/β1/γ23.22023-11-29doi.org/10.1038/s41594-023-01175-5
8K2X (No Gprot) AProteinChemokineCXCR3Homo sapiensCXCL10-3.22023-11-29doi.org/10.1038/s41594-023-01175-5
8XXYAProteinChemokineCXCR3Homo sapiens---3.682025-02-26doi.org/10.1038/s41467-025-58264-w
8XXZAProteinChemokineCXCR3Homo sapiens--Go/β1/γ23.32025-02-26doi.org/10.1038/s41467-025-58264-w
8XXZ (No Gprot) AProteinChemokineCXCR3Homo sapiens--3.32025-02-26doi.org/10.1038/s41467-025-58264-w
8XYIAProteinChemokineCXCR3Homo sapiensVUF10661--3.162025-02-26doi.org/10.1038/s41467-025-58264-w
8XYKAProteinChemokineCXCR3Homo sapiensVUF10661-Go/β1/γ23.032025-02-26doi.org/10.1038/s41467-025-58264-w
8XYK (No Gprot) AProteinChemokineCXCR3Homo sapiensVUF10661-3.032025-02-26doi.org/10.1038/s41467-025-58264-w
8Y0HAProteinChemokineCXCR3Homo sapiensVUF11418--3.532025-02-26doi.org/10.1038/s41467-025-58264-w
8Y0NAProteinChemokineCXCR3Homo sapiensVUF11418-Go/β1/γ23.072025-02-26doi.org/10.1038/s41467-025-58264-w
8Y0N (No Gprot) AProteinChemokineCXCR3Homo sapiensVUF11418-3.072025-02-26doi.org/10.1038/s41467-025-58264-w
8YU7AProteinChemokineCXCR4Homo sapiens---3.012025-03-05doi.org/10.1016/j.celrep.2025.115255
8U4NAProteinChemokineCXCR4Homo sapiens--Gi1/β1/γ22.722024-03-13doi.org/10.1101/2024.02.09.579708
8U4N (No Gprot) AProteinChemokineCXCR4Homo sapiens--2.722024-03-13doi.org/10.1101/2024.02.09.579708
8U4OAProteinChemokineCXCR4Homo sapiensCXCL12-Gi1/β1/γ23.292024-03-13doi.org/10.1101/2024.02.09.579708
8U4O (No Gprot) AProteinChemokineCXCR4Homo sapiensCXCL12-3.292024-03-13doi.org/10.1101/2024.02.09.579708
8U4PAProteinChemokineCXCR4Homo sapiensAMD3100-Gi1/β1/γ23.152024-03-13doi.org/10.1101/2024.02.09.579708
8U4P (No Gprot) AProteinChemokineCXCR4Homo sapiensAMD3100-3.152024-03-13doi.org/10.1101/2024.02.09.579708
8U4QAProteinChemokineCXCR4Homo sapiensREGN7663-Fab-Gi1/β1/γ23.362024-03-13doi.org/10.1101/2024.02.09.579708
8U4Q (No Gprot) AProteinChemokineCXCR4Homo sapiensREGN7663-Fab-3.362024-03-13doi.org/10.1101/2024.02.09.579708
8U4RAProteinChemokineCXCR4Homo sapiensREGN7663-Fab--3.12024-03-13doi.org/10.1101/2024.02.09.579708
3ODUAProteinChemokineCXCR4Homo sapiensIT1t--2.52010-10-27doi.org/10.1126/science.1194396
3OE0AProteinChemokineCXCR4Homo sapiensCVX15--2.92010-10-27doi.org/10.1126/science.1194396
3OE6AProteinChemokineCXCR4Homo sapiensIT1t--3.22010-10-27doi.org/10.1126/science.1194396
3OE8AProteinChemokineCXCR4Homo sapiensIT1t--3.12010-10-27doi.org/10.1126/science.1194396
3OE9AProteinChemokineCXCR4Homo sapiensIT1t--3.12010-10-27doi.org/10.1126/science.1194396
4RWSAProteinChemokineCXCR4Homo sapiensvMIP-II--3.12015-02-11doi.org/10.1126/science.1261064
8K3ZAProteinChemokineCXCR4Homo sapiensCXCL12-Gi1/β1/γ12.812024-07-17doi.org/10.1016/j.celrep.2024.114578
8K3Z (No Gprot) AProteinChemokineCXCR4Homo sapiensCXCL12-2.812024-07-17doi.org/10.1016/j.celrep.2024.114578
8U4SAProteinChemokineCXCR4Homo sapiensREGN7663-Fab--3.352024-03-13doi.org/10.1038/s41594-024-01397-1
8U4TAProteinChemokineCXCR4Homo sapiensREGN7663-Fab--3.382024-03-13doi.org/10.1038/s41594-024-01397-1
8ZPLAProteinChemokineCXCR4Homo sapiensHF51116--3.012025-02-26doi.org/10.1073/pnas.2425795122
8ZPMAProteinChemokineCXCR4Homo sapiensAMD070--3.22025-02-26doi.org/10.1073/pnas.2425795122
8ZPNAProteinChemokineCXCR4Homo sapiensAMD3100--3.312025-02-26doi.org/10.1073/pnas.2425795122
9ASTAProteinChemokineXCR1Homo sapiensLymphotactin-Gi1/β1/γ23.072024-12-11doi.org/10.1073/pnas.2405732121
9AST (No Gprot) AProteinChemokineXCR1Homo sapiensLymphotactin-3.072024-12-11doi.org/10.1073/pnas.2405732121
7XOUAPeptideCholecystokininCCKAHomo sapiensCholecystokinin-8-Gs/β1/γ23.22022-07-20doi.org/10.1038/s41421-022-00420-3
7XOU (No Gprot) APeptideCholecystokininCCKAHomo sapiensCholecystokinin-8-3.22022-07-20doi.org/10.1038/s41421-022-00420-3
7XOVAPeptideCholecystokininCCKAHomo sapiensSR146131-Gs/β1/γ232022-07-20doi.org/10.1038/s41421-022-00420-3
7XOV (No Gprot) APeptideCholecystokininCCKAHomo sapiensSR146131-32022-07-20doi.org/10.1038/s41421-022-00420-3
7EZHAPeptideCholecystokininCCKAHomo sapiensCholecystokinin-8-Gi1/β1/γ23.22021-08-25doi.org/10.1038/s41589-021-00841-3
7EZH (No Gprot) APeptideCholecystokininCCKAHomo sapiensCholecystokinin-8-3.22021-08-25doi.org/10.1038/s41589-021-00841-3
7EZKAPeptideCholecystokininCCKAHomo sapiensCholecystokinin-8-chim(NtGi1-Gs)/β1/γ23.12021-08-25doi.org/10.1038/s41589-021-00841-3
7EZK (No Gprot) APeptideCholecystokininCCKAHomo sapiensCholecystokinin-8-3.12021-08-25doi.org/10.1038/s41589-021-00841-3
7EZMAPeptideCholecystokininCCKAHomo sapiensCholecystokinin-8-chim(NtGsL-Gq)/β1/γ22.92021-08-25doi.org/10.1038/s41589-021-00841-3
7EZM (No Gprot) APeptideCholecystokininCCKAHomo sapiensCholecystokinin-8-2.92021-08-25doi.org/10.1038/s41589-021-00841-3
7F8UAPeptideCholecystokininCCKAHomo sapiensLintitript--2.82021-10-13doi.org/10.1038/s41589-021-00866-8
7F8YAPeptideCholecystokininCCKAHomo sapiensDevazepide--2.52021-10-13doi.org/10.1038/s41589-021-00866-8
7F8XAPeptideCholecystokininCCKAHomo sapiensNN9056--32021-12-29doi.org/10.1038/s41589-021-00866-8
7MBXAPeptideCholecystokininCCKAHomo sapiensCholecystokinin-8-Gs/β1/γ11.952021-05-26doi.org/10.1371/journal.pbio.3001295
7MBX (No Gprot) APeptideCholecystokininCCKAHomo sapiensCholecystokinin-8-1.952021-05-26doi.org/10.1371/journal.pbio.3001295
7MBYAPeptideCholecystokininCCKAHomo sapiensCholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ22.442021-05-26doi.org/10.1371/journal.pbio.3001295
7MBY (No Gprot) APeptideCholecystokininCCKAHomo sapiensCholecystokinin-8-2.442021-05-26doi.org/10.1371/journal.pbio.3001295
9BKJAPeptideCholecystokininCCKAHomo sapiensCholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ22.592024-05-22doi.org/10.1371/journal.pbio.3002673
9BKJ (No Gprot) APeptideCholecystokininCCKAHomo sapiensCholecystokinin-8-2.592024-05-22doi.org/10.1371/journal.pbio.3002673
9BKKAPeptideCholecystokininCCKAHomo sapiensCholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ22.512024-05-22doi.org/10.1371/journal.pbio.3002673
9BKK (No Gprot) APeptideCholecystokininCCKAHomo sapiensCholecystokinin-8-2.512024-05-22doi.org/10.1371/journal.pbio.3002673
7XOWAPeptideCholecystokininCCKBHomo sapiensGastrin-chim(NtGi1-Gq)/β1/γ23.12022-07-20doi.org/10.1038/s41421-022-00420-3
7XOW (No Gprot) APeptideCholecystokininCCKBHomo sapiensGastrin-3.12022-07-20doi.org/10.1038/s41421-022-00420-3
8IA7APeptideCholecystokininCCKBHomo sapiensCholecystokinin-8-chim(NtGi1L-Gq)/β1/γ23.12023-12-06doi.org/10.1038/s41421-022-00420-3
8IA7 (No Gprot) APeptideCholecystokininCCKBHomo sapiensCholecystokinin-8-3.12023-12-06doi.org/10.1038/s41421-022-00420-3
7F8VAPeptideCholecystokininCCKBHomo sapiensGastrin-17-Gi2/β1/γ23.32021-10-13doi.org/10.1038/s41589-021-00866-8
7F8V (No Gprot) APeptideCholecystokininCCKBHomo sapiensGastrin-17-3.32021-10-13doi.org/10.1038/s41589-021-00866-8
7F8WAPeptideCholecystokininCCKBHomo sapiensGastrin-17-chim(NtGsL-Gq)/β1/γ23.12021-10-13doi.org/10.1038/s41589-021-00866-8
7F8W (No Gprot) APeptideCholecystokininCCKBHomo sapiensGastrin-17-3.12021-10-13doi.org/10.1038/s41589-021-00866-8
5O9HAPeptideComplement PeptideC5a1Homo sapiens-NDT9513727-2.72018-01-10doi.org/10.1038/nature25025
6C1QAPeptideComplement PeptideC5a1Homo sapiensPMX53NDT9513727-2.92018-05-30doi.org/10.1038/s41594-018-0067-z
6C1RAPeptideComplement PeptideC5a1Homo sapiensPMX53Avacopan; Na-2.22018-05-30doi.org/10.1038/s41594-018-0067-z
8I95APeptideComplement PeptideC3aBHomo sapiensEP54-Go/β1/γ22.882023-10-18doi.org/10.1016/j.cell.2023.09.020
8I95 (No Gprot) APeptideComplement PeptideC3aBHomo sapiensEP54-2.882023-10-18doi.org/10.1016/j.cell.2023.09.020
8I97APeptideComplement PeptideC3aBHomo sapiens--Go/β1/γ23.12023-10-18doi.org/10.1016/j.cell.2023.09.020
8I97 (No Gprot) APeptideComplement PeptideC3aBHomo sapiens--3.12023-10-18doi.org/10.1016/j.cell.2023.09.020
8I9AAPeptideComplement PeptideC3aBHomo sapiensEP54-chim(NtGi1-Gs-CtGq)/β1/γ23.572023-10-18doi.org/10.1016/j.cell.2023.09.020
8I9A (No Gprot) APeptideComplement PeptideC3aBHomo sapiensEP54-3.572023-10-18doi.org/10.1016/j.cell.2023.09.020
8I9LAPeptideComplement PeptideC3aBHomo sapiensC3a anaphylatoxin-Go/β1/γ23.182023-10-18doi.org/10.1016/j.cell.2023.09.020
8I9L (No Gprot) APeptideComplement PeptideC3aBHomo sapiensC3a anaphylatoxin-3.182023-10-18doi.org/10.1016/j.cell.2023.09.020
8I9SAPeptideComplement PeptideC3aBHomo sapiens--Go/β1/γ23.262023-10-18doi.org/10.1016/j.cell.2023.09.020
8I9S (No Gprot) APeptideComplement PeptideC3aBHomo sapiens--3.262023-10-18doi.org/10.1016/j.cell.2023.09.020
8J6DAPeptideComplement PeptideC3aBHomo sapiensEP141-Go/β1/γ23.12023-10-18doi.org/10.1016/j.cell.2023.09.020
8J6D (No Gprot) APeptideComplement PeptideC3aBHomo sapiensEP141-3.12023-10-18doi.org/10.1016/j.cell.2023.09.020
8HK2APeptideComplement PeptideC3aBHomo sapiensC3a anaphylatoxin-Gi1/β1/γ22.92023-05-10doi.org/10.1038/s41589-023-01339-w
8HK2 (No Gprot) APeptideComplement PeptideC3aBHomo sapiensC3a anaphylatoxin-2.92023-05-10doi.org/10.1038/s41589-023-01339-w
8HK3APeptideComplement PeptideC3aBHomo sapiens--Gi1/β1/γ23.22023-05-10doi.org/10.1038/s41589-023-01339-w
8HK3 (No Gprot) APeptideComplement PeptideC3aBHomo sapiens--3.22023-05-10doi.org/10.1038/s41589-023-01339-w
8ZWFAPeptideComplement PeptideC3aBHomo sapiensJR14a--32025-05-14doi.org/10.1038/s41421-024-00765-x
8ZWGAPeptideComplement PeptideC3aBHomo sapiensJR14a-Gi1/β1/γ22.872025-05-14doi.org/10.1038/s41421-024-00765-x
8ZWG (No Gprot) APeptideComplement PeptideC3aBHomo sapiensJR14a-2.872025-05-14doi.org/10.1038/s41421-024-00765-x
9IPVAPeptideComplement PeptideC3aBHomo sapiensJR14a-Gi1/β1/γ22.532025-04-23doi.org/10.1038/s44318-025-00429-w
9IPV (No Gprot) APeptideComplement PeptideC3aBHomo sapiensJR14a-2.532025-04-23doi.org/10.1038/s44318-025-00429-w
9IPYAPeptideComplement PeptideC3aBHomo sapiensJR14a--3.552025-04-23doi.org/10.1038/s44318-025-00429-w
9ISIAPeptideComplement PeptideC3aBHomo sapiens---3.562025-04-23doi.org/10.1038/s44318-025-00429-w
8IA8APeptideComplement PeptideC3aBHomo sapiensE7 peptide-Gi1/β1/γ22.862023-05-24To be published
8IA8 (No Gprot) APeptideComplement PeptideC3aBHomo sapiensE7 peptide-2.862023-05-24To be published
8HPTAPeptideComplement PeptideC5a1Mus musculusC5a anaphylatoxin C-terminal peptide-Go/β1/γ23.392023-10-18doi.org/10.1016/j.cell.2023.09.020
8HPT (No Gprot) APeptideComplement PeptideC5a1Mus musculusC5a anaphylatoxin C-terminal peptide-3.392023-10-18doi.org/10.1016/j.cell.2023.09.020
8HQCAPeptideComplement PeptideC5a1Mus musculusC5a anaphylatoxin-Go/β1/γ23.892023-10-18doi.org/10.1016/j.cell.2023.09.020
8HQC (No Gprot) APeptideComplement PeptideC5a1Mus musculusC5a anaphylatoxin-3.892023-10-18doi.org/10.1016/j.cell.2023.09.020
8IA2APeptideComplement PeptideC5a1Homo sapiensC5a anaphylatoxin-Go/β1/γ23.212023-10-18doi.org/10.1016/j.cell.2023.09.020
8IA2 (No Gprot) APeptideComplement PeptideC5a1Homo sapiensC5a anaphylatoxin-3.212023-10-18doi.org/10.1016/j.cell.2023.09.020
8JZZAPeptideComplement PeptideC5a1Homo sapiensC5a-desArg-Go/β1/γ23.312023-10-18doi.org/10.1016/j.cell.2023.09.020
8JZZ (No Gprot) APeptideComplement PeptideC5a1Homo sapiensC5a-desArg-3.312023-10-18doi.org/10.1016/j.cell.2023.09.020
7Y64APeptideComplement PeptideC5a1Homo sapiensC5a anaphylatoxin-Gi1/β1/γ22.92023-03-01doi.org/10.1038/s41422-023-00779-2
7Y64 (No Gprot) APeptideComplement PeptideC5a1Homo sapiensC5a anaphylatoxin-2.92023-03-01doi.org/10.1038/s41422-023-00779-2
7Y65APeptideComplement PeptideC5a1Homo sapiensC5a peptide-Gi1/β1/γ23.22023-03-01doi.org/10.1038/s41422-023-00779-2
7Y65 (No Gprot) APeptideComplement PeptideC5a1Homo sapiensC5a peptide-3.22023-03-01doi.org/10.1038/s41422-023-00779-2
7Y66APeptideComplement PeptideC5a1Homo sapiensBM213-Gi1/β1/γ22.92023-03-01doi.org/10.1038/s41422-023-00779-2
7Y66 (No Gprot) APeptideComplement PeptideC5a1Homo sapiensBM213-2.92023-03-01doi.org/10.1038/s41422-023-00779-2
7Y67APeptideComplement PeptideC5a1Homo sapiensC089 peptide-Gi1/β1/γ22.82023-03-01doi.org/10.1038/s41422-023-00779-2
7Y67 (No Gprot) APeptideComplement PeptideC5a1Homo sapiensC089 peptide-2.82023-03-01doi.org/10.1038/s41422-023-00779-2
8HK5APeptideComplement PeptideC5a1Homo sapiensComplement C5-Gi1/β1/γ232023-05-10doi.org/10.1038/s41589-023-01339-w
8HK5 (No Gprot) APeptideComplement PeptideC5a1Homo sapiensComplement C5-32023-05-10doi.org/10.1038/s41589-023-01339-w
8JZPAPeptideComplement PeptideC5a1Homo sapiensC5A anaphylatoxin-Go/β1/γ23.542025-01-15To be published
8JZP (No Gprot) APeptideComplement PeptideC5a1Homo sapiensC5A anaphylatoxin-3.542025-01-15To be published
4K5YB1PeptideCorticotropin Releasing FactorCRF1Homo sapiens-CP-376395-2.982013-07-17doi.org/10.1038/nature12357
4Z9GB1PeptideCorticotropin Releasing FactorCRF1Homo sapiens-CP-376395-3.182016-06-29doi.org/10.2174/1874467210666170110114727
8GTGB1PeptideCorticotropin Releasing FactorCRF1Homo sapiens-BMK-I152-2.752023-09-13doi.org/10.1038/s12276-023-01082-1
8GTIB1PeptideCorticotropin Releasing FactorCRF1Homo sapiens-BMK-C205-2.22023-09-13doi.org/10.1038/s12276-023-01082-1
8GTMB1PeptideCorticotropin Releasing FactorCRF1Homo sapiens-BMK-C203-2.62023-09-13doi.org/10.1038/s12276-023-01082-1
6P9XB1PeptideCorticotropin Releasing FactorCRF1Homo sapiensCorticoliberin-Gs/β1/γ22.912020-02-05doi.org/10.1016/j.molcel.2020.01.012
6P9X (No Gprot) B1PeptideCorticotropin Releasing FactorCRF1Homo sapiensCorticoliberin-2.912020-02-05doi.org/10.1016/j.molcel.2020.01.012
6PB0B1PeptideCorticotropin Releasing FactorCRF1Homo sapiensUrocortin-chim(NtGi1-Gs)/β1/γ232020-02-12doi.org/10.1016/j.molcel.2020.01.013
6PB0 (No Gprot) B1PeptideCorticotropin Releasing FactorCRF1Homo sapiensUrocortin-32020-02-12doi.org/10.1016/j.molcel.2020.01.013
6PB1B1PeptideCorticotropin Releasing FactorCRF2Homo sapiensUrocortin-chim(NtGi1-Gs)/β1/γ22.82020-02-12doi.org/10.1016/j.molcel.2020.01.013
6PB1 (No Gprot) B1PeptideCorticotropin Releasing FactorCRF2Homo sapiensUrocortin-2.82020-02-12doi.org/10.1016/j.molcel.2020.01.013
7TRYB1PeptideCorticotropin Releasing FactorCRF2Homo sapiensUrocortin-chim(NtGi1-G11)/β1/γ23.72022-11-09doi.org/10.1038/s41467-022-33851-3
7TRY (No Gprot) B1PeptideCorticotropin Releasing FactorCRF2Homo sapiensUrocortin-3.72022-11-09doi.org/10.1038/s41467-022-33851-3
7TS0B1PeptideCorticotropin Releasing FactorCRF2Homo sapiensUrocortin-chim(NtGi1L-Go)/β1/γ22.82022-11-09doi.org/10.1038/s41467-022-33851-3
7TS0 (No Gprot) B1PeptideCorticotropin Releasing FactorCRF2Homo sapiensUrocortin-2.82022-11-09doi.org/10.1038/s41467-022-33851-3
5WIVAAmineDopamineD4Homo sapiensNemonaprideNa-2.142017-10-18doi.org/10.1126/science.aan5468
7CKZAAmineDopamineD1Homo sapiensDopamineMevidalenGs/β1/γ23.12021-03-03doi.org/10.1016/j.cell.2021.01.028
7CKZ (No Gprot) AAmineDopamineD1Homo sapiensDopamineMevidalen3.12021-03-03doi.org/10.1016/j.cell.2021.01.028
7LJCAAmineDopamineD1Homo sapiensSKF-81297MevidalenGs/β1/γ232021-03-03doi.org/10.1038/s41422-021-00482-0
7LJC (No Gprot) AAmineDopamineD1Homo sapiensSKF-81297Mevidalen32021-03-03doi.org/10.1038/s41422-021-00482-0
7LJDAAmineDopamineD1Homo sapiensDopamineMevidalenGs/β1/γ13.22021-03-03doi.org/10.1038/s41422-021-00482-0
7LJD (No Gprot) AAmineDopamineD1Homo sapiensDopamineMevidalen3.22021-03-03doi.org/10.1038/s41422-021-00482-0
7X2FAAmineDopamineD1Homo sapiensDopamineMevidalenGs/β1/γ232022-06-15doi.org/10.1038/s41467-022-30929-w
7X2F (No Gprot) AAmineDopamineD1Homo sapiensDopamineMevidalen32022-06-15doi.org/10.1038/s41467-022-30929-w
7F1OAAmineDopamineD1Homo sapiensDopamineGDP; MgGs/β1/γ23.132022-06-15doi.org/10.1126/sciadv.abo4158
7F1O (No Gprot) AAmineDopamineD1Homo sapiensDopamineGDP; Mg3.132022-06-15doi.org/10.1126/sciadv.abo4158
7F1ZAAmineDopamineD1Homo sapiensDopamineGDPGs/β1/γ23.462022-06-15doi.org/10.1126/sciadv.abo4158
7F1Z (No Gprot) AAmineDopamineD1Homo sapiensDopamineGDP3.462022-06-15doi.org/10.1126/sciadv.abo4158
7F23AAmineDopamineD1Homo sapiensDopamineGDPGs/β1/γ23.582022-06-15doi.org/10.1126/sciadv.abo4158
7F23 (No Gprot) AAmineDopamineD1Homo sapiensDopamineGDP3.582022-06-15doi.org/10.1126/sciadv.abo4158
7F24AAmineDopamineD1Homo sapiensDopamineGDPGs/β1/γ24.162022-06-15doi.org/10.1126/sciadv.abo4158
7F24 (No Gprot) AAmineDopamineD1Homo sapiensDopamineGDP4.162022-06-15doi.org/10.1126/sciadv.abo4158
7X2CAAmineDopamineD1Homo sapiensFenoldopamFenoldopamGs/β1/γ23.22022-06-29doi.org/10.1038/s41467-022-30929-w
7X2C (No Gprot) AAmineDopamineD1Homo sapiensFenoldopamFenoldopam3.22022-06-29doi.org/10.1038/s41467-022-30929-w
7JV5AAmineDopamineD1Homo sapiensSKF81297-Gs/β1/γ232021-02-24doi.org/10.1016/j.cell.2021.01.027
7JV5 (No Gprot) AAmineDopamineD1Homo sapiensSKF81297-32021-02-24doi.org/10.1016/j.cell.2021.01.027
7JVPAAmineDopamineD1Homo sapiensSKF83959-Gs/β1/γ22.92021-02-24doi.org/10.1016/j.cell.2021.01.027
7JVP (No Gprot) AAmineDopamineD1Homo sapiensSKF83959-2.92021-02-24doi.org/10.1016/j.cell.2021.01.027
7JVQAAmineDopamineD1Homo sapiensApomorphine-Gs/β1/γ232021-02-24doi.org/10.1016/j.cell.2021.01.027
7JVQ (No Gprot) AAmineDopamineD1Homo sapiensApomorphine-32021-02-24doi.org/10.1016/j.cell.2021.01.027
7CKWAAmineDopamineD1Homo sapiensFenoldopam-Gs/β1/γ23.222021-03-03doi.org/10.1016/j.cell.2021.01.028
7CKW (No Gprot) AAmineDopamineD1Homo sapiensFenoldopam-3.222021-03-03doi.org/10.1016/j.cell.2021.01.028
7CKXAAmineDopamineD1Homo sapiensA77636-Gs/β1/γ23.542021-03-03doi.org/10.1016/j.cell.2021.01.028
7CKX (No Gprot) AAmineDopamineD1Homo sapiensA77636-3.542021-03-03doi.org/10.1016/j.cell.2021.01.028
7CKYAAmineDopamineD1Homo sapiensPW0464-Gs/β1/γ23.22021-03-03doi.org/10.1016/j.cell.2021.01.028
7CKY (No Gprot) AAmineDopamineD1Homo sapiensPW0464-3.22021-03-03doi.org/10.1016/j.cell.2021.01.028
7CRHAAmineDopamineD1Homo sapiensSKF83959-Gs/β1/γ23.32021-03-03doi.org/10.1016/j.cell.2021.01.028
7CRH (No Gprot) AAmineDopamineD1Homo sapiensSKF83959-3.32021-03-03doi.org/10.1016/j.cell.2021.01.028
8IRRAAmineDopamineD1Homo sapiensRotigotine-Gs/β1/γ23.22023-06-07doi.org/10.1038/s41422-023-00808-0
8IRR (No Gprot) AAmineDopamineD1Homo sapiensRotigotine-3.22023-06-07doi.org/10.1038/s41422-023-00808-0
7JOZAAmineDopamineD1Homo sapiensVFP-Gs/β1/γ23.82021-04-14doi.org/10.1038/s41467-021-23519-9
7JOZ (No Gprot) AAmineDopamineD1Homo sapiensVFP-3.82021-04-14doi.org/10.1038/s41467-021-23519-9
7X2DAAmineDopamineD1Homo sapiensTavapadon-Gs/β1/γ23.32022-06-15doi.org/10.1038/s41467-022-30929-w
7X2D (No Gprot) AAmineDopamineD1Homo sapiensTavapadon-3.32022-06-15doi.org/10.1038/s41467-022-30929-w
7F0TAAmineDopamineD1Homo sapiensDopamine-Gs/β1/γ23.12022-06-15doi.org/10.1126/sciadv.abo4158
7F0T (No Gprot) AAmineDopamineD1Homo sapiensDopamine-3.12022-06-15doi.org/10.1126/sciadv.abo4158
8JXRAAmineDopamineD1Homo sapiensLSD--3.572024-09-04doi.org/10.1016/j.neuron.2024.07.003
8JXSAAmineDopamineD1Homo sapiensPF-6142--32024-09-04doi.org/10.1016/j.neuron.2024.07.003
7JVRAAmineDopamineD2Homo sapiensBromoergocryptine-Gi1/β1/γ22.82021-02-24doi.org/10.1016/j.cell.2021.01.027
7JVR (No Gprot) AAmineDopamineD2Homo sapiensBromoergocryptine-2.82021-02-24doi.org/10.1016/j.cell.2021.01.027
6CM4AAmineDopamineD2Homo sapiensRisperidone--2.872018-03-14doi.org/10.1038/nature25758
8IRSAAmineDopamineD2Homo sapiensRotigotine-Gi1/β1/γ232023-06-07doi.org/10.1038/s41422-023-00808-0
8IRS (No Gprot) AAmineDopamineD2Homo sapiensRotigotine-32023-06-07doi.org/10.1038/s41422-023-00808-0
6LUQAAmineDopamineD2Homo sapiensHaloperidol--3.12020-03-04doi.org/10.1038/s41467-020-14884-y
7DFPAAmineDopamineD2Homo sapiensSpiperone--3.12020-12-30doi.org/10.1038/s41467-020-20221-0
6VMSAAmineDopamineD2Homo sapiensBromoergocryptine-Gi1/β1/γ23.82020-06-17doi.org/10.1038/s41586-020-2379-5
6VMS (No Gprot) AAmineDopamineD2Homo sapiensBromoergocryptine-3.82020-06-17doi.org/10.1038/s41586-020-2379-5
8TZQAAmineDopamineD2Homo sapiensL-Dopamine-Go/β1/γ23.22024-08-21doi.org/10.1038/s41467-024-50964-z
8TZQ (No Gprot) AAmineDopamineD2Homo sapiensL-Dopamine-3.22024-08-21doi.org/10.1038/s41467-024-50964-z
8U02AAmineDopamineD2Homo sapiensL-Dopamine-Go/β1/γ23.282024-08-21doi.org/10.1038/s41467-024-50964-z
8U02 (No Gprot) AAmineDopamineD2Homo sapiensL-Dopamine-3.282024-08-21doi.org/10.1038/s41467-024-50964-z
7CMUAAmineDopamineD3Homo sapiensPramipexole-Gi1/β1/γ232021-03-10doi.org/10.1016/j.molcel.2021.01.003
7CMU (No Gprot) AAmineDopamineD3Homo sapiensPramipexole-32021-03-10doi.org/10.1016/j.molcel.2021.01.003
7CMVAAmineDopamineD3Homo sapiensPD128907-Gi1/β1/γ22.72021-03-10doi.org/10.1016/j.molcel.2021.01.003
7CMV (No Gprot) AAmineDopamineD3Homo sapiensPD128907-2.72021-03-10doi.org/10.1016/j.molcel.2021.01.003
8IRTAAmineDopamineD3Homo sapiensRotigotine-Gi1/β1/γ22.72023-06-07doi.org/10.1038/s41422-023-00808-0
8IRT (No Gprot) AAmineDopamineD3Homo sapiensRotigotine-2.72023-06-07doi.org/10.1038/s41422-023-00808-0
9F33AAmineDopamineD3Homo sapiensFOB02-04A-Go/β1/γ23.052024-09-18doi.org/10.1038/s41467-024-51993-4
9F33 (No Gprot) AAmineDopamineD3Homo sapiensFOB02-04A-3.052024-09-18doi.org/10.1038/s41467-024-51993-4
9F34AAmineDopamineD3Homo sapiensFOB02-04A-Go/β1/γ23.052024-09-18doi.org/10.1038/s41467-024-51993-4
9F34 (No Gprot) AAmineDopamineD3Homo sapiensFOB02-04A-3.052024-09-18doi.org/10.1038/s41467-024-51993-4
3PBLAAmineDopamineD3Homo sapiensEticlopride--2.892010-11-03doi.org/10.1126/science.1197410
8IRUAAmineDopamineD4Homo sapiensRotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ23.22023-06-07doi.org/10.1038/s41422-023-00808-0
8IRU (No Gprot) AAmineDopamineD4Homo sapiensRotigotine-3.22023-06-07doi.org/10.1038/s41422-023-00808-0
5WIUAAmineDopamineD4Homo sapiensNemonapride--1.962017-10-18doi.org/10.1126/science.aan5468
6IQLAAmineDopamineD4Mus musculusL745870--3.52019-12-04doi.org/10.7554/eLife.48822
8IRVAAmineDopamineD5Homo sapiensRotigotine-chim(NtGi1-Gs)/β1/γ23.12023-06-07doi.org/10.1038/s41422-023-00808-0
8IRV (No Gprot) AAmineDopamineD5Homo sapiensRotigotine-3.12023-06-07doi.org/10.1038/s41422-023-00808-0
8HCQAPeptideEndothelinETAHomo sapiensEndothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ23.012023-03-22doi.org/10.1038/s41467-023-36998-9
8HCQ (No Gprot) APeptideEndothelinETAHomo sapiensEndothelin-1-3.012023-03-22doi.org/10.1038/s41467-023-36998-9
8XVIAPeptideEndothelinETAHomo sapiensEndothelin-1-chim(Gs-CtGq)/β1/γ23.322024-08-28doi.org/10.1038/s41421-024-00705-9
8XVI (No Gprot) APeptideEndothelinETAHomo sapiensEndothelin-1-3.322024-08-28doi.org/10.1038/s41421-024-00705-9
8XVJAPeptideEndothelinETAHomo sapiensMacitentan--3.262024-08-28doi.org/10.1038/s41421-024-00705-9
8XVKAPeptideEndothelinETAHomo sapiensAmbrisentan--3.212024-08-28doi.org/10.1038/s41421-024-00705-9
8XVLAPeptideEndothelinETAHomo sapiensZibotentan--3.222024-08-28doi.org/10.1038/s41421-024-00705-9
6LRYAPeptideEndothelinETBHomo sapiensSarafotoxin-B--32020-02-12doi.org/10.1016/j.bbrc.2019.12.091
5GLHAPeptideEndothelinETBHomo sapiensEndothelin-1--2.82016-09-07doi.org/10.1038/nature19319
5GLIAPeptideEndothelinETBHomo sapiens---2.52016-09-07doi.org/10.1038/nature19319
5X93APeptideEndothelinETBHomo sapiensK-8794--2.22017-08-16doi.org/10.1038/nsmb.3450
5XPRAPeptideEndothelinETBHomo sapiensBosentan--3.62017-08-16doi.org/10.1038/nsmb.3450
6IGKAPeptideEndothelinETBHomo sapiensEndothelin-3--22018-11-21doi.org/10.1038/s41467-018-07094-0
6IGLAPeptideEndothelinETBHomo sapiensIRL1620--2.72018-11-21doi.org/10.1038/s41467-018-07094-0
8HBDAPeptideEndothelinETBHomo sapiensIRL1620-Gi1/β1/γ22.992023-03-22doi.org/10.1038/s41467-023-36998-9
8HBD (No Gprot) APeptideEndothelinETBHomo sapiensIRL1620-2.992023-03-22doi.org/10.1038/s41467-023-36998-9
8HCXAPeptideEndothelinETBHomo sapiensEndothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ23.52023-03-22doi.org/10.1038/s41467-023-36998-9
8HCX (No Gprot) APeptideEndothelinETBHomo sapiensEndothelin-1-3.52023-03-22doi.org/10.1038/s41467-023-36998-9
6K1QAPeptideEndothelinETBHomo sapiensIRL2500--2.72019-07-17doi.org/10.1038/s42003-019-0482-7
8IY5APeptideEndothelinETBHomo sapiensEndothelin-1-Gi1/β1/γ22.82023-08-16doi.org/10.7554/eLife.85821
8IY5 (No Gprot) APeptideEndothelinETBHomo sapiensEndothelin-1-2.82023-08-16doi.org/10.7554/eLife.85821
8IY6APeptideEndothelinETBHomo sapiensEndothelin-1--3.132023-08-16doi.org/10.7554/eLife.85821
8XVEAPeptideEndothelinETBHomo sapiensBQ3020-chim(Gs-CtGq)/β1/γ232024-08-28doi.org/10.1038/s41421-024-00705-9
8XVE (No Gprot) APeptideEndothelinETBHomo sapiensBQ3020-32024-08-28doi.org/10.1038/s41421-024-00705-9
8XVHAPeptideEndothelinETBHomo sapiensEndothelin-1-chim(Gs-CtGq)/β1/γ23.262024-08-28doi.org/10.1038/s41421-024-00705-9
8XVH (No Gprot) APeptideEndothelinETBHomo sapiensEndothelin-1-3.262024-08-28doi.org/10.1038/s41421-024-00705-9
9KDFAPeptideEndothelinETBHomo sapiensRES-701-3--3.32025-05-07doi.org/10.1038/s41467-025-57960-x
9KDGAPeptideEndothelinETBHomo sapiens---3.332025-05-07doi.org/10.1038/s41467-025-57960-x
8XWPAPeptideEndothelinETBHomo sapiensEndothelin-1-Gi1/β1/γ23.212024-10-02doi.org/10.1038/s42003-024-06905-z
8XWP (No Gprot) APeptideEndothelinETBHomo sapiensEndothelin-1-3.212024-10-02doi.org/10.1038/s42003-024-06905-z
8XWQAPeptideEndothelinETBHomo sapiensEndothelin-1-Gi1/β1/γ24.62024-10-02doi.org/10.1038/s42003-024-06905-z
8XWQ (No Gprot) APeptideEndothelinETBHomo sapiensEndothelin-1-4.62024-10-02doi.org/10.1038/s42003-024-06905-z
8ZRTAPeptideEndothelinETBHomo sapiensET-1--3.622024-10-02doi.org/10.1038/s42003-024-06905-z
7T6TAPeptideFormylpeptideFPR1-ALXHomo sapiensfMLFII-Gi1/β1/γ23.22022-03-30doi.org/10.1038/s41467-022-28586-0
7T6T (No Gprot) APeptideFormylpeptideFPR1-ALXHomo sapiensfMLFII-3.22022-03-30doi.org/10.1038/s41467-022-28586-0
7WVUAPeptideFormylpeptideFPR1-ALXHomo sapiensfMLF-Gi1/β1/γ23.32022-04-13doi.org/10.1038/s41467-022-29361-x
7WVU (No Gprot) APeptideFormylpeptideFPR1-ALXHomo sapiensfMLF-3.32022-04-13doi.org/10.1038/s41467-022-29361-x
7EUOAPeptideFormylpeptideFPR1-ALXHomo sapiensfMLF-Gi1/β1/γ22.92022-05-25doi.org/10.1038/s41467-022-32822-y
7EUO (No Gprot) APeptideFormylpeptideFPR1-ALXHomo sapiensfMLF-2.92022-05-25doi.org/10.1038/s41467-022-32822-y
7VFXAPeptideFormylpeptideFPR1-ALXHomo sapiensfMLF-Gi1/β1/γ22.82022-09-21doi.org/10.1038/s41467-022-32822-y
7VFX (No Gprot) APeptideFormylpeptideFPR1-ALXHomo sapiensfMLF-2.82022-09-21doi.org/10.1038/s41467-022-32822-y
6OMMAPeptideFormylpeptideFPR2-ALXHomo sapiensWKYMVX-Gi1/β1/γ23.172020-02-26doi.org/10.1038/s41467-020-14728-9
6OMM (No Gprot) APeptideFormylpeptideFPR2-ALXHomo sapiensWKYMVX-3.172020-02-26doi.org/10.1038/s41467-020-14728-9
6LW5APeptideFormylpeptideFPR2-ALXHomo sapiensWKYMVm--2.82020-03-25doi.org/10.1038/s41467-020-15009-1
7T6SAPeptideFormylpeptideFPR2-ALXHomo sapiensPubChem 24776341-Gi1/β1/γ232022-03-30doi.org/10.1038/s41467-022-28586-0
7T6S (No Gprot) APeptideFormylpeptideFPR2-ALXHomo sapiensPubChem 24776341-32022-03-30doi.org/10.1038/s41467-022-28586-0
7T6UAPeptideFormylpeptideFPR2-ALXHomo sapiensCGEN-855A-Gi1/β1/γ22.92022-03-30doi.org/10.1038/s41467-022-28586-0
7T6U (No Gprot) APeptideFormylpeptideFPR2-ALXHomo sapiensCGEN-855A-2.92022-03-30doi.org/10.1038/s41467-022-28586-0
7T6VAPeptideFormylpeptideFPR2-ALXHomo sapiensfMLFII-Gi1/β1/γ23.12022-03-30doi.org/10.1038/s41467-022-28586-0
7T6V (No Gprot) APeptideFormylpeptideFPR2-ALXHomo sapiensfMLFII-3.12022-03-30doi.org/10.1038/s41467-022-28586-0
7WVVAPeptideFormylpeptideFPR2-ALXHomo sapiensfMLFII-Gi2/β1/γ22.92022-04-13doi.org/10.1038/s41467-022-29361-x
7WVV (No Gprot) APeptideFormylpeptideFPR2-ALXHomo sapiensfMLFII-2.92022-04-13doi.org/10.1038/s41467-022-29361-x
7WVWAPeptideFormylpeptideFPR2-ALXHomo sapiensfMYFINILTL-Gi2/β1/γ23.12022-04-13doi.org/10.1038/s41467-022-29361-x
7WVW (No Gprot) APeptideFormylpeptideFPR2-ALXHomo sapiensfMYFINILTL-3.12022-04-13doi.org/10.1038/s41467-022-29361-x
7WVXAPeptideFormylpeptideFPR2-ALXHomo sapiensHumanin-Gi2/β1/γ22.82022-04-13doi.org/10.1038/s41467-022-29361-x
7WVX (No Gprot) APeptideFormylpeptideFPR2-ALXHomo sapiensHumanin-2.82022-04-13doi.org/10.1038/s41467-022-29361-x
7WVYAPeptideFormylpeptideFPR2-ALXHomo sapiensAmyloid-β42-Gi2/β1/γ232022-04-13doi.org/10.1038/s41467-022-29361-x
7WVY (No Gprot) APeptideFormylpeptideFPR2-ALXHomo sapiensAmyloid-β42-32022-04-13doi.org/10.1038/s41467-022-29361-x
8Y62APeptideFormylpeptideFPR2-ALXHomo sapiensC16:0 Ceramide-Gi1/β1/γ23.22025-02-05doi.org/10.1126/science.ado4188
8Y62 (No Gprot) APeptideFormylpeptideFPR2-ALXHomo sapiensC16:0 Ceramide-3.22025-02-05doi.org/10.1126/science.ado4188
8Y63APeptideFormylpeptideFPR2-ALXHomo sapiensC20:0 Ceramide-Gi1/β1/γ23.22025-02-05doi.org/10.1126/science.ado4188
8Y63 (No Gprot) APeptideFormylpeptideFPR2-ALXHomo sapiensC20:0 Ceramide-3.22025-02-05doi.org/10.1126/science.ado4188
9JHJAPeptideFormylpeptideFPR2-ALXHomo sapiensC18:0 Ceramide-Gi1/β1/γ23.22025-03-19doi.org/10.1126/science.ado4188
9JHJ (No Gprot) APeptideFormylpeptideFPR2-ALXHomo sapiensC18:0 Ceramide-3.22025-03-19doi.org/10.1126/science.ado4188
5KW2ALipidFree Fatty AcidFFA1Homo sapiens-PubChem 133053953-2.762018-05-02doi.org/10.1038/s41467-017-01240-w
5TZYALipidFree Fatty AcidFFA1Homo sapiens-MK8666; AP8-3.222017-06-07doi.org/10.1038/nsmb.3417
5TZRALipidFree Fatty AcidFFA1Homo sapiens-MK8666-2.22017-06-07doi.org/10.1038/nsmb.3417
8IYSALipidFree Fatty AcidFFA4Homo sapiensTUG-891GDPchim(NtGi1L-Gq)/β1/γ22.952023-06-21doi.org/10.1038/s41422-023-00835-x
8IYS (No Gprot) ALipidFree Fatty AcidFFA4Homo sapiensTUG-891GDP2.952023-06-21doi.org/10.1038/s41422-023-00835-x
4PHUALipidFree Fatty AcidFFA1Homo sapiens-Fasiglifam-2.332014-07-16doi.org/10.1038/nature13494
9K1CALipidFree Fatty AcidFFA1Homo sapiens-DHAGi1/β1/γ23.22024-12-11doi.org/10.1016/j.celrep.2024.115024
9K1C (No Gprot) ALipidFree Fatty AcidFFA1Homo sapiens-DHA3.22024-12-11doi.org/10.1016/j.celrep.2024.115024
9CM3ALipidFree Fatty AcidFFA2Homo sapiensTUG-1375Compound 187chim(NtGi1L-Gs-CtGq)/β1/γ23.062025-06-25doi.org/10.1038/s41586-025-09186-6
9CM3 (No Gprot) ALipidFree Fatty AcidFFA2Homo sapiensTUG-1375Compound 1873.062025-06-25doi.org/10.1038/s41586-025-09186-6
9NS9ALipidFree Fatty AcidFFA2Homo sapiensTUG-1375Compound 187Gi1/β1/γ23.32025-06-25doi.org/10.1038/s41586-025-09186-6
9NS9 (No Gprot) ALipidFree Fatty AcidFFA2Homo sapiensTUG-1375Compound 1873.32025-06-25doi.org/10.1038/s41586-025-09186-6
9CM7ALipidFree Fatty AcidFFA2Homo sapiensTUG-1375AZ-1729Gi1/β1/γ23.292025-06-25doi.org/10.1038/s41586-025-09186-6
9CM7 (No Gprot) ALipidFree Fatty AcidFFA2Homo sapiensTUG-1375AZ-17293.292025-06-25doi.org/10.1038/s41586-025-09186-6
8J20ALipidFree Fatty AcidFFA3Homo sapiensValeric acidAR420626Gi1/β1/γ23.22024-01-24doi.org/10.1038/s41422-023-00914-z
8J20 (No Gprot) ALipidFree Fatty AcidFFA3Homo sapiensValeric acidAR4206263.22024-01-24doi.org/10.1038/s41422-023-00914-z
8Y6WALipidFree Fatty AcidFFA2Homo sapiensTUG-13754-CMTBGi1/β1/γ23.192025-04-02doi.org/10.1038/s41467-025-57983-4
8Y6W (No Gprot) ALipidFree Fatty AcidFFA2Homo sapiensTUG-13754-CMTB3.192025-04-02doi.org/10.1038/s41467-025-57983-4
9CLWALipidFree Fatty AcidFFA2Homo sapiensTUG-13754-CMTBchim(NtGi1L-Gs-CtGq)/β1/γ23.192025-06-25doi.org/10.1038/s41586-025-09186-6
9CLW (No Gprot) ALipidFree Fatty AcidFFA2Homo sapiensTUG-13754-CMTB3.192025-06-25doi.org/10.1038/s41586-025-09186-6
8EITALipidFree Fatty AcidFFA1Homo sapiensDoconexent-chim(NtGi1L-Gs-CtGq)/β1/γ22.82023-05-24doi.org/10.1073/pnas.2219569120
8EIT (No Gprot) ALipidFree Fatty AcidFFA1Homo sapiensDoconexent-2.82023-05-24doi.org/10.1073/pnas.2219569120
8EJCALipidFree Fatty AcidFFA1Homo sapiensTAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ232023-05-24doi.org/10.1073/pnas.2219569120
8EJC (No Gprot) ALipidFree Fatty AcidFFA1Homo sapiensTAK-875-32023-05-24doi.org/10.1073/pnas.2219569120
8EJKALipidFree Fatty AcidFFA1Homo sapiensTAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ23.42023-05-24doi.org/10.1073/pnas.2219569120
8EJK (No Gprot) ALipidFree Fatty AcidFFA1Homo sapiensTAK-875-3.42023-05-24doi.org/10.1073/pnas.2219569120
8T3VALipidFree Fatty AcidFFA1Homo sapiensDocosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ23.392024-01-24doi.org/10.1126/sciadv.adj2384
8T3V (No Gprot) ALipidFree Fatty AcidFFA1Homo sapiensDocosa-4,7,10,13,16,19-Hexaenoic acid-3.392024-01-24doi.org/10.1126/sciadv.adj2384
9K1DALipidFree Fatty AcidFFA2Homo sapiensButanoic acid-Gi1/β1/γ23.342024-12-11doi.org/10.1016/j.celrep.2024.115024
9K1D (No Gprot) ALipidFree Fatty AcidFFA2Homo sapiensButanoic acid-3.342024-12-11doi.org/10.1016/j.celrep.2024.115024
8J22ALipidFree Fatty AcidFFA2Homo sapiensTUG-1375-Gi1/β1/γ23.22024-01-24doi.org/10.1038/s41422-023-00914-z
8J22 (No Gprot) ALipidFree Fatty AcidFFA2Homo sapiensTUG-1375-3.22024-01-24doi.org/10.1038/s41422-023-00914-z
8J24ALipidFree Fatty AcidFFA2Homo sapiensAcetic acid-Gi1/β1/γ22.62024-01-24doi.org/10.1038/s41422-023-00914-z
8J24 (No Gprot) ALipidFree Fatty AcidFFA2Homo sapiensAcetic acid-2.62024-01-24doi.org/10.1038/s41422-023-00914-z
8T3SALipidFree Fatty AcidFFA2Homo sapiensButyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ23.072024-01-24doi.org/10.1126/sciadv.adj2384
8T3S (No Gprot) ALipidFree Fatty AcidFFA2Homo sapiensButyric acid-3.072024-01-24doi.org/10.1126/sciadv.adj2384
8Y6YALipidFree Fatty AcidFFA2Homo sapiensGLPG0974--3.362025-04-02doi.org/10.1038/s41467-025-57983-4
8J23ALipidFree Fatty AcidFFA2Homo sapiens--Gi1/β1/γ23.22024-04-17To be published
8J23 (No Gprot) ALipidFree Fatty AcidFFA2Homo sapiens--3.22024-04-17To be published
8J21ALipidFree Fatty AcidFFA3Homo sapiensButyric acid-Gi1/β1/γ23.32024-01-24doi.org/10.1038/s41422-023-00914-z
8J21 (No Gprot) ALipidFree Fatty AcidFFA3Homo sapiensButyric acid-3.32024-01-24doi.org/10.1038/s41422-023-00914-z
8H4IALipidFree Fatty AcidFFA4Homo sapiensDoconexent-chim(NtGi1-Gs)/β1/γ23.062023-06-21doi.org/10.1038/s41422-023-00835-x
8H4I (No Gprot) ALipidFree Fatty AcidFFA4Homo sapiensDoconexent-3.062023-06-21doi.org/10.1038/s41422-023-00835-x
8H4KALipidFree Fatty AcidFFA4Homo sapiensGW9508-chim(NtGi1-Gs-CtGq)/β1/γ23.12023-06-21doi.org/10.1038/s41422-023-00835-x
8H4K (No Gprot) ALipidFree Fatty AcidFFA4Homo sapiensGW9508-3.12023-06-21doi.org/10.1038/s41422-023-00835-x
8H4LALipidFree Fatty AcidFFA4Homo sapiensDoconexent-chim(NtGi1-Gs-CtGq)/β1/γ23.072023-06-21doi.org/10.1038/s41422-023-00835-x
8H4L (No Gprot) ALipidFree Fatty AcidFFA4Homo sapiensDoconexent-3.072023-06-21doi.org/10.1038/s41422-023-00835-x
8T3OALipidFree Fatty AcidFFA4Homo sapiensTUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ23.062024-01-17doi.org/10.1126/sciadv.adj2384
8T3O (No Gprot) ALipidFree Fatty AcidFFA4Homo sapiensTUG-891-3.062024-01-17doi.org/10.1126/sciadv.adj2384
8T3QALipidFree Fatty AcidFFA4Homo sapiensDocosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ23.142024-01-24doi.org/10.1126/sciadv.adj2384
8T3Q (No Gprot) ALipidFree Fatty AcidFFA4Homo sapiensDocosa-4,7,10,13,16,19-Hexaenoic acid-3.142024-01-24doi.org/10.1126/sciadv.adj2384
8G59ALipidFree Fatty AcidFFA4Homo sapiensTUG-891-chim(Gi1-CtGq)/β1/γ22.642023-03-08doi.org/10.1126/science.add6220
8G59 (No Gprot) ALipidFree Fatty AcidFFA4Homo sapiensTUG-891-2.642023-03-08doi.org/10.1126/science.add6220
8ID3ALipidFree Fatty AcidFFA4Homo sapiens9-Hydroxystearic acid-Gi1/β1/γ23.12023-03-15doi.org/10.1126/science.add6220
8ID3 (No Gprot) ALipidFree Fatty AcidFFA4Homo sapiens9-Hydroxystearic acid-3.12023-03-15doi.org/10.1126/science.add6220
8ID4ALipidFree Fatty AcidFFA4Homo sapiensLinoleic acid-Gi1/β1/γ23.12023-03-15doi.org/10.1126/science.add6220
8ID4 (No Gprot) ALipidFree Fatty AcidFFA4Homo sapiensLinoleic acid-3.12023-03-15doi.org/10.1126/science.add6220
8ID6ALipidFree Fatty AcidFFA4Homo sapiensOleic acid-Gi1/β1/γ22.82023-03-15doi.org/10.1126/science.add6220
8ID6 (No Gprot) ALipidFree Fatty AcidFFA4Homo sapiensOleic acid-2.82023-03-15doi.org/10.1126/science.add6220
8ID8ALipidFree Fatty AcidFFA4Homo sapiensTUG-891-Gi1/β1/γ232023-03-15doi.org/10.1126/science.add6220
8ID8 (No Gprot) ALipidFree Fatty AcidFFA4Homo sapiensTUG-891-32023-03-15doi.org/10.1126/science.add6220
8ID9ALipidFree Fatty AcidFFA4Homo sapiensEicosapentaenoic acid-Gi1/β1/γ232023-03-15doi.org/10.1126/science.add6220
8ID9 (No Gprot) ALipidFree Fatty AcidFFA4Homo sapiensEicosapentaenoic acid-32023-03-15doi.org/10.1126/science.add6220
4N4WFProteinFrizzledSMOHomo sapiens-SANT-1-2.82014-01-22doi.org/10.1038/ncomms5355
6D32FProteinFrizzledSMOXenopus laevisCyclopamineCyclopamine-3.752018-05-23doi.org/10.1016/j.cell.2018.04.029
6D35FProteinFrizzledSMOXenopus laevis-Cholesterol-3.92018-05-23doi.org/10.1016/j.cell.2018.04.029
5L7DFProteinFrizzledSMOHomo sapiens-Cholesterol-3.22016-07-20doi.org/10.1038/nature18934
6O3CFProteinFrizzledSMOMus musculusSAG21kCholesterol-2.82019-07-03doi.org/10.1038/s41586-019-1355-4
6XBJFProteinFrizzledSMOHomo sapiens-CholesterolGi1/β1/γ23.882020-09-30doi.org/10.1038/s41589-020-0646-2
6XBJ (No Gprot) FProteinFrizzledSMOHomo sapiens-Cholesterol3.882020-09-30doi.org/10.1038/s41589-020-0646-2
6XBKFProteinFrizzledSMOHomo sapiens-CholesterolGi1/β1/γ23.242020-09-30doi.org/10.1038/s41589-020-0646-2
6XBK (No Gprot) FProteinFrizzledSMOHomo sapiens-Cholesterol3.242020-09-30doi.org/10.1038/s41589-020-0646-2
6XBLFProteinFrizzledSMOHomo sapiensSAGCholesterolGi1/β1/γ23.962020-09-30doi.org/10.1038/s41589-020-0646-2
6XBL (No Gprot) FProteinFrizzledSMOHomo sapiensSAGCholesterol3.962020-09-30doi.org/10.1038/s41589-020-0646-2
7ZI0FProteinFrizzledSMOHomo sapiensSAGCholesterol-32022-06-15doi.org/10.1126/sciadv.abm5563
6XBMFProteinFrizzledSMOHomo sapiens-5LWEGi1/β1/γ23.142020-09-30doi.org/10.1038/s41589-020-0646-2
6XBM (No Gprot) FProteinFrizzledSMOHomo sapiens-5LWE3.142020-09-30doi.org/10.1038/s41589-020-0646-2
6OT0FProteinFrizzledSMOHomo sapiens-25(S)-EpoxycholesterolGi1/β1/γ23.842019-06-12doi.org/10.1038/s41586-019-1286-0
6OT0 (No Gprot) FProteinFrizzledSMOHomo sapiens-25(S)-Epoxycholesterol3.842019-06-12doi.org/10.1038/s41586-019-1286-0
8J9NFProteinFrizzledFZD1Homo sapiens--chim(Gs-CtGq)/β1/γ23.52024-01-17doi.org/10.1038/s41421-023-00627-y
8J9N (No Gprot) FProteinFrizzledFZD1Homo sapiens--3.52024-01-17doi.org/10.1038/s41421-023-00627-y
8J9OFProteinFrizzledFZD1Homo sapiens---3.42024-01-17doi.org/10.1038/s41421-023-00627-y
8JHCFProteinFrizzledFZD3Homo sapiens---3.32024-01-17doi.org/10.1038/s41421-023-00627-y
8JHIFProteinFrizzledFZD3Homo sapiens--chim(NtGsXLas-Gs)/β1/γ23.22024-01-17doi.org/10.1038/s41421-023-00627-y
8JHI (No Gprot) FProteinFrizzledFZD3Homo sapiens--3.22024-01-17doi.org/10.1038/s41421-023-00627-y
8QW4FProteinFrizzledFZD3Homo sapiens---2.92024-09-04doi.org/10.1038/s41467-024-51451-1
6BD4FProteinFrizzledFZD4Homo sapiens---2.42018-08-22doi.org/10.1038/s41586-018-0447-x
8WM9FProteinFrizzledFZD4Homo sapiens--DVL-23.532024-09-11doi.org/10.1038/s41467-024-52174-z
8WMAFProteinFrizzledFZD4Homo sapiens--DVL-23.472024-09-11doi.org/10.1038/s41467-024-52174-z
6WW2FProteinFrizzledFZD5Homo sapiens---3.72020-08-19doi.org/10.7554/eLife.58464
8JH7FProteinFrizzledFZD6Homo sapiens---3.22024-01-17doi.org/10.1038/s41421-023-00627-y
8JHBFProteinFrizzledFZD6Homo sapiens--chim(NtGsXLas-Gs)/β1/γ23.32024-01-17doi.org/10.1038/s41421-023-00627-y
8JHB (No Gprot) FProteinFrizzledFZD6Homo sapiens--3.32024-01-17doi.org/10.1038/s41421-023-00627-y
8YY8FProteinFrizzledFZD7Homo sapiens--Gs/β1/γ23.222024-04-24doi.org/10.1038/s41422-021-00525-6
8YY8 (No Gprot) FProteinFrizzledFZD7Homo sapiens--3.222024-04-24doi.org/10.1038/s41422-021-00525-6
9EPOFProteinFrizzledFZD7Homo sapiens---1.92024-10-02doi.org/10.1038/s41467-024-51664-4
9EW2FProteinFrizzledFZD7Homo sapiens--Gs/β1/γ23.22024-10-02doi.org/10.1038/s41467-024-51664-4
9EW2 (No Gprot) FProteinFrizzledFZD7Homo sapiens--3.22024-10-02doi.org/10.1038/s41467-024-51664-4
4JKVFProteinFrizzledSMOHomo sapiensTaladegib--2.452013-04-24doi.org/10.1038/nature12167
5L7IFProteinFrizzledSMOHomo sapiensVismodegib--3.32016-07-20doi.org/10.1038/nature18934
5V56FProteinFrizzledSMOHomo sapiensTC114--2.92017-05-24doi.org/10.1038/ncomms15383
5V57FProteinFrizzledSMOHomo sapiensTC114--32017-05-24doi.org/10.1038/ncomms15383
4O9RFProteinFrizzledSMOHomo sapiensCyclopamine--3.22014-03-05doi.org/10.1038/ncomms4309
4QIMFProteinFrizzledSMOHomo sapiensANTA XV--2.612014-07-23doi.org/10.1038/ncomms5355
4QINFProteinFrizzledSMOHomo sapiensSAG1.5--2.62014-07-23doi.org/10.1038/ncomms5355
8CXOFProteinFrizzledSMOMus musculus---3.72022-08-03doi.org/10.1038/s41467-022-32125-2
7CA3CAminoacidGABABGABAB1, GABAB2Homo sapiens-rac-BHFF-4.52020-11-11doi.org/10.1016/j.jmb.2020.09.023
7EB2CAminoacidGABABGABAB2; GABAB1Homo sapiensBaclofenrac-BHFFGi1/β1/γ23.52021-05-05doi.org/10.1038/s41586-021-03507-1
7EB2 (No Gprot) CAminoacidGABABGABAB2; GABAB1Homo sapiensBaclofenrac-BHFF3.52021-05-05doi.org/10.1038/s41586-021-03507-1
6WIVCAminoacidGABABGABAB1, GABAB2Homo sapiens-PubChem 52923113; PubChem 52924645-3.32020-07-01doi.org/10.1038/s41586-020-2452-0
6UO8CAminoacidGABABGABAB1, GABAB2Homo sapiensSKF97541GS39783-3.632020-06-10doi.org/10.1038/s41586-020-2408-4
7C7QCAminoacidGABABGABAB1, GABAB2Homo sapiensBaclofenBHFF-32020-07-01doi.org/10.1038/s41422-020-0350-5
6W2YCAminoacidGABABGABAB1; GABAB1Homo sapiensPubChem 5311042--3.22020-07-01doi.org/10.1038/s41586-020-2469-4
7CA5CAminoacidGABABGABAB1, GABAB2Homo sapiens---7.62020-11-11doi.org/10.1016/j.jmb.2020.09.023
7CUMCAminoacidGABABGABAB1, GABAB2Homo sapiensCGP54626--3.522020-11-11doi.org/10.1016/j.jmb.2020.09.023
7C7SCAminoacidGABABGABAB1, GABAB2Homo sapiensCGP54626--2.92020-07-01doi.org/10.1038/s41422-020-0350-5
6UO9CAminoacidGABABGABAB1, GABAB2Homo sapiensSKF97541--4.82020-06-10doi.org/10.1038/s41586-020-2408-4
6UOACAminoacidGABABGABAB1, GABAB2Homo sapiens---6.32020-06-10doi.org/10.1038/s41586-020-2408-4
6VJMCAminoacidGABABGABAB1, GABAB2Homo sapiens---3.972020-06-10doi.org/10.1038/s41586-020-2408-4
6W2XCAminoacidGABABGABAB1, GABAB2Homo sapiensPubChem 5311042--3.62020-07-01doi.org/10.1038/s41586-020-2469-4
7WQ3APeptideGalaninGAL1Homo sapiensGalanin-Gi1/β1/γ22.72022-04-20doi.org/10.1038/s41467-022-29072-3
7WQ3 (No Gprot) APeptideGalaninGAL1Homo sapiensGalanin-2.72022-04-20doi.org/10.1038/s41467-022-29072-3
7XJJAPeptideGalaninGAL1Homo sapiensGalanin-Go/β1/γ23.32023-05-03doi.org/10.1073/pnas.2121465119
7XJJ (No Gprot) APeptideGalaninGAL1Homo sapiensGalanin-3.32023-05-03doi.org/10.1073/pnas.2121465119
7WQ4APeptideGalaninGAL2Homo sapiensGalanin-chim(NtGi1-Gs-CtGq)/β1/γ22.62022-04-20doi.org/10.1038/s41467-022-29072-3
7WQ4 (No Gprot) APeptideGalaninGAL2Homo sapiensGalanin-2.62022-04-20doi.org/10.1038/s41467-022-29072-3
7XJKAPeptideGalaninGAL2Homo sapiensGalanin-chim(NtGi2L-Gs-CtGq)/β1/γ23.32022-06-29doi.org/10.1073/pnas.2121465119
7XJK (No Gprot) APeptideGalaninGAL2Homo sapiensGalanin-3.32022-06-29doi.org/10.1073/pnas.2121465119
7XJLAPeptideGalaninGAL2Homo sapiensSpexin-chim(NtGi2L-Gs-CtGq)/β1/γ23.52022-06-29doi.org/10.1073/pnas.2121465119
7XJL (No Gprot) APeptideGalaninGAL2Homo sapiensSpexin-3.52022-06-29doi.org/10.1073/pnas.2121465119
7XBDAPeptideGalaninGAL2Homo sapiensGalanin-chim(NtGi2L-Gs-CtGq)/β1/γ23.112022-07-13doi.org/10.1371/journal.pbio.3001714
7XBD (No Gprot) APeptideGalaninGAL2Homo sapiensGalanin-3.112022-07-13doi.org/10.1371/journal.pbio.3001714
6KO5APeptideGhrelinGhrelinHomo sapiensPubChem 57400002--3.32020-08-12doi.org/10.1038/s41467-020-17554-1
7F9YAPeptideGhrelinGhrelinHomo sapiensGhrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ22.92021-08-18doi.org/10.1038/s41467-021-25364-2
7F9Y (No Gprot) APeptideGhrelinGhrelinHomo sapiensGhrelin-28-2.92021-08-18doi.org/10.1038/s41467-021-25364-2
7F9ZAPeptideGhrelinGhrelinHomo sapiensGHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ23.22021-08-18doi.org/10.1038/s41467-021-25364-2
7F9Z (No Gprot) APeptideGhrelinGhrelinHomo sapiensGHRP-6-3.22021-08-18doi.org/10.1038/s41467-021-25364-2
7NA7APeptideGhrelinGhrelinHomo sapiensGhrelin-27-Gi1/β1/γ22.72021-12-15doi.org/10.1038/s41467-021-26735-5
7NA7 (No Gprot) APeptideGhrelinGhrelinHomo sapiensGhrelin-27-2.72021-12-15doi.org/10.1038/s41467-021-26735-5
7NA8APeptideGhrelinGhrelinHomo sapiensPubChem 178024-Gi1/β1/γ22.72021-12-15doi.org/10.1038/s41467-021-26735-5
7NA8 (No Gprot) APeptideGhrelinGhrelinHomo sapiensPubChem 178024-2.72021-12-15doi.org/10.1038/s41467-021-26735-5
7F83APeptideGhrelinGhrelinHomo sapiensPF-05190457--2.942022-01-19doi.org/10.1038/s41467-022-27975-9
7W2ZAPeptideGhrelinGhrelinHomo sapiensGhrelin-Go/β1/γ22.82022-01-19doi.org/10.1038/s41467-022-27975-9
7W2Z (No Gprot) APeptideGhrelinGhrelinHomo sapiensGhrelin-2.82022-01-19doi.org/10.1038/s41467-022-27975-9
8JSRAPeptideGhrelinGhrelinHomo sapiensAnamorelin-chim(NtGi1-Gs-CtGq)/β1/γ22.92025-01-22doi.org/10.1038/s41594-024-01481-6
8JSR (No Gprot) APeptideGhrelinGhrelinHomo sapiensAnamorelin-2.92025-01-22doi.org/10.1038/s41594-024-01481-6
9UY3APeptideGhrelinGhrelinHomo sapiensAnamorelin-chim(NtGi1-Gs-CtGq)/β1/γ22.522025-07-02doi.org/10.1038/s41401-025-01606-7
9UY3 (No Gprot) APeptideGhrelinGhrelinHomo sapiensAnamorelin-2.522025-07-02doi.org/10.1038/s41401-025-01606-7
9V2NAPeptideGhrelinGhrelinHomo sapiensMacimorelin-chim(NtGi1-Gs-CtGq)/β1/γ22.632025-07-02doi.org/10.1038/s41401-025-01606-7
9V2N (No Gprot) APeptideGhrelinGhrelinHomo sapiensMacimorelin-2.632025-07-02doi.org/10.1038/s41401-025-01606-7
6ORVB1PeptideGlucagonGLP-1Homo sapiens-TT-OAD2Gs/β1/γ232020-01-08doi.org/10.1038/s41586-019-1902-z
6ORV (No Gprot) B1PeptideGlucagonGLP-1Homo sapiens-TT-OAD232020-01-08doi.org/10.1038/s41586-019-1902-z
7E14B1PeptideGlucagonGLP-1Homo sapiensOrforglipronPubChem 156022738Gs/β1/γ22.92021-07-07doi.org/10.1038/s41467-021-24058-z
7E14 (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensOrforglipronPubChem 1560227382.92021-07-07doi.org/10.1038/s41467-021-24058-z
7DUQB1PeptideGlucagonGLP-1Homo sapiensGLP-1PubChem 156022738Gs/β1/γ22.52021-07-14doi.org/10.1038/s41467-021-24058-z
7DUQ (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensGLP-1PubChem 1560227382.52021-07-14doi.org/10.1038/s41467-021-24058-z
7DURB1PeptideGlucagonGLP-1Homo sapiens-PubChem 156022738Gs/β1/γ23.32021-08-11doi.org/10.1038/s41467-021-24058-z
7DUR (No Gprot) B1PeptideGlucagonGLP-1Homo sapiens-PubChem 1560227383.32021-08-11doi.org/10.1038/s41467-021-24058-z
7EVMB1PeptideGlucagonGLP-1Homo sapiens-PubChem 156022738Gs/β1/γ22.52021-08-11doi.org/10.1038/s41467-021-24058-z
7EVM (No Gprot) B1PeptideGlucagonGLP-1Homo sapiens-PubChem 1560227382.52021-08-11doi.org/10.1038/s41467-021-24058-z
5VEWB1PeptideGlucagonGLP-1Homo sapiens-PF-06372222-2.72017-05-24doi.org/10.1038/nature22378
6LN2B1PeptideGlucagonGLP-1Homo sapiens-PF-06372222-3.22020-03-18doi.org/10.1038/s41467-020-14934-5
6KJVB1PeptideGlucagonGLP-1Homo sapiens-PF-06372222-2.82019-11-13doi.org/10.1107/S2052252519013496
6KK1B1PeptideGlucagonGLP-1Homo sapiens-PF-06372222-2.82019-11-13doi.org/10.1107/S2052252519013496
6KK7B1PeptideGlucagonGLP-1Homo sapiens-PF-06372222-3.12019-11-13doi.org/10.1107/S2052252519013496
8WG8B1PeptideGlucagonGlucagonHomo sapiens-Peptidechim(NtGi1-Gs)/β1/γ22.712024-03-06doi.org/10.1038/s41421-024-00649-0
8WG8 (No Gprot) B1PeptideGlucagonGlucagonHomo sapiens-Peptide2.712024-03-06doi.org/10.1038/s41421-024-00649-0
5VEXB1PeptideGlucagonGLP-1Homo sapiens-NNC0640-32017-05-17doi.org/10.1038/nature22378
5XEZB1PeptideGlucagonGlucagonHomo sapiens-NNC0640-32017-05-24doi.org/10.1038/nature22363
5XF1B1PeptideGlucagonGlucagonHomo sapiens-NNC0640-3.192017-05-24doi.org/10.1038/nature22363
5EE7B1PeptideGlucagonGlucagonHomo sapiens-MK0893-2.52016-04-20doi.org/10.1038/nature17414
7RBTB1PeptideGlucagonGIPHomo sapiensTirzepatideLSN3556672chim(NtGi1-Gs)/β1/γ23.082022-04-13doi.org/10.1073/pnas.2116506119
7RBT (No Gprot) B1PeptideGlucagonGIPHomo sapiensTirzepatideLSN35566723.082022-04-13doi.org/10.1073/pnas.2116506119
9IVMB1PeptideGlucagonGLP-1Homo sapiensGLP-1 (Truncated)LSN3318839chim(NtGi1-Gs)/β2/γ23.222024-11-13doi.org/10.1016/j.apsb.2024.09.002
9IVM (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensGLP-1 (Truncated)LSN33188393.222024-11-13doi.org/10.1016/j.apsb.2024.09.002
6VCBB1PeptideGlucagonGLP-1Homo sapiensGLP-1LSN3160440Gs/β1/γ23.32020-07-22doi.org/10.1038/s41589-020-0589-7
6VCB (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensGLP-1LSN31604403.32020-07-22doi.org/10.1038/s41589-020-0589-7
7CZ5B1PeptideGlucagonGHRHHomo sapiensSomatoliberin-Gs/β1/γ22.62020-11-18doi.org/10.1038/s41467-020-18945-0
7CZ5 (No Gprot) B1PeptideGlucagonGHRHHomo sapiensSomatoliberin-2.62020-11-18doi.org/10.1038/s41467-020-18945-0
7V9MB1PeptideGlucagonGHRH (SV1)Homo sapiensSomatoliberin-Gs/β1/γ23.292021-10-20doi.org/10.1073/pnas.2106606118
7V9M (No Gprot) B1PeptideGlucagonGHRH (SV1)Homo sapiensSomatoliberin-3.292021-10-20doi.org/10.1073/pnas.2106606118
7V9LB1PeptideGlucagonGHRH (SV1)Homo sapiens--chim(NtGi1-Gs)/β1/γ22.62022-04-06doi.org/10.1073/pnas.2106606118
7V9L (No Gprot) B1PeptideGlucagonGHRH (SV1)Homo sapiens--2.62022-04-06doi.org/10.1073/pnas.2106606118
8WA3B1PeptideGlucagonGIPHomo sapiens--Gs/β1/γ22.862024-03-06doi.org/10.1038/s41421-024-00649-0
8WA3 (No Gprot) B1PeptideGlucagonGIPHomo sapiens--2.862024-03-06doi.org/10.1038/s41421-024-00649-0
7FINB1PeptideGlucagonGIPHomo sapiensPeptide-20; GGL-Gs/β1/γ23.12022-02-23doi.org/10.1038/s41467-022-28683-0
7FIN (No Gprot) B1PeptideGlucagonGIPHomo sapiensPeptide-20; GGL-3.12022-02-23doi.org/10.1038/s41467-022-28683-0
7FIYB1PeptideGlucagonGIPHomo sapiensTirzepatide-Gs/β1/γ23.42022-03-02doi.org/10.1038/s41467-022-28683-0
7FIY (No Gprot) B1PeptideGlucagonGIPHomo sapiensTirzepatide-3.42022-03-02doi.org/10.1038/s41467-022-28683-0
7VABB1PeptideGlucagonGIPHomo sapiensNon-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ23.22022-03-02doi.org/10.1038/s41467-022-28683-0
7VAB (No Gprot) B1PeptideGlucagonGIPHomo sapiensNon-Acylated Tirzepatide-3.22022-03-02doi.org/10.1038/s41467-022-28683-0
7RA3B1PeptideGlucagonGIPHomo sapiensGIP-chim(NtGi1-Gs)/β1/γ23.242022-04-13doi.org/10.1073/pnas.2116506119
7RA3 (No Gprot) B1PeptideGlucagonGIPHomo sapiensGIP-3.242022-04-13doi.org/10.1073/pnas.2116506119
8ITLB1PeptideGlucagonGIPHomo sapiens--Gs/β1/γ23.232023-10-18doi.org/10.1073/pnas.2306145120
8ITL (No Gprot) B1PeptideGlucagonGIPHomo sapiens--3.232023-10-18doi.org/10.1073/pnas.2306145120
8ITMB1PeptideGlucagonGIPHomo sapiens--Gs/β1/γ23.132023-10-18doi.org/10.1073/pnas.2306145120
8ITM (No Gprot) B1PeptideGlucagonGIPHomo sapiens--3.132023-10-18doi.org/10.1073/pnas.2306145120
7DTYB1PeptideGlucagonGIPHomo sapiensGIP-Gs/β1/γ22.982021-08-04doi.org/10.7554/eLife.68719
7DTY (No Gprot) B1PeptideGlucagonGIPHomo sapiensGIP-2.982021-08-04doi.org/10.7554/eLife.68719
8YW4B1PeptideGlucagonGIPHomo sapiensRetatrutide-chim(NtGi1-Gs)/β1/γ23.262024-09-18doi.org/10.1038/s41421-024-00700-0
8YW4 (No Gprot) B1PeptideGlucagonGIPHomo sapiensRetatrutide-3.262024-09-18doi.org/10.1038/s41421-024-00700-0
9IVGB1PeptideGlucagonGLP-1Homo sapiensGLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ232024-11-27doi.org/10.1016/j.apsb.2024.09.002
9IVG (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensGLP-1 (Truncated)-32024-11-27doi.org/10.1016/j.apsb.2024.09.002
7RTBB1PeptideGlucagonGLP-1Homo sapiensPeptide-19-Gs/β1/γ22.142021-10-06doi.org/10.1016/j.bbrc.2021.09.016
7RTB (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensPeptide-19-2.142021-10-06doi.org/10.1016/j.bbrc.2021.09.016
7KI0B1PeptideGlucagonGLP-1Homo sapiensSemaglutide-Gs/β1/γ22.52021-08-04doi.org/10.1016/j.celrep.2021.109374
7KI0 (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensSemaglutide-2.52021-08-04doi.org/10.1016/j.celrep.2021.109374
7KI1B1PeptideGlucagonGLP-1Homo sapiensTaspoglutide-Gs/β1/γ22.52021-08-04doi.org/10.1016/j.celrep.2021.109374
7KI1 (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensTaspoglutide-2.52021-08-04doi.org/10.1016/j.celrep.2021.109374
6X18B1PeptideGlucagonGLP-1Homo sapiensGLP-1-Gs/β1/γ22.12020-09-09doi.org/10.1016/j.molcel.2020.09.020
6X18 (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensGLP-1-2.12020-09-09doi.org/10.1016/j.molcel.2020.09.020
6X19B1PeptideGlucagonGLP-1Homo sapiensCHU-128-Gs/β1/γ22.12020-09-09doi.org/10.1016/j.molcel.2020.09.020
6X19 (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensCHU-128-2.12020-09-09doi.org/10.1016/j.molcel.2020.09.020
6X1AB1PeptideGlucagonGLP-1Homo sapiensDanuglipron-Gs/β1/γ22.52020-09-09doi.org/10.1016/j.molcel.2020.09.020
6X1A (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensDanuglipron-2.52020-09-09doi.org/10.1016/j.molcel.2020.09.020
7LCIB1PeptideGlucagonGLP-1Homo sapiensDanuglipron-Gs/β1/γ22.92021-01-20doi.org/10.1016/j.str.2021.04.008
7LCI (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensDanuglipron-2.92021-01-20doi.org/10.1016/j.str.2021.04.008
7LCJB1PeptideGlucagonGLP-1Homo sapiensDanuglipron--2.822021-01-20doi.org/10.1016/j.str.2021.04.008
7LCKB1PeptideGlucagonGLP-1Homo sapiensDanuglipron--3.242021-01-20doi.org/10.1016/j.str.2021.04.008
7S15B1PeptideGlucagonGLP-1Homo sapiensPubChem 134611223--3.82022-06-08doi.org/10.1021/acs.jmedchem.1c01856
9J1PB1PeptideGlucagonGLP-1Homo sapiensg1:Ox-chim(NtGi1-Gs)/β1/γ22.992025-02-26doi.org/10.1021/jacs.4c12808
9J1P (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensg1:Ox-2.992025-02-26doi.org/10.1021/jacs.4c12808
5VAIB1PeptideGlucagonGLP-1Oryctolagus cuniculusGLP-1-Gs/β1/γ24.12017-05-24doi.org/10.1038/nature22394
5VAI (No Gprot) B1PeptideGlucagonGLP-1Oryctolagus cuniculusGLP-1-4.12017-05-24doi.org/10.1038/nature22394
5NX2B1PeptideGlucagonGLP-1Homo sapiensGLP-1 (Truncated)--3.72017-06-14doi.org/10.1038/nature22800
6B3JB1PeptideGlucagonGLP-1Homo sapiensExendin-P5-Gs/β1/γ23.32018-02-21doi.org/10.1038/nature25773
6B3J (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensExendin-P5-3.32018-02-21doi.org/10.1038/nature25773
8WG7B1PeptideGlucagonGLP-1Homo sapiens--Gs/β1/γ22.542024-03-06doi.org/10.1038/s41421-024-00649-0
8WG7 (No Gprot) B1PeptideGlucagonGLP-1Homo sapiens--2.542024-03-06doi.org/10.1038/s41421-024-00649-0
7C2EB1PeptideGlucagonGLP-1Homo sapiensPubChem 149050799-Gs/β1/γ24.22020-08-26doi.org/10.1038/s41422-020-0384-8
7C2E (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensPubChem 149050799-4.22020-08-26doi.org/10.1038/s41422-020-0384-8
7LLLB1PeptideGlucagonGLP-1Homo sapiensExendin-4-Gs/β1/γ23.72022-01-12doi.org/10.1038/s41467-021-27760-0
7LLL (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensExendin-4-3.72022-01-12doi.org/10.1038/s41467-021-27760-0
7LLYB1PeptideGlucagonGLP-1Homo sapiensOxyntomodulin-Gs/β1/γ23.32022-01-12doi.org/10.1038/s41467-021-27760-0
7LLY (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensOxyntomodulin-3.32022-01-12doi.org/10.1038/s41467-021-27760-0
7FIMB1PeptideGlucagonGLP-1Homo sapiensTirzepatide-Gs/β1/γ23.42022-03-02doi.org/10.1038/s41467-022-28683-0
7FIM (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensTirzepatide-3.42022-03-02doi.org/10.1038/s41467-022-28683-0
7VBIB1PeptideGlucagonGLP-1Homo sapiensNon-Acylated Tirzepatide-Gs/β1/γ232022-03-02doi.org/10.1038/s41467-022-28683-0
7VBI (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensNon-Acylated Tirzepatide-32022-03-02doi.org/10.1038/s41467-022-28683-0
7VBHB1PeptideGlucagonGLP-1Homo sapiensPeptide-20-Gs/β1/γ232022-04-06doi.org/10.1038/s41467-022-28683-0
7VBH (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensPeptide-20-32022-04-06doi.org/10.1038/s41467-022-28683-0
7S1MB1PeptideGlucagonGLP-1Homo sapiensEx4-D-Ala-Gs/β1/γ22.412022-01-05doi.org/10.1038/s41589-021-00945-w
7S1M (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensEx4-D-Ala-2.412022-01-05doi.org/10.1038/s41589-021-00945-w
7S3IB1PeptideGlucagonGLP-1Homo sapiens--Gs/β1/γ22.512022-01-05doi.org/10.1038/s41589-021-00945-w
7S3I (No Gprot) B1PeptideGlucagonGLP-1Homo sapiens--2.512022-01-05doi.org/10.1038/s41589-021-00945-w
6XOXB1PeptideGlucagonGLP-1Homo sapiensOrforglipron-chim(NtGi1-Gs)/β1/γ23.12020-11-18doi.org/10.1073/pnas.2014879117
6XOX (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensOrforglipron-3.12020-11-18doi.org/10.1073/pnas.2014879117
7RG9B1PeptideGlucagonGLP-1Homo sapiens--chim(NtGi1-Gs)/β1/γ23.22022-04-13doi.org/10.1073/pnas.2116506119
7RG9 (No Gprot) B1PeptideGlucagonGLP-1Homo sapiens--3.22022-04-13doi.org/10.1073/pnas.2116506119
7RGPB1PeptideGlucagonGLP-1Homo sapiensTirzepatide-chim(NtGi1-Gs)/β1/γ22.92022-04-13doi.org/10.1073/pnas.2116506119
7RGP (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensTirzepatide-2.92022-04-13doi.org/10.1073/pnas.2116506119
7X8RB1PeptideGlucagonGLP-1Homo sapiensBOC5-Gs/β1/γ22.612022-06-29doi.org/10.1073/pnas.2200155119
7X8R (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensBOC5-2.612022-06-29doi.org/10.1073/pnas.2200155119
7X8SB1PeptideGlucagonGLP-1Homo sapiensWB4-24-Gs/β1/γ23.092022-06-29doi.org/10.1073/pnas.2200155119
7X8S (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensWB4-24-3.092022-06-29doi.org/10.1073/pnas.2200155119
8JIPB1PeptideGlucagonGLP-1Homo sapiensMEDI0382-chim(NtGi1-Gs)/β1/γ22.852023-09-06doi.org/10.1073/pnas.2303696120
8JIP (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensMEDI0382-2.852023-09-06doi.org/10.1073/pnas.2303696120
8JIRB1PeptideGlucagonGLP-1Homo sapiensSAR425899-chim(NtGi1-Gs)/β1/γ22.572023-09-06doi.org/10.1073/pnas.2303696120
8JIR (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensSAR425899-2.572023-09-06doi.org/10.1073/pnas.2303696120
8JISB1PeptideGlucagonGLP-1Homo sapiensPeptide-15-chim(NtGi1-Gs)/β1/γ22.462023-11-08doi.org/10.1073/pnas.2303696120
8JIS (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensPeptide-15-2.462023-11-08doi.org/10.1073/pnas.2303696120
8YW3B1PeptideGlucagonGLP-1Homo sapiensRetatrutide-Gs/β1/γ22.682024-09-18doi.org/10.1038/s41421-024-00700-0
8YW3 (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensRetatrutide-2.682024-09-18doi.org/10.1038/s41421-024-00700-0
9EBNB1PeptideGlucagonGLP-1Homo sapiens--Gs/β1/γ23.442025-03-26doi.org/10.1073/pnas.2407574122
9EBN (No Gprot) B1PeptideGlucagonGLP-1Homo sapiens--3.442025-03-26doi.org/10.1073/pnas.2407574122
9EBOB1PeptideGlucagonGLP-1Homo sapiensGLP-1 (ACPC18)-Gs/β1/γ23.132025-03-26doi.org/10.1073/pnas.2407574122
9EBO (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensGLP-1 (ACPC18)-3.132025-03-26doi.org/10.1073/pnas.2407574122
9EBQB1PeptideGlucagonGLP-1Homo sapiens--Gs/β1/γ23.162025-03-26doi.org/10.1073/pnas.2407574122
9EBQ (No Gprot) B1PeptideGlucagonGLP-1Homo sapiens--3.162025-03-26doi.org/10.1073/pnas.2407574122
8YWFB1PeptideGlucagonGLP-1Homo sapiensRetatrutide-chim(NtGi1-Gs)/β1/γ22.742025-04-16To be published
8YWF (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensRetatrutide-2.742025-04-16To be published
9BYOB1PeptideGlucagonGLP-1Homo sapiensExendin-3-Gs/β1/γ22.312025-06-11To be published
9BYO (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensExendin-3-2.312025-06-11To be published
9C0KB1PeptideGlucagonGLP-1Homo sapiensExendin-4-Gs/β1/γ22.722025-06-11To be published
9C0K (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensExendin-4-2.722025-06-11To be published
7D68B1PeptideGlucagonGLP-2Homo sapiensGLP-2-Gs/β1/γ232020-12-16doi.org/10.1038/s41422-020-00442-0
7D68 (No Gprot) B1PeptideGlucagonGLP-2Homo sapiensGLP-2-32020-12-16doi.org/10.1038/s41422-020-00442-0
8FU6B1PeptideGlucagonGlucagonHomo sapiensGlucagon derivative ZP3780-Gs/β1/γ22.92023-04-12doi.org/10.1016/j.cell.2023.02.028
8FU6 (No Gprot) B1PeptideGlucagonGlucagonHomo sapiensGlucagon derivative ZP3780-2.92023-04-12doi.org/10.1016/j.cell.2023.02.028
4L6RB1PeptideGlucagonGlucagonHomo sapiens---3.32013-07-24doi.org/10.1038/nature12393
5YQZB1PeptideGlucagonGlucagonHomo sapiensGlucagon analogue--32018-01-17doi.org/10.1038/nature25153
7V35B1PeptideGlucagonGlucagonHomo sapiensPeptide-20-Gs/β1/γ23.52022-03-02doi.org/10.1038/s41467-022-28683-0
7V35 (No Gprot) B1PeptideGlucagonGlucagonHomo sapiensPeptide-20-3.52022-03-02doi.org/10.1038/s41467-022-28683-0
8JRUB1PeptideGlucagonGlucagonHomo sapiens--Arrestin23.52023-08-16doi.org/10.1038/s41586-023-06420-x
8JRVB1PeptideGlucagonGlucagonHomo sapiensGlucagon-Arrestin23.32023-08-16doi.org/10.1038/s41586-023-06420-x
8JITB1PeptideGlucagonGlucagonHomo sapiensMEDI0382-Gs/β1/γ22.912023-09-06doi.org/10.1073/pnas.2303696120
8JIT (No Gprot) B1PeptideGlucagonGlucagonHomo sapiensMEDI0382-2.912023-09-06doi.org/10.1073/pnas.2303696120
8JIQB1PeptideGlucagonGlucagonHomo sapiensPeptide-15-Gs/β1/γ23.42023-09-13doi.org/10.1073/pnas.2303696120
8JIQ (No Gprot) B1PeptideGlucagonGlucagonHomo sapiensPeptide-15-3.42023-09-13doi.org/10.1073/pnas.2303696120
8JIUB1PeptideGlucagonGlucagonHomo sapiensSAR425899-Gs/β1/γ22.762023-09-13doi.org/10.1073/pnas.2303696120
8JIU (No Gprot) B1PeptideGlucagonGlucagonHomo sapiensSAR425899-2.762023-09-13doi.org/10.1073/pnas.2303696120
6WHCB1PeptideGlucagonGlucagonHomo sapiensGlu16 analog of GCG-Gs/β1/γ23.42020-05-27doi.org/10.1074/jbc.RA120.013793
6WHC (No Gprot) B1PeptideGlucagonGlucagonHomo sapiensGlu16 analog of GCG-3.42020-05-27doi.org/10.1074/jbc.RA120.013793
6LMKB1PeptideGlucagonGlucagonHomo sapiensGlucagon-Gs/β1/γ23.72020-04-01doi.org/10.1126/science.aaz5346
6LMK (No Gprot) B1PeptideGlucagonGlucagonHomo sapiensGlucagon-3.72020-04-01doi.org/10.1126/science.aaz5346
6LMLB1PeptideGlucagonGlucagonHomo sapiensGlucagon-Gi1/β1/γ13.92020-04-01doi.org/10.1126/science.aaz5346
6LML (No Gprot) B1PeptideGlucagonGlucagonHomo sapiensGlucagon-3.92020-04-01doi.org/10.1126/science.aaz5346
6WPWB1PeptideGlucagonGlucagonHomo sapiensGlucagon derivative ZP3780-Gs/β1/γ23.12020-08-12doi.org/10.1126/science.aba3373
6WPW (No Gprot) B1PeptideGlucagonGlucagonHomo sapiensGlucagon derivative ZP3780-3.12020-08-12doi.org/10.1126/science.aba3373
8YW5B1PeptideGlucagonGlucagonHomo sapiensRetatrutide-Gs/β1/γ22.842024-09-18doi.org/10.1038/s41421-024-00700-0
8YW5 (No Gprot) B1PeptideGlucagonGlucagonHomo sapiensRetatrutide-2.842024-09-18doi.org/10.1038/s41421-024-00700-0
7D3SB1PeptideGlucagonSecretinHomo sapiensSecretin-Gs/β1/γ22.92020-11-04doi.org/10.1016/j.bbrc.2020.08.042
7D3S (No Gprot) B1PeptideGlucagonSecretinHomo sapiensSecretin-2.92020-11-04doi.org/10.1016/j.bbrc.2020.08.042
6WI9B1PeptideGlucagonSecretinHomo sapiensSecretin-Gs/β1/γ24.32020-08-12doi.org/10.1038/s41467-020-17791-4
6WI9 (No Gprot) B1PeptideGlucagonSecretinHomo sapiensSecretin-4.32020-08-12doi.org/10.1038/s41467-020-17791-4
6WZGB1PeptideGlucagonSecretinHomo sapiensSecretin-Gs/β1/γ22.32020-08-12doi.org/10.1038/s41467-020-17791-4
6WZG (No Gprot) B1PeptideGlucagonSecretinHomo sapiensSecretin-2.32020-08-12doi.org/10.1038/s41467-020-17791-4
7FIHAProteinGlycoprotein HormoneLHHomo sapienshCGOrg43553chim(NtGi1-Gs)/β1/γ23.22021-09-29doi.org/10.1038/s41586-021-03924-2
7FIH (No Gprot) AProteinGlycoprotein HormoneLHHomo sapienshCGOrg435533.22021-09-29doi.org/10.1038/s41586-021-03924-2
7XW6AProteinGlycoprotein HormoneTSHHomo sapiensM22 FabML109Gs/β1/γ22.782022-08-17doi.org/10.1038/s41586-022-05173-3
7XW6 (No Gprot) AProteinGlycoprotein HormoneTSHHomo sapiensM22 FabML1092.782022-08-17doi.org/10.1038/s41586-022-05173-3
7XW5AProteinGlycoprotein HormoneTSHHomo sapiensTSHML109Gs/β1/γ22.962022-08-24doi.org/10.1038/s41586-022-05173-3
7XW5 (No Gprot) AProteinGlycoprotein HormoneTSHHomo sapiensTSHML1092.962022-08-24doi.org/10.1038/s41586-022-05173-3
7T9NAProteinGlycoprotein HormoneTSHHomo sapiensM22 FabDPPCGs/β1/γ22.92022-08-03doi.org/10.1038/s41586-022-05159-1
7T9N (No Gprot) AProteinGlycoprotein HormoneTSHHomo sapiensM22 FabDPPC2.92022-08-03doi.org/10.1038/s41586-022-05159-1
7UTZAProteinGlycoprotein HormoneTSHHomo sapiensTR1402DPPCGs/β1/γ22.42022-08-03doi.org/10.1038/s41586-022-05159-1
7UTZ (No Gprot) AProteinGlycoprotein HormoneTSHHomo sapiensTR1402DPPC2.42022-08-03doi.org/10.1038/s41586-022-05159-1
7T9MAProteinGlycoprotein HormoneTSHHomo sapiens-CS-17 Antibody-3.12022-08-10doi.org/10.1038/s41586-022-05159-1
8I2GAProteinGlycoprotein HormoneFSHHomo sapiensGlycoprotein hormones α chainCompound 716340Gs/β1/γ22.82023-03-29doi.org/10.1038/s41467-023-36170-3
8I2G (No Gprot) AProteinGlycoprotein HormoneFSHHomo sapiensGlycoprotein hormones α chainCompound 7163402.82023-03-29doi.org/10.1038/s41467-023-36170-3
8I2HAProteinGlycoprotein HormoneFSHHomo sapiens---62023-03-22doi.org/10.1038/s41467-023-36170-3
7FIGAProteinGlycoprotein HormoneLHHomo sapienshCG-chim(NtGi1L-Gs)/β1/γ23.92021-09-29doi.org/10.1038/s41586-021-03924-2
7FIG (No Gprot) AProteinGlycoprotein HormoneLHHomo sapienshCG-3.92021-09-29doi.org/10.1038/s41586-021-03924-2
7FIIAProteinGlycoprotein HormoneLHHomo sapienshCG-chim(NtGi1-Gs)/β1/γ24.32021-09-29doi.org/10.1038/s41586-021-03924-2
7FII (No Gprot) AProteinGlycoprotein HormoneLHHomo sapienshCG-4.32021-09-29doi.org/10.1038/s41586-021-03924-2
7FIJAProteinGlycoprotein HormoneLHHomo sapiens---3.82021-09-29doi.org/10.1038/s41586-021-03924-2
7T9IAProteinGlycoprotein HormoneTSHHomo sapiensTSH-Gs/β1/γ22.92022-08-03doi.org/10.1038/s41586-022-05159-1
7T9I (No Gprot) AProteinGlycoprotein HormoneTSHHomo sapiensTSH-2.92022-08-03doi.org/10.1038/s41586-022-05159-1
7XW7AProteinGlycoprotein HormoneTSHHomo sapiensK1-70--5.52022-08-17doi.org/10.1038/s41586-022-05173-3
7BR3APeptideGonadotrophin Releasing HormoneGnRH1Homo sapiensElagolix--2.792020-10-07doi.org/10.1038/s41467-020-19109-w
9U4WAPeptideGonadotrophin Releasing HormoneGnRH1Sus scrofaGonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ23.182025-06-11doi.org/10.1073/pnas.2500112122
9U4W (No Gprot) APeptideGonadotrophin Releasing HormoneGnRH1Sus scrofaGonadoliberin-1-3.182025-06-11doi.org/10.1073/pnas.2500112122
9U4YAPeptideGonadotrophin Releasing HormoneGnRH1Xenopus laevisGonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ23.182025-06-11doi.org/10.1073/pnas.2500112122
9U4Y (No Gprot) APeptideGonadotrophin Releasing HormoneGnRH1Xenopus laevisGonadoliberin-1-3.182025-06-11doi.org/10.1073/pnas.2500112122
7WCMALipidGPR119GPR119Homo sapiensMBX-2982-Gs/β1/γ22.332022-12-21doi.org/10.1038/s41467-022-34696-6
7WCM (No Gprot) ALipidGPR119GPR119Homo sapiensMBX-2982-2.332022-12-21doi.org/10.1038/s41467-022-34696-6
7WCNALipidGPR119GPR119Homo sapiensAR231453-Gs/β1/γ22.872022-12-21doi.org/10.1038/s41467-022-34696-6
7WCN (No Gprot) ALipidGPR119GPR119Homo sapiensAR231453-2.872022-12-21doi.org/10.1038/s41467-022-34696-6
7XZ5ALipidGPR119GPR119Homo sapiensLysophosphatidylcholine-Gs/β1/γ23.12022-08-24doi.org/10.1038/s41594-022-00816-5
7XZ5 (No Gprot) ALipidGPR119GPR119Homo sapiensLysophosphatidylcholine-3.12022-08-24doi.org/10.1038/s41594-022-00816-5
7XZ6ALipidGPR119GPR119Homo sapiensAPD668-Gs/β1/γ22.82022-08-24doi.org/10.1038/s41594-022-00816-5
7XZ6 (No Gprot) ALipidGPR119GPR119Homo sapiensAPD668-2.82022-08-24doi.org/10.1038/s41594-022-00816-5
8VHFALipidGPR119GPR119Homo sapiensMBX-2982-Gs/β1/γ23.512024-10-30doi.org/10.1016/j.str.2024.10.004
8VHF (No Gprot) ALipidGPR119GPR119Homo sapiensMBX-2982-3.512024-10-30doi.org/10.1016/j.str.2024.10.004
8ZR5ALipidGPR119GPR119Homo sapiensFiruglipel-Gs/β1/γ23.312024-06-19To be published
8ZR5 (No Gprot) ALipidGPR119GPR119Homo sapiensFiruglipel-3.312024-06-19To be published
8ZRKALipidGPR119GPR119Homo sapiensGSK-1292263-Gs/β1/γ22.822024-06-19To be published
8ZRK (No Gprot) ALipidGPR119GPR119Homo sapiensGSK-1292263-2.822024-06-19To be published
8ZX4ALipidGPR55GPR55Homo sapiensLysophosphatidylinositol-chim(NtGi1-G13)/β1/γ23.032024-11-13doi.org/10.1038/s41422-024-01044-w
8ZX4 (No Gprot) ALipidGPR55GPR55Homo sapiensLysophosphatidylinositol-3.032024-11-13doi.org/10.1038/s41422-024-01044-w
8ZX5ALipidGPR55GPR55Homo sapiensAM251-chim(NtGi1-G13)/β1/γ22.852024-11-13doi.org/10.1038/s41422-024-01044-w
8ZX5 (No Gprot) ALipidGPR55GPR55Homo sapiensAM251-2.852024-11-13doi.org/10.1038/s41422-024-01044-w
9IYAALipidGPR55GPR55Homo sapiensONO-9710531--3.042025-01-01doi.org/10.1038/s41422-024-01046-8
8JXTAAmineHistamineH4Homo sapiensHistaminePO4Gi1/β1/γ23.072024-03-20doi.org/10.1038/s41467-024-46840-5
8JXT (No Gprot) AAmineHistamineH4Homo sapiensHistaminePO43.072024-03-20doi.org/10.1038/s41467-024-46840-5
3RZEAAmineHistamineH1Homo sapiensCidoxepin--3.12011-06-15doi.org/10.1038/nature10236
7DFLAAmineHistamineH1Homo sapiensHistamine-chim(NtGi1L-Gq)/β1/γ23.32021-03-31doi.org/10.1038/s41467-021-22427-2
7DFL (No Gprot) AAmineHistamineH1Homo sapiensHistamine-3.32021-03-31doi.org/10.1038/s41467-021-22427-2
8X5XAAmineHistamineH1Homo sapiens---3.52024-01-17doi.org/10.1038/s41467-023-44477-4
8X5YAAmineHistamineH1Homo sapiensAstemizole--32024-01-17doi.org/10.1038/s41467-023-44477-4
8X63AAmineHistamineH1Homo sapiensMepyramine--3.22024-01-17doi.org/10.1038/s41467-023-44477-4
8X64AAmineHistamineH1Homo sapiensDesloratadine--3.42024-01-17doi.org/10.1038/s41467-023-44477-4
8YN2AAmineHistamineH1Homo sapiensHistamine-chim(NtGi1L-Gs-CtGq)/β1/γ22.662024-10-09doi.org/10.1038/s41467-024-52585-y
8YN2 (No Gprot) AAmineHistamineH1Homo sapiensHistamine-2.662024-10-09doi.org/10.1038/s41467-024-52585-y
9LRDAAmineHistamineH1Homo sapiensHistamine-Gi1/β1/γ23.232025-06-11To be published
9LRD (No Gprot) AAmineHistamineH1Homo sapiensHistamine-3.232025-06-11To be published
9LRBAAmineHistamineH1Homo sapiensHistamine-Gs/β1/γ22.772025-06-11To be published
9LRB (No Gprot) AAmineHistamineH1Homo sapiensHistamine-2.772025-06-11To be published
8YUTAAmineHistamineH2Homo sapiensAmthamine-Gs/β1/γ22.72024-06-05doi.org/10.1002/advs.202310120
8YUT (No Gprot) AAmineHistamineH2Homo sapiensAmthamine-2.72024-06-05doi.org/10.1002/advs.202310120
8POKAAmineHistamineH2Homo sapiensHistamine-Gs/β1/γ23.42024-03-06doi.org/10.1038/s41467-024-46096-z
8POK (No Gprot) AAmineHistamineH2Homo sapiensHistamine-3.42024-03-06doi.org/10.1038/s41467-024-46096-z
8YN3AAmineHistamineH2Homo sapiensHistamine-Gs/β1/γ22.562024-10-09doi.org/10.1038/s41467-024-52585-y
8YN3 (No Gprot) AAmineHistamineH2Homo sapiensHistamine-2.562024-10-09doi.org/10.1038/s41467-024-52585-y
8YN4AAmineHistamineH2Homo sapiensHistamine-chim(NtGi1L-Gs-CtGq)/β1/γ22.972024-10-09doi.org/10.1038/s41467-024-52585-y
8YN4 (No Gprot) AAmineHistamineH2Homo sapiensHistamine-2.972024-10-09doi.org/10.1038/s41467-024-52585-y
7UL3AAmineHistamineH2Homo sapiensFamotidine--32022-06-29doi.org/10.1038/s41594-022-00859-8
8YUVAAmineHistamineH3Homo sapiensImmepip-Gi1/β1/γ232024-06-05doi.org/10.1002/advs.202310120
8YUV (No Gprot) AAmineHistamineH3Homo sapiensImmepip-32024-06-05doi.org/10.1002/advs.202310120
7F61AAmineHistamineH3Homo sapiensPF-03654746--2.62022-10-26doi.org/10.1038/s41467-022-33880-y
8YN7AAmineHistamineH3Homo sapiensImmethridine-Go/β1/γ22.772024-10-16doi.org/10.2210/pdb8YN7/pdb
8YN7 (No Gprot) AAmineHistamineH3Homo sapiensImmethridine-2.772024-10-16doi.org/10.2210/pdb8YN7/pdb
8YN8AAmineHistamineH3Homo sapiensProxyfan-Go/β1/γ22.772024-10-16doi.org/10.2210/pdb8YN7/pdb
8YN8 (No Gprot) AAmineHistamineH3Homo sapiensProxyfan-2.772024-10-16doi.org/10.2210/pdb8YN7/pdb
8YUUAAmineHistamineH3Homo sapiensHistamine-Gi1/β1/γ12.72024-06-05doi.org/10.1002/advs.202310120
8YUU (No Gprot) AAmineHistamineH3Homo sapiensHistamine-2.72024-06-05doi.org/10.1002/advs.202310120
8YN5AAmineHistamineH3Homo sapiensHistamine-Gi1/β1/γ22.72024-10-09doi.org/10.1038/s41467-024-52585-y
8YN5 (No Gprot) AAmineHistamineH3Homo sapiensHistamine-2.72024-10-09doi.org/10.1038/s41467-024-52585-y
8YN6AAmineHistamineH3Homo sapiensImetit-Gi1/β1/γ22.772024-10-09doi.org/10.1038/s41467-024-52585-y
8YN6 (No Gprot) AAmineHistamineH3Homo sapiensImetit-2.772024-10-09doi.org/10.1038/s41467-024-52585-y
7YFCAAmineHistamineH4Homo sapiensHistamine-chim(NtGi1-Gs-CtGq)/β1/γ232023-10-25doi.org/10.1038/s41467-023-42260-z
7YFC (No Gprot) AAmineHistamineH4Homo sapiensHistamine-32023-10-25doi.org/10.1038/s41467-023-42260-z
7YFDAAmineHistamineH4Homo sapiensImetit-chim(NtGi1-Gs-CtGq)/β1/γ23.12023-10-25doi.org/10.1038/s41467-023-42260-z
7YFD (No Gprot) AAmineHistamineH4Homo sapiensImetit-3.12023-10-25doi.org/10.1038/s41467-023-42260-z
8JXVAAmineHistamineH4Homo sapiensClozapine-Gi1/β1/γ23.212024-03-20doi.org/10.1038/s41467-024-46840-5
8JXV (No Gprot) AAmineHistamineH4Homo sapiensClozapine-3.212024-03-20doi.org/10.1038/s41467-024-46840-5
8JXWAAmineHistamineH4Homo sapiensVUF6884-Gi1/β1/γ23.012024-03-20doi.org/10.1038/s41467-024-46840-5
8JXW (No Gprot) AAmineHistamineH4Homo sapiensVUF6884-3.012024-03-20doi.org/10.1038/s41467-024-46840-5
8JXXAAmineHistamineH4Homo sapiensClobenpropit-Gi1/β1/γ23.062024-03-20doi.org/10.1038/s41467-024-46840-5
8JXX (No Gprot) AAmineHistamineH4Homo sapiensClobenpropit-3.062024-03-20doi.org/10.1038/s41467-024-46840-5
8YNAAAmineHistamineH4Homo sapiensImmepip-Gi1/β1/γ22.632024-10-16doi.org/10.2210/pdb8YN7/pdb
8YNA (No Gprot) AAmineHistamineH4Homo sapiensImmepip-2.632024-10-16doi.org/10.2210/pdb8YN7/pdb
8YN9AAmineHistamineH4Homo sapiensHistamine-Gi1/β1/γ22.32024-10-09doi.org/10.1038/s41467-024-52585-y
8YN9 (No Gprot) AAmineHistamineH4Homo sapiensHistamine-2.32024-10-09doi.org/10.1038/s41467-024-52585-y
8HN8AAmineHistamineH4Homo sapiensHistamine-Gi1/β1/γ232023-12-20To be published
8HN8 (No Gprot) AAmineHistamineH4Homo sapiensHistamine-32023-12-20To be published
8HOCAAmineHistamineH4Homo sapiensImetit-Gi1/β1/γ232023-12-20To be published
8HOC (No Gprot) AAmineHistamineH4Homo sapiensImetit-32023-12-20To be published
9LRCAAmineHistamineH4Homo sapiensHistamine--2.842025-06-11To be published
9LREAAmineHistamineH4Homo sapiensHistamine-Gi1/β1/γ22.842025-06-11To be published
9LRE (No Gprot) AAmineHistamineH4Homo sapiensHistamine-2.842025-06-11To be published
8JHYAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiens-Compound 9nGi1/β1/γ22.872023-09-06doi.org/10.1016/j.molcel.2023.07.030
8JHY (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiens-Compound 9n2.872023-09-06doi.org/10.1016/j.molcel.2023.07.030
8JIIAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensNiacinCompound 9nGi1/β1/γ23.172023-09-06doi.org/10.1016/j.molcel.2023.07.030
8JII (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensNiacinCompound 9n3.172023-09-06doi.org/10.1016/j.molcel.2023.07.030
8J6PAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensNiacinCompound 9nGi1/β1/γ22.552023-12-06doi.org/10.1038/s41467-023-43537-z
8J6P (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensNiacinCompound 9n2.552023-12-06doi.org/10.1038/s41467-023-43537-z
8J6QAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensβ-HydroxybutyrateCompound 9nGi1/β1/γ22.62023-12-06doi.org/10.1038/s41467-023-43537-z
8J6Q (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensβ-HydroxybutyrateCompound 9n2.62023-12-06doi.org/10.1038/s41467-023-43537-z
9IZDAAlicarboxylic acidHydroxycarboxylic acidHCA1Homo sapiensCHBA-Gi1/β1/γ23.162025-04-02To be published
9IZD (No Gprot) AAlicarboxylic acidHydroxycarboxylic acidHCA1Homo sapiensCHBA-3.162025-04-02To be published
9J8ZAAlicarboxylic acidHydroxycarboxylic acidHCA1Homo sapiens--Gi1/β1/γ23.362025-04-02To be published
9J8Z (No Gprot) AAlicarboxylic acidHydroxycarboxylic acidHCA1Homo sapiens--3.362025-04-02To be published
8UTDAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensMK1903-Gi1/β1/γ23.242025-02-26doi.org/10.1016/j.cell.2024.11.001
8UTD (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensMK1903-3.242025-02-26doi.org/10.1016/j.cell.2024.11.001
8UUJAAlicarboxylic acidHydroxycarboxylic AcidHCA2Mus musculusFCH-2296413-Gi1/β1/γ22.622025-02-26doi.org/10.1016/j.cell.2024.11.001
8UUJ (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Mus musculusFCH-2296413-2.622025-02-26doi.org/10.1016/j.cell.2024.11.001
8J6JAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensGSK256073-Gi1/β1/γ22.82024-01-10doi.org/10.1016/j.celrep.2023.113406
8J6J (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensGSK256073-2.82024-01-10doi.org/10.1016/j.celrep.2023.113406
8J6IAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensMK6892-Gi1/β1/γ22.922024-04-03doi.org/10.1016/j.celrep.2023.113406
8J6I (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensMK6892-2.922024-04-03doi.org/10.1016/j.celrep.2023.113406
8J6LAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensNiacin-Gi1/β1/γ23.052024-04-03doi.org/10.1016/j.celrep.2023.113406
8J6L (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensNiacin-3.052024-04-03doi.org/10.1016/j.celrep.2023.113406
8JILAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensNiacin-Gi1/β1/γ23.52023-09-06doi.org/10.1016/j.molcel.2023.07.030
8JIL (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensNiacin-3.52023-09-06doi.org/10.1016/j.molcel.2023.07.030
8JIMAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensMMF-Gi1/β1/γ22.982023-09-06doi.org/10.1016/j.molcel.2023.07.030
8JIM (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensMMF-2.982023-09-06doi.org/10.1016/j.molcel.2023.07.030
8JZ7AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensMK6892-Gi1/β1/γ22.62023-10-04doi.org/10.1038/s41392-023-01625-y
8JZ7 (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensMK6892-2.62023-10-04doi.org/10.1038/s41392-023-01625-y
8IJ3AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiens--Gi1/β1/γ23.282024-01-03doi.org/10.1038/s41421-023-00610-7
8IJ3 (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiens--3.282024-01-03doi.org/10.1038/s41421-023-00610-7
8IJAAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensNiacin-Gi1/β1/γ22.692024-01-03doi.org/10.1038/s41421-023-00610-7
8IJA (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensNiacin-2.692024-01-03doi.org/10.1038/s41421-023-00610-7
8IJBAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensAcipimox-Gi1/β1/γ23.232024-01-03doi.org/10.1038/s41421-023-00610-7
8IJB (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensAcipimox-3.232024-01-03doi.org/10.1038/s41421-023-00610-7
8IJDAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensMK6892-Gi1/β1/γ23.252024-01-03doi.org/10.1038/s41421-023-00610-7
8IJD (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensMK6892-3.252024-01-03doi.org/10.1038/s41421-023-00610-7
7XK2AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensMK6892-Gi1/β1/γ23.12023-02-22doi.org/10.1038/s41467-023-37177-6
7XK2 (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensMK6892-3.12023-02-22doi.org/10.1038/s41467-023-37177-6
7ZL9AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiens---2.72023-04-12doi.org/10.1038/s41467-023-37177-6
7ZLYAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiens---2.72023-04-12doi.org/10.1038/s41467-023-37177-6
8IHFAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensMK6892-Gi1/β1/γ22.972023-08-30doi.org/10.1038/s41467-023-41650-7
8IHF (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensMK6892-2.972023-08-30doi.org/10.1038/s41467-023-41650-7
8IHHAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensLUF6283-Gi1/β1/γ23.062023-08-30doi.org/10.1038/s41467-023-41650-7
8IHH (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensLUF6283-3.062023-08-30doi.org/10.1038/s41467-023-41650-7
8IHIAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensAcifran-Gi1/β1/γ23.112023-08-30doi.org/10.1038/s41467-023-41650-7
8IHI (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensAcifran-3.112023-08-30doi.org/10.1038/s41467-023-41650-7
8IHBAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensGSK256073-Gi1/β1/γ22.852023-09-13doi.org/10.1038/s41467-023-41650-7
8IHB (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensGSK256073-2.852023-09-13doi.org/10.1038/s41467-023-41650-7
8K5BAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensNiacin--3.432023-11-22doi.org/10.1038/s41467-023-42764-8
8K5CAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensAcipimox--3.132023-11-22doi.org/10.1038/s41467-023-42764-8
8K5DAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensGSK256073--3.742023-11-22doi.org/10.1038/s41467-023-42764-8
8I7VAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensAcipimox-Gi1/β1/γ22.772024-02-07doi.org/10.1038/s41467-023-42764-8
8I7V (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensAcipimox-2.772024-02-07doi.org/10.1038/s41467-023-42764-8
8I7WAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensGSK256073-Gi1/β1/γ23.392024-02-07doi.org/10.1038/s41467-023-42764-8
8I7W (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensGSK256073-3.392024-02-07doi.org/10.1038/s41467-023-42764-8
8J6RAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensMK6892-Gi1/β1/γ22.762023-12-06doi.org/10.1038/s41467-023-43537-z
8J6R (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensMK6892-2.762023-12-06doi.org/10.1038/s41467-023-43537-z
8IY9AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensNiacin-Go/β1/γ23.372024-03-06doi.org/10.1038/s41467-024-46239-2
8IY9 (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensNiacin-3.372024-03-06doi.org/10.1038/s41467-024-46239-2
8IYHAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensMK6892-Go/β1/γ23.32024-03-06doi.org/10.1038/s41467-024-46239-2
8IYH (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensMK6892-3.32024-03-06doi.org/10.1038/s41467-024-46239-2
8IYWAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensGSK256073-Go/β1/γ23.452024-03-06doi.org/10.1038/s41467-024-46239-2
8IYW (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensGSK256073-3.452024-03-06doi.org/10.1038/s41467-024-46239-2
8JERAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensAcipimox-Go/β1/γ23.452024-03-06doi.org/10.1038/s41467-024-46239-2
8JER (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensAcipimox-3.452024-03-06doi.org/10.1038/s41467-024-46239-2
8JHNAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensMMF-Go/β1/γ23.752024-03-06doi.org/10.1038/s41467-024-46239-2
8JHN (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensMMF-3.752024-03-06doi.org/10.1038/s41467-024-46239-2
9CIBAAlicarboxylic acidHydroxycarboxylic acidHCA2Mus musculusFCH-2296413--2.622025-05-14doi.org/10.1016/j.cell.2024.11.001
9IQTAAlicarboxylic acidHydroxycarboxylic acidHCA2Homo sapiensNiacin-Gi1/β1/γ22.92024-10-02doi.org/10.1016/j.jmb.2024.168795
9IQT (No Gprot) AAlicarboxylic acidHydroxycarboxylic acidHCA2Homo sapiensNiacin-2.92024-10-02doi.org/10.1016/j.jmb.2024.168795
8H2GAAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensNiacin-Gi1/β1/γ23.012023-10-11doi.org/10.1038/s41467-023-42764-8
8H2G (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA2Homo sapiensNiacin-3.012023-10-11doi.org/10.1038/s41467-023-42764-8
9IZAAAlicarboxylic acidHydroxycarboxylic acidHCA2Homo sapiensSCH900271-Gi1/β1/γ23.062025-04-02To be published
9IZA (No Gprot) AAlicarboxylic acidHydroxycarboxylic acidHCA2Homo sapiensSCH900271-3.062025-04-02To be published
9IZCAAlicarboxylic acidHydroxycarboxylic acidHCA2Homo sapiensMK1903-Gi1/β1/γ22.682025-04-02To be published
9IZC (No Gprot) AAlicarboxylic acidHydroxycarboxylic acidHCA2Homo sapiensMK1903-2.682025-04-02To be published
8IHJAAlicarboxylic acidHydroxycarboxylic AcidHCA3Homo sapiensAcifran-Gi1/β1/γ23.072023-08-30doi.org/10.1038/s41467-023-41650-7
8IHJ (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA3Homo sapiensAcifran-3.072023-08-30doi.org/10.1038/s41467-023-41650-7
8IHKAAlicarboxylic acidHydroxycarboxylic AcidHCA3Homo sapiensAcifran--3.212023-08-30doi.org/10.1038/s41467-023-41650-7
8JEFAAlicarboxylic acidHydroxycarboxylic AcidHCA3Homo sapiens(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ22.962024-12-18doi.org/10.1016/j.celrep.2024.114895
8JEF (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCA3Homo sapiens(3S)-3-hydroxyoctanoic acid-2.962024-12-18doi.org/10.1016/j.celrep.2024.114895
8JEIAAlicarboxylic acidHydroxycarboxylic AcidHCAR3Homo sapiens3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ22.732024-11-20doi.org/10.2210/pdb8JEI/pdb
8JEI (No Gprot) AAlicarboxylic acidHydroxycarboxylic AcidHCAR3Homo sapiens3-nitro-4-(propylamino)benzoic acid-2.732024-11-20doi.org/10.2210/pdb8JEI/pdb
8ZJDAPeptideKisspeptinKiss1Homo sapiensKisspeptin-10-chim(NtGi1-Gq)/β1/γ13.062024-07-03doi.org/10.1016/j.celrep.2024.114389
8ZJD (No Gprot) APeptideKisspeptinKiss1Homo sapiensKisspeptin-10-3.062024-07-03doi.org/10.1016/j.celrep.2024.114389
8ZJEAPeptideKisspeptinKiss1Homo sapiensTAK-448-chim(NtGi1-Gq)/β1/γ13.072024-07-03doi.org/10.1016/j.celrep.2024.114389
8ZJE (No Gprot) APeptideKisspeptinKiss1Homo sapiensTAK-448-3.072024-07-03doi.org/10.1016/j.celrep.2024.114389
8XGOAPeptideKisspeptinKiss1Homo sapiensTAK448-chim(NtGi1-Gq)/β1/γ22.682024-10-30doi.org/10.1126/sciadv.adn7771
8XGO (No Gprot) APeptideKisspeptinKiss1Homo sapiensTAK448-2.682024-10-30doi.org/10.1126/sciadv.adn7771
8XGSAPeptideKisspeptinKiss1Homo sapiensMetastin-chim(NtGi1-Gq)/β1/γ22.952024-10-30doi.org/10.1126/sciadv.adn7771
8XGS (No Gprot) APeptideKisspeptinKiss1Homo sapiensMetastin-2.952024-10-30doi.org/10.1126/sciadv.adn7771
8XGUAPeptideKisspeptinKiss1Homo sapiensTAK448-Gi1/β1/γ232024-10-30doi.org/10.1126/sciadv.adn7771
8XGU (No Gprot) APeptideKisspeptinKiss1Homo sapiensTAK448-32024-10-30doi.org/10.1126/sciadv.adn7771
7K15ALipidLeukotrieneBLT1Homo sapiensMKD046Na-2.882021-02-17doi.org/10.1038/s41467-021-23149-1
6RZ4ALipidLeukotrieneCysLT1Homo sapiensPranlukastNa-2.72019-10-30doi.org/10.1126/sciadv.aax2518
6RZ5ALipidLeukotrieneCysLT1Homo sapiensZafirlukastNa-2.532019-10-30doi.org/10.1126/sciadv.aax2518
5X33ALipidLeukotrieneBLT1Cavia porcellusBIIL260--3.72018-01-03doi.org/10.1038/nchembio.2547
7VKTALipidLeukotrieneBLT1Homo sapiensLTB4-Gi1/β1/γ22.92022-03-09doi.org/10.1038/s41467-022-28820-9
7VKT (No Gprot) ALipidLeukotrieneBLT1Homo sapiensLTB4-2.92022-03-09doi.org/10.1038/s41467-022-28820-9
6RZ6ALipidLeukotrieneCysLT2Homo sapiensONO-2570366--2.432019-12-11doi.org/10.1038/s41467-019-13348-2
6RZ7ALipidLeukotrieneCysLT2Homo sapiensONO-2570366--2.432019-12-11doi.org/10.1038/s41467-019-13348-2
6RZ8ALipidLeukotrieneCysLT2Homo sapiensONO-2080365--2.72019-12-11doi.org/10.1038/s41467-019-13348-2
6RZ9ALipidLeukotrieneCysLT2Homo sapiensONO-2770372--2.732019-12-11doi.org/10.1038/s41467-019-13348-2
9JH5ALipidLeukotrieneCysLT2Homo sapiensC16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ22.762025-04-23doi.org/10.1038/s41586-025-08792-8
9JH5 (No Gprot) ALipidLeukotrieneCysLT2Homo sapiensC16:0 Ceramide-2.762025-04-23doi.org/10.1038/s41586-025-08792-8
9JH6ALipidLeukotrieneCysLT2Homo sapiensC20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ22.892025-04-23doi.org/10.1038/s41586-025-08792-8
9JH6 (No Gprot) ALipidLeukotrieneCysLT2Homo sapiensC20:0 Ceramide-2.892025-04-23doi.org/10.1038/s41586-025-08792-8
9IXXALipidLeukotrieneCysLT2Homo sapiensLTD4-chim(NtGi1-Gs-CtGq)/β1/γ23.152025-04-02doi.org/10.1073/pnas.2417148122
9IXX (No Gprot) ALipidLeukotrieneCysLT2Homo sapiensLTD4-3.152025-04-02doi.org/10.1073/pnas.2417148122
8G94ALipidLysophospholipidS1P1Homo sapiens-CD69Gi1/β1/γ23.152023-04-19doi.org/10.7554/eLife.88204
8G94 (No Gprot) ALipidLysophospholipidS1P1Homo sapiens-CD693.152023-04-19doi.org/10.7554/eLife.88204
4Z34ALipidLysophospholipidLPA1Homo sapiensONO-9780307--32015-06-03doi.org/10.1016/j.cell.2015.06.002
4Z35ALipidLysophospholipidLPA1Homo sapiensONO-9910539--2.92015-06-03doi.org/10.1016/j.cell.2015.06.002
4Z36ALipidLysophospholipidLPA1Homo sapiensONO-3080573--2.92015-06-03doi.org/10.1016/j.cell.2015.06.002
9IZFALipidLysophospholipidLPA1Homo sapiensNKP-Gi1/β1/γ23.142025-01-01doi.org/10.1016/j.jsb.2024.108164
9IZF (No Gprot) ALipidLysophospholipidLPA1Homo sapiensNKP-3.142025-01-01doi.org/10.1016/j.jsb.2024.108164
9IZGALipidLysophospholipidLPA1Homo sapiensNKP-chim(NtGi1-Gs-CtGq)/β1/γ23.042025-01-01doi.org/10.1016/j.jsb.2024.108164
9IZG (No Gprot) ALipidLysophospholipidLPA1Homo sapiensNKP-3.042025-01-01doi.org/10.1016/j.jsb.2024.108164
7TD0ALipidLysophospholipidLPA1Homo sapiensLPA-Gi1/β1/γ22.832022-02-09doi.org/10.1038/s41467-022-28417-2
7TD0 (No Gprot) ALipidLysophospholipidLPA1Homo sapiensLPA-2.832022-02-09doi.org/10.1038/s41467-022-28417-2
7TD1ALipidLysophospholipidLPA1Homo sapiensLPA-Gi1/β1/γ23.082022-02-09doi.org/10.1038/s41467-022-28417-2
7TD1 (No Gprot) ALipidLysophospholipidLPA1Homo sapiensLPA-3.082022-02-09doi.org/10.1038/s41467-022-28417-2
7TD2ALipidLysophospholipidLPA1Homo sapiensLPA-Gi1/β1/γ23.112022-02-09doi.org/10.1038/s41467-022-28417-2
7TD2 (No Gprot) ALipidLysophospholipidLPA1Homo sapiensLPA-3.112022-02-09doi.org/10.1038/s41467-022-28417-2
7YU3ALipidLysophospholipidLPA1Homo sapiensONO-0740556-Gi1/β1/γ23.52022-10-05doi.org/10.1038/s41467-022-33121-2
7YU3 (No Gprot) ALipidLysophospholipidLPA1Homo sapiensONO-0740556-3.52022-10-05doi.org/10.1038/s41467-022-33121-2
7YU4ALipidLysophospholipidLPA1Homo sapiensONO-0740556--3.72022-10-05doi.org/10.1038/s41467-022-33121-2
7YU5ALipidLysophospholipidLPA1Homo sapiensONO-0740556-Gi1/β1/γ23.72022-10-05doi.org/10.1038/s41467-022-33121-2
7YU5 (No Gprot) ALipidLysophospholipidLPA1Homo sapiensONO-0740556-3.72022-10-05doi.org/10.1038/s41467-022-33121-2
7YU6ALipidLysophospholipidLPA1Homo sapiensONO-0740556-Gi1/β1/γ23.92022-10-05doi.org/10.1038/s41467-022-33121-2
7YU6 (No Gprot) ALipidLysophospholipidLPA1Homo sapiensONO-0740556-3.92022-10-05doi.org/10.1038/s41467-022-33121-2
7YU7ALipidLysophospholipidLPA1Homo sapiensONO-0740556-Gi1/β1/γ24.52022-10-05doi.org/10.1038/s41467-022-33121-2
7YU7 (No Gprot) ALipidLysophospholipidLPA1Homo sapiensONO-0740556-4.52022-10-05doi.org/10.1038/s41467-022-33121-2
7YU8ALipidLysophospholipidLPA1Homo sapiensONO-0740556-Gi1/β1/γ25.62022-10-05doi.org/10.1038/s41467-022-33121-2
7YU8 (No Gprot) ALipidLysophospholipidLPA1Homo sapiensONO-0740556-5.62022-10-05doi.org/10.1038/s41467-022-33121-2
9J5VALipidLysophospholipidLPA1Homo sapiensCpY-Gi1/β1/γ22.862024-11-27doi.org/10.1038/s42003-024-07152-y
9J5V (No Gprot) ALipidLysophospholipidLPA1Homo sapiensCpY-2.862024-11-27doi.org/10.1038/s42003-024-07152-y
9IZHALipidLysophospholipidLPA1Homo sapiensLPA-chim(NtGi2-G13)/β1/γ23.042025-01-01doi.org/10.1016/j.jsb.2024.108164
9IZH (No Gprot) ALipidLysophospholipidLPA1Homo sapiensLPA-3.042025-01-01doi.org/10.1016/j.jsb.2024.108164
5XSZALipidLysophospholipidLPA6Danio rerioGlyceryl-mono-oleate--3.22017-08-16doi.org/10.1038/nature23448
9ITBALipidLysophospholipidLPA6Homo sapiensLPA-chim(NtGi1-Gs-CtGq)/β1/γ22.892025-01-15doi.org/10.1073/pnas.2415426122
9ITB (No Gprot) ALipidLysophospholipidLPA6Homo sapiensLPA-2.892025-01-15doi.org/10.1073/pnas.2415426122
9ITEALipidLysophospholipidLPA6Homo sapiensLPA-chim(NtGi2-G13)/β1/γ23.062025-01-15doi.org/10.1073/pnas.2415426122
9ITE (No Gprot) ALipidLysophospholipidLPA6Homo sapiensLPA-3.062025-01-15doi.org/10.1073/pnas.2415426122
7EVYALipidLysophospholipidS1P1Homo sapiensSiponimod-Gi1/β1/γ22.982021-09-29doi.org/10.1038/s41422-021-00566-x
7EVY (No Gprot) ALipidLysophospholipidS1P1Homo sapiensSiponimod-2.982021-09-29doi.org/10.1038/s41422-021-00566-x
7EVZALipidLysophospholipidS1P1Homo sapiensCenerimod-Gi1/β1/γ23.072021-09-29doi.org/10.1038/s41422-021-00566-x
7EVZ (No Gprot) ALipidLysophospholipidS1P1Homo sapiensCenerimod-3.072021-09-29doi.org/10.1038/s41422-021-00566-x
7EW0ALipidLysophospholipidS1P1Homo sapiensOzanimod-Gi1/β1/γ23.422021-09-29doi.org/10.1038/s41422-021-00566-x
7EW0 (No Gprot) ALipidLysophospholipidS1P1Homo sapiensOzanimod-3.422021-09-29doi.org/10.1038/s41422-021-00566-x
7EW7ALipidLysophospholipidS1P1Homo sapiensSEW2871-Gi1/β1/γ23.272021-09-29doi.org/10.1038/s41422-021-00566-x
7EW7 (No Gprot) ALipidLysophospholipidS1P1Homo sapiensSEW2871-3.272021-09-29doi.org/10.1038/s41422-021-00566-x
7TD3ALipidLysophospholipidS1P1Homo sapiensS1P-Gi1/β1/γ232022-02-09doi.org/10.1038/s41467-022-28417-2
7TD3 (No Gprot) ALipidLysophospholipidS1P1Homo sapiensS1P-32022-02-09doi.org/10.1038/s41467-022-28417-2
7TD4ALipidLysophospholipidS1P1Homo sapiensSiponimod-Gi1/β1/γ22.62022-02-09doi.org/10.1038/s41467-022-28417-2
7TD4 (No Gprot) ALipidLysophospholipidS1P1Homo sapiensSiponimod-2.62022-02-09doi.org/10.1038/s41467-022-28417-2
7EO2ALipidLysophospholipidS1P1Homo sapiensFTY720-P-Gi1/β1/γ22.892022-01-05doi.org/10.1038/s41589-021-00930-3
7EO2 (No Gprot) ALipidLysophospholipidS1P1Homo sapiensFTY720-P-2.892022-01-05doi.org/10.1038/s41589-021-00930-3
7EO4ALipidLysophospholipidS1P1Homo sapiensBAF312-Gi1/β1/γ22.862022-01-05doi.org/10.1038/s41589-021-00930-3
7EO4 (No Gprot) ALipidLysophospholipidS1P1Homo sapiensBAF312-2.862022-01-05doi.org/10.1038/s41589-021-00930-3
7WF7ALipidLysophospholipidS1P1Homo sapiensS1P-Gi1/β1/γ23.42022-01-05doi.org/10.1038/s41589-021-00930-3
7WF7 (No Gprot) ALipidLysophospholipidS1P1Homo sapiensS1P-3.42022-01-05doi.org/10.1038/s41589-021-00930-3
7VIEALipidLysophospholipidS1P1Homo sapiensS1P-Gi1/β1/γ22.862022-09-28doi.org/10.1073/pnas.2117716119
7VIE (No Gprot) ALipidLysophospholipidS1P1Homo sapiensS1P-2.862022-09-28doi.org/10.1073/pnas.2117716119
7VIFALipidLysophospholipidS1P1Homo sapiensS-FTY720-P-Gi1/β1/γ22.832022-09-28doi.org/10.1073/pnas.2117716119
7VIF (No Gprot) ALipidLysophospholipidS1P1Homo sapiensS-FTY720-P-2.832022-09-28doi.org/10.1073/pnas.2117716119
7VIGALipidLysophospholipidS1P1Homo sapiensCBP-307-Gi1/β1/γ22.892022-09-28doi.org/10.1073/pnas.2117716119
7VIG (No Gprot) ALipidLysophospholipidS1P1Homo sapiensCBP-307-2.892022-09-28doi.org/10.1073/pnas.2117716119
7VIHALipidLysophospholipidS1P1Homo sapiensCBP-307-Gi1/β1/γ22.982022-09-28doi.org/10.1073/pnas.2117716119
7VIH (No Gprot) ALipidLysophospholipidS1P1Homo sapiensCBP-307-2.982022-09-28doi.org/10.1073/pnas.2117716119
3V2WALipidLysophospholipidS1P1Homo sapiensPubChem 51892645--3.352012-02-15doi.org/10.1126/science.1215904
3V2YALipidLysophospholipidS1P1Homo sapiensPubChem 51892645--2.82012-02-15doi.org/10.1126/science.1215904
8YICALipidLysophospholipidS1P1Homo sapiensSAR247799-Gi1/β1/γ23.472024-12-11To be published
8YIC (No Gprot) ALipidLysophospholipidS1P1Homo sapiensSAR247799-3.472024-12-11To be published
7T6BALipidLysophospholipidS1P2Homo sapiensS1P-chim(NtGi1L-G13)/β1/γ23.192022-04-06doi.org/10.1126/sciadv.abn0067
7T6B (No Gprot) ALipidLysophospholipidS1P2Homo sapiensS1P-3.192022-04-06doi.org/10.1126/sciadv.abn0067
7EW2ALipidLysophospholipidS1P3Homo sapiensFingolimod-Gi1/β1/γ23.12021-09-29doi.org/10.1038/s41422-021-00567-w
7EW2 (No Gprot) ALipidLysophospholipidS1P3Homo sapiensFingolimod-3.12021-09-29doi.org/10.1038/s41422-021-00567-w
7EW3ALipidLysophospholipidS1P3Homo sapiensS1P-Gi1/β1/γ23.12021-09-29doi.org/10.1038/s41422-021-00567-w
7EW3 (No Gprot) ALipidLysophospholipidS1P3Homo sapiensS1P-3.12021-09-29doi.org/10.1038/s41422-021-00567-w
7EW4ALipidLysophospholipidS1P3Homo sapiensCYM5541-Gi1/β1/γ23.22021-09-29doi.org/10.1038/s41422-021-00567-w
7EW4 (No Gprot) ALipidLysophospholipidS1P3Homo sapiensCYM5541-3.22021-09-29doi.org/10.1038/s41422-021-00567-w
7C4SALipidLysophospholipidS1P3Homo sapiensS1P--3.22021-06-09doi.org/10.1126/sciadv.abf5325
7EW1ALipidLysophospholipidS1P5Homo sapiensSiponimod-Gi1/β1/γ23.42021-09-29doi.org/10.1038/s41422-021-00566-x
7EW1 (No Gprot) ALipidLysophospholipidS1P5Homo sapiensSiponimod-3.42021-09-29doi.org/10.1038/s41422-021-00566-x
7YXAALipidLysophospholipidS1P5Homo sapiensONO-5430608--2.22022-08-10doi.org/10.1038/s41467-022-32447-1
8WSSAPeptideMelanin Concentrating HormoneMCH1Homo sapiensPro-MCH-Gi1/β1/γ13.012024-06-19doi.org/10.1038/s41421-024-00679-8
8WSS (No Gprot) APeptideMelanin Concentrating HormoneMCH1Homo sapiensPro-MCH-3.012024-06-19doi.org/10.1038/s41421-024-00679-8
8YNSAPeptideMelanin Concentrating HormoneMCH1Homo sapiensSNAP-94847--3.332024-12-18doi.org/10.1038/s41421-024-00754-0
8YNTAPeptideMelanin Concentrating HormoneMCH1Homo sapiensSNAP-94847--3.432024-12-18doi.org/10.1038/s41421-024-00754-0
8WWKAPeptideMelanin Concentrating HormoneMCH1Homo sapiensMCH-Gi1/β1/γ22.612024-11-13doi.org/10.1038/s41421-024-00754-0
8WWK (No Gprot) APeptideMelanin Concentrating HormoneMCH1Homo sapiensMCH-2.612024-11-13doi.org/10.1038/s41421-024-00754-0
8WWLAPeptideMelanin Concentrating HormoneMCH1Homo sapiensMCH-Gi1/β1/γ22.782024-11-13doi.org/10.1038/s41421-024-00754-0
8WWL (No Gprot) APeptideMelanin Concentrating HormoneMCH1Homo sapiensMCH-2.782024-11-13doi.org/10.1038/s41421-024-00754-0
8WWMAPeptideMelanin Concentrating HormoneMCH1Homo sapiensMCH-Gi1/β1/γ22.812024-11-13doi.org/10.1038/s41421-024-00754-0
8WWM (No Gprot) APeptideMelanin Concentrating HormoneMCH1Homo sapiensMCH-2.812024-11-13doi.org/10.1038/s41421-024-00754-0
8WWNAPeptideMelanin Concentrating HormoneMCH1Homo sapiensMCH-Gi1/β1/γ22.652024-11-13doi.org/10.1038/s41421-024-00754-0
8WWN (No Gprot) APeptideMelanin Concentrating HormoneMCH1Homo sapiensMCH-2.652024-11-13doi.org/10.1038/s41421-024-00754-0
8WWHAPeptideMelanin Concentrating HormoneMCH1Homo sapiens--Gi1/β1/γ22.842024-11-13To be published
8WWH (No Gprot) APeptideMelanin Concentrating HormoneMCH1Homo sapiens--2.842024-11-13To be published
8WWIAPeptideMelanin Concentrating HormoneMCH1Homo sapiens--Gi1/β1/γ23.432024-11-13To be published
8WWI (No Gprot) APeptideMelanin Concentrating HormoneMCH1Homo sapiens--3.432024-11-13To be published
8WWJAPeptideMelanin Concentrating HormoneMCH1Homo sapiens--Gi1/β1/γ23.032024-11-13To be published
8WWJ (No Gprot) APeptideMelanin Concentrating HormoneMCH1Homo sapiens--3.032024-11-13To be published
8WSTAPeptideMelanin Concentrating HormoneMCH2Homo sapiensPro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ22.42024-06-19doi.org/10.1038/s41421-024-00679-8
8WST (No Gprot) APeptideMelanin Concentrating HormoneMCH2Homo sapiensPro-MCH-2.42024-06-19doi.org/10.1038/s41421-024-00679-8
8GY7APeptideMelanocortinMC2Homo sapiensCorticotropinCachim(NtGi1-Gs)/β1/γ2; MRAP13.32023-01-11doi.org/10.1038/s41422-022-00751-6
8GY7 (No Gprot) APeptideMelanocortinMC2Homo sapiensCorticotropinCa3.32023-01-11doi.org/10.1038/s41422-022-00751-6
8IOCAPeptideMelanocortinMC3Homo sapiensγ-MSHCachim(NtGi1-Gs)/β1/γ22.862023-09-20doi.org/10.1038/s41421-023-00586-4
8IOC (No Gprot) APeptideMelanocortinMC3Homo sapiensγ-MSHCa2.862023-09-20doi.org/10.1038/s41421-023-00586-4
8KIGAPeptideMelanocortinMC3Homo sapiensSHU9119Ca-3.12025-02-26doi.org/10.2210/pdb8KIG/pdb
8W8WAPeptideMelanocortinMC3Homo sapiensα-MSHCaGs/β1/γ22.92025-03-19To be published
8W8W (No Gprot) APeptideMelanocortinMC3Homo sapiensα-MSHCa2.92025-03-19To be published
8W8XAPeptideMelanocortinMC3Homo sapiensβ-MSHCaGs/β1/γ22.92025-03-19To be published
8W8X (No Gprot) APeptideMelanocortinMC3Homo sapiensβ-MSHCa2.92025-03-19To be published
8W8YAPeptideMelanocortinMC3Homo sapiensγ-MSHCaGs/β1/γ22.92025-03-19To be published
8W8Y (No Gprot) APeptideMelanocortinMC3Homo sapiensγ-MSHCa2.92025-03-19To be published
6W25APeptideMelanocortinMC4Homo sapiensSHU9119Ca-2.752020-04-29doi.org/10.1126/science.aaz8995
8INRAPeptideMelanocortinMC5Homo sapiensα-MSHCachim(NtGi1-Gs)/β1/γ22.732023-09-20doi.org/10.1038/s41421-023-00586-4
8INR (No Gprot) APeptideMelanocortinMC5Homo sapiensα-MSHCa2.732023-09-20doi.org/10.1038/s41421-023-00586-4
8IODAPeptideMelanocortinMC5Homo sapiensPG-901Cachim(NtGi1-Gs)/β1/γ22.592023-09-20doi.org/10.1038/s41421-023-00586-4
8IOD (No Gprot) APeptideMelanocortinMC5Homo sapiensPG-901Ca2.592023-09-20doi.org/10.1038/s41421-023-00586-4
7F4DAPeptideMelanocortinMC1Homo sapiensα-MSH-chim(NtGi1-Gs)/β1/γ232021-09-08doi.org/10.1038/s41422-021-00557-y
7F4D (No Gprot) APeptideMelanocortinMC1Homo sapiensα-MSH-32021-09-08doi.org/10.1038/s41422-021-00557-y
7F4FAPeptideMelanocortinMC1Homo sapiensAfamelanotide-chim(NtGi1-Gs)/β1/γ22.92021-09-08doi.org/10.1038/s41422-021-00557-y
7F4F (No Gprot) APeptideMelanocortinMC1Homo sapiensAfamelanotide-2.92021-09-08doi.org/10.1038/s41422-021-00557-y
7F4HAPeptideMelanocortinMC1Homo sapiensAfamelanotide-chim(NtGi1-Gs)/β1/γ22.72021-09-08doi.org/10.1038/s41422-021-00557-y
7F4H (No Gprot) APeptideMelanocortinMC1Homo sapiensAfamelanotide-2.72021-09-08doi.org/10.1038/s41422-021-00557-y
7F4IAPeptideMelanocortinMC1Homo sapiensSHU9119-chim(NtGi1-Gs)/β1/γ23.12021-09-08doi.org/10.1038/s41422-021-00557-y
7F4I (No Gprot) APeptideMelanocortinMC1Homo sapiensSHU9119-3.12021-09-08doi.org/10.1038/s41422-021-00557-y
7F53APeptideMelanocortinMC4Homo sapiensα-MSH-Gs/β1/γ232021-11-03doi.org/10.1038/s41422-021-00552-3
7F53 (No Gprot) APeptideMelanocortinMC4Homo sapiensα-MSH-32021-11-03doi.org/10.1038/s41422-021-00552-3
7F54APeptideMelanocortinMC4Homo sapiensAfamelanotide-Gs/β1/γ232021-11-03doi.org/10.1038/s41422-021-00552-3
7F54 (No Gprot) APeptideMelanocortinMC4Homo sapiensAfamelanotide-32021-11-03doi.org/10.1038/s41422-021-00552-3
7F55APeptideMelanocortinMC4Homo sapiensBremelanotide-Gs/β1/γ23.12021-11-03doi.org/10.1038/s41422-021-00552-3
7F55 (No Gprot) APeptideMelanocortinMC4Homo sapiensBremelanotide-3.12021-11-03doi.org/10.1038/s41422-021-00552-3
7F58APeptideMelanocortinMC4Homo sapiensTHIQ-Gs/β1/γ23.12021-11-03doi.org/10.1038/s41422-021-00552-3
7F58 (No Gprot) APeptideMelanocortinMC4Homo sapiensTHIQ-3.12021-11-03doi.org/10.1038/s41422-021-00552-3
7PIUAPeptideMelanocortinMC4Homo sapiensSetmelanotide-Gs/β1/γ22.582021-11-17doi.org/10.1038/s41422-021-00569-8
7PIU (No Gprot) APeptideMelanocortinMC4Homo sapiensSetmelanotide-2.582021-11-17doi.org/10.1038/s41422-021-00569-8
7PIVAPeptideMelanocortinMC4Homo sapiensSetmelanotide-Gs/β1/γ22.862021-11-17doi.org/10.1038/s41422-021-00569-8
7PIV (No Gprot) APeptideMelanocortinMC4Homo sapiensSetmelanotide-2.862021-11-17doi.org/10.1038/s41422-021-00569-8
7AUEAPeptideMelanocortinMC4Homo sapiensSetmelanotide-chim(NtGi1L-Gs)/β1/γ22.972021-04-28doi.org/10.1126/science.abf7958
7AUE (No Gprot) APeptideMelanocortinMC4Homo sapiensSetmelanotide-2.972021-04-28doi.org/10.1126/science.abf7958
8WKYAPeptideMelanocortinMC4Homo sapiensPG-934--2.92024-08-07doi.org/10.1021/acs.jmedchem.3c01822
8WKZAPeptideMelanocortinMC4Homo sapiensSBL-MC-31--3.32024-08-07doi.org/10.1021/acs.jmedchem.3c01822
8QJ2APeptideMelanocortinMC4Homo sapienspN162-Gs3.42024-09-25doi.org/10.1038/s41467-024-50827-7
8QJ2 (No Gprot) APeptideMelanocortinMC4Homo sapienspN162-3.42024-09-25doi.org/10.1038/s41467-024-50827-7
7VGYAMelatoninMelatoninMT1Homo sapiens2-Iodomelatonin-Gi1/β1/γ23.12022-03-02doi.org/10.1038/s41467-022-28111-3
7VGY (No Gprot) AMelatoninMelatoninMT1Homo sapiens2-Iodomelatonin-3.12022-03-02doi.org/10.1038/s41467-022-28111-3
7VGZAMelatoninMelatoninMT1Homo sapiensRemalteon-Gi1/β1/γ23.32022-03-02doi.org/10.1038/s41467-022-28111-3
7VGZ (No Gprot) AMelatoninMelatoninMT1Homo sapiensRemalteon-3.32022-03-02doi.org/10.1038/s41467-022-28111-3
6ME2AMelatoninMelatoninMT1Homo sapiensRamelteon--2.82019-04-24doi.org/10.1038/s41586-019-1141-3
6ME3AMelatoninMelatoninMT1Homo sapiens2-Phenylmelatonin--2.92019-04-24doi.org/10.1038/s41586-019-1141-3
6ME4AMelatoninMelatoninMT1Homo sapiens2-Iodomelatonin--3.22019-04-24doi.org/10.1038/s41586-019-1141-3
6ME5AMelatoninMelatoninMT1Homo sapiensAgomelatine--3.22019-04-24doi.org/10.1038/s41586-019-1141-3
7DB6AMelatoninMelatoninMT1Homo sapiensRamelteon-Gi1/β1/γ23.32021-08-18doi.org/10.1038/s41594-021-00634-1
7DB6 (No Gprot) AMelatoninMelatoninMT1Homo sapiensRamelteon-3.32021-08-18doi.org/10.1038/s41594-021-00634-1
6PS8AMelatoninMelatoninMT1Homo sapiens2-Phenylmelatonin--3.32019-11-13doi.org/10.1107/S2052252519013137
7VH0AMelatoninMelatoninMT2Homo sapiensRamelteon-Gi1/β1/γ13.462022-03-02doi.org/10.1038/s41467-022-28111-3
7VH0 (No Gprot) AMelatoninMelatoninMT2Homo sapiensRamelteon-3.462022-03-02doi.org/10.1038/s41467-022-28111-3
6ME6AMelatoninMelatoninMT2Homo sapiens2-Phenylmelatonin--2.82019-04-24doi.org/10.1038/s41586-019-1144-0
6ME7AMelatoninMelatoninMT2Homo sapiens2-Phenylmelatonin--3.22019-04-24doi.org/10.1038/s41586-019-1144-0
6ME8AMelatoninMelatoninMT2Homo sapiens2-Phenylmelatonin--3.12019-04-24doi.org/10.1038/s41586-019-1144-0
6ME9AMelatoninMelatoninMT2Homo sapiensRamelteon--3.32019-04-24doi.org/10.1038/s41586-019-1144-0
8X0BCAminoacidMetabotropic GlutamatemGlu5; mGlu5Homo sapiensQuisqualateVU0424465-3.12024-11-06doi.org/10.1038/s41467-024-55439-9
8X0CCAminoacidMetabotropic GlutamatemGlu5; mGlu5Homo sapiensQuisqualateVU0424465-3.22024-11-06doi.org/10.1038/s41467-024-55439-9
8X0DCAminoacidMetabotropic GlutamatemGlu5; mGlu5Homo sapiensQuisqualateVU0424465-3.52024-11-06doi.org/10.1038/s41467-024-55439-9
8X0FCAminoacidMetabotropic GlutamatemGlu5; mGlu5Homo sapiensQuisqualateVU0424465-3.32024-11-06doi.org/10.1038/s41467-024-55439-9
8JD6CAminoacidMetabotropic GlutamatemGlu4; mGlu4Homo sapiensPhosphoserineVU0364770Gi3/β1/γ23.42023-06-21doi.org/10.1038/s41422-023-00830-2
8JD6 (No Gprot) CAminoacidMetabotropic GlutamatemGlu4; mGlu4Homo sapiensPhosphoserineVU03647703.42023-06-21doi.org/10.1038/s41422-023-00830-2
8WGBCAminoacidMetabotropic GlutamatemGlu4; mGlu2Homo sapiensGlutammateVU0155041Gi3/β1/γ23.72024-10-30doi.org/10.1038/s41467-024-54744-7
8WGB (No Gprot) CAminoacidMetabotropic GlutamatemGlu4; mGlu2Homo sapiensGlutammateVU01550413.72024-10-30doi.org/10.1038/s41467-024-54744-7
7EPFCAminoacidMetabotropic GlutamatemGlu2; mGlu2Homo sapiens-NAM597-2.72021-06-23doi.org/10.1038/s41586-021-03641-w
7EPECAminoacidMetabotropic GlutamatemGlu2; mGlu2Homo sapiens-NAM563-2.52021-06-23doi.org/10.1038/s41586-021-03641-w
8JD0CAminoacidMetabotropic GlutamatemGlu2; mGlu3Homo sapiensGlutamateNAM563-3.32023-06-21doi.org/10.1038/s41422-023-00830-2
6FFICAminoacidMetabotropic GlutamatemGlu5Homo sapiens-MMPEP-2.22018-03-07doi.org/10.1021/acs.jmedchem.7b01722
4OO9CAminoacidMetabotropic GlutamatemGlu5Homo sapiens-Mavoglurant-2.62014-07-02doi.org/10.1038/nature13396
8JD5CAminoacidMetabotropic GlutamatemGlu2; mGlu4Homo sapiensGlutamateJNJ-40411813; ADX88178Gi1/β1/γ23.62023-06-21doi.org/10.1038/s41422-023-00830-2
8JD5 (No Gprot) CAminoacidMetabotropic GlutamatemGlu2; mGlu4Homo sapiensGlutamateJNJ-40411813; ADX881783.62023-06-21doi.org/10.1038/s41422-023-00830-2
7E9GCAminoacidMetabotropic GlutamatemGlu2; mGlu2Homo sapiensEglumetadJNJ-40411813Gi1/β1/γ23.52021-06-23doi.org/10.1038/s41586-021-03495-2
7E9G (No Gprot) CAminoacidMetabotropic GlutamatemGlu2; mGlu2Homo sapiensEglumetadJNJ-404118133.52021-06-23doi.org/10.1038/s41586-021-03495-2
8JD3CAminoacidMetabotropic GlutamatemGlu2; mGlu3Homo sapiensGlutamateJNJ-40411813Gi1/β1/γ23.32023-06-21doi.org/10.1038/s41422-023-00830-2
8JD3 (No Gprot) CAminoacidMetabotropic GlutamatemGlu2; mGlu3Homo sapiensGlutamateJNJ-404118133.32023-06-21doi.org/10.1038/s41422-023-00830-2
5CGCCAminoacidMetabotropic GlutamatemGlu5Homo sapiens-HTL14242-3.12015-08-12doi.org/10.1021/acs.jmedchem.5b00892
5CGDCAminoacidMetabotropic GlutamatemGlu5Homo sapiens-HTL14242-2.62015-08-12doi.org/10.1021/acs.jmedchem.5b00892
4OR2CAminoacidMetabotropic GlutamatemGlu1; mGlu1Homo sapiens-FITM-2.82014-03-19doi.org/10.1126/science.1249489
6FFHCAminoacidMetabotropic GlutamatemGlu5Homo sapiens-Fenobam-2.652018-03-07doi.org/10.1021/acs.jmedchem.7b01722
8T6JCAminoacidMetabotropic GlutamatemGlu5; mGlu5Homo sapiens-CDPPB-3.52023-10-11doi.org/10.1101/2023.08.29.555158
8TAOCAminoacidMetabotropic GlutamatemGlu5; mGlu5Homo sapiensQuisqualateCDPPB-2.92023-10-11doi.org/10.1101/2023.08.29.555158
8TQBCAminoacidMetabotropic GlutamatemGlu3; mGlu3Rattus norvegicusCa; PAM VU6023326Ca-3.32024-07-31doi.org/10.1101/2023.08.13.552748
8TR2CAminoacidMetabotropic GlutamatemGlu3; mGlu3Rattus norvegicusCa; LY379268Ca-3.52024-07-31doi.org/10.1101/2023.08.13.552748
7MTRCAminoacidMetabotropic GlutamatemGlu2; mGlu2Homo sapiensGlutamateADX55164-3.32021-07-07doi.org/10.1038/s41586-021-03680-3
7MTSCAminoacidMetabotropic GlutamatemGlu2; mGlu2Homo sapiensGlutamateADX55164Gi1/β1/γ23.22021-07-07doi.org/10.1038/s41586-021-03680-3
7MTS (No Gprot) CAminoacidMetabotropic GlutamatemGlu2; mGlu2Homo sapiensGlutamateADX551643.22021-07-07doi.org/10.1038/s41586-021-03680-3
7P2LCAminoacidMetabotropic GlutamatemGlu5Homo sapiens-4YI-2.542021-09-08doi.org/10.1016/j.celrep.2021.109648
9HC0CAminoacidMetabotropic GlutamatemGlu5Homo sapiens-4YI-2.332025-06-25doi.org/10.1002/pro.70104
7DGDCAminoacidMetabotropic GlutamatemGlu1; mGlu1Homo sapiens---3.962021-09-22doi.org/10.1007/s13238-020-00808-5
7DGECAminoacidMetabotropic GlutamatemGlu1; mGlu1Homo sapiensQuisqualate--3.652021-09-22doi.org/10.1007/s13238-020-00808-5
7EPACAminoacidMetabotropic GlutamatemGlu2; mGlu2Homo sapiens---3.62021-06-23doi.org/10.1038/s41586-021-03641-w
7EPBCAminoacidMetabotropic GlutamatemGlu2; mGlu2Homo sapiensEglumetad--3.12021-06-23doi.org/10.1038/s41586-021-03641-w
7MTQCAminoacidMetabotropic GlutamatemGlu2; mGlu2Homo sapiensLY341495--3.652021-07-07doi.org/10.1038/s41586-021-03680-3
8JCUCAminoacidMetabotropic GlutamatemGlu2; mGlu3Homo sapiensLY341495--2.82023-06-21doi.org/10.1038/s41422-023-00830-2
8JCVCAminoacidMetabotropic GlutamatemGlu2; mGlu3Homo sapiensLY341495--3.42023-06-21doi.org/10.1038/s41422-023-00830-2
8JCWCAminoacidMetabotropic GlutamatemGlu2; mGlu3Homo sapiensLY341495--32023-06-21doi.org/10.1038/s41422-023-00830-2
8JCXCAminoacidMetabotropic GlutamatemGlu2; mGlu3Homo sapiensLY341495--32023-06-21doi.org/10.1038/s41422-023-00830-2
8JCYCAminoacidMetabotropic GlutamatemGlu2; mGlu3Homo sapiensLY341495--2.92023-06-21doi.org/10.1038/s41422-023-00830-2
8JCZCAminoacidMetabotropic GlutamatemGlu2; mGlu3Homo sapiensLY341495--32023-06-21doi.org/10.1038/s41422-023-00830-2
8JD1CAminoacidMetabotropic GlutamatemGlu2; mGlu3Homo sapiensGlutamate--3.72023-06-21doi.org/10.1038/s41422-023-00830-2
8JD2CAminoacidMetabotropic GlutamatemGlu2; mGlu3Homo sapiensGlutamate--2.82023-06-21doi.org/10.1038/s41422-023-00830-2
8JD4CAminoacidMetabotropic GlutamatemGlu2; mGlu4Homo sapiensGlutamate--2.92023-06-21doi.org/10.1038/s41422-023-00830-2
7EPDCAminoacidMetabotropic GlutamatemGlu2, mGlu7Homo sapiens---3.92021-06-23doi.org/10.1038/s41586-021-03641-w
7WI6CAminoacidMetabotropic GlutamatemGlu3; mGlu3Homo sapiensLY341495--3.712022-03-16doi.org/10.1038/s41422-022-00623-z
7WI8CAminoacidMetabotropic GlutamatemGlu3; mGlu3Homo sapiensLY341495--4.172022-03-16doi.org/10.1038/s41422-022-00623-z
7WIHCAminoacidMetabotropic GlutamatemGlu3; mGlu3Homo sapiensLY2794193--3.682022-03-16doi.org/10.1038/s41422-022-00623-z
8TR0CAminoacidMetabotropic GlutamatemGlu3; mGlu3Rattus norvegicusLY341495--3.22024-07-31doi.org/10.1101/2023.08.13.552748
8TRCCAminoacidMetabotropic GlutamatemGlu3; mGlu3Rattus norvegicusLY341495--3.32024-07-31doi.org/10.1101/2023.08.13.552748
8TRDCAminoacidMetabotropic GlutamatemGlu3; mGlu3Rattus norvegicusLY341495--3.42024-07-31doi.org/10.1038/s41467-024-50548-x
9II2CAminoacidMetabotropic GlutamatemGlu3; mGlu3Homo sapiensGlutamate-Arrestin23.72025-03-05doi.org/10.1038/s41589-025-01858-8
9II3CAminoacidMetabotropic GlutamatemGlu3; mGlu3Homo sapiensGlutamate-Arrestin23.92025-03-05doi.org/10.1038/s41589-025-01858-8
8WG9CAminoacidMetabotropic GlutamatemGlu4; mGlu2Homo sapiens(2S)-2-amino-4-phosphonobutanoic acid--4.462024-11-27doi.org/10.1038/s41467-024-54744-7
8WGCCAminoacidMetabotropic GlutamatemGlu4; mGlu2Homo sapiensLY379268--5.952024-11-27doi.org/10.1038/s41467-024-54744-7
8WGDCAminoacidMetabotropic GlutamatemGlu4; mGlu2Homo sapiensWAG; WA6--4.452024-11-27doi.org/10.1038/s41467-024-54744-7
7E9HCAminoacidMetabotropic GlutamatemGlu4; mGlu4Homo sapiensPhosphoserine-Gi3/β1/γ242021-06-23doi.org/10.1038/s41586-021-03495-2
7E9H (No Gprot) CAminoacidMetabotropic GlutamatemGlu4; mGlu4Homo sapiensPhosphoserine-42021-06-23doi.org/10.1038/s41586-021-03495-2
9HC3CAminoacidMetabotropic GlutamatemGlu5Homo sapiens---2.92025-06-25doi.org/10.1002/pro.70104
7FD8CAminoacidMetabotropic GlutamatemGlu5; mGlu5Homo sapiensQuisqualate--3.82021-09-08doi.org/10.1016/j.celrep.2021.109648
7FD9CAminoacidMetabotropic GlutamatemGlu5; mGlu5Homo sapiensLY341495--42021-09-08doi.org/10.1016/j.celrep.2021.109648
6N51CAminoacidMetabotropic GlutamatemGlu5; mGlu5Homo sapiensQuisqualate--42019-01-23doi.org/10.1038/s41586-019-0881-4
6N52CAminoacidMetabotropic GlutamatemGlu5; mGlu5Homo sapiens---42019-01-23doi.org/10.1038/s41586-019-0881-4
8T7HCAminoacidMetabotropic GlutamatemGlu5; mGlu5Homo sapiensQuisqualate--3.32023-10-11doi.org/10.1101/2023.08.29.555158
8T8MCAminoacidMetabotropic GlutamatemGlu5; mGlu5Homo sapiensQuisqualate--32023-10-11doi.org/10.1101/2023.08.29.555158
8X0ECAminoacidMetabotropic GlutamatemGlu5; mGlu5Homo sapiensQuisqualate--3.42024-11-06doi.org/10.1038/s41467-024-55439-9
8X0GCAminoacidMetabotropic GlutamatemGlu5; mGlu5Homo sapiensQuisqualate--32024-11-06doi.org/10.1038/s41467-024-55439-9
8X0HCAminoacidMetabotropic GlutamatemGlu5; mGlu5Homo sapiensQuisqualate--4.12024-11-06doi.org/10.1038/s41467-024-55439-9
7EPCCAminoacidMetabotropic GlutamatemGlu7; mGlu7Homo sapiens---42021-06-23doi.org/10.1038/s41586-021-03641-w
9OMOCAminoacidMetabotropic GlutamatemGlu7; mGlu7Homo sapiens---4.12025-07-09doi.org/10.1073/pnas.2507112122
9OMPCAminoacidMetabotropic GlutamatemGlu7; mGlu7Homo sapiens---4.32025-07-09doi.org/10.1073/pnas.2507112122
8IBUAPeptideMotilinMotilinHomo sapiensErythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ23.512023-04-12doi.org/10.1126/sciadv.ade9020
8IBU (No Gprot) APeptideMotilinMotilinHomo sapiensErythromycin-A-3.512023-04-12doi.org/10.1126/sciadv.ade9020
8IBVAPeptideMotilinMotilinHomo sapiensMotilin-chim(NtGi1-Gs-CtGq)/β1/γ23.192023-04-12doi.org/10.1126/sciadv.ade9020
8IBV (No Gprot) APeptideMotilinMotilinHomo sapiensMotilin-3.192023-04-12doi.org/10.1126/sciadv.ade9020
9JMCAPeptideMotilinMotilinHomo sapiensDS-3801b-chim(Gs-CtGq)/β1/γ22.572025-05-28doi.org/10.1016/j.celrep.2025.115329
9JMC (No Gprot) APeptideMotilinMotilinHomo sapiensDS-3801b-2.572025-05-28doi.org/10.1016/j.celrep.2025.115329
9JMDAPeptideMotilinMotilinHomo sapiensAzithromycin-chim(Gs-CtGq)/β1/γ22.742025-05-28doi.org/10.1016/j.celrep.2025.115329
9JMD (No Gprot) APeptideMotilinMotilinHomo sapiensAzithromycin-2.742025-05-28doi.org/10.1016/j.celrep.2025.115329
7W53APeptideNeuromedin UNMUR1Homo sapiensNeuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ23.22022-04-20doi.org/10.1038/s41467-022-29683-w
7W53 (No Gprot) APeptideNeuromedin UNMUR1Homo sapiensNeuromedin-U-25-3.22022-04-20doi.org/10.1038/s41467-022-29683-w
7W56APeptideNeuromedin UNMUR1Homo sapiensNeuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ22.92022-04-20doi.org/10.1038/s41467-022-29683-w
7W56 (No Gprot) APeptideNeuromedin UNMUR1Homo sapiensNeuromedin-S-2.92022-04-20doi.org/10.1038/s41467-022-29683-w
7W55APeptideNeuromedin UNMUR2Homo sapiensNeuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ22.82022-04-20doi.org/10.1038/s41467-022-29683-w
7W55 (No Gprot) APeptideNeuromedin UNMUR2Homo sapiensNeuromedin-U-25-2.82022-04-20doi.org/10.1038/s41467-022-29683-w
7W57APeptideNeuromedin UNMUR2Homo sapiensNeuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ23.22022-04-20doi.org/10.1038/s41467-022-29683-w
7W57 (No Gprot) APeptideNeuromedin UNMUR2Homo sapiensNeuromedin-S-3.22022-04-20doi.org/10.1038/s41467-022-29683-w
7XK8APeptideNeuromedin UNMUR2Homo sapiensNeuromedin-U-25-Gi1/β1/γ23.32023-02-22doi.org/10.1038/s41467-022-34814-4
7XK8 (No Gprot) APeptideNeuromedin UNMUR2Homo sapiensNeuromedin-U-25-3.32023-02-22doi.org/10.1038/s41467-022-34814-4
9JFYAPeptideNeuropeptide FFNPFF2Homo sapienshNPSF-Gi1/β1/γ23.212025-04-09doi.org/10.1038/s44319-025-00428-2
9JFY (No Gprot) APeptideNeuropeptide FFNPFF2Homo sapienshNPSF-3.212025-04-09doi.org/10.1038/s44319-025-00428-2
9JG0APeptideNeuropeptide FFNPFF2Homo sapiens---2.912025-04-09doi.org/10.1038/s44319-025-00428-2
7VGXAPeptideNeuropeptide YY1Homo sapiensNeuropeptide-Y-Gi1/β1/γ23.22022-02-23doi.org/10.1038/s41467-022-28510-6
7VGX (No Gprot) APeptideNeuropeptide YY1Homo sapiensNeuropeptide-Y-3.22022-02-23doi.org/10.1038/s41467-022-28510-6
5ZBHAPeptideNeuropeptide YY1Homo sapiensBMS-193885--32018-04-25doi.org/10.1038/s41586-018-0046-x
5ZBQAPeptideNeuropeptide YY1Homo sapiensUR-MK-299--2.72018-04-25doi.org/10.1038/s41586-018-0046-x
7X9AAPeptideNeuropeptide YY1Homo sapiensNeuropeptide-Y-Gi1/β1/γ23.22022-05-18doi.org/10.1126/sciadv.abm1232
7X9A (No Gprot) APeptideNeuropeptide YY1Homo sapiensNeuropeptide-Y-3.22022-05-18doi.org/10.1126/sciadv.abm1232
8K6MAPeptideNeuropeptide YY1Homo sapiensNeuropeptide-Y-Gi2/β1/γ13.32024-07-31doi.org/10.1002/mco2.565
8K6M (No Gprot) APeptideNeuropeptide YY1Homo sapiensNeuropeptide-Y-3.32024-07-31doi.org/10.1002/mco2.565
8K6OAPeptideNeuropeptide YY1Homo sapiensPro-neuropeptide-Y-Gi2/β1/γ13.32024-07-31doi.org/10.1002/mco2.565
8K6O (No Gprot) APeptideNeuropeptide YY1Homo sapiensPro-neuropeptide-Y-3.32024-07-31doi.org/10.1002/mco2.565
7YONAPeptideNeuropeptide YY2Homo sapiensPeptide-YY(3-36)-Gi1/β1/γ22.952023-03-22doi.org/10.1016/j.str.2022.11.010
7YON (No Gprot) APeptideNeuropeptide YY2Homo sapiensPeptide-YY(3-36)-2.952023-03-22doi.org/10.1016/j.str.2022.11.010
7YOOAPeptideNeuropeptide YY2Homo sapiensNeuropeptide-Y-Gi1/β1/γ23.112023-03-22doi.org/10.1016/j.str.2022.11.010
7YOO (No Gprot) APeptideNeuropeptide YY2Homo sapiensNeuropeptide-Y-3.112023-03-22doi.org/10.1016/j.str.2022.11.010
7DDZAPeptideNeuropeptide YY2Homo sapiensJNJ-31020028--2.82021-01-27doi.org/10.1038/s41467-021-21030-9
7X9BAPeptideNeuropeptide YY2Homo sapiensNeuropeptide-Y-Gi1/β1/γ23.42022-05-18doi.org/10.1126/sciadv.abm1232
7X9B (No Gprot) APeptideNeuropeptide YY2Homo sapiensNeuropeptide-Y-3.42022-05-18doi.org/10.1126/sciadv.abm1232
8K6NAPeptideNeuropeptide YY2Homo sapiensPro-neuropeptide-Y-Gi2/β1/γ13.22024-07-31doi.org/10.1002/mco2.565
8K6N (No Gprot) APeptideNeuropeptide YY2Homo sapiensPro-neuropeptide-Y-3.22024-07-31doi.org/10.1002/mco2.565
7X9CAPeptideNeuropeptide YY4Homo sapiensPancreatic Hormone-Gi1/β1/γ232022-05-18doi.org/10.1126/sciadv.abm1232
7X9C (No Gprot) APeptideNeuropeptide YY4Homo sapiensPancreatic Hormone-32022-05-18doi.org/10.1126/sciadv.abm1232
8JPBAPeptideNeurotensinNTS1Homo sapiensNeurotensin-(8-13)SBI-553; GDP; MgGq; GRK23.072023-08-09doi.org/10.1038/s41586-023-06395-9
8JPB (No Gprot) APeptideNeurotensinNTS1Homo sapiensNeurotensin-(8-13)SBI-553; GDP; Mg3.072023-08-09doi.org/10.1038/s41586-023-06395-9
8JPCAPeptideNeurotensinNTS1Homo sapiensNeurotensin-(8-13)SBI-553; GDP; MgGq; GRK23.072023-08-09doi.org/10.1038/s41586-023-06395-9
8JPC (No Gprot) APeptideNeurotensinNTS1Homo sapiensNeurotensin-(8-13)SBI-553; GDP; Mg3.072023-08-09doi.org/10.1038/s41586-023-06395-9
8FN0APeptideNeurotensinNTS1Rattus norvegicusNeurotensin/Neuromedin-NSBI-553chim(NtGi1-Go)/β1/γ22.892023-03-29doi.org/10.1021/acs.biochem.3c00029
8FN0 (No Gprot) APeptideNeurotensinNTS1Rattus norvegicusNeurotensin/Neuromedin-NSBI-5532.892023-03-29doi.org/10.1021/acs.biochem.3c00029
8JPFAPeptideNeurotensinNTS1Homo sapiensNeurotensinSBI-553-3.022023-08-09doi.org/10.1038/s41586-023-06395-9
8ZYTAPeptideNeurotensinNTS1Homo sapiensNeurotensin peptide 8-13SBI-553Arrestin22.652025-04-09doi.org/10.1038/s41422-025-01095-7
8ZYYAPeptideNeurotensinNTS1Homo sapiensNeurotensin peptide 8-13SBI-553Arrestin22.832025-04-09doi.org/10.1038/s41422-025-01095-7
8ZYUAPeptideNeurotensinNTS1Homo sapiensNeurotensin peptide 8-13SBI-553Arrestin22.652025-04-16doi.org/10.1038/s41422-025-01095-7
7UL2APeptideNeurotensinNTS1Homo sapiensSR48692Na-2.42022-06-29doi.org/10.1038/s41594-022-00859-8
8FMZAPeptideNeurotensinNTS1Rattus norvegicusNeurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ22.592023-03-29doi.org/10.1021/acs.biochem.3c00029
8FMZ (No Gprot) APeptideNeurotensinNTS1Rattus norvegicusNeurotensin/Neuromedin-N-2.592023-03-29doi.org/10.1021/acs.biochem.3c00029
8FN1APeptideNeurotensinNTS1Rattus norvegicusNeurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ22.882023-03-29doi.org/10.1021/acs.biochem.3c00029
8FN1 (No Gprot) APeptideNeurotensinNTS1Rattus norvegicusNeurotensin/Neuromedin-N-2.882023-03-29doi.org/10.1021/acs.biochem.3c00029
4GRVAPeptideNeurotensinNTS1Rattus norvegicusNeurotensin-(8-13)--2.82012-10-17doi.org/10.1038/nature11558
4XEEAPeptideNeurotensinNTS1Rattus norvegicusNeurotensin--2.92015-07-29doi.org/10.1038/ncomms8895
4XESAPeptideNeurotensinNTS1Rattus norvegicusNeurotensin--2.62015-07-29doi.org/10.1038/ncomms8895
6PWCAPeptideNeurotensinNTS1Homo sapiensNeurotensin-Arrestin24.92019-12-04doi.org/10.1038/s41422-019-0256-2
6OS9APeptideNeurotensinNTS1Homo sapiensJMV449-Gi1/β1/γ232019-07-10doi.org/10.1038/s41586-019-1337-6
6OS9 (No Gprot) APeptideNeurotensinNTS1Homo sapiensJMV449-32019-07-10doi.org/10.1038/s41586-019-1337-6
6OSAAPeptideNeurotensinNTS1Homo sapiensJMV449-Gi1/β1/γ232019-07-10doi.org/10.1038/s41586-019-1337-6
6OSA (No Gprot) APeptideNeurotensinNTS1Homo sapiensJMV449-32019-07-10doi.org/10.1038/s41586-019-1337-6
6UP7APeptideNeurotensinNTS1Homo sapiensNeurotensin-Arrestin24.22020-02-26doi.org/10.1038/s41586-020-1953-1
7L0PAPeptideNeurotensinNTS1Rattus norvegicusNeurotensin-Gi1/β1/γ14.12021-01-06doi.org/10.1038/s41594-020-00554-6
7L0P (No Gprot) APeptideNeurotensinNTS1Rattus norvegicusNeurotensin-4.12021-01-06doi.org/10.1038/s41594-020-00554-6
7L0QAPeptideNeurotensinNTS1Rattus norvegicusNeurotensin-Gi1/β1/γ14.32021-01-06doi.org/10.1038/s41594-020-00554-6
7L0Q (No Gprot) APeptideNeurotensinNTS1Rattus norvegicusNeurotensin-4.32021-01-06doi.org/10.1038/s41594-020-00554-6
7L0RAPeptideNeurotensinNTS1Rattus norvegicusNeurotensin-Gi1/β1/γ14.22021-01-06doi.org/10.1038/s41594-020-00554-6
7L0R (No Gprot) APeptideNeurotensinNTS1Rattus norvegicusNeurotensin-4.22021-01-06doi.org/10.1038/s41594-020-00554-6
7L0SAPeptideNeurotensinNTS1Rattus norvegicusNeurotensin-Gi1/β1/γ14.52021-01-06doi.org/10.1038/s41594-020-00554-6
7L0S (No Gprot) APeptideNeurotensinNTS1Rattus norvegicusNeurotensin-4.52021-01-06doi.org/10.1038/s41594-020-00554-6
5T04APeptideNeurotensinNTS1Rattus norvegicusNeurotensin--3.32016-12-21doi.org/10.1038/srep38564
3ZEVAPeptideNeurotensinNTS1Rattus norvegicusNeurotensin--32014-01-29doi.org/10.1073/pnas.1317903111
4BUOAPeptideNeurotensinNTS1Rattus norvegicusNeurotensin--2.752014-01-29doi.org/10.1073/pnas.1317903111
4BV0APeptideNeurotensinNTS1Rattus norvegicusNeurotensin--3.12014-01-29doi.org/10.1073/pnas.1317903111
4BWBAPeptideNeurotensinNTS1Rattus norvegicusNeurotensin--3.572014-01-29doi.org/10.1073/pnas.1317903111
6YVRAPeptideNeurotensinNTS1Rattus norvegicusNTS8-13--2.462021-02-10doi.org/10.1126/sciadv.abe5504
6Z4QAPeptideNeurotensinNTS1Rattus norvegicusSR142948A--2.922021-02-10doi.org/10.1126/sciadv.abe5504
6Z4SAPeptideNeurotensinNTS1Rattus norvegicusSR48692--2.712021-02-10doi.org/10.1126/sciadv.abe5504
6Z4VAPeptideNeurotensinNTS1Rattus norvegicusNTS8-13--2.62021-02-10doi.org/10.1126/sciadv.abe5504
6Z66APeptideNeurotensinNTS1Rattus norvegicus---3.192021-02-10doi.org/10.1126/sciadv.abe5504
6Z8NAPeptideNeurotensinNTS1Rattus norvegicusSRI-9829--2.82021-02-10doi.org/10.1126/sciadv.abe5504
6ZA8APeptideNeurotensinNTS1Rattus norvegicusRTI-3a--2.722021-02-10doi.org/10.1126/sciadv.abe5504
6ZINAPeptideNeurotensinNTS1Rattus norvegicusSR48692--2.642021-02-10doi.org/10.1126/sciadv.abe5504
9M0DAPeptideNeurotensinNTS1Homo sapiens--Arrestin23.412025-04-09doi.org/10.1038/s41422-025-01095-7
8UXYO2Odorant receptorsOdorant family 1consOR1Homo sapiensL-menthol-Gs/β1/γ23.32024-10-30doi.org/10.1038/s41586-024-08126-0
8UXY (No Gprot) O2Odorant receptorsOdorant family 1consOR1Homo sapiensL-menthol-3.32024-10-30doi.org/10.1038/s41586-024-08126-0
8UY0O2Odorant receptorsOdorant family 2consOR2Homo sapiensS-carvone-Gs/β1/γ23.22024-10-30doi.org/10.1038/s41586-024-08126-0
8UY0 (No Gprot) O2Odorant receptorsOdorant family 2consOR2Homo sapiensS-carvone-3.22024-10-30doi.org/10.1038/s41586-024-08126-0
8UYQO2Odorant receptorsOdorant family 4consOR4Homo sapiens2-methylthiazoline-Gs/β1/γ23.52024-10-30doi.org/10.1038/s41586-024-08126-0
8UYQ (No Gprot) O2Odorant receptorsOdorant family 4consOR4Homo sapiens2-methylthiazoline-3.52024-10-30doi.org/10.1038/s41586-024-08126-0
8UXVO1Odorant receptorsOdorant family 51consOR51Homo sapiens--Gs/β1/γ23.22024-10-30doi.org/10.1038/s41586-024-08126-0
8UXV (No Gprot) O1Odorant receptorsOdorant family 51consOR51Homo sapiens--3.22024-10-30doi.org/10.1038/s41586-024-08126-0
8F76O1Odorant receptorsOdorant family 51OR51E2Homo sapiensPropanoic acid-Gs/β1/γ23.12023-03-22doi.org/10.1038/s41586-023-05798-y
8F76 (No Gprot) O1Odorant receptorsOdorant family 51OR51E2Homo sapiensPropanoic acid-3.12023-03-22doi.org/10.1038/s41586-023-05798-y
8HTIO1Odorant receptorsOdorant family 52OR52CHomo sapiensOcatnoic acid-Gs/β1/γ22.972023-12-20doi.org/10.1038/s41467-023-43983-9
8HTI (No Gprot) O1Odorant receptorsOdorant family 52OR52CHomo sapiensOcatnoic acid-2.972023-12-20doi.org/10.1038/s41467-023-43983-9
8J46O1Odorant receptorsOdorant family 52OR52CHomo sapiens---3.662023-12-20doi.org/10.1038/s41467-023-43983-9
8W77O1Odorant receptorsOdorant family 52OR52CHomo sapiens---3.612023-12-20doi.org/10.1038/s41467-023-43983-9
9BJKAPeptideOpioidμMus musculusNaloxoneNAM-3.262024-07-17doi.org/10.1038/s41586-024-07587-7
4N6HAPeptideOpioidδHomo sapiensNaltrindoleNa-1.82013-12-25doi.org/10.1038/nature12944
4RWDAPeptideOpioidδHomo sapiensDIPP-NH2Na-2.72015-01-14doi.org/10.1038/nsmb.2965
8K9LAPeptideOpioidμHomo sapiensDamgoBMS-986122Gi3/β1/γ13.052024-05-29doi.org/10.1038/s41467-024-47792-6
8K9L (No Gprot) APeptideOpioidμHomo sapiensDamgoBMS-9861223.052024-05-29doi.org/10.1038/s41467-024-47792-6
8F7SAPeptideOpioidδHomo sapiensDeltorphin-Gi1/β1/γ232022-12-14doi.org/10.1016/j.cell.2022.12.026
8F7S (No Gprot) APeptideOpioidδHomo sapiensDeltorphin-32022-12-14doi.org/10.1016/j.cell.2022.12.026
4EJ4APeptideOpioidδMus musculusNaltrindole--3.42012-05-16doi.org/10.1038/nature11111
4RWAAPeptideOpioidδHomo sapiensDIPP-NH2--3.282015-01-14doi.org/10.1038/nsmb.2965
6PT2APeptideOpioidδHomo sapiensKGCHM07--2.82019-12-11doi.org/10.1126/sciadv.aax9115
6PT3APeptideOpioidδHomo sapiensDPI-287--3.32019-12-11doi.org/10.1126/sciadv.aax9115
8Y45APeptideOpioidδHomo sapiensADL5859-Gi2/β1/γ23.452024-11-27doi.org/10.1038/s41467-024-52601-1
8Y45 (No Gprot) APeptideOpioidδHomo sapiensADL5859-3.452024-11-27doi.org/10.1038/s41467-024-52601-1
9CGJAPeptideOpioidδHomo sapiensC6-Quino-Gi1/β1/γ22.82025-04-02doi.org/10.1038/s41467-025-57734-5
9CGJ (No Gprot) APeptideOpioidδHomo sapiensC6-Quino-2.82025-04-02doi.org/10.1038/s41467-025-57734-5
9CGKAPeptideOpioidδHomo sapiensC5-Quino-Gi1/β1/γ22.622025-04-02doi.org/10.1038/s41467-025-57734-5
9CGK (No Gprot) APeptideOpioidδHomo sapiensC5-Quino-2.622025-04-02doi.org/10.1038/s41467-025-57734-5
6B73APeptideOpioidκHomo sapiensMP1104--3.12018-01-17doi.org/10.1016/j.cell.2017.12.011
8F7WAPeptideOpioidκHomo sapiensDynorphin-Gi1/β1/γ23.192022-12-14doi.org/10.1016/j.cell.2022.12.026
8F7W (No Gprot) APeptideOpioidκHomo sapiensDynorphin-3.192022-12-14doi.org/10.1016/j.cell.2022.12.026
4DJHAPeptideOpioidκHomo sapiensJDTic--2.92012-03-21doi.org/10.1038/nature10939
6VI4APeptideOpioidκHomo sapiensJDTic--3.32020-03-18doi.org/10.1038/s41467-020-14889-7
7YITAPeptideOpioidκHomo sapiensNalfurafine--3.32023-04-12doi.org/10.1038/s41467-023-37041-7
8FEGAPeptideOpioidκHomo sapiens(DNCP)-β-Naloxamine-Gi1/β1/γ22.542023-12-06doi.org/10.1038/s41467-023-43718-w
8FEG (No Gprot) APeptideOpioidκHomo sapiens(DNCP)-β-Naloxamine-2.542023-12-06doi.org/10.1038/s41467-023-43718-w
8DZPAPeptideOpioidκHomo sapiensmomSalB-Gi1/β1/γ22.712023-05-03doi.org/10.1038/s41586-023-06030-7
8DZP (No Gprot) APeptideOpioidκHomo sapiensmomSalB-2.712023-05-03doi.org/10.1038/s41586-023-06030-7
8DZQAPeptideOpioidκHomo sapiensmomSalB-Go/β1/γ22.822023-05-03doi.org/10.1038/s41586-023-06030-7
8DZQ (No Gprot) APeptideOpioidκHomo sapiensmomSalB-2.822023-05-03doi.org/10.1038/s41586-023-06030-7
8DZRAPeptideOpioidκHomo sapiensGR89,696-chim(NtGi2-Gt3)/β1/γ22.612023-05-03doi.org/10.1038/s41586-023-06030-7
8DZR (No Gprot) APeptideOpioidκHomo sapiensGR89,696-2.612023-05-03doi.org/10.1038/s41586-023-06030-7
8DZSAPeptideOpioidκHomo sapiensGR89,696-chim(NtGi2-Gz)/β1/γ22.652023-05-03doi.org/10.1038/s41586-023-06030-7
8DZS (No Gprot) APeptideOpioidκHomo sapiensGR89,696-2.652023-05-03doi.org/10.1038/s41586-023-06030-7
7Y1FAPeptideOpioidκHomo sapiensDynorphin-Gi1/β1/γ23.32023-05-24doi.org/10.1093/procel/pwac033
7Y1F (No Gprot) APeptideOpioidκHomo sapiensDynorphin-3.32023-05-24doi.org/10.1093/procel/pwac033
9MQKAPeptideOpioidκHomo sapiensIsoquinuclidine--3.182025-02-12doi.org/10.1101/2025.01.09.632033
9MQLAPeptideOpioidκHomo sapiensIsoquinuclidine--2.962025-02-12doi.org/10.1101/2025.01.09.632033
8VVEAPeptideOpioidκHomo sapiensnorBNI-Gi1/β1/γ23.32025-01-15doi.org/10.1038/s41589-024-01812-0
8VVE (No Gprot) APeptideOpioidκHomo sapiensnorBNI-3.32025-01-15doi.org/10.1038/s41589-024-01812-0
8VVFAPeptideOpioidκHomo sapiensJDTic-Gi1/β1/γ232025-01-15doi.org/10.1038/s41589-024-01812-0
8VVF (No Gprot) APeptideOpioidκHomo sapiensJDTic-32025-01-15doi.org/10.1038/s41589-024-01812-0
8VVGAPeptideOpioidκHomo sapiensGB18-Gi1/β1/γ23.32025-01-15doi.org/10.1038/s41589-024-01812-0
8VVG (No Gprot) APeptideOpioidκHomo sapiensGB18-3.32025-01-15doi.org/10.1038/s41589-024-01812-0
9D61APeptideOpioidκHomo sapiensJDTic-Gi1/β1/γ23.582025-01-15doi.org/10.1038/s41589-024-01812-0
9D61 (No Gprot) APeptideOpioidκHomo sapiensJDTic-3.582025-01-15doi.org/10.1038/s41589-024-01812-0
7SBFAPeptideOpioidμMus musculusPZM21-Gi1/β1/γ22.92022-04-20doi.org/10.1002/anie.202200269
7SBF (No Gprot) APeptideOpioidμMus musculusPZM21-2.92022-04-20doi.org/10.1002/anie.202200269
7SCGAPeptideOpioidμMus musculusFH210-Gi1/β1/γ232022-04-20doi.org/10.1002/anie.202200269
7SCG (No Gprot) APeptideOpioidμMus musculusFH210-32022-04-20doi.org/10.1002/anie.202200269
8EF5APeptideOpioidμHomo sapiensFentanyl-Gi1/β1/γ23.32022-11-09doi.org/10.1016/j.cell.2022.09.041
8EF5 (No Gprot) APeptideOpioidμHomo sapiensFentanyl-3.32022-11-09doi.org/10.1016/j.cell.2022.09.041
8EF6APeptideOpioidμHomo sapiensMorphine-Gi1/β1/γ23.22022-11-09doi.org/10.1016/j.cell.2022.09.041
8EF6 (No Gprot) APeptideOpioidμHomo sapiensMorphine-3.22022-11-09doi.org/10.1016/j.cell.2022.09.041
8EFBAPeptideOpioidμHomo sapiensOliceridine-Gi1/β1/γ23.22022-11-09doi.org/10.1016/j.cell.2022.09.041
8EFB (No Gprot) APeptideOpioidμHomo sapiensOliceridine-3.22022-11-09doi.org/10.1016/j.cell.2022.09.041
8EFLAPeptideOpioidμHomo sapiensSR17018-Gi1/β1/γ23.22022-11-09doi.org/10.1016/j.cell.2022.09.041
8EFL (No Gprot) APeptideOpioidμHomo sapiensSR17018-3.22022-11-09doi.org/10.1016/j.cell.2022.09.041
8EFOAPeptideOpioidμHomo sapiensPZM21-Gi1/β1/γ22.82022-11-09doi.org/10.1016/j.cell.2022.09.041
8EFO (No Gprot) APeptideOpioidμHomo sapiensPZM21-2.82022-11-09doi.org/10.1016/j.cell.2022.09.041
8EFQAPeptideOpioidμHomo sapiensDamgo-Gi1/β1/γ23.32022-11-09doi.org/10.1016/j.cell.2022.09.041
8EFQ (No Gprot) APeptideOpioidμHomo sapiensDamgo-3.32022-11-09doi.org/10.1016/j.cell.2022.09.041
8F7QAPeptideOpioidμHomo sapiensβ-Endorphin-Gi1/β1/γ23.222022-12-14doi.org/10.1016/j.cell.2022.12.026
8F7Q (No Gprot) APeptideOpioidμHomo sapiensβ-Endorphin-3.222022-12-14doi.org/10.1016/j.cell.2022.12.026
8F7RAPeptideOpioidμHomo sapiensEndomorphin-Gi1/β1/γ23.282022-12-14doi.org/10.1016/j.cell.2022.12.026
8F7R (No Gprot) APeptideOpioidμHomo sapiensEndomorphin-3.282022-12-14doi.org/10.1016/j.cell.2022.12.026
9BQJAPeptideOpioidμMus musculusRO76-Gi1/β1/γ23.32024-09-11doi.org/10.1021/acscentsci.4c00525
9BQJ (No Gprot) APeptideOpioidμMus musculusRO76-3.32024-09-11doi.org/10.1021/acscentsci.4c00525
4DKLAPeptideOpioidμMus musculusβ-Funaltrexamine--2.82012-03-21doi.org/10.1038/nature10954
5C1MAPeptideOpioidμMus musculusBU72--2.072015-08-05doi.org/10.1038/nature14886
8K9KAPeptideOpioidμHomo sapiensDamgo-Gi3/β1/γ12.982024-05-29doi.org/10.1038/s41467-024-47792-6
8K9K (No Gprot) APeptideOpioidμHomo sapiensDamgo-2.982024-05-29doi.org/10.1038/s41467-024-47792-6
6DDEAPeptideOpioidμMus musculusDamgo-Gi1/β1/γ23.52018-06-13doi.org/10.1038/s41586-018-0219-7
6DDE (No Gprot) APeptideOpioidμMus musculusDamgo-3.52018-06-13doi.org/10.1038/s41586-018-0219-7
6DDFAPeptideOpioidμMus musculusDamgo-Gi1/β1/γ23.52018-06-13doi.org/10.1038/s41586-018-0219-7
6DDF (No Gprot) APeptideOpioidμMus musculusDamgo-3.52018-06-13doi.org/10.1038/s41586-018-0219-7
7U2LAPeptideOpioidμMus musculusPubChem 163201242-Gi1/β1/γ23.22022-05-04doi.org/10.1038/s41586-022-05588-y
7U2L (No Gprot) APeptideOpioidμMus musculusPubChem 163201242-3.22022-05-04doi.org/10.1038/s41586-022-05588-y
7U2KAPeptideOpioidμMus musculusC6-guano-Gi1/β1/γ23.32022-12-07doi.org/10.1038/s41586-022-05588-y
7U2K (No Gprot) APeptideOpioidμMus musculusC6-guano-3.32022-12-07doi.org/10.1038/s41586-022-05588-y
7T2GAPeptideOpioidμMus musculusMitragynine Pseudoindoxyl-Gi1/β1/γ22.52022-12-07doi.org/10.1038/s41589-022-01208-y
7T2G (No Gprot) APeptideOpioidμMus musculusMitragynine Pseudoindoxyl-2.52022-12-07doi.org/10.1038/s41589-022-01208-y
7T2HAPeptideOpioidμMus musculusLofentanil-Gi1/β1/γ22.52022-12-07doi.org/10.1038/s41589-022-01208-y
7T2H (No Gprot) APeptideOpioidμMus musculusLofentanil-2.52022-12-07doi.org/10.1038/s41589-022-01208-y
7UL4APeptideOpioidμMus musculusAlvimopan--2.82022-06-29doi.org/10.1038/s41594-022-00859-8
8QOTAPeptideOpioidμMus musculusNanobody-E--3.22023-12-27doi.org/10.1101/2023.12.06.570395
9MQHAPeptideOpioidμHomo sapiens---3.92025-02-12doi.org/10.1101/2025.01.09.632033
9MQIAPeptideOpioidμHomo sapiensIsoquinuclidine--3.32025-02-12doi.org/10.1101/2025.01.09.632033
9MQJAPeptideOpioidμHomo sapiensIsoquinuclidine--3.232025-02-12doi.org/10.1101/2025.01.09.632033
8E0GAPeptideOpioidμMus musculusBU72--2.12023-10-18doi.org/10.1186/s12915-023-01689-w
8F7XAPeptideOpioidNOPHomo sapiensNociceptin-Gi1/β1/γ23.282022-12-14doi.org/10.1016/j.cell.2022.12.026
8F7X (No Gprot) APeptideOpioidNOPHomo sapiensNociceptin-3.282022-12-14doi.org/10.1016/j.cell.2022.12.026
5DHGAPeptideOpioidNOPHomo sapiensC-35--32015-10-21doi.org/10.1016/j.str.2015.07.024
5DHHAPeptideOpioidNOPHomo sapiensSB-612111--32015-10-21doi.org/10.1016/j.str.2015.07.024
4EA3APeptideOpioidNOPHomo sapiensPubChem 10296561--3.012012-04-25doi.org/10.1038/nature11085
8P13ASensoryOpsinRhodopsinBos taurus--Gi1/β1/γT15.22024-11-20To be published
8P13 (No Gprot) ASensoryOpsinRhodopsinBos taurus--5.22024-11-20To be published
8P15ASensoryOpsinRhodopsinBos taurus--Gi1/β1/γT15.92024-11-20To be published
8P15 (No Gprot) ASensoryOpsinRhodopsinBos taurus--5.92024-11-20To be published
6FKDASensoryOpsinsRhodopsinBos taurus-PubChem 137349183-2.492018-04-04doi.org/10.1073/pnas.1718084115
6FKCASensoryOpsinsRhodopsinBos taurus-PubChem 132473039-2.462018-04-04doi.org/10.1073/pnas.1718084115
6FKBASensoryOpsinsRhodopsinBos taurus-PubChem 132473038-3.032018-04-04doi.org/10.1073/pnas.1718084115
6FKAASensoryOpsinsRhodopsinBos taurus-PubChem 132473037-2.72018-04-04doi.org/10.1073/pnas.1718084115
6FK9ASensoryOpsinsRhodopsinBos taurus-PubChem 132473036-2.632018-04-04doi.org/10.1073/pnas.1718084115
6FK8ASensoryOpsinsRhodopsinBos taurus-PubChem 132473035-2.872018-04-04doi.org/10.1073/pnas.1718084115
6FK7ASensoryOpsinsRhodopsinBos taurus-PubChem 132473034-2.622018-04-04doi.org/10.1073/pnas.1718084115
6FK6ASensoryOpsinsRhodopsinBos taurus-PubChem 132473033-2.362018-04-04doi.org/10.1073/pnas.1718084115
6PH7ASensoryOpsinsRhodopsinBos taurus-NerolGt(CT)2.92020-07-01To be published
6PH7 (No Gprot) ASensoryOpsinsRhodopsinBos taurus-Nerol2.92020-07-01To be published
6PGSASensoryOpsinsRhodopsinBos taurus-GeraniolGt(CT)2.92020-07-01To be published
6PGS (No Gprot) ASensoryOpsinsRhodopsinBos taurus-Geraniol2.92020-07-01To be published
6PELASensoryOpsinsRhodopsinBos taurus-CitronellolGt(CT)3.192020-06-24To be published
6PEL (No Gprot) ASensoryOpsinsRhodopsinBos taurus-Citronellol3.192020-06-24To be published
8Y02ASensoryOpsinsOPN1SWHomo sapiensRetinal-Gi1/β1/γ22.612025-06-11To be published
8Y02 (No Gprot) ASensoryOpsinsOPN1SWHomo sapiensRetinal-2.612025-06-11To be published
8IU2ASensoryOpsinsOpsin1LWHomo sapiensRetinal-Gi1/β1/γ23.352024-03-27To be published
8IU2 (No Gprot) ASensoryOpsinsOpsin1LWHomo sapiensRetinal-3.352024-03-27To be published
8Y01ASensoryOpsinsOpsin1MWHomo sapiensRetinal-Gi1/β1/γ22.482025-02-12To be published
8Y01 (No Gprot) ASensoryOpsinsOpsin1MWHomo sapiensRetinal-2.482025-02-12To be published
2G87ASensoryOpsinsRhodopsinBos taurusAll-trans-Retinal--2.62006-09-02doi.org/10.1002/anie.200600595
4J4QASensoryOpsinsRhodopsinBos taurusOctyl β-D-Glucopyranoside-Gt(CT)2.652013-10-30doi.org/10.1002/anie.201302374
4J4Q (No Gprot) ASensoryOpsinsRhodopsinBos taurusOctyl β-D-Glucopyranoside-2.652013-10-30doi.org/10.1002/anie.201302374
3OAXASensoryOpsinsRhodopsinBos taurus11-cis-Retinal--2.62011-01-19doi.org/10.1016/j.bpj.2010.08.003
5W0PASensoryOpsinsRhodopsinHomo sapiens--Arrestin13.012017-08-09doi.org/10.1016/j.cell.2017.07.002
1U19ASensoryOpsinsRhodopsinBos taurus11-cis-Retinal--2.22004-10-12doi.org/10.1016/j.jmb.2004.07.044
1GZMASensoryOpsinsRhodopsinBos taurus11-cis-Retinal--2.652003-11-20doi.org/10.1016/j.jmb.2004.08.090
2J4YASensoryOpsinsRhodopsinBos taurus11-cis-Retinal--3.42007-09-25doi.org/10.1016/j.jmb.2007.03.007
3AYMASensoryOpsinsRhodopsinTodarodes pacificusAll-trans-Retinal--2.82011-08-17doi.org/10.1016/j.jmb.2011.08.044
3AYNASensoryOpsinsRhodopsinTodarodes pacificus9-cis-Retinal--2.72011-08-17doi.org/10.1016/j.jmb.2011.08.044
6OY9ASensoryOpsinsRhodopsinBos taurusAll-trans-Retinal-Gt/β1/γ13.92019-07-24doi.org/10.1016/j.molcel.2019.06.007
6OY9 (No Gprot) ASensoryOpsinsRhodopsinBos taurusAll-trans-Retinal-3.92019-07-24doi.org/10.1016/j.molcel.2019.06.007
6OYAASensoryOpsinsRhodopsinBos taurusAll-trans-Retinal-Gt/β1/γ13.32019-07-24doi.org/10.1016/j.molcel.2019.06.007
6OYA (No Gprot) ASensoryOpsinsRhodopsinBos taurusAll-trans-Retinal-3.32019-07-24doi.org/10.1016/j.molcel.2019.06.007
4X1HASensoryOpsinsRhodopsinBos taurusNonyl-β-D-Glucopyranoside-Gt(CT)2.292015-11-04doi.org/10.1016/j.str.2015.09.015
4X1H (No Gprot) ASensoryOpsinsRhodopsinBos taurusNonyl-β-D-Glucopyranoside-2.292015-11-04doi.org/10.1016/j.str.2015.09.015
1HZXASensoryOpsinsRhodopsinBos taurus11-cis-Retinal--2.82001-07-04doi.org/10.1021/bi0155091
4BEZASensoryOpsinsRhodopsinBos taurus---3.32013-04-24doi.org/10.1038/embor.2013.44
4BEYASensoryOpsinsRhodopsinBos taurus--Gt(CT)2.92013-05-08doi.org/10.1038/embor.2013.44
4BEY (No Gprot) ASensoryOpsinsRhodopsinBos taurus--2.92013-05-08doi.org/10.1038/embor.2013.44
2Z73ASensoryOpsinsRhodopsinTodarodes pacificus11-cis-Retinal--2.52008-05-13doi.org/10.1038/nature06925
3CAPASensoryOpsinsRhodopsinBos taurus---2.92008-06-24doi.org/10.1038/nature07063
3DQBASensoryOpsinsRhodopsinBos taurus--Gt(CT)3.22008-09-23doi.org/10.1038/nature07330
3DQB (No Gprot) ASensoryOpsinsRhodopsinBos taurus--3.22008-09-23doi.org/10.1038/nature07330
3PQRASensoryOpsinsRhodopsinBos taurusAll-trans-Retinal-Gt(CT)2.852011-03-09doi.org/10.1038/nature09789
3PQR (No Gprot) ASensoryOpsinsRhodopsinBos taurusAll-trans-Retinal-2.852011-03-09doi.org/10.1038/nature09789
3PXOASensoryOpsinsRhodopsinBos taurusAll-trans-Retinal--32011-03-09doi.org/10.1038/nature09789
2X72ASensoryOpsinsRhodopsinBos taurusAll-trans-Retinal-Gt(CT)32011-03-16doi.org/10.1038/nature09795
2X72 (No Gprot) ASensoryOpsinsRhodopsinBos taurusAll-trans-Retinal-32011-03-16doi.org/10.1038/nature09795
4ZWJASensoryOpsinsRhodopsinHomo sapiens--Arrestin13.32015-07-29doi.org/10.1038/nature14656
4PXFASensoryOpsinsRhodopsinBos taurusOctyl-β-D-Glucopyranoside-Arrestin1 Finger Loop2.752014-09-17doi.org/10.1038/ncomms5801
5WKTASensoryOpsinsRhodopsinBos taurusOctyl-β-D-Glucopyranoside-Gt(CT)3.22017-12-13doi.org/10.1038/nprot.2017.135
5WKT (No Gprot) ASensoryOpsinsRhodopsinBos taurusOctyl-β-D-Glucopyranoside-3.22017-12-13doi.org/10.1038/nprot.2017.135
8FCZASensoryOpsinsRhodopsinBos taurus11-cis-Retinal--3.72023-08-30doi.org/10.1038/s41467-023-40911-9
8FD0ASensoryOpsinsRhodopsinBos taurus---3.712023-08-30doi.org/10.1038/s41467-023-40911-9
8FD1ASensoryOpsinsRhodopsinBos taurus---4.252023-08-30doi.org/10.1038/s41467-023-40911-9
9EPPASensoryOpsinsRhodopsinHasarius adansoni11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ24.062024-10-23doi.org/10.1038/s41467-024-53208-2
9EPP (No Gprot) ASensoryOpsinsRhodopsinHasarius adansoni11,20-Ethanoretinal-4.062024-10-23doi.org/10.1038/s41467-024-53208-2
9EPQASensoryOpsinsRhodopsinHasarius adansoni11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ24.152024-10-23doi.org/10.1038/s41467-024-53208-2
9EPQ (No Gprot) ASensoryOpsinsRhodopsinHasarius adansoni11,20-Ethanoretinal-4.152024-10-23doi.org/10.1038/s41467-024-53208-2
6CMOASensoryOpsinsRhodopsinHomo sapiens--Gi1/β1/γ24.52018-06-20doi.org/10.1038/s41586-018-0215-y
6CMO (No Gprot) ASensoryOpsinsRhodopsinHomo sapiens--4.52018-06-20doi.org/10.1038/s41586-018-0215-y
7MT8ASensoryOpsinsRhodopsinBos taurusAll-trans-Retinal-GRK15.82021-07-07doi.org/10.1038/s41586-021-03721-x
7MT9ASensoryOpsinsRhodopsinBos taurusAll-trans-Retinal-GRK172021-07-07doi.org/10.1038/s41586-021-03721-x
7MTAASensoryOpsinsRhodopsinBos taurusAll-trans-Retinal-GRK14.12021-07-07doi.org/10.1038/s41586-021-03721-x
7MTBASensoryOpsinsRhodopsinBos taurusAll-trans-Retinal-GRK142021-07-07doi.org/10.1038/s41586-021-03721-x
7ZBCASensoryOpsinsRhodopsinBos taurus11-cis-Retinal--1.82023-03-29doi.org/10.1038/s41586-023-05863-6
7ZBEASensoryOpsinsRhodopsinBos taurus11-cis-Retinal--1.82023-03-29doi.org/10.1038/s41586-023-05863-6
8A6CASensoryOpsinsRhodopsinBos taurusAll-trans-Retinal--1.82023-03-29doi.org/10.1038/s41586-023-05863-6
8A6DASensoryOpsinsRhodopsinBos taurusAll-trans-Retinal--1.82023-03-29doi.org/10.1038/s41586-023-05863-6
8A6EASensoryOpsinsRhodopsinBos taurusAll-trans-Retinal--1.82023-03-29doi.org/10.1038/s41586-023-05863-6
5DGYASensoryOpsinsRhodopsinHomo sapiens--Arrestin17.72016-03-23doi.org/10.1038/sdata.2016.21
2HPYASensoryOpsinsRhodopsinBos taurusAll-trans-Retinal--2.82006-08-22doi.org/10.1073/pnas.0601765103
2I35ASensoryOpsinsRhodopsinBos taurus11-cis-Retinal--3.82006-10-17doi.org/10.1073/pnas.0608022103
2I36ASensoryOpsinsRhodopsinBos taurus---4.12006-10-17doi.org/10.1073/pnas.0608022103
2I37ASensoryOpsinsRhodopsinBos taurus---4.152006-10-17doi.org/10.1073/pnas.0608022103
1L9HASensoryOpsinsRhodopsinBos taurus11-cis-Retinal--2.62002-05-15doi.org/10.1073/pnas.082666399
4A4MASensoryOpsinsRhodopsinBos taurusAll-trans-Retinal-Gt(CT)3.32012-01-25doi.org/10.1073/pnas.1114089108
4A4M (No Gprot) ASensoryOpsinsRhodopsinBos taurusAll-trans-Retinal-3.32012-01-25doi.org/10.1073/pnas.1114089108
5TE3ASensoryOpsinsRhodopsinBos taurusOctyl-β-D-Glucopyranoside--2.72017-03-15doi.org/10.1073/pnas.1617446114
5TE5ASensoryOpsinsRhodopsinBos taurus20-Methanoretinal--4.012017-03-15doi.org/10.1073/pnas.1617446114
6I9KASensoryOpsinsRhodopsinHasarius adansoni9-cis-Retinal--2.152019-07-03doi.org/10.1073/pnas.1902192116
2ZIYASensoryOpsinsRhodopsinTodarodes pacificus11-cis-Retinal--3.72008-05-06doi.org/10.1074/jbc.C800040200
6OFJASensoryOpsinsRhodopsinBos taurus---4.52019-08-21doi.org/10.1074/jbc.RA119.010089
3C9LASensoryOpsinsRhodopsinBos taurus11-cis-Retinal--2.652008-08-05doi.org/10.1107/S0907444908017162
3C9MASensoryOpsinsRhodopsinBos taurus11-cis-Retinal--3.42008-08-05doi.org/10.1107/S0907444908017162
6FUFASensoryOpsinsRhodopsinBos taurusAll-trans-Retinal-Go3.122018-10-03doi.org/10.1126/sciadv.aat7052
6FUF (No Gprot) ASensoryOpsinsRhodopsinBos taurusAll-trans-Retinal-3.122018-10-03doi.org/10.1126/sciadv.aat7052
1F88ASensoryOpsinsRhodopsinBos taurus11-cis-Retinal--2.82000-08-04doi.org/10.1126/science.289.5480.739
4WW3ASensoryOpsinsRhodopsinTodarodes pacificusAll-trans-Retinal--2.82015-06-17doi.org/10.1371/journal.pone.0126970
5DYSASensoryOpsinsRhodopsinBos taurusAll-trans-Retinal--2.32016-08-10doi.org/10.15252/embr.201642671
5EN0ASensoryOpsinsRhodopsinBos taurusAll-trans-Retinal-Gt(CT)2.812016-08-10doi.org/10.15252/embr.201642671
5EN0 (No Gprot) ASensoryOpsinsRhodopsinBos taurusAll-trans-Retinal-2.812016-08-10doi.org/10.15252/embr.201642671
2PEDASensoryOpsinsRhodopsinBos taurus9-cis-Retinal--2.952007-10-30doi.org/10.1529/biophysj.107.108225
6QNOASensoryOpsinsRhodopsinBos taurusAll-trans-Retinal-Gi1/β1/γ14.382019-07-10doi.org/10.7554/eLife.46041
6QNO (No Gprot) ASensoryOpsinsRhodopsinBos taurusAll-trans-Retinal-4.382019-07-10doi.org/10.7554/eLife.46041
9EPRASensoryOpsinsRhodopsinHasarius adansoniRetinal-Gi1/β1/γ24.92024-10-30doi.org/10.1038/s41467-024-53208-2
9EPR (No Gprot) ASensoryOpsinsRhodopsinHasarius adansoniRetinal-4.92024-10-30doi.org/10.1038/s41467-024-53208-2
6NWEASensoryOpsinsRhodopsinBos taurusOctyl-β-D-Glucopyranoside-Gt(CT)2.712020-02-12To be published
6NWE (No Gprot) ASensoryOpsinsRhodopsinBos taurusOctyl-β-D-Glucopyranoside-2.712020-02-12To be published
8P12ASensoryOpsinsRhodopsinBos taurus--Gi1/β1/γT13.212024-11-20To be published
8P12 (No Gprot) ASensoryOpsinsRhodopsinBos taurus--3.212024-11-20To be published
6TO7APeptideOrexinOX1Homo sapiensSuvorexantNa-2.262020-01-01doi.org/10.1021/acs.jmedchem.9b01787
6TODAPeptideOrexinOX1Homo sapiensEMPANa-2.112020-01-01doi.org/10.1021/acs.jmedchem.9b01787
6TQ4APeptideOrexinOX1Homo sapiensPubChem 16046844Na-2.32020-01-01doi.org/10.1021/acs.jmedchem.9b01787
6TOSAPeptideOrexinOX1Homo sapiensGSK1059865Na-2.132020-01-15doi.org/10.1021/acs.jmedchem.9b01787
6TP3APeptideOrexinOX1Homo sapiensNemorexant--3.042020-01-01doi.org/10.1021/acs.jmedchem.9b01787
6TP4APeptideOrexinOX1Homo sapiensACT-462206--3.012020-01-01doi.org/10.1021/acs.jmedchem.9b01787
6TP6APeptideOrexinOX1Homo sapiensFilorexant--2.342020-01-01doi.org/10.1021/acs.jmedchem.9b01787
6TQ6APeptideOrexinOX1Homo sapiensPubChem 145714283--2.552020-01-01doi.org/10.1021/acs.jmedchem.9b01787
6TQ7APeptideOrexinOX1Homo sapiensSB-334867--2.662020-01-01doi.org/10.1021/acs.jmedchem.9b01787
6TQ9APeptideOrexinOX1Homo sapiensSB-408124--2.652020-01-01doi.org/10.1021/acs.jmedchem.9b01787
6TOTAPeptideOrexinOX1Homo sapiensLemborexant--2.222020-01-15doi.org/10.1021/acs.jmedchem.9b01787
4ZJ8APeptideOrexinOX1Homo sapiensSuvorexant--2.752016-03-09doi.org/10.1038/nsmb.3183
4ZJCAPeptideOrexinOX1Homo sapiensSB-674042--2.832016-03-09doi.org/10.1038/nsmb.3183
6V9SAPeptideOrexinOX1Homo sapiensGTPL11403--3.52020-07-15doi.org/10.1073/pnas.2002704117
5WQCAPeptideOrexinOX2Homo sapiensEMPA--1.962017-11-29doi.org/10.1016/j.str.2017.11.005
5WS3APeptideOrexinOX2Homo sapiensEMPA--2.32017-12-13doi.org/10.1016/j.str.2017.11.005
7XRRAPeptideOrexinOX2Homo sapiensLemborexant--2.892022-11-23doi.org/10.1016/j.str.2022.11.001
6TPGAPeptideOrexinOX2Homo sapiensEMPA--2.742020-01-01doi.org/10.1021/acs.jmedchem.9b01787
6TPJAPeptideOrexinOX2Homo sapiensSuvorexant--2.742020-01-01doi.org/10.1021/acs.jmedchem.9b01787
6TPNAPeptideOrexinOX2Homo sapiensHTL6641--2.612020-01-01doi.org/10.1021/acs.jmedchem.9b01787
4S0VAPeptideOrexinOX2Homo sapiensSuvorexant--2.52015-01-14doi.org/10.1038/nature14035
7L1UAPeptideOrexinOX2Homo sapiensOrexin-chim(NtGi1-Gs-CtGq)/β1/γ23.22021-02-10doi.org/10.1038/s41467-021-21087-6
7L1U (No Gprot) APeptideOrexinOX2Homo sapiensOrexin-3.22021-02-10doi.org/10.1038/s41467-021-21087-6
7L1VAPeptideOrexinOX2Homo sapiensPubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ232021-02-10doi.org/10.1038/s41467-021-21087-6
7L1V (No Gprot) APeptideOrexinOX2Homo sapiensPubChem 155491009-32021-02-10doi.org/10.1038/s41467-021-21087-6
7SQOAPeptideOrexinOX2Homo sapiensTAK-925-Gi1/β1/γ23.172022-05-25doi.org/10.1038/s41467-022-30601-3
7SQO (No Gprot) APeptideOrexinOX2Homo sapiensTAK-925-3.172022-05-25doi.org/10.1038/s41467-022-30601-3
7SR8APeptideOrexinOX2Homo sapiensTAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ23.32022-06-08doi.org/10.1038/s41467-022-30601-3
7SR8 (No Gprot) APeptideOrexinOX2Homo sapiensTAK-925-3.32022-06-08doi.org/10.1038/s41467-022-30601-3
8TB7AOrphanOrphanGPR61Homo sapiens-PubChem 168510218-2.942023-10-04doi.org/10.1038/s41467-023-41646-3
8T1VAOrphanOrphanGPR6Homo sapiensPubChem 118310209Na-2.62024-12-04doi.org/10.1126/scisignal.ado8741
8DWGAOrphanOrphanMRGPRX1Homo sapiensProenkephalin-AML382chim(NtGi2L-Gs-CtGq)/β1/γ22.712022-11-02doi.org/10.1038/s41589-022-01173-6
8DWG (No Gprot) AOrphanOrphanMRGPRX1Homo sapiensProenkephalin-AML3822.712022-11-02doi.org/10.1038/s41589-022-01173-6
9JCPAOrphanOrphanGPR4Homo sapiens-LPCchim(NtGi1-Gs-CtGq)/β1/γ22.552025-07-09doi.org/10.1038/s41421-025-00807-y
9JCP (No Gprot) AOrphanOrphanGPR4Homo sapiens-LPC2.552025-07-09doi.org/10.1038/s41421-025-00807-y
9JCOAOrphanOrphanGPR4Homo sapiens-LPCchim(NtGi1-Gs)/β1/γ22.362025-07-09doi.org/10.1038/s41421-025-00807-y
9JCO (No Gprot) AOrphanOrphanGPR4Homo sapiens-LPC2.362025-07-09doi.org/10.1038/s41421-025-00807-y
9JCQAOrphanOrphanGPR4Homo sapiens-LPCchim(NtGi1-Gs)/β1/γ22.592025-07-09doi.org/10.1038/s41421-025-00807-y
9JCQ (No Gprot) AOrphanOrphanGPR4Homo sapiens-LPC2.592025-07-09doi.org/10.1038/s41421-025-00807-y
7VUIAOrphanOrphanGPR139Homo sapiensJNJ-63533054GTPchim(Gs-CtGq)/β1/γ23.32021-12-29doi.org/10.1038/s41422-021-00591-w
7VUI (No Gprot) AOrphanOrphanGPR139Homo sapiensJNJ-63533054GTP3.32021-12-29doi.org/10.1038/s41422-021-00591-w
7VUJAOrphanOrphanGPR139Homo sapiensJNJ-63533054GDPchim(Gs-CtGq)/β1/γ23.82021-12-29doi.org/10.1038/s41422-021-00591-w
7VUJ (No Gprot) AOrphanOrphanGPR139Homo sapiensJNJ-63533054GDP3.82021-12-29doi.org/10.1038/s41422-021-00591-w
8H8JAOrphanOrphanGPR35Homo sapiensLodoxamideCachim(NtGi1L-G13)/β1/γ23.22023-02-08doi.org/10.1038/s41421-022-00499-8
8H8J (No Gprot) AOrphanOrphanGPR35Homo sapiensLodoxamideCa3.22023-02-08doi.org/10.1038/s41421-022-00499-8
8HMPAOrphanOrphanGPR52Homo sapiens-C17Gs/β1/γ22.772023-06-21doi.org/10.1002/mco2.260
8HMP (No Gprot) AOrphanOrphanGPR52Homo sapiens-C172.772023-06-21doi.org/10.1002/mco2.260
6LI0AOrphanOrphanGPR52Homo sapiens-C17-2.22020-02-26doi.org/10.1038/s41586-020-2019-0
8W8RAOrphanOrphanGPR101Homo sapiens-AA-14chim(NtGi1-Gs)/β1/γ23.32024-01-03doi.org/10.1038/s41589-023-01456-6
8W8R (No Gprot) AOrphanOrphanGPR101Homo sapiens-AA-143.32024-01-03doi.org/10.1038/s41589-023-01456-6
8W8SAOrphanOrphanGPR101Homo sapiens-AA-14-3.32024-01-03doi.org/10.1038/s41589-023-01456-6
7EJXAOrphanOrphanGPR88Homo sapiens-(1R;2R)-2-PCCAGi1/β1/γ22.42022-04-13doi.org/10.1038/s41467-022-30081-5
7EJX (No Gprot) AOrphanOrphanGPR88Homo sapiens-(1R;2R)-2-PCCA2.42022-04-13doi.org/10.1038/s41467-022-30081-5
8W8QAOrphanOrphanGPR101Homo sapiens--Gs/β1/γ22.892024-01-03doi.org/10.1038/s41589-023-01456-6
8W8Q (No Gprot) AOrphanOrphanGPR101Homo sapiens--2.892024-01-03doi.org/10.1038/s41589-023-01456-6
7Y3GAOrphanOrphanGPR12Homo sapiens--Gs/β1/γ22.772023-06-07doi.org/10.1016/j.scib.2022.12.023
7Y3G (No Gprot) AOrphanOrphanGPR12Homo sapiens--2.772023-06-07doi.org/10.1016/j.scib.2022.12.023
8HQEAOrphanOrphanGPR132Homo sapiens--Gi1/β1/γ22.972023-10-11doi.org/10.1038/s42255-023-00899-4
8HQE (No Gprot) AOrphanOrphanGPR132Homo sapiens--2.972023-10-11doi.org/10.1038/s42255-023-00899-4
8HQMAOrphanOrphanGPR132Homo sapiensNPGLY-Gi1/β1/γ22.952023-10-11doi.org/10.1038/s42255-023-00899-4
8HQM (No Gprot) AOrphanOrphanGPR132Homo sapiensNPGLY-2.952023-10-11doi.org/10.1038/s42255-023-00899-4
8HQNAOrphanOrphanGPR132Homo sapiens9-S-HODE-Gi1/β1/γ232023-10-11doi.org/10.1038/s42255-023-00899-4
8HQN (No Gprot) AOrphanOrphanGPR132Homo sapiens9-S-HODE-32023-10-11doi.org/10.1038/s42255-023-00899-4
8HVIAOrphanOrphanGPR132Homo sapiensNOX-6-7-Gi1/β1/γ23.042023-10-11doi.org/10.1038/s42255-023-00899-4
8HVI (No Gprot) AOrphanOrphanGPR132Homo sapiensNOX-6-7-3.042023-10-11doi.org/10.1038/s42255-023-00899-4
7VUGAOrphanOrphanGPR139Homo sapiensJNJ-63533054-Gi1/β1/γ23.22021-12-29doi.org/10.1038/s41422-021-00591-w
7VUG (No Gprot) AOrphanOrphanGPR139Homo sapiensJNJ-63533054-3.22021-12-29doi.org/10.1038/s41422-021-00591-w
7VUHAOrphanOrphanGPR139Homo sapiensJNJ-63533054-chim(Gs-CtGq)/β1/γ23.222021-12-29doi.org/10.1038/s41422-021-00591-w
7VUH (No Gprot) AOrphanOrphanGPR139Homo sapiensJNJ-63533054-3.222021-12-29doi.org/10.1038/s41422-021-00591-w
8ZQEAOrphanOrphanGPR15Homo sapiensGPR15L(C11)-Gi1/β1/γ12.92024-07-10doi.org/10.1038/s41421-024-00698-5
8ZQE (No Gprot) AOrphanOrphanGPR15Homo sapiensGPR15L(C11)-2.92024-07-10doi.org/10.1038/s41421-024-00698-5
8KH4AOrphanOrphanGPR161Homo sapiens--Gs/β1/γ23.12023-10-11doi.org/10.1038/s41467-023-41654-3
8KH4 (No Gprot) AOrphanOrphanGPR161Homo sapiens--3.12023-10-11doi.org/10.1038/s41467-023-41654-3
8SMVAOrphanOrphanGPR161Homo sapiens--Gs/β1/γ22.742024-02-21doi.org/10.1038/s41594-024-01223-8
8SMV (No Gprot) AOrphanOrphanGPR161Homo sapiens--2.742024-02-21doi.org/10.1038/s41594-024-01223-8
7Y89AOrphanOrphanGPR17 (CysLT)Homo sapiens--Gi1/β1/γ23.022022-10-12doi.org/10.1002/mco2.159
7Y89 (No Gprot) AOrphanOrphanGPR17 (CysLT)Homo sapiens--3.022022-10-12doi.org/10.1002/mco2.159
7XV3AOrphanOrphanGPR174Homo sapiensLysophosphatidylserine-chim(NtGi1-Gs)/β1/γ22.762023-02-15doi.org/10.1038/s41467-023-36575-0
7XV3 (No Gprot) AOrphanOrphanGPR174Homo sapiensLysophosphatidylserine-2.762023-02-15doi.org/10.1038/s41467-023-36575-0
8KH5AOrphanOrphanGPR174Homo sapiensLysophosphatidylserine-Gs/β1/γ22.832023-10-11doi.org/10.1038/s41467-023-41654-3
8KH5 (No Gprot) AOrphanOrphanGPR174Homo sapiensLysophosphatidylserine-2.832023-10-11doi.org/10.1038/s41467-023-41654-3
8IZBAOrphanOrphanGPR174Homo sapiensLysophosphatidylserine-Gs/β1/γ23.062023-11-01doi.org/10.1371/journal.pbio.3002387
8IZB (No Gprot) AOrphanOrphanGPR174Homo sapiensLysophosphatidylserine-3.062023-11-01doi.org/10.1371/journal.pbio.3002387
7TUYAOrphanOrphanGPR183Homo sapiensGSK682753A--2.982022-04-13doi.org/10.1016/j.str.2022.04.006
7TUZAOrphanOrphanGPR183Homo sapiens7-α,25-dihydroxycholesterol-Gi1/β1/γ23.122022-04-13doi.org/10.1016/j.str.2022.04.006
7TUZ (No Gprot) AOrphanOrphanGPR183Homo sapiens7-α,25-dihydroxycholesterol-3.122022-04-13doi.org/10.1016/j.str.2022.04.006
8HS2AOrphanOrphanGPR20Homo sapiensFab046--3.082023-03-08doi.org/10.1038/s41421-023-00520-8
8HS3AOrphanOrphanGPR20Homo sapiens--Gi1/β1/γ23.142023-03-08doi.org/10.1038/s41421-023-00520-8
8HS3 (No Gprot) AOrphanOrphanGPR20Homo sapiens--3.142023-03-08doi.org/10.1038/s41421-023-00520-8
8HSCAOrphanOrphanGPR20Homo sapiensFab046-Gi1/β1/γ23.222023-03-08doi.org/10.1038/s41421-023-00520-8
8HSC (No Gprot) AOrphanOrphanGPR20Homo sapiensFab046-3.222023-03-08doi.org/10.1038/s41421-023-00520-8
8HMVAOrphanOrphanGPR21Homo sapiens--Gs/β1/γ22.912023-03-01doi.org/10.1002/mco2.205
8HMV (No Gprot) AOrphanOrphanGPR21Homo sapiens--2.912023-03-01doi.org/10.1002/mco2.205
8HIXAOrphanOrphanGPR21Homo sapiens--Gs/β1/γ23.122023-03-15doi.org/10.1038/s41467-023-35882-w
8HIX (No Gprot) AOrphanOrphanGPR21Homo sapiens--3.122023-03-15doi.org/10.1038/s41467-023-35882-w
8HJ0AOrphanOrphanGPR21Homo sapiens--chim(Gs-CtG15)/β1/γ23.122023-03-15doi.org/10.1038/s41467-023-35882-w
8HJ0 (No Gprot) AOrphanOrphanGPR21Homo sapiens--3.122023-03-15doi.org/10.1038/s41467-023-35882-w
8HJ2AOrphanOrphanGPR21Homo sapiens--chim(Gs-CtG15)/β1/γ23.82023-03-15doi.org/10.1038/s41467-023-35882-w
8HJ2 (No Gprot) AOrphanOrphanGPR21Homo sapiens--3.82023-03-15doi.org/10.1038/s41467-023-35882-w
8HJ1AOrphanOrphanGPR21Homo sapiens--Gs/β1/γ23.272023-12-27doi.org/10.1038/s41467-023-35882-w
8HJ1 (No Gprot) AOrphanOrphanGPR21Homo sapiens--3.272023-12-27doi.org/10.1038/s41467-023-35882-w
8U8FAOrphanOrphanGPR3Homo sapiensPalmitic Acid-Gs/β1/γ23.492024-03-06doi.org/10.1021/acs.biochem.3c00647
8U8F (No Gprot) AOrphanOrphanGPR3Homo sapiensPalmitic Acid-3.492024-03-06doi.org/10.1021/acs.biochem.3c00647
8WW2AOrphanOrphanGPR3Homo sapiens--chim(NtGi1-Gs)/β1/γ22.792024-02-14doi.org/10.1038/s41422-024-00932-5
8WW2 (No Gprot) AOrphanOrphanGPR3Homo sapiens--2.792024-02-14doi.org/10.1038/s41422-024-00932-5
9LYBAOrphanOrphanGPR3Homo sapiens--Gs/β1/γ23.162025-04-09doi.org/10.1016/j.celrep.2025.115478
9LYB (No Gprot) AOrphanOrphanGPR3Homo sapiens--3.162025-04-09doi.org/10.1016/j.celrep.2025.115478
9LYCAOrphanOrphanGPR3Homo sapiens--Gs/β1/γ23.062025-04-09doi.org/10.1016/j.celrep.2025.115478
9LYC (No Gprot) AOrphanOrphanGPR3Homo sapiens--3.062025-04-09doi.org/10.1016/j.celrep.2025.115478
9LYDAOrphanOrphanGPR3Homo sapiens---3.662025-04-09doi.org/10.1016/j.celrep.2025.115478
8X2KAOrphanOrphanGPR3Homo sapiensOleic monoethanolamide-chim(NtGi1-Gs)/β1/γ23.032024-04-03doi.org/10.1038/s41422-023-00919-8
8X2K (No Gprot) AOrphanOrphanGPR3Homo sapiensOleic monoethanolamide-3.032024-04-03doi.org/10.1038/s41422-023-00919-8
8XOFAOrphanOrphanGPR30Homo sapiensLys05-chim(NtGi1-Gs-CtGq)/β1/γ22.62024-04-10doi.org/10.1038/s41422-024-00963-y
8XOF (No Gprot) AOrphanOrphanGPR30Homo sapiensLys05-2.62024-04-10doi.org/10.1038/s41422-024-00963-y
8XOGAOrphanOrphanGPR30Homo sapiens--chim(NtGi1-Gs-CtGq)/β1/γ22.92024-04-10doi.org/10.1038/s41422-024-00963-y
8XOG (No Gprot) AOrphanOrphanGPR30Homo sapiens--2.92024-04-10doi.org/10.1038/s41422-024-00963-y
8XOHAOrphanOrphanGPR30Homo sapiens--chim(NtGi1-Gs-CtGq)/β1/γ23.22024-04-10doi.org/10.1038/s41422-024-00963-y
8XOH (No Gprot) AOrphanOrphanGPR30Homo sapiens--3.22024-04-10doi.org/10.1038/s41422-024-00963-y
8XOIAOrphanOrphanGPR30Homo sapiens--chim(NtGi1-Gs-CtGq)/β1/γ23.22024-04-10doi.org/10.1038/s41422-024-00963-y
8XOI (No Gprot) AOrphanOrphanGPR30Homo sapiens--3.22024-04-10doi.org/10.1038/s41422-024-00963-y
8XOJAOrphanOrphanGPR30Homo sapiens--chim(NtGi1-Gs-CtGq)/β1/γ23.12024-04-10doi.org/10.1038/s41422-024-00963-y
8XOJ (No Gprot) AOrphanOrphanGPR30Homo sapiens--3.12024-04-10doi.org/10.1038/s41422-024-00963-y
8XBEAOrphanOrphanGPR34Homo sapiensS3E-LysoPS-Gi1/β1/γ13.42024-05-15doi.org/10.1038/s41467-024-45046-z
8XBE (No Gprot) AOrphanOrphanGPR34Homo sapiensS3E-LysoPS-3.42024-05-15doi.org/10.1038/s41467-024-45046-z
8XBGAOrphanOrphanGPR34Homo sapiensS3E-LysoPS--3.432024-05-15doi.org/10.1038/s41467-024-45046-z
8SAIAOrphanOrphanGPR34Homo sapiens1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ23.272023-10-04doi.org/10.1073/pnas.2308435120
8SAI (No Gprot) AOrphanOrphanGPR34Homo sapiens1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-3.272023-10-04doi.org/10.1073/pnas.2308435120
8IYXAOrphanOrphanGPR34Homo sapiensYL-365--3.342024-03-20doi.org/10.1073/pnas.2308435120
8WRBAOrphanOrphanGPR34Homo sapiensLysophosphatidylserine-Gi1/β1/γ22.912023-11-08doi.org/10.1371/journal.pbio.3002387
8WRB (No Gprot) AOrphanOrphanGPR34Homo sapiensLysophosphatidylserine-2.912023-11-08doi.org/10.1371/journal.pbio.3002387
8XBHAOrphanOrphanGPR34Homo sapiensS3E-LysoPS-Gi1/β1/γ22.832023-12-27doi.org/10.1038/s41467-024-45046-z
8XBH (No Gprot) AOrphanOrphanGPR34Homo sapiensS3E-LysoPS-2.832023-12-27doi.org/10.1038/s41467-024-45046-z
8XBIAOrphanOrphanGPR34Homo sapiensS3E-LysoPS--3.062023-12-27doi.org/10.1038/s41467-024-45046-z
8K4NAOrphanOrphanGPR34Homo sapiensVF0-Gi1/β1/γ22.832023-10-25To be published
8K4N (No Gprot) AOrphanOrphanGPR34Homo sapiensVF0-2.832023-10-25To be published
8IZ4AOrphanOrphanGPR34Homo sapiensLysophosphatidylserine-Gi1/β1/γ22.942024-04-10To be published
8IZ4 (No Gprot) AOrphanOrphanGPR34Homo sapiensLysophosphatidylserine-2.942024-04-10To be published
8ZD1AOrphanOrphanGPR4Xenopus tropicalis--chim(NtGi1-Gs)/β1/γ22.62025-02-26doi.org/10.1016/j.cell.2024.12.001
8ZD1 (No Gprot) AOrphanOrphanGPR4Xenopus tropicalis--2.62025-02-26doi.org/10.1016/j.cell.2024.12.001
8ZF4AOrphanOrphanGPR4Xenopus tropicalis---3.052025-02-26doi.org/10.1016/j.cell.2024.12.001
8ZF6AOrphanOrphanGPR4Xenopus tropicalis--chim(NtGi1-Gs)/β1/γ22.982025-02-26doi.org/10.1016/j.cell.2024.12.001
8ZF6 (No Gprot) AOrphanOrphanGPR4Xenopus tropicalis--2.982025-02-26doi.org/10.1016/j.cell.2024.12.001
8ZF7AOrphanOrphanGPR4Xenopus tropicalis---3.152025-02-26doi.org/10.1016/j.cell.2024.12.001
8ZF9AOrphanOrphanGPR4Mus musculus--chim(NtGi1-Gs)/β1/γ22.562025-02-26doi.org/10.1016/j.cell.2024.12.001
8ZF9 (No Gprot) AOrphanOrphanGPR4Mus musculus--2.562025-02-26doi.org/10.1016/j.cell.2024.12.001
8ZFAAOrphanOrphanGPR4Xenopus tropicalis--chim(NtGi1-Gs)/β1/γ22.962025-02-26doi.org/10.1016/j.cell.2024.12.001
8ZFA (No Gprot) AOrphanOrphanGPR4Xenopus tropicalis--2.962025-02-26doi.org/10.1016/j.cell.2024.12.001
8ZFBAOrphanOrphanGPR4Xenopus tropicalis---3.782025-02-26doi.org/10.1016/j.cell.2024.12.001
8ZFCAOrphanOrphanGPR4Mus musculus--chim(NtGi1-Gs)/β1/γ22.682025-02-26doi.org/10.1016/j.cell.2024.12.001
8ZFC (No Gprot) AOrphanOrphanGPR4Mus musculus--2.682025-02-26doi.org/10.1016/j.cell.2024.12.001
8ZFDAOrphanOrphanGPR4Mus musculus---2.562025-02-26doi.org/10.1016/j.cell.2024.12.001
8ZFEAOrphanOrphanGPR4Mus musculus---2.562025-02-26doi.org/10.1016/j.cell.2024.12.001
9JVGAOrphanOrphanGPR4Mus musculus--chim(NtGi1-Gs)/β1/γ22.762025-02-26doi.org/10.1016/j.cell.2024.12.001
9JVG (No Gprot) AOrphanOrphanGPR4Mus musculus--2.762025-02-26doi.org/10.1016/j.cell.2024.12.001
9JVHAOrphanOrphanGPR4Mus musculus---2.762025-02-26doi.org/10.1016/j.cell.2024.12.001
9JVMAOrphanOrphanGPR4Xenopus tropicalis---2.362025-02-26doi.org/10.1016/j.cell.2024.12.001
9BIPAOrphanOrphanGPR4Homo sapiens--Gs/β1/γ22.82025-01-22doi.org/10.1016/j.cell.2024.11.036
9BIP (No Gprot) AOrphanOrphanGPR4Homo sapiens--2.82025-01-22doi.org/10.1016/j.cell.2024.11.036
8ZCEAOrphanOrphanGPR4Homo sapiens--Gs/β1/γ23.12025-04-23doi.org/10.1038/s41422-025-01092-w
8ZCE (No Gprot) AOrphanOrphanGPR4Homo sapiens--3.12025-04-23doi.org/10.1038/s41422-025-01092-w
8ZCFAOrphanOrphanGPR4Homo sapiens--Gs/β1/γ22.92025-04-23doi.org/10.1038/s41422-025-01092-w
8ZCF (No Gprot) AOrphanOrphanGPR4Homo sapiens--2.92025-04-23doi.org/10.1038/s41422-025-01092-w
9JFUAOrphanOrphanGPR4Homo sapiensNE52-QQ57--3.232025-04-23doi.org/10.1038/s41422-025-01092-w
9JFVAOrphanOrphanGPR4Homo sapiens--chim(Gs-CtGq)/β1/γ22.672025-04-23doi.org/10.1038/s41422-025-01092-w
9JFV (No Gprot) AOrphanOrphanGPR4Homo sapiens--2.672025-04-23doi.org/10.1038/s41422-025-01092-w
9JFWAOrphanOrphanGPR4Homo sapiens--Gs/β1/γ23.132025-04-23doi.org/10.1038/s41422-025-01092-w
9JFW (No Gprot) AOrphanOrphanGPR4Homo sapiens--3.132025-04-23doi.org/10.1038/s41422-025-01092-w
9JFXAOrphanOrphanGPR4Homo sapiens--chim(Gs-CtGq)/β1/γ22.872025-04-23doi.org/10.1038/s41422-025-01092-w
9JFX (No Gprot) AOrphanOrphanGPR4Homo sapiens--2.872025-04-23doi.org/10.1038/s41422-025-01092-w
9JFZAOrphanOrphanGPR4Homo sapiens--chim(Gs-CtGq)/β1/γ22.92025-04-23doi.org/10.1038/s41422-025-01092-w
9JFZ (No Gprot) AOrphanOrphanGPR4Homo sapiens--2.92025-04-23doi.org/10.1038/s41422-025-01092-w
9JHPAOrphanOrphanGPR4Homo sapiens--chim(NtGi2-G13)/β1/γ23.352025-04-23doi.org/10.1038/s41422-025-01092-w
9JHP (No Gprot) AOrphanOrphanGPR4Homo sapiens--3.352025-04-23doi.org/10.1038/s41422-025-01092-w
9LGMAOrphanOrphanGPR4Homo sapiens--Gs/β1/γ22.842025-04-23doi.org/10.1038/s41422-025-01092-w
9LGM (No Gprot) AOrphanOrphanGPR4Homo sapiens--2.842025-04-23doi.org/10.1038/s41422-025-01092-w
8ZFZAOrphanOrphanGPR4Danio rerio--chim(NtGi1-Gs)/β1/γ23.32025-01-22doi.org/10.1038/s41467-025-55901-2
8ZFZ (No Gprot) AOrphanOrphanGPR4Danio rerio--3.32025-01-22doi.org/10.1038/s41467-025-55901-2
9J31AOrphanOrphanGPR4Danio rerio--chim(NtGi1-Gs)/β1/γ23.052025-01-22doi.org/10.1038/s41467-025-55901-2
9J31 (No Gprot) AOrphanOrphanGPR4Danio rerio--3.052025-01-22doi.org/10.1038/s41467-025-55901-2
8Z3MAOrphanOrphanGPR4Homo sapiens--chim(NtGi1-Gs-CtGq)/β1/γ22.92025-04-23To be published
8Z3M (No Gprot) AOrphanOrphanGPR4Homo sapiens--2.92025-04-23To be published
8Z3QAOrphanOrphanGPR4Homo sapiens--chim(NtGi1-Gs)/β1/γ22.762025-04-23To be published
8Z3Q (No Gprot) AOrphanOrphanGPR4Homo sapiens--2.762025-04-23To be published
8Z65AOrphanOrphanGPR4Homo sapiens--chim(NtGi1-Gs)/β1/γ22.982025-04-23To be published
8Z65 (No Gprot) AOrphanOrphanGPR4Homo sapiens--2.982025-04-23To be published
8Z66AOrphanOrphanGPR4Homo sapiens---3.062025-04-23To be published
8Z67AOrphanOrphanGPR4Homo sapiens---3.22025-04-23To be published
9LMOAOrphanOrphanGPR4Homo sapiens---3.22025-07-09To be published
9LMPAOrphanOrphanGPR4Homo sapiensNE52-QQ57--2.652025-07-02To be published
8Z3YAOrphanOrphanGPR4Homo sapiens--chim(NtGi1-Gs)/β1/γ23.22025-06-04To be published
8Z3Y (No Gprot) AOrphanOrphanGPR4Homo sapiens--3.22025-06-04To be published
8Z9PAOrphanOrphanGPR4Homo sapiens--Gi1/β1/γ22.52025-07-09To be published
8Z9P (No Gprot) AOrphanOrphanGPR4Homo sapiens--2.52025-07-09To be published
6LI1AOrphanOrphanGPR52Homo sapiens---2.92020-02-26doi.org/10.1038/s41586-020-2019-0
6LI2AOrphanOrphanGPR52Homo sapiens---2.82020-02-26doi.org/10.1038/s41586-020-2019-0
6LI3AOrphanOrphanGPR52Homo sapiens--Gs/β1/γ23.322020-02-26doi.org/10.1038/s41586-020-2019-0
6LI3 (No Gprot) AOrphanOrphanGPR52Homo sapiens--3.322020-02-26doi.org/10.1038/s41586-020-2019-0
9IY8AOrphanOrphanGPR55Homo sapiens--chim(NtGi1-G13)/β1/γ23.012025-01-01doi.org/10.1038/s41422-024-01046-8
9IY8 (No Gprot) AOrphanOrphanGPR55Homo sapiens--3.012025-01-01doi.org/10.1038/s41422-024-01046-8
9GE2AOrphanOrphanGPR55Homo sapiensML184-chim(NtGi1-G13)/β1/γ22.512025-03-05doi.org/10.1038/s41467-025-57204-y
9GE2 (No Gprot) AOrphanOrphanGPR55Homo sapiensML184-2.512025-03-05doi.org/10.1038/s41467-025-57204-y
9GE3AOrphanOrphanGPR55Homo sapiensLysophosphatidylinositol-chim(NtGi1-G13)/β1/γ22.872025-03-05doi.org/10.1038/s41467-025-57204-y
9GE3 (No Gprot) AOrphanOrphanGPR55Homo sapiensLysophosphatidylinositol-2.872025-03-05doi.org/10.1038/s41467-025-57204-y
8T1WAOrphanOrphanGPR6Homo sapiensCVN424--3.492024-12-04doi.org/10.1126/scisignal.ado8741
8TF5AOrphanOrphanGPR6Homo sapiensOleic acid--2.12024-12-04doi.org/10.2210/pdb8TF5/pdb
8TYWAOrphanOrphanGPR6Homo sapiens--Gs/β1/γ23.432024-12-04doi.org/10.2210/pdb8TF5/pdb
8TYW (No Gprot) AOrphanOrphanGPR6Homo sapiens--3.432024-12-04doi.org/10.2210/pdb8TF5/pdb
8TB0AOrphanOrphanGPR61Homo sapiens--chim(NtGi1-Gs)/β1/γ23.472023-10-04doi.org/10.1038/s41467-023-41646-3
8TB0 (No Gprot) AOrphanOrphanGPR61Homo sapiens--3.472023-10-04doi.org/10.1038/s41467-023-41646-3
8KGKAOrphanOrphanGPR61Homo sapiens--Gs/β1/γ23.162023-10-11doi.org/10.1038/s41467-023-41654-3
8KGK (No Gprot) AOrphanOrphanGPR61Homo sapiens--3.162023-10-11doi.org/10.1038/s41467-023-41654-3
9BHLAOrphanOrphanGPR65Homo sapiens--Gs/β12.82025-01-22doi.org/10.1016/j.cell.2024.11.036
9BHL (No Gprot) AOrphanOrphanGPR65Homo sapiens--2.82025-01-22doi.org/10.1016/j.cell.2024.11.036
9BHMAOrphanOrphanGPR68Homo sapiens--Gs/β12.92025-01-22doi.org/10.1016/j.cell.2024.11.036
9BHM (No Gprot) AOrphanOrphanGPR68Homo sapiens--2.92025-01-22doi.org/10.1016/j.cell.2024.11.036
9BI6AOrphanOrphanGPR68Homo sapiens--chim(Gs-CtGq)/β1/γ22.92025-01-22doi.org/10.1016/j.cell.2024.11.036
9BI6 (No Gprot) AOrphanOrphanGPR68Homo sapiens--2.92025-01-22doi.org/10.1016/j.cell.2024.11.036
8Z3OAOrphanOrphanGPR68Homo sapiens---3.32025-04-23To be published
8Z5HAOrphanOrphanGPR68Homo sapiens--chim(NtGi1-Gs)/β1/γ23.32025-04-23To be published
8Z5H (No Gprot) AOrphanOrphanGPR68Homo sapiens--3.32025-04-23To be published
8Z68AOrphanOrphanGPR68Homo sapiens--chim(NtGi1-Gs)/β1/γ22.642025-04-23To be published
8Z68 (No Gprot) AOrphanOrphanGPR68Homo sapiens--2.642025-04-23To be published
8J18AOrphanOrphanGPR84Homo sapiens(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ22.892023-06-21doi.org/10.1038/s41467-023-38985-6
8J18 (No Gprot) AOrphanOrphanGPR84Homo sapiens(3R)-3-Hydroxydodecanoic acid-2.892023-06-21doi.org/10.1038/s41467-023-38985-6
8J19AOrphanOrphanGPR84Homo sapiensLY237-Gi1/β1/γ23.232023-06-21doi.org/10.1038/s41467-023-38985-6
8J19 (No Gprot) AOrphanOrphanGPR84Homo sapiensLY237-3.232023-06-21doi.org/10.1038/s41467-023-38985-6
8J1AAOrphanOrphanGPR84Homo sapiens--Gi1/β1/γ23.242023-06-21doi.org/10.1038/s41467-023-38985-6
8J1A (No Gprot) AOrphanOrphanGPR84Homo sapiens--3.242023-06-21doi.org/10.1038/s41467-023-38985-6
8G05AOrphanOrphanGPR84Homo sapiens6-OAU-Gi1/β1/γ232023-11-01doi.org/10.1038/s41467-023-41201-0
8G05 (No Gprot) AOrphanOrphanGPR84Homo sapiens6-OAU-32023-11-01doi.org/10.1038/s41467-023-41201-0
7WZ4AOrphanOrphanGPR88Homo sapiens--Gi1/β1/γ232022-10-26doi.org/10.1038/s41467-022-30081-5
7WZ4 (No Gprot) AOrphanOrphanGPR88Homo sapiens--32022-10-26doi.org/10.1038/s41467-022-30081-5
8XT9AOrphanOrphanLGR4Homo sapiens---3.12025-01-15doi.org/10.1016/j.molcel.2025.01.024
8XUMAOrphanOrphanLGR4Homo sapiensR-spondin-2--2.92025-01-15doi.org/10.1016/j.molcel.2025.01.024
8XFPAOrphanOrphanLGR4Homo sapiensR-spondin-2-ZNRF33.212024-12-04doi.org/10.1038/s41467-024-55431-3
8XFSAOrphanOrphanLGR4Homo sapiensR-spondin-2-ZNRF33.22024-12-04doi.org/10.1038/s41467-024-55431-3
8XFTAOrphanOrphanLGR4Homo sapiensR-spondin-2-ZNRF33.242024-12-04doi.org/10.1038/s41467-024-55431-3
8Y69AOrphanOrphanLGR4Homo sapiensR-spondin-2-ZNRF33.382024-12-04doi.org/10.1038/s41467-024-55431-3
8WVUAOrphanOrphanLGR4Homo sapiensR-spondin-1-RNF433.612024-10-30To be published
8WVVAOrphanOrphanLGR4Homo sapiens---3.352024-10-30To be published
8WVWAOrphanOrphanLGR4Homo sapiens---3.532024-10-30To be published
8WVXAOrphanOrphanLGR4Homo sapiensNorrin--3.322024-10-30To be published
8WVYAOrphanOrphanLGR4Homo sapiensNorrin--3.292024-10-30To be published
9DQHAOrphanOrphanMRGPRDHomo sapiensEP-2825-chim(NtGi1-Gs-CtGq)/β1/γ22.922024-12-11doi.org/10.1016/j.celrep.2024.114942
9DQH (No Gprot) AOrphanOrphanMRGPRDHomo sapiensEP-2825-2.922024-12-11doi.org/10.1016/j.celrep.2024.114942
9DQJAOrphanOrphanMRGPRDHomo sapiensEP-3945-chim(NtGi1-Gs-CtGq)/β1/γ22.92024-12-11doi.org/10.1016/j.celrep.2024.114942
9DQJ (No Gprot) AOrphanOrphanMRGPRDHomo sapiensEP-3945-2.92024-12-11doi.org/10.1016/j.celrep.2024.114942
7Y12AOrphanOrphanMRGPRDHomo sapiensβ-Alanine-Gi1/β1/γ23.12022-07-20doi.org/10.1038/s42003-022-03668-3
7Y12 (No Gprot) AOrphanOrphanMRGPRDHomo sapiensβ-Alanine-3.12022-07-20doi.org/10.1038/s42003-022-03668-3
7Y13AOrphanOrphanMRGPRDHomo sapiens---3.12022-07-20doi.org/10.1038/s42003-022-03668-3
7Y14AOrphanOrphanMRGPRDHomo sapiensβ-Alanine--3.22022-07-20doi.org/10.1038/s42003-022-03668-3
7Y15AOrphanOrphanMRGPRDHomo sapiens--Gi1/β1/γ22.92022-07-20doi.org/10.1038/s42003-022-03668-3
7Y15 (No Gprot) AOrphanOrphanMRGPRDHomo sapiens--2.92022-07-20doi.org/10.1038/s42003-022-03668-3
8YFSAOrphanOrphanMRGPREEquus quaggaA1D6H-chim(NtGi1-Gs-CtGq)/β1/γ22.82025-03-05To be published
8YFS (No Gprot) AOrphanOrphanMRGPREEquus quaggaA1D6H-2.82025-03-05To be published
9USTAOrphanOrphanMRGPREEquus quaggaA1D6H-chim(NtGi1-Gs-CtGq)/β1/γ23.022025-07-02To be published
9UST (No Gprot) AOrphanOrphanMRGPREEquus quaggaA1D6H-3.022025-07-02To be published
8JGBAOrphanOrphanMRGPRX1Homo sapiensConorfamide-Tx2-Gi1/β1/γ22.842024-01-10doi.org/10.1038/s41467-023-40705-z
8JGB (No Gprot) AOrphanOrphanMRGPRX1Homo sapiensConorfamide-Tx2-2.842024-01-10doi.org/10.1038/s41467-023-40705-z
8JGFAOrphanOrphanMRGPRX1Homo sapiensBAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ22.72024-01-10doi.org/10.1038/s41467-023-40705-z
8JGF (No Gprot) AOrphanOrphanMRGPRX1Homo sapiensBAM8-22-2.72024-01-10doi.org/10.1038/s41467-023-40705-z
8JGGAOrphanOrphanMRGPRX1Homo sapiensBAM8-22-Gi1/β1/γ232024-01-10doi.org/10.1038/s41467-023-40705-z
8JGG (No Gprot) AOrphanOrphanMRGPRX1Homo sapiensBAM8-22-32024-01-10doi.org/10.1038/s41467-023-40705-z
8DWCAOrphanOrphanMRGPRX1Homo sapiensProenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ22.872022-11-02doi.org/10.1038/s41589-022-01173-6
8DWC (No Gprot) AOrphanOrphanMRGPRX1Homo sapiensProenkephalin-A-2.872022-11-02doi.org/10.1038/s41589-022-01173-6
8DWHAOrphanOrphanMRGPRX1Homo sapiensPubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ23.252022-11-02doi.org/10.1038/s41589-022-01173-6
8DWH (No Gprot) AOrphanOrphanMRGPRX1Homo sapiensPubChem 139030531-3.252022-11-02doi.org/10.1038/s41589-022-01173-6
8HJ5AOrphanOrphanMRGPRX1Homo sapiensPubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ232023-05-31doi.org/10.1371/journal.pbio.3001975
8HJ5 (No Gprot) AOrphanOrphanMRGPRX1Homo sapiensPubChem 139030531-32023-05-31doi.org/10.1371/journal.pbio.3001975
7VDHAOrphanOrphanMRGPRX2Homo sapiensC48/80-Gi1/β1/γ22.92021-12-01doi.org/10.1038/s41586-021-04077-y
7VDH (No Gprot) AOrphanOrphanMRGPRX2Homo sapiensC48/80-2.92021-12-01doi.org/10.1038/s41586-021-04077-y
7VDLAOrphanOrphanMRGPRX2Homo sapiensCortistatin-14-Gi1/β1/γ23.222021-12-01doi.org/10.1038/s41586-021-04077-y
7VDL (No Gprot) AOrphanOrphanMRGPRX2Homo sapiensCortistatin-14-3.222021-12-01doi.org/10.1038/s41586-021-04077-y
7VDMAOrphanOrphanMRGPRX2Homo sapiensSubstance-P-Gi1/β1/γ22.982021-12-01doi.org/10.1038/s41586-021-04077-y
7VDM (No Gprot) AOrphanOrphanMRGPRX2Homo sapiensSubstance-P-2.982021-12-01doi.org/10.1038/s41586-021-04077-y
7VUYAOrphanOrphanMRGPRX2Homo sapiens--Gi1/β1/γ22.842021-12-01doi.org/10.1038/s41586-021-04077-y
7VUY (No Gprot) AOrphanOrphanMRGPRX2Homo sapiens--2.842021-12-01doi.org/10.1038/s41586-021-04077-y
7VUZAOrphanOrphanMRGPRX2Homo sapiens--Gi1/β1/γ22.892021-12-01doi.org/10.1038/s41586-021-04077-y
7VUZ (No Gprot) AOrphanOrphanMRGPRX2Homo sapiens--2.892021-12-01doi.org/10.1038/s41586-021-04077-y
7VV0AOrphanOrphanMRGPRX2Homo sapiensPAMP-12--3.52021-12-01doi.org/10.1038/s41586-021-04077-y
7VV3AOrphanOrphanMRGPRX2Homo sapiens--Gi1/β1/γ22.972021-12-01doi.org/10.1038/s41586-021-04077-y
7VV3 (No Gprot) AOrphanOrphanMRGPRX2Homo sapiens--2.972021-12-01doi.org/10.1038/s41586-021-04077-y
7VV4AOrphanOrphanMRGPRX2Homo sapiensCortistatin-14--2.972021-12-01doi.org/10.1038/s41586-021-04077-y
7VV5AOrphanOrphanMRGPRX2Homo sapiensC48/80-Gi1/β1/γ22.762021-12-01doi.org/10.1038/s41586-021-04077-y
7VV5 (No Gprot) AOrphanOrphanMRGPRX2Homo sapiensC48/80-2.762021-12-01doi.org/10.1038/s41586-021-04077-y
7VV6AOrphanOrphanMRGPRX2Homo sapiensC48/80--3.32021-12-01doi.org/10.1038/s41586-021-04077-y
7S8LAOrphanOrphanMRGPRX2Homo sapiensCortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ22.452021-11-17doi.org/10.1038/s41586-021-04126-6
7S8L (No Gprot) AOrphanOrphanMRGPRX2Homo sapiensCortistatin-14-2.452021-11-17doi.org/10.1038/s41586-021-04126-6
7S8MAOrphanOrphanMRGPRX2Homo sapiensCortistatin-14-Gi1/β1/γ22.542021-11-17doi.org/10.1038/s41586-021-04126-6
7S8M (No Gprot) AOrphanOrphanMRGPRX2Homo sapiensCortistatin-14-2.542021-11-17doi.org/10.1038/s41586-021-04126-6
7S8NAOrphanOrphanMRGPRX2Homo sapiensR-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ22.92021-11-17doi.org/10.1038/s41586-021-04126-6
7S8N (No Gprot) AOrphanOrphanMRGPRX2Homo sapiensR-Zinc-3573-2.92021-11-17doi.org/10.1038/s41586-021-04126-6
7S8OAOrphanOrphanMRGPRX2Homo sapiensR-Zinc-3573-Gi1/β1/γ22.582021-11-17doi.org/10.1038/s41586-021-04126-6
7S8O (No Gprot) AOrphanOrphanMRGPRX2Homo sapiensR-Zinc-3573-2.582021-11-17doi.org/10.1038/s41586-021-04126-6
7S8PAOrphanOrphanMRGPRX4Homo sapiensMS47134-chim(NtGi2L-Gs-CtGq)/β1/γ22.62021-11-17doi.org/10.1038/s41586-021-04126-6
7S8P (No Gprot) AOrphanOrphanMRGPRX4Homo sapiensMS47134-2.62021-11-17doi.org/10.1038/s41586-021-04126-6
8YRGAOrphanOrphanMRGPRX4Homo sapiensFospropofol-chim(NtGi1-Gs-CtGq)/β1/γ23.142024-05-22doi.org/10.1126/scitranslmed.adk8198
8YRG (No Gprot) AOrphanOrphanMRGPRX4Homo sapiensFospropofol-3.142024-05-22doi.org/10.1126/scitranslmed.adk8198
8K4SAOrphanOrphanMRGPRX4Homo sapiensDCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ22.92024-11-06doi.org/10.1016/j.cell.2024.10.001
8K4S (No Gprot) AOrphanOrphanMRGPRX4Homo sapiensDCA-3P-2.92024-11-06doi.org/10.1016/j.cell.2024.10.001
8KEXAOrphanOrphanMRGPRX4Homo sapiensDCA-3P--3.22024-11-06doi.org/10.1016/j.cell.2024.10.001
8ITFAOrphanOrphanTA9Mus musculusDMCHA-chim(NtGi1-Gs)/β1/γ23.462023-05-31doi.org/10.1038/s41586-023-06106-4
8ITF (No Gprot) AOrphanOrphanTA9Mus musculusDMCHA-3.462023-05-31doi.org/10.1038/s41586-023-06106-4
8IW1AOrphanOrphanTA9Mus musculus--chim(NtGi1-Gs)/β1/γ23.42023-05-31doi.org/10.1038/s41586-023-06106-4
8IW1 (No Gprot) AOrphanOrphanTA9Mus musculus--3.42023-05-31doi.org/10.1038/s41586-023-06106-4
8IW4AOrphanOrphanTA9Mus musculusSpermidine-chim(NtGi1-Gs)/β1/γ23.492023-05-31doi.org/10.1038/s41586-023-06106-4
8IW4 (No Gprot) AOrphanOrphanTA9Mus musculusSpermidine-3.492023-05-31doi.org/10.1038/s41586-023-06106-4
8IW7AOrphanOrphanTA9Mus musculus2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ22.972023-05-31doi.org/10.1038/s41586-023-06106-4
8IW7 (No Gprot) AOrphanOrphanTA9Mus musculus2-Phenylethylamine-2.972023-05-31doi.org/10.1038/s41586-023-06106-4
8IW9AOrphanOrphanTA9Mus musculus--chim(NtGi1-Gs)/β1/γ23.082023-05-31doi.org/10.1038/s41586-023-06106-4
8IW9 (No Gprot) AOrphanOrphanTA9Mus musculus--3.082023-05-31doi.org/10.1038/s41586-023-06106-4
8IWEAOrphanOrphanTA9Mus musculusSpermidine--3.42023-05-31doi.org/10.1038/s41586-023-06106-4
8IWMAOrphanOrphanTA9Mus musculus2-Phenylethylamine--3.172023-05-31doi.org/10.1038/s41586-023-06106-4
8YJPCOrphanOrphanGPR156Homo sapiens---3.092025-02-05doi.org/10.1038/s41467-024-54681-5
8YK0COrphanOrphanGPR156Homo sapiens--Gi3/β1/γ22.42025-02-05doi.org/10.1038/s41467-024-54681-5
8YK0 (No Gprot) COrphanOrphanGPR156Homo sapiens--2.42025-02-05doi.org/10.1038/s41467-024-54681-5
8IEBCOrphanOrphanGPR156Homo sapiensA1LYA--3.032024-02-14doi.org/10.1038/s41594-024-01224-7
8IEDCOrphanOrphanGPR156Homo sapiensA1LYA-Go/β1/γ23.332024-02-14doi.org/10.1038/s41594-024-01224-7
8IED (No Gprot) COrphanOrphanGPR156Homo sapiensA1LYA-3.332024-02-14doi.org/10.1038/s41594-024-01224-7
8IEICOrphanOrphanGPR156Homo sapiensA1LYA--2.622024-02-14doi.org/10.1038/s41594-024-01224-7
8IEPCOrphanOrphanGPR156Homo sapiensA1LYA--2.612024-02-14doi.org/10.1038/s41594-024-01224-7
7EWLCOrphanOrphanGPR158Homo sapiens---3.522021-12-01doi.org/10.1038/s41467-021-27147-1
7EWPCOrphanOrphanGPR158Homo sapiens--B5; RGS74.32021-12-01doi.org/10.1038/s41467-021-27147-1
7EWRCOrphanOrphanGPR158Homo sapiens--B5; RGS74.72021-12-01doi.org/10.1038/s41467-021-27147-1
7SHECOrphanOrphanGPR158Homo sapiens---3.42021-12-01doi.org/10.1126/science.abl4732
7SHFCOrphanOrphanGPR158Homo sapiens--B5; RGS73.42021-12-01doi.org/10.1126/science.abl4732
8IRJCOrphanOrphanGPR179Homo sapiens---3.492024-09-18To be published
8YZKCOrphanOrphanGPRC5DHomo sapiens---3.42024-07-03doi.org/10.1038/s41467-024-49625-y
9IMACOrphanOrphanGPRC5DHomo sapiensTalquetamab--2.652024-09-11doi.org/10.1016/j.jmb.2024.168748
8YYXAAlicarboxylic acidOxoglutarateOxoglutarateHomo sapiens-Leukotriene e4chim(Gi1-CtGq)/β1/γ22.842025-04-09To be published
8YYX (No Gprot) AAlicarboxylic acidOxoglutarateOxoglutarateHomo sapiens-Leukotriene e42.842025-04-09To be published
8YYWAAlicarboxylic acidOxoglutarateOxoglutarateHomo sapiensα-ketoglutarateα-ketoglutaratechim(Gi1-CtGq)/β1/γ23.192025-04-09To be published
8YYW (No Gprot) AAlicarboxylic acidOxoglutarateOxoglutarateHomo sapiensα-ketoglutarateα-ketoglutarate3.192025-04-09To be published
4XNVANucleotideP2YP2Y1Homo sapiens-BPTU-2.22015-04-01doi.org/10.1038/nature14287
4XNWANucleotideP2YP2Y1Homo sapiensMRS2500--2.72015-04-01doi.org/10.1038/nature14287
7XXHANucleotideP2YP2Y1Homo sapiens2MeSADP-chim(NtGi1-G11)/β1/γ22.92023-06-07doi.org/10.1093/procel/pwac025
7XXH (No Gprot) ANucleotideP2YP2Y1Homo sapiens2MeSADP-2.92023-06-07doi.org/10.1093/procel/pwac025
8WJXANucleotideP2YP2Y1Homo sapiensADP-chim(Gs-CtGq)/β1/γ23.22024-10-02To be published
8WJX (No Gprot) ANucleotideP2YP2Y1Homo sapiensADP-3.22024-10-02To be published
8KGGANucleotideP2YP2Y10Homo sapiensLPS-chim(NtGi2-G13)/β1/γ23.062024-07-31doi.org/10.1016/j.chembiol.2024.08.005
8KGG (No Gprot) ANucleotideP2YP2Y10Homo sapiensLPS-3.062024-07-31doi.org/10.1016/j.chembiol.2024.08.005
7PP1ANucleotideP2YP2Y12Homo sapiensSelatogrel--2.782022-11-02doi.org/10.1016/j.bcp.2022.115291
4NTJANucleotideP2YP2Y12Homo sapiensAZD1283--2.622014-03-26doi.org/10.1038/nature13083
4PXZANucleotideP2YP2Y12Homo sapiens2MeSADP--2.52014-04-30doi.org/10.1038/nature13288
4PY0ANucleotideP2YP2Y12Homo sapiens2MeSATP--3.12014-04-30doi.org/10.1038/nature13288
7XXIANucleotideP2YP2Y12Homo sapiens2MeSADP-Gi2/β1/γ232023-06-07doi.org/10.1093/procel/pwac025
7XXI (No Gprot) ANucleotideP2YP2Y12Homo sapiens2MeSADP-32023-06-07doi.org/10.1093/procel/pwac025
9J0FANucleotideP2YP2Y14Homo sapiensNADH-Gi1/β1/γ22.762025-06-04doi.org/10.1038/s41421-025-00799-9
9J0F (No Gprot) ANucleotideP2YP2Y14Homo sapiensNADH-2.762025-06-04doi.org/10.1038/s41421-025-00799-9
9J0IANucleotideP2YP2Y14Homo sapiensUDP-Glucuronic acid-Gi1/β1/γ22.762025-06-04doi.org/10.1038/s41421-025-00799-9
9J0I (No Gprot) ANucleotideP2YP2Y14Homo sapiensUDP-Glucuronic acid-2.762025-06-04doi.org/10.1038/s41421-025-00799-9
9K20ANucleotideP2YP2Y2Homo sapiensATP-chim(NtGi1-Go)/β1/γ22.652025-06-11doi.org/10.1038/s41421-025-00797-x
9K20 (No Gprot) ANucleotideP2YP2Y2Homo sapiensATP-2.652025-06-11doi.org/10.1038/s41421-025-00797-x
9K0XANucleotideP2YP2Y2Homo sapiensATP-chim(NtGi1-Gs-CtGq)/β1/γ22.832025-06-11doi.org/10.1038/s41421-025-00797-x
9K0X (No Gprot) ANucleotideP2YP2Y2Homo sapiensATP-2.832025-06-11doi.org/10.1038/s41421-025-00797-x
9K25ANucleotideP2YP2Y2Homo sapiens--chim(NtGi1-Gs-CtGq)/β1/γ23.312025-06-11doi.org/10.1038/s41421-025-00797-x
9K25 (No Gprot) ANucleotideP2YP2Y2Homo sapiens--3.312025-06-11doi.org/10.1038/s41421-025-00797-x
9K0KANucleotideP2YP2Y4Homo sapiensUTP-chim(NtGi1-Gs-CtGq)/β1/γ23.142025-06-11doi.org/10.1038/s41421-025-00797-x
9K0K (No Gprot) ANucleotideP2YP2Y4Homo sapiensUTP-3.142025-06-11doi.org/10.1038/s41421-025-00797-x
8WZ2APeptideP518QRFPHomo sapiensOrexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ22.732024-06-19doi.org/10.1038/s41421-024-00670-3
8WZ2 (No Gprot) APeptideP518QRFPHomo sapiensOrexigenic Neuropeptide QRFP-2.732024-06-19doi.org/10.1038/s41421-024-00670-3
8ZH8APeptideP518QRFPHomo sapiensQRF-Amide-Gq/β1/γ13.192024-07-03doi.org/10.1038/s41467-024-49030-5
8ZH8 (No Gprot) APeptideP518QRFPHomo sapiensQRF-Amide-3.192024-07-03doi.org/10.1038/s41467-024-49030-5
8GW8B1PeptideParathyroid HormonePTH1Homo sapiens-PCO371Gs/β1/γ22.92023-06-14doi.org/10.1038/s41586-023-06169-3
8GW8 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiens-PCO3712.92023-06-14doi.org/10.1038/s41586-023-06169-3
8JR9B1PeptideParathyroid HormonePTH1Homo sapiens-PCO371chim(NtGi1-Gs)/β1/γ22.572023-08-02doi.org/10.1038/s41586-023-06467-w
8JR9 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiens-PCO3712.572023-08-02doi.org/10.1038/s41586-023-06467-w
7VVJB1PeptideParathyroid HormonePTH1Homo sapiensPTHrP(1-36)-Gs/β1/γ23.22022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVJ (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTHrP(1-36)-3.22022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVKB1PeptideParathyroid HormonePTH1Homo sapiensPTH-Gs/β1/γ23.32022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVK (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-3.32022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVLB1PeptideParathyroid HormonePTH1Homo sapiensPTH-Gs/β1/γ22.82022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVL (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-2.82022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVMB1PeptideParathyroid HormonePTH1Homo sapiensPTH-Gs/β1/γ23.22022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVM (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-3.22022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVNB1PeptideParathyroid HormonePTH1Homo sapiensPTH-Gs/β1/γ23.82022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVN (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-3.82022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVOB1PeptideParathyroid HormonePTH1Homo sapiensPTH-Gs/β1/γ24.12022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVO (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-4.12022-08-03doi.org/10.1016/j.molcel.2022.07.003
8FLQB1PeptideParathyroid HormonePTH1Homo sapiensPTH-Gs/β1/γ22.552023-04-26doi.org/10.1016/j.str.2023.04.002
8FLQ (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-2.552023-04-26doi.org/10.1016/j.str.2023.04.002
8FLRB1PeptideParathyroid HormonePTH1Homo sapiensPTHrP(1-36)-Gs/β1/γ22.942023-04-26doi.org/10.1016/j.str.2023.04.002
8FLR (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTHrP(1-36)-2.942023-04-26doi.org/10.1016/j.str.2023.04.002
8FLSB1PeptideParathyroid HormonePTH1Homo sapiensAbaloparatide-Gs/β1/γ23.092023-04-26doi.org/10.1016/j.str.2023.04.002
8FLS (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensAbaloparatide-3.092023-04-26doi.org/10.1016/j.str.2023.04.002
8FLTB1PeptideParathyroid HormonePTH1Homo sapiensM-PTH(1-14)-Gs/β1/γ23.032023-04-26doi.org/10.1016/j.str.2023.04.002
8FLT (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensM-PTH(1-14)-3.032023-04-26doi.org/10.1016/j.str.2023.04.002
8FLUB1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH-Gs/β1/γ22.762023-04-26doi.org/10.1016/j.str.2023.04.002
8FLU (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH-2.762023-04-26doi.org/10.1016/j.str.2023.04.002
8HA0B1PeptideParathyroid HormonePTH1Homo sapiensPTH-chim(NtGi1-Gs)/β1/γ22.622022-12-21doi.org/10.1038/s41401-022-01032-z
8HA0 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-2.622022-12-21doi.org/10.1038/s41401-022-01032-z
8HAFB1PeptideParathyroid HormonePTH1Homo sapiensPTHrP(1-36)-chim(NtGi1-Gs)/β1/γ23.252022-12-21doi.org/10.1038/s41401-022-01032-z
8HAF (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTHrP(1-36)-3.252022-12-21doi.org/10.1038/s41401-022-01032-z
8HAOB1PeptideParathyroid HormonePTH1Homo sapiensPTH-chim(NtGi1-Gs)/β1/γ23.762022-12-21doi.org/10.1038/s41401-022-01032-z
8HAO (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-3.762022-12-21doi.org/10.1038/s41401-022-01032-z
6FJ3B1PeptideParathyroid HormonePTH1Homo sapiensPTH--2.52018-11-21doi.org/10.1038/s41594-018-0151-4
6NBFB1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH Analog-Gs/β1/γ232019-04-17doi.org/10.1126/science.aav7942
6NBF (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH Analog-32019-04-17doi.org/10.1126/science.aav7942
6NBHB1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH Analog-Gs/β1/γ23.52019-04-17doi.org/10.1126/science.aav7942
6NBH (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH Analog-3.52019-04-17doi.org/10.1126/science.aav7942
6NBIB1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH Analog-Gs/β1/γ242019-04-17doi.org/10.1126/science.aav7942
6NBI (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH Analog-42019-04-17doi.org/10.1126/science.aav7942
9B5YB1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH-chim(NtGi1-Gq)/β1/γ23.492025-03-19doi.org/10.1073/pnas.2426178122
9B5Y (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH-3.492025-03-19doi.org/10.1073/pnas.2426178122
7Y35B1PeptideParathyroid HormonePTH1Homo sapiensAbaloparatide-Gs/β1/γ22.92023-07-05To be published
7Y35 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensAbaloparatide-2.92023-07-05To be published
7Y36B1PeptideParathyroid HormonePTH1Homo sapiensTeriparatide-Gs/β1/γ22.82023-07-05To be published
7Y36 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensTeriparatide-2.82023-07-05To be published
9JR2B1PeptideParathyroid HormonePTH1Homo sapiensPTH-chim(NtGi1L-Gs-CtGq)/β1/γ22.82024-10-16To be published
9JR2 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-2.82024-10-16To be published
9JR3B1PeptideParathyroid HormonePTH1Homo sapiensPTH-chim(NtGi1L-Gs-CtGq)/β1/γ22.82024-10-16To be published
9JR3 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-2.82024-10-16To be published
7F16B1PeptideParathyroid HormonePTH2Homo sapiensTIP39-Gs/β1/γ22.82021-08-18doi.org/10.1073/pnas.2101279118
7F16 (No Gprot) B1PeptideParathyroid HormonePTH2Homo sapiensTIP39-2.82021-08-18doi.org/10.1073/pnas.2101279118
8XYDALipidPlatelet Activating FactorPAFHomo sapiensPlatelet Activating Factor-Gi1/β1/γ22.92024-11-13doi.org/10.1016/j.celrep.2024.114422
8XYD (No Gprot) ALipidPlatelet Activating FactorPAFHomo sapiensPlatelet Activating Factor-2.92024-11-13doi.org/10.1016/j.celrep.2024.114422
5ZKPALipidPlatelet Activating FactorPAFHomo sapiensForopafant (SR27417)--2.812018-06-20doi.org/10.1038/s41594-018-0068-y
5ZKQALipidPlatelet Activating FactorPAFHomo sapiensABT-491--2.92018-06-20doi.org/10.1038/s41594-018-0068-y
8ZPSAPeptideProlactin-releasing peptidePrRPHomo sapiensPrRP20-chim(NtGi1-Gs-CtGq)/β1/γ22.972024-09-25doi.org/10.1038/s41421-024-00724-6
8ZPS (No Gprot) APeptideProlactin-releasing peptidePrRPHomo sapiensPrRP20-2.972024-09-25doi.org/10.1038/s41421-024-00724-6
8ZPTAPeptideProlactin-releasing peptidePrRPHomo sapiensPrRP20-chim(NtGi1-Gs-CtGq)/β1/γ22.962024-09-25doi.org/10.1038/s41421-024-00724-6
8ZPT (No Gprot) APeptideProlactin-releasing peptidePrRPHomo sapiensPrRP20-2.962024-09-25doi.org/10.1038/s41421-024-00724-6
9K26APeptideProlactin-releasing peptidePrRPHomo sapiensPrRP31-Gi1/β1/γ232025-01-29To be published
9K26 (No Gprot) APeptideProlactin-releasing peptidePrRPHomo sapiensPrRP31-32025-01-29To be published
9K27APeptideProlactin-releasing peptidePrRPHomo sapiensPrRP31-chim(NtGi1-Gq)/β1/γ22.682025-01-29To be published
9K27 (No Gprot) APeptideProlactin-releasing peptidePrRPHomo sapiensPrRP31-2.682025-01-29To be published
9UWDALipidProstaglandinDP1Homo sapiens----2025-04-09doi.org/10.1073/pnas.2501902122
8ZVZALipidProstaglandinDP1Homo sapiensBW245C-Gs/β1/γ22.352025-05-28doi.org/10.1073/pnas.2501902122
8ZVZ (No Gprot) ALipidProstaglandinDP1Homo sapiensBW245C-2.352025-05-28doi.org/10.1073/pnas.2501902122
8ZW0ALipidProstaglandinDP1Homo sapiensPGD2-Gs/β1/γ22.722025-05-28doi.org/10.1073/pnas.2501902122
8ZW0 (No Gprot) ALipidProstaglandinDP1Homo sapiensPGD2-2.722025-05-28doi.org/10.1073/pnas.2501902122
7M8WALipidProstanoidDP2Homo sapiens15r-Methyl-Prostaglandin D2Na-2.612021-08-25doi.org/10.1073/pnas.2102813118
9IYBALipidProstanoidDP2Homo sapiensProstaglandinA1D5QGi1/β1/γ22.822024-12-04doi.org/10.1073/pnas.2403304121
9IYB (No Gprot) ALipidProstanoidDP2Homo sapiensProstaglandinA1D5Q2.822024-12-04doi.org/10.1073/pnas.2403304121
8XXUALipidProstanoidDP2Homo sapiens-A1D5QGi1/β1/γ22.542024-12-04doi.org/10.1073/pnas.2403304121
8XXU (No Gprot) ALipidProstanoidDP2Homo sapiens-A1D5Q2.542024-12-04doi.org/10.1073/pnas.2403304121
8XXVALipidProstanoidDP2Homo sapiensIndomethacinA1D5QGi1/β1/γ22.332024-12-04doi.org/10.1073/pnas.2403304121
8XXV (No Gprot) ALipidProstanoidDP2Homo sapiensIndomethacinA1D5Q2.332024-12-04doi.org/10.1073/pnas.2403304121
6D26ALipidProstanoidDP2Homo sapiensFevipiprant--2.82018-10-03doi.org/10.1016/j.molcel.2018.08.009
6D27ALipidProstanoidDP2Homo sapiensCAY10471--2.742018-10-03doi.org/10.1016/j.molcel.2018.08.009
9M1HALipidProstanoidEP1Homo sapiensProstaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ22.552025-04-09To be published
9M1H (No Gprot) ALipidProstanoidEP1Homo sapiensProstaglandin E2-2.552025-04-09To be published
7CX2ALipidProstanoidEP2Homo sapiensPGE2-Gs/β1/γ22.82021-05-05doi.org/10.1126/sciadv.abf1268
7CX2 (No Gprot) ALipidProstanoidEP2Homo sapiensPGE2-2.82021-05-05doi.org/10.1126/sciadv.abf1268
7CX3ALipidProstanoidEP2Homo sapiensTaprenepag-Gs/β1/γ22.82021-05-05doi.org/10.1126/sciadv.abf1268
7CX3 (No Gprot) ALipidProstanoidEP2Homo sapiensTaprenepag-2.82021-05-05doi.org/10.1126/sciadv.abf1268
7CX4ALipidProstanoidEP2Homo sapiensEvatanepag-Gs/β1/γ22.92021-05-05doi.org/10.1126/sciadv.abf1268
7CX4 (No Gprot) ALipidProstanoidEP2Homo sapiensEvatanepag-2.92021-05-05doi.org/10.1126/sciadv.abf1268
7WU9ALipidProstanoidEP3Homo sapiens--Gi1/β1/γ23.382022-08-17doi.org/10.1016/j.celrep.2022.111323
7WU9 (No Gprot) ALipidProstanoidEP3Homo sapiens--3.382022-08-17doi.org/10.1016/j.celrep.2022.111323
6M9TALipidProstanoidEP3Homo sapiensMisoprostol-FA--2.52018-12-05doi.org/10.1038/s41589-018-0160-y
6AK3ALipidProstanoidEP3Homo sapiensDinoprostone IPGE2--2.92018-12-05doi.org/10.1038/s41589-018-0171-8
8GDCALipidProstanoidEP3Homo sapiensPGE2-Gi1/β1/γ23.52024-01-03doi.org/10.1073/pnas.2216329120
8GDC (No Gprot) ALipidProstanoidEP3Homo sapiensPGE2-3.52024-01-03doi.org/10.1073/pnas.2216329120
7D7MALipidProstanoidEP4Homo sapiensDinoprostone-Gs/β1/γ13.32020-11-18doi.org/10.1016/j.str.2020.11.007
7D7M (No Gprot) ALipidProstanoidEP4Homo sapiensDinoprostone-3.32020-11-18doi.org/10.1016/j.str.2020.11.007
5YHLALipidProstanoidEP4Homo sapiensPubChem 135121352--4.22018-12-05doi.org/10.1038/s41589-018-0131-3
5YWYALipidProstanoidEP4Homo sapiensONO-AE3-208--3.22018-12-05doi.org/10.1038/s41589-018-0131-3
8GCMALipidProstanoidEP4Homo sapiensL902688-Gi1/β1/γ23.52024-01-03doi.org/10.1073/pnas.2216329120
8GCM (No Gprot) ALipidProstanoidEP4Homo sapiensL902688-3.52024-01-03doi.org/10.1073/pnas.2216329120
8GCPALipidProstanoidEP4Homo sapiensPGE2-Gi1/β1/γ23.12024-01-03doi.org/10.1073/pnas.2216329120
8GCP (No Gprot) ALipidProstanoidEP4Homo sapiensPGE2-3.12024-01-03doi.org/10.1073/pnas.2216329120
8GD9ALipidProstanoidEP4Homo sapiensRivenprost-Gs/β1/γ23.22024-01-03doi.org/10.1073/pnas.2216329120
8GD9 (No Gprot) ALipidProstanoidEP4Homo sapiensRivenprost-3.22024-01-03doi.org/10.1073/pnas.2216329120
8GDAALipidProstanoidEP4Homo sapiensL902688-Gs/β1/γ23.32024-01-03doi.org/10.1073/pnas.2216329120
8GDA (No Gprot) ALipidProstanoidEP4Homo sapiensL902688-3.32024-01-03doi.org/10.1073/pnas.2216329120
8GDBALipidProstanoidEP4Homo sapiensPGE2-Gs/β1/γ23.12024-01-03doi.org/10.1073/pnas.2216329120
8GDB (No Gprot) ALipidProstanoidEP4Homo sapiensPGE2-3.12024-01-03doi.org/10.1073/pnas.2216329120
8IUKALipidProstanoidFP-alphaHomo sapiensPGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ22.672023-07-12doi.org/10.1038/s41467-023-38411-x
8IUK (No Gprot) ALipidProstanoidFP-alphaHomo sapiensPGF2-α-2.672023-07-12doi.org/10.1038/s41467-023-38411-x
8IULALipidProstanoidFP-alphaHomo sapiensLatanoprost-chim(NtGi1-Gs-CtGq)/β1/γ22.782023-07-12doi.org/10.1038/s41467-023-38411-x
8IUL (No Gprot) ALipidProstanoidFP-alphaHomo sapiensLatanoprost-2.782023-07-12doi.org/10.1038/s41467-023-38411-x
8IUMALipidProstanoidFP-alphaHomo sapiensTafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ23.142023-07-12doi.org/10.1038/s41467-023-38411-x
8IUM (No Gprot) ALipidProstanoidFP-alphaHomo sapiensTafluprost acid-3.142023-07-12doi.org/10.1038/s41467-023-38411-x
8IQ4ALipidProstanoidFP-alphaHomo sapiensCarboprost-chim(NtGi1-Gs-CtGq)/β1/γ22.72024-01-31doi.org/10.1038/s41467-023-43922-8
8IQ4 (No Gprot) ALipidProstanoidFP-alphaHomo sapiensCarboprost-2.72024-01-31doi.org/10.1038/s41467-023-43922-8
8IQ6ALipidProstanoidFP-alphaHomo sapiensLatanoprost-chim(NtGi1-Gs-CtGq)/β1/γ23.42024-01-31doi.org/10.1038/s41467-023-43922-8
8IQ6 (No Gprot) ALipidProstanoidFP-alphaHomo sapiensLatanoprost-3.42024-01-31doi.org/10.1038/s41467-023-43922-8
8XJKALipidProstanoidFP-alphaHomo sapiensCloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ22.632024-02-28doi.org/10.1016/j.celrep.2024.113893
8XJK (No Gprot) ALipidProstanoidFP-alphaHomo sapiensCloprosetnol-2.632024-02-28doi.org/10.1016/j.celrep.2024.113893
8XJLALipidProstanoidFP-alphaHomo sapiensPGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ22.772024-02-28doi.org/10.1016/j.celrep.2024.113893
8XJL (No Gprot) ALipidProstanoidFP-alphaHomo sapiensPGF2-α-2.772024-02-28doi.org/10.1016/j.celrep.2024.113893
8XJMALipidProstanoidFP-alphaHomo sapiensLatanoprost-chim(NtGi2-Gs-CtGq)/β1/γ22.852024-02-28doi.org/10.1016/j.celrep.2024.113893
8XJM (No Gprot) ALipidProstanoidFP-alphaHomo sapiensLatanoprost-2.852024-02-28doi.org/10.1016/j.celrep.2024.113893
8X79ALipidProstanoidI2Homo sapiensMRE-269-Gs/β1/γ22.412024-03-06doi.org/10.1126/sciadv.adk5184
8X79 (No Gprot) ALipidProstanoidI2Homo sapiensMRE-269-2.412024-03-06doi.org/10.1126/sciadv.adk5184
8X7AALipidProstanoidI2Homo sapiensTreprostinil-Gs/β1/γ22.562024-03-06doi.org/10.1126/sciadv.adk5184
8X7A (No Gprot) ALipidProstanoidI2Homo sapiensTreprostinil-2.562024-03-06doi.org/10.1126/sciadv.adk5184
6IIUALipidProstanoidTXA2Homo sapiensRamatroban--2.52018-12-19doi.org/10.1038/s41589-018-0170-9
6IIVALipidProstanoidTXA2Homo sapiensDaltroban--32018-12-19doi.org/10.1038/s41589-018-0170-9
8XJNALipidProstanoidTXA2Homo sapiensCloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ23.062024-02-28doi.org/10.1016/j.celrep.2024.113893
8XJN (No Gprot) ALipidProstanoidTXA2Homo sapiensCloprosetnol-3.062024-02-28doi.org/10.1016/j.celrep.2024.113893
8XJOALipidProstanoidTXA2Homo sapiensU46619-chim(NtGi1-Gs-CtGq)/β1/γ23.112024-02-28doi.org/10.1016/j.celrep.2024.113893
8XJO (No Gprot) ALipidProstanoidTXA2Homo sapiensU46619-3.112024-02-28doi.org/10.1016/j.celrep.2024.113893
3VW7APeptideProteinase ActivatedPAR1Homo sapiens-Vorapaxar; Na-2.22012-12-12doi.org/10.1038/nature11701
5NDDAPeptideProteinase ActivatedPAR2Homo sapiens-AZ8838; Na-2.82017-05-03doi.org/10.1038/nature22309
5NDZAPeptideProteinase ActivatedPAR2Homo sapiens-AZ3451; Na-3.62017-05-03doi.org/10.1038/nature22309
8XORAPeptideProteinase ActivatedPAR1Homo sapiens--chim(NtGi1-Gs-CtGq)/β1/γ232024-09-18doi.org/10.1038/s41422-024-00997-2
8XOR (No Gprot) APeptideProteinase ActivatedPAR1Homo sapiens--32024-09-18doi.org/10.1038/s41422-024-00997-2
8XOSAPeptideProteinase ActivatedPAR1Homo sapiens--Gi1/β1/γ23.22024-09-18doi.org/10.1038/s41422-024-00997-2
8XOS (No Gprot) APeptideProteinase ActivatedPAR1Homo sapiens--3.22024-09-18doi.org/10.1038/s41422-024-00997-2
9D4ZAPeptideProteinase ActivatedPAR1Homo sapiens--chim(NtGi1L-Gs-CtGq)/β1/γ22.742025-05-07doi.org/10.1038/s41467-025-59138-x
9D4Z (No Gprot) APeptideProteinase ActivatedPAR1Homo sapiens--2.742025-05-07doi.org/10.1038/s41467-025-59138-x
5NJ6APeptideProteinase ActivatedPAR2Homo sapiens---42017-05-03doi.org/10.1038/nature22309
9D0AAPeptideProteinase ActivatedPAR2Homo sapiens--chim(NtGi1L-Gs-CtGq)/β1/γ23.12025-05-07doi.org/10.1038/s41467-025-59138-x
9D0A (No Gprot) APeptideProteinase ActivatedPAR2Homo sapiens--3.12025-05-07doi.org/10.1038/s41467-025-59138-x
9E7RAPeptideProteinase ActivatedPAR2Homo sapiensGB88-chim(NtGi1L-Gs-CtGq)/β1/γ23.182025-05-07doi.org/10.1038/s41467-025-59138-x
9E7R (No Gprot) APeptideProteinase ActivatedPAR2Homo sapiensGB88-3.182025-05-07doi.org/10.1038/s41467-025-59138-x
8ZMDAPeptideProteinase ActivatedPAR2Homo sapiens--chim(NtGi1L-Gs-CtGq)/β1/γ23.252025-05-28To be published
8ZMD (No Gprot) APeptideProteinase ActivatedPAR2Homo sapiens--3.252025-05-28To be published
8ZMEAPeptideProteinase ActivatedPAR2Homo sapiens--chim(NtGi1-G13)/β1/γ23.22025-05-28To be published
8ZME (No Gprot) APeptideProteinase ActivatedPAR2Homo sapiens--3.22025-05-28To be published
7TMWAPeptideRelaxinRXFP1Homo sapiens--Gs/β1/γ23.22023-02-15doi.org/10.1101/2022.01.22.477343
7TMW (No Gprot) APeptideRelaxinRXFP1Homo sapiens--3.22023-02-15doi.org/10.1101/2022.01.22.477343
7YJ4APeptideRelaxinRXFP4Homo sapiensINSL5-Gi2/β1/γ23.192023-03-01doi.org/10.1038/s41467-023-36182-z
7YJ4 (No Gprot) APeptideRelaxinRXFP4Homo sapiensINSL5-3.192023-03-01doi.org/10.1038/s41467-023-36182-z
7YK6APeptideRelaxinRXFP4Homo sapiensPubChem 138319674-Gi2/β1/γ23.032023-03-01doi.org/10.1038/s41467-023-36182-z
7YK6 (No Gprot) APeptideRelaxinRXFP4Homo sapiensPubChem 138319674-3.032023-03-01doi.org/10.1038/s41467-023-36182-z
7YK7APeptideRelaxinRXFP4Homo sapiensDC591053-Gi2/β1/γ22.752023-03-01doi.org/10.1038/s41467-023-36182-z
7YK7 (No Gprot) APeptideRelaxinRXFP4Homo sapiensDC591053-2.752023-03-01doi.org/10.1038/s41467-023-36182-z
9IK8APeptideSomatostatinSST1Homo sapiensSST analogue-Gi1/β1/γ22.822025-04-30doi.org/10.1016/j.apsb.2025.03.043
9IK8 (No Gprot) APeptideSomatostatinSST1Homo sapiensSST analogue-2.822025-04-30doi.org/10.1016/j.apsb.2025.03.043
9IK9APeptideSomatostatinSST1Homo sapiensSST analogue-Gi1/β1/γ23.372025-04-30doi.org/10.1016/j.apsb.2025.03.043
9IK9 (No Gprot) APeptideSomatostatinSST1Homo sapiensSST analogue-3.372025-04-30doi.org/10.1016/j.apsb.2025.03.043
8XIOAPeptideSomatostatinSST1Homo sapiensL797591-chim(NtGi1-Gs-CtGi1)/β1/γ22.652024-07-03doi.org/10.1073/pnas.2400298121
8XIO (No Gprot) APeptideSomatostatinSST1Homo sapiensL797591-2.652024-07-03doi.org/10.1073/pnas.2400298121
8XIPAPeptideSomatostatinSST1Homo sapiensPasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ23.292024-07-03doi.org/10.1073/pnas.2400298121
8XIP (No Gprot) APeptideSomatostatinSST1Homo sapiensPasireotide-3.292024-07-03doi.org/10.1073/pnas.2400298121
7XATAPeptideSomatostatinSST2Homo sapiensSomatostatin-14-Gi1/β1/γ22.852022-08-31doi.org/10.1038/s41421-022-00405-2
7XAT (No Gprot) APeptideSomatostatinSST2Homo sapiensSomatostatin-14-2.852022-08-31doi.org/10.1038/s41421-022-00405-2
7XAUAPeptideSomatostatinSST2Homo sapiensOctreotide-Gi1/β1/γ22.972022-08-31doi.org/10.1038/s41421-022-00405-2
7XAU (No Gprot) APeptideSomatostatinSST2Homo sapiensOctreotide-2.972022-08-31doi.org/10.1038/s41421-022-00405-2
7XAVAPeptideSomatostatinSST2Homo sapiensLanreotide-Gi1/β1/γ22.872022-08-31doi.org/10.1038/s41421-022-00405-2
7XAV (No Gprot) APeptideSomatostatinSST2Homo sapiensLanreotide-2.872022-08-31doi.org/10.1038/s41421-022-00405-2
7WICAPeptideSomatostatinSST2Homo sapiensSomatostatin-14-Gi1/β1/γ22.82022-06-01doi.org/10.1038/s41422-022-00669-z
7WIC (No Gprot) APeptideSomatostatinSST2Homo sapiensSomatostatin-14-2.82022-06-01doi.org/10.1038/s41422-022-00669-z
7WIGAPeptideSomatostatinSST2Homo sapiensL-054,264-Gi1/β1/γ22.72022-06-01doi.org/10.1038/s41422-022-00669-z
7WIG (No Gprot) APeptideSomatostatinSST2Homo sapiensL-054,264-2.72022-06-01doi.org/10.1038/s41422-022-00669-z
7XMRAPeptideSomatostatinSST2Homo sapiensSomatostatin-14-Gi1/β1/γ23.12022-08-03doi.org/10.1038/s41422-022-00679-x
7XMR (No Gprot) APeptideSomatostatinSST2Homo sapiensSomatostatin-14-3.12022-08-03doi.org/10.1038/s41422-022-00679-x
7XN9APeptideSomatostatinSST2Homo sapiensL-054,522--2.62022-08-03doi.org/10.1038/s41422-022-00679-x
7XNAAPeptideSomatostatinSST2Homo sapiensCYN154806--2.652022-08-03doi.org/10.1038/s41422-022-00679-x
7YACAPeptideSomatostatinSST2Homo sapiensPaltusotine-Gi1/β1/γ23.242023-04-19doi.org/10.1038/s41467-023-36673-z
7YAC (No Gprot) APeptideSomatostatinSST2Homo sapiensPaltusotine-3.242023-04-19doi.org/10.1038/s41467-023-36673-z
7YAEAPeptideSomatostatinSST2Homo sapiensOctreotide-Gi1/β1/γ23.372023-04-19doi.org/10.1038/s41467-023-36673-z
7YAE (No Gprot) APeptideSomatostatinSST2Homo sapiensOctreotide-3.372023-04-19doi.org/10.1038/s41467-023-36673-z
7Y24APeptideSomatostatinSST2Homo sapiensOctreotide-Go/β1/γ23.252022-10-19doi.org/10.1038/s41589-022-01130-3
7Y24 (No Gprot) APeptideSomatostatinSST2Homo sapiensOctreotide-3.252022-10-19doi.org/10.1038/s41589-022-01130-3
7Y26APeptideSomatostatinSST2Homo sapiensOctreotide-chim(NtGi2L-Gs-CtGq)/β1/γ23.32022-10-19doi.org/10.1038/s41589-022-01130-3
7Y26 (No Gprot) APeptideSomatostatinSST2Homo sapiensOctreotide-3.32022-10-19doi.org/10.1038/s41589-022-01130-3
7Y27APeptideSomatostatinSST2Homo sapiensSomatostatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ23.482022-10-19doi.org/10.1038/s41589-022-01130-3
7Y27 (No Gprot) APeptideSomatostatinSST2Homo sapiensSomatostatin-14-3.482022-10-19doi.org/10.1038/s41589-022-01130-3
7UL5APeptideSomatostatinSST2Homo sapiens---3.12022-06-29doi.org/10.1038/s41594-022-00859-8
7WJ5APeptideSomatostatinSST2Homo sapiensSomatostatin-14-Gi1/β1/γ23.722022-07-13doi.org/10.7554/eLife.76823
7WJ5 (No Gprot) APeptideSomatostatinSST2Homo sapiensSomatostatin-14-3.722022-07-13doi.org/10.7554/eLife.76823
7T10APeptideSomatostatinSST2Homo sapiensSomatostatin-14-Gi3/β1/γ22.52022-03-09doi.org/10.1038/s41594-022-00727-5
7T10 (No Gprot) APeptideSomatostatinSST2Homo sapiensSomatostatin-14-2.52022-03-09doi.org/10.1038/s41594-022-00727-5
7T11APeptideSomatostatinSST2Homo sapiensOctreotide-Gi3/β1/γ22.72022-03-09doi.org/10.1038/s41594-022-00727-5
7T11 (No Gprot) APeptideSomatostatinSST2Homo sapiensOctreotide-2.72022-03-09doi.org/10.1038/s41594-022-00727-5
8XIQAPeptideSomatostatinSST3Homo sapiensL796778-chim(NtGi1-Gs-CtGi1)/β1/γ22.712024-07-03doi.org/10.1073/pnas.2400298121
8XIQ (No Gprot) APeptideSomatostatinSST3Homo sapiensL796778-2.712024-07-03doi.org/10.1073/pnas.2400298121
8XIRAPeptideSomatostatinSST3Homo sapiensPasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ22.522024-07-03doi.org/10.1073/pnas.2400298121
8XIR (No Gprot) APeptideSomatostatinSST3Homo sapiensPasireotide-2.522024-07-03doi.org/10.1073/pnas.2400298121
8ZBIAPeptideSomatostatinSST3Homo sapiensSomatostatin-14-Gi1/β1/γ22.792025-04-30To be published
8ZBI (No Gprot) APeptideSomatostatinSST3Homo sapiensSomatostatin-14-2.792025-04-30To be published
7XMSAPeptideSomatostatinSST4Homo sapiensSomatostatin-14-Gi1/β1/γ22.92022-08-03doi.org/10.1038/s41422-022-00679-x
7XMS (No Gprot) APeptideSomatostatinSST4Homo sapiensSomatostatin-14-2.92022-08-03doi.org/10.1038/s41422-022-00679-x
7XMTAPeptideSomatostatinSST4Homo sapiensJ-2156-Gi1/β1/γ22.82022-08-03doi.org/10.1038/s41422-022-00679-x
7XMT (No Gprot) APeptideSomatostatinSST4Homo sapiensJ-2156-2.82022-08-03doi.org/10.1038/s41422-022-00679-x
8ZBEAPeptideSomatostatinSST5Homo sapiensOctreotide-Gi1/β1/γ13.242024-07-10doi.org/10.1038/s41401-024-01314-8
8ZBE (No Gprot) APeptideSomatostatinSST5Homo sapiensOctreotide-3.242024-07-10doi.org/10.1038/s41401-024-01314-8
8ZCJAPeptideSomatostatinSST5Homo sapiensPasireotide-Gi1/β1/γ13.092024-07-10doi.org/10.1038/s41401-024-01314-8
8ZCJ (No Gprot) APeptideSomatostatinSST5Homo sapiensPasireotide-3.092024-07-10doi.org/10.1038/s41401-024-01314-8
8X8LAPeptideSomatostatinSST5Homo sapiensCortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ22.72024-06-12doi.org/10.1073/pnas.2321710121
8X8L (No Gprot) APeptideSomatostatinSST5Homo sapiensCortistatin-2.72024-06-12doi.org/10.1073/pnas.2321710121
8X8NAPeptideSomatostatinSST5Homo sapiensOctreotide-chim(NtGi1-Gs-CtGi1)/β1/γ22.92024-06-12doi.org/10.1073/pnas.2321710121
8X8N (No Gprot) APeptideSomatostatinSST5Homo sapiensOctreotide-2.92024-06-12doi.org/10.1073/pnas.2321710121
8ZBJAPeptideSomatostatinSST5Homo sapiensSomatostatin-14-Gi1/β1/γ22.942025-04-30To be published
8ZBJ (No Gprot) APeptideSomatostatinSST5Homo sapiensSomatostatin-14-2.942025-04-30To be published
7AD3D1Ste2-likeSTE2STE2Saccharomyces cerevisiaeα-factor mating pheromone-Gi1/STE4/γ23.32020-12-09doi.org/10.1038/s41586-020-2994-1
7AD3 (No Gprot) D1Ste2-likeSTE2STE2Saccharomyces cerevisiaeα-factor mating pheromone-3.32020-12-09doi.org/10.1038/s41586-020-2994-1
7QA8D1Ste2-likeSTE2STE2Saccharomyces cerevisiaePeptide--2.72022-03-16doi.org/10.1038/s41586-022-04498-3
7QB9D1Ste2-likeSTE2STE2Saccharomyces cerevisiae---3.12022-03-16doi.org/10.1038/s41586-022-04498-3
7QBCD1Ste2-likeSTE2STE2Saccharomyces cerevisiaeα-factor mating pheromone--3.532022-03-16doi.org/10.1038/s41586-022-04498-3
7QBID1Ste2-likeSTE2STE2Saccharomyces cerevisiaeα-factor mating pheromone--3.462022-03-16doi.org/10.1038/s41586-022-04498-3
6Z10AAlicarboxylic acidSuccinateSuccinateRattus norvegicusPubChem 154585554--2.272020-09-16doi.org/10.1021/acs.jmedchem.0c01020
8JPNAAlicarboxylic acidSuccinateSuccinateHomo sapiensCis-Epoxysuccinic acid-Gi1/β1/γ12.92024-05-22doi.org/10.1038/s41422-024-00968-7
8JPN (No Gprot) AAlicarboxylic acidSuccinateSuccinateHomo sapiensCis-Epoxysuccinic acid-2.92024-05-22doi.org/10.1038/s41422-024-00968-7
8JPPAAlicarboxylic acidSuccinateSuccinateHomo sapiensSuccinic acid-chim(Gs-CtGq)/β1/γ13.22024-05-22doi.org/10.1038/s41422-024-00968-7
8JPP (No Gprot) AAlicarboxylic acidSuccinateSuccinateHomo sapiensSuccinic acid-3.22024-05-22doi.org/10.1038/s41422-024-00968-7
8YKWAAlicarboxylic acidSuccinateSuccinateHomo sapiensSuccinic acid-Gi1/β1/γ12.752024-05-29doi.org/10.1038/s41422-024-00984-7
8YKW (No Gprot) AAlicarboxylic acidSuccinateSuccinateHomo sapiensSuccinic acid-2.752024-05-29doi.org/10.1038/s41422-024-00984-7
8YKXAAlicarboxylic acidSuccinateSuccinateHomo sapiensMaleic acid-Gi1/β1/γ12.692024-05-29doi.org/10.1038/s41422-024-00984-7
8YKX (No Gprot) AAlicarboxylic acidSuccinateSuccinateHomo sapiensMaleic acid-2.692024-05-29doi.org/10.1038/s41422-024-00984-7
6IBBAAlicarboxylic acidSuccinateSuccinateRattus norvegicus---2.122019-08-14doi.org/10.1038/s41586-019-1663-8
6RNKAAlicarboxylic acidSuccinateSuccinateRattus norvegicusNF-56-EJ40--1.942019-08-14doi.org/10.1038/s41586-019-1663-8
8WOGAAlicarboxylic acidSuccinateSuccinateHomo sapiensSuccinic acid-Gi1/β1/γ22.972024-09-11doi.org/10.1016/j.celrep.2024.114381
8WOG (No Gprot) AAlicarboxylic acidSuccinateSuccinateHomo sapiensSuccinic acid-2.972024-09-11doi.org/10.1016/j.celrep.2024.114381
8WP1AAlicarboxylic acidSuccinateSuccinateHomo sapiensCis-Epoxysuccinic acid-Gi1/β1/γ23.152024-09-11doi.org/10.1016/j.celrep.2024.114381
8WP1 (No Gprot) AAlicarboxylic acidSuccinateSuccinateHomo sapiensCis-Epoxysuccinic acid-3.152024-09-11doi.org/10.1016/j.celrep.2024.114381
8YKVAAlicarboxylic acidSuccinateSuccinateHomo sapiensPubChem 137553168-Gi1/β1/γ22.482024-05-29doi.org/10.1038/s41422-024-00984-7
8YKV (No Gprot) AAlicarboxylic acidSuccinateSuccinateHomo sapiensPubChem 137553168-2.482024-05-29doi.org/10.1038/s41422-024-00984-7
6HLLAPeptideTachykininNK1Homo sapiensCP99994--3.272019-01-16doi.org/10.1038/s41467-018-07939-8
6HLOAPeptideTachykininNK1Homo sapiensAprepitant--2.42019-01-16doi.org/10.1038/s41467-018-07939-8
6HLPAPeptideTachykininNK1Homo sapiensNetupitant--2.22019-01-16doi.org/10.1038/s41467-018-07939-8
6J20APeptideTachykininNK1Homo sapiensAprepitant--2.72019-03-06doi.org/10.1038/s41467-019-08568-5
6J21APeptideTachykininNK1Homo sapiensAprepitant--3.22019-03-06doi.org/10.1038/s41467-019-08568-5
7RMGAPeptideTachykininNK1Homo sapiensSubstance-P-chim(Gs-CtGq)/β1/γ232021-11-03doi.org/10.1038/s41589-021-00890-8
7RMG (No Gprot) APeptideTachykininNK1Homo sapiensSubstance-P-32021-11-03doi.org/10.1038/s41589-021-00890-8
7RMHAPeptideTachykininNK1Homo sapiensSubstance-P-Gs/β1/γ23.12021-11-03doi.org/10.1038/s41589-021-00890-8
7RMH (No Gprot) APeptideTachykininNK1Homo sapiensSubstance-P-3.12021-11-03doi.org/10.1038/s41589-021-00890-8
7RMIAPeptideTachykininNK1Homo sapiensSubstance-P-chim(Gs-CtGq)/β1/γ23.22021-11-03doi.org/10.1038/s41589-021-00890-8
7RMI (No Gprot) APeptideTachykininNK1Homo sapiensSubstance-P-3.22021-11-03doi.org/10.1038/s41589-021-00890-8
8U26APeptideTachykininNK1Homo sapiensProtachykinin-1-Gs/β1/γ22.52023-11-15doi.org/10.1038/s41592-023-02082-9
8U26 (No Gprot) APeptideTachykininNK1Homo sapiensProtachykinin-1-2.52023-11-15doi.org/10.1038/s41592-023-02082-9
6E59APeptideTachykininNK1Homo sapiensL-760735--3.42018-12-12doi.org/10.1073/pnas.1812717115
7P00APeptideTachykininNK1Homo sapiensSubstance-P-chim(NtGi1-Gs-CtGq)/β1/γ22.712021-12-15doi.org/10.1126/sciadv.abk2872
7P00 (No Gprot) APeptideTachykininNK1Homo sapiensSubstance-P-2.712021-12-15doi.org/10.1126/sciadv.abk2872
7P02APeptideTachykininNK1Homo sapiensProtachykinin-1-chim(NtGi1-Gs)/β1/γ22.872021-12-15doi.org/10.1126/sciadv.abk2872
7P02 (No Gprot) APeptideTachykininNK1Homo sapiensProtachykinin-1-2.872021-12-15doi.org/10.1126/sciadv.abk2872
7XWOAPeptideTachykininNK2Homo sapiensNeurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ22.72023-05-31doi.org/10.1038/s41421-022-00437-8
7XWO (No Gprot) APeptideTachykininNK2Homo sapiensNeurokinin-A-2.72023-05-31doi.org/10.1038/s41421-022-00437-8
8JBFAPeptideTachykininNK3Homo sapiensSenktide-chim(NtGi1-Gs-CtGq)/β1/γ232024-02-28doi.org/10.1038/s41421-023-00564-w
8JBF (No Gprot) APeptideTachykininNK3Homo sapiensSenktide-32024-02-28doi.org/10.1038/s41421-023-00564-w
8JBGAPeptideTachykininNK3Homo sapiensNeurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ22.82024-02-07doi.org/10.1038/s41421-023-00564-w
8JBG (No Gprot) APeptideTachykininNK3Homo sapiensNeurokinin-B-2.82024-02-07doi.org/10.1038/s41421-023-00564-w
8JBHAPeptideTachykininNK3Homo sapiensSubstance-P-chim(NtGi1-Gs-CtGq)/β1/γ22.92024-02-07doi.org/10.1038/s41421-023-00564-w
8JBH (No Gprot) APeptideTachykininNK3Homo sapiensSubstance-P-2.92024-02-07doi.org/10.1038/s41421-023-00564-w
9NOXCSensoryTaste1TAS1R2Homo sapiens--chim(Gs-CtGt3)/β1/γ232025-04-09doi.org/10.1016/j.cell.2025.04.021
9NOX (No Gprot) CSensoryTaste1TAS1R2Homo sapiens--32025-04-09doi.org/10.1016/j.cell.2025.04.021
9NOYCSensoryTaste1TAS1R2Homo sapiens---3.72025-04-09doi.org/10.1016/j.cell.2025.04.021
9NORCSensoryTaste1TAS1R2; TAS1R3Homo sapiens---3.42025-04-09doi.org/10.1016/j.cell.2025.04.021
9NOSCSensoryTaste1TAS1R2; TAS1R3Homo sapiens---3.52025-04-09doi.org/10.1016/j.cell.2025.04.021
9NOTCSensoryTaste1TAS1R2; TAS1R3Homo sapiens---3.82025-04-09doi.org/10.1016/j.cell.2025.04.021
9O38CSensoryTaste1TAS1R2; TAS1R3Homo sapiens--chim(Gs-CtGt3)/β1/γ232025-04-09doi.org/10.1016/j.cell.2025.04.021
9O38 (No Gprot) CSensoryTaste1TAS1R2; TAS1R3Homo sapiens--32025-04-09doi.org/10.1016/j.cell.2025.04.021
8RQLT2SensoryTaste2TAS2R14Homo sapiensFlufenamic acidFlufenamic acidchim(NtGi1-Gt3)/β1/γ23.032024-11-27doi.org/10.1038/s41467-024-54157-6
8RQL (No Gprot) T2SensoryTaste2TAS2R14Homo sapiensFlufenamic acidFlufenamic acid3.032024-11-27doi.org/10.1038/s41467-024-54157-6
8XQRT2SensoryTaste2TAS2R14Homo sapiens-Flufenamic acidGt3/β1/γ13.22024-07-10doi.org/10.1038/s41586-024-07569-9
8XQR (No Gprot) T2SensoryTaste2TAS2R14Homo sapiens-Flufenamic acid3.22024-07-10doi.org/10.1038/s41586-024-07569-9
8XQST2SensoryTaste2TAS2R14Homo sapiensCholesterolFlufenamic acidGi1/β1/γ13.32024-07-10doi.org/10.1038/s41586-024-07569-9
8XQS (No Gprot) T2SensoryTaste2TAS2R14Homo sapiensCholesterolFlufenamic acid3.32024-07-10doi.org/10.1038/s41586-024-07569-9
8XQLT2SensoryTaste2TAS2R14Homo sapiensCholesterolAristolochic acid AGt3/β1/γ12.992024-07-10doi.org/10.1038/s41586-024-07569-9
8XQL (No Gprot) T2SensoryTaste2TAS2R14Homo sapiensCholesterolAristolochic acid A2.992024-07-10doi.org/10.1038/s41586-024-07569-9
8XQNT2SensoryTaste2TAS2R14Homo sapiensCholesterolAristolochic acid AGi1/β1/γ13.052024-07-10doi.org/10.1038/s41586-024-07569-9
8XQN (No Gprot) T2SensoryTaste2TAS2R14Homo sapiensCholesterolAristolochic acid A3.052024-07-10doi.org/10.1038/s41586-024-07569-9
8XQOT2SensoryTaste2TAS2R14Homo sapiensCholesterolAristolochic acid AGi1/β1/γ12.772024-07-10doi.org/10.1038/s41586-024-07569-9
8XQO (No Gprot) T2SensoryTaste2TAS2R14Homo sapiensCholesterolAristolochic acid A2.772024-07-10doi.org/10.1038/s41586-024-07569-9
8XQPT2SensoryTaste2TAS2R14Homo sapiensCholesterolAristolochic acid AGt3/β1/γ13.292024-07-10doi.org/10.1038/s41586-024-07569-9
8XQP (No Gprot) T2SensoryTaste2TAS2R14Homo sapiensCholesterolAristolochic acid A3.292024-07-10doi.org/10.1038/s41586-024-07569-9
8XQTT2SensoryTaste2TAS2R14Homo sapiensCholesterol-Gi1/β1/γ12.942024-07-10doi.org/10.1038/s41586-024-07569-9
8XQT (No Gprot) T2SensoryTaste2TAS2R14Homo sapiensCholesterol-2.942024-07-10doi.org/10.1038/s41586-024-07569-9
9K6LT2SensoryTaste2TAS2R16Homo sapiensSA0-Gi2/β1/γ22.772025-04-02To be published
9K6L (No Gprot) T2SensoryTaste2TAS2R16Homo sapiensSA0-2.772025-04-02To be published
9KPDT2SensoryTaste2TAS2R16Homo sapiensSA0-chim(Gs-CtGt3)/β1/γ22.842025-04-02To be published
9KPD (No Gprot) T2SensoryTaste2TAS2R16Homo sapiensSA0-2.842025-04-02To be published
9KPET2SensoryTaste2TAS2R16Homo sapiensSA0-Gi1/β1/γ23.352025-04-02To be published
9KPE (No Gprot) T2SensoryTaste2TAS2R16Homo sapiensSA0-3.352025-04-02To be published
9KPFT2SensoryTaste2TAS2R16Homo sapiensSA0-Gi1/β1/γ23.152025-04-02To be published
9KPF (No Gprot) T2SensoryTaste2TAS2R16Homo sapiensSA0-3.152025-04-02To be published
7XP4T2SensoryTaste2TAS2R46Homo sapiens--chim(Gs-CtGt3)/β1/γ23.012022-10-12doi.org/10.1126/science.abo1633
7XP4 (No Gprot) T2SensoryTaste2TAS2R46Homo sapiens--3.012022-10-12doi.org/10.1126/science.abo1633
7XP5T2SensoryTaste2TAS2R46Homo sapiens--chim(Gs-CtGt3)/β1/γ23.082022-10-12doi.org/10.1126/science.abo1633
7XP5 (No Gprot) T2SensoryTaste2TAS2R46Homo sapiens--3.082022-10-12doi.org/10.1126/science.abo1633
7XP6T2SensoryTaste2TAS2R46Homo sapiensStrychnine-chim(Gs-CtGt3)/β1/γ23.012022-10-12doi.org/10.1126/science.abo1633
7XP6 (No Gprot) T2SensoryTaste2TAS2R46Homo sapiensStrychnine-3.012022-10-12doi.org/10.1126/science.abo1633
7XW9APeptideThyrotropin Releasing HormoneTRHHomo sapiensTRH-chim(NtGi1L-Gs-CtGq)/β1/γ22.72022-12-28doi.org/10.1038/s41421-022-00477-0
7XW9 (No Gprot) APeptideThyrotropin Releasing HormoneTRHHomo sapiensTRH-2.72022-12-28doi.org/10.1038/s41421-022-00477-0
7WKDAPeptideThyrotropin Releasing HormoneTRHHomo sapiensTRH-chim(NtGi1-Gs-CtGq)/β1/γ23.012022-06-15doi.org/10.1038/s41422-022-00641-x
7WKD (No Gprot) APeptideThyrotropin Releasing HormoneTRHHomo sapiensTRH-3.012022-06-15doi.org/10.1038/s41422-022-00641-x
7X1TAPeptideThyrotropin Releasing HormoneTRHHomo sapiensTaltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ23.262022-08-31doi.org/10.1038/s41422-022-00646-6
7X1T (No Gprot) APeptideThyrotropin Releasing HormoneTRHHomo sapiensTaltirelin-3.262022-08-31doi.org/10.1038/s41422-022-00646-6
7X1UAPeptideThyrotropin Releasing HormoneTRHHomo sapiensTRH-chim(NtGi2L-Gs-CtGq)/β1/γ23.192022-08-31doi.org/10.1038/s41422-022-00646-6
7X1U (No Gprot) APeptideThyrotropin Releasing HormoneTRHHomo sapiensTRH-3.192022-08-31doi.org/10.1038/s41422-022-00646-6
8WC3AAmineTrace Amine ReceptorsTA1Mus musculusSEP-363856-chim(NtGi1-Gs)/β1/γ232023-12-27doi.org/10.1016/j.cell.2023.10.014
8WC3 (No Gprot) AAmineTrace Amine ReceptorsTA1Mus musculusSEP-363856-32023-12-27doi.org/10.1016/j.cell.2023.10.014
8WC4AAmineTrace Amine ReceptorsTA1Mus musculusZH8651-chim(NtGi1-Gs)/β1/γ23.12023-12-27doi.org/10.1016/j.cell.2023.10.014
8WC4 (No Gprot) AAmineTrace Amine ReceptorsTA1Mus musculusZH8651-3.12023-12-27doi.org/10.1016/j.cell.2023.10.014
8WC5AAmineTrace Amine ReceptorsTA1Mus musculusTetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ23.32023-12-27doi.org/10.1016/j.cell.2023.10.014
8WC5 (No Gprot) AAmineTrace Amine ReceptorsTA1Mus musculusTetramethylammonium Ion-3.32023-12-27doi.org/10.1016/j.cell.2023.10.014
8WC6AAmineTrace Amine ReceptorsTA1Mus musculus2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ23.22023-12-27doi.org/10.1016/j.cell.2023.10.014
8WC6 (No Gprot) AAmineTrace Amine ReceptorsTA1Mus musculus2-Phenylethylamine-3.22023-12-27doi.org/10.1016/j.cell.2023.10.014
8WC7AAmineTrace Amine ReceptorsTA1Mus musculusZH8667-chim(NtGi1-Gs)/β1/γ23.12023-12-27doi.org/10.1016/j.cell.2023.10.014
8WC7 (No Gprot) AAmineTrace Amine ReceptorsTA1Mus musculusZH8667-3.12023-12-27doi.org/10.1016/j.cell.2023.10.014
8WC8AAmineTrace Amine ReceptorsTA1Homo sapiensZH8651-chim(NtGi1-Gs)/β1/γ22.92023-12-27doi.org/10.1016/j.cell.2023.10.014
8WC8 (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensZH8651-2.92023-12-27doi.org/10.1016/j.cell.2023.10.014
8WC9AAmineTrace Amine ReceptorsTA1Mus musculusZH8651-chim(NtGi1-Gs-CtGq)/β1/γ23.22023-12-27doi.org/10.1016/j.cell.2023.10.014
8WC9 (No Gprot) AAmineTrace Amine ReceptorsTA1Mus musculusZH8651-3.22023-12-27doi.org/10.1016/j.cell.2023.10.014
8WCAAAmineTrace Amine ReceptorsTA1Homo sapiens2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ23.482023-12-27doi.org/10.1016/j.cell.2023.10.014
8WCA (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiens2-Phenylethylamine-3.482023-12-27doi.org/10.1016/j.cell.2023.10.014
8WCBAAmineTrace Amine ReceptorsTA1Mus musculusCyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ23.12023-12-27doi.org/10.1016/j.cell.2023.10.014
8WCB (No Gprot) AAmineTrace Amine ReceptorsTA1Mus musculusCyclohexylammonium Ion-3.12023-12-27doi.org/10.1016/j.cell.2023.10.014
8WCCAAmineTrace Amine ReceptorsTA1Mus musculusCyclohexylammonium Ion--3.042023-12-27doi.org/10.1016/j.cell.2023.10.014
8ZSJAAmineTrace Amine ReceptorsTA1Homo sapiens--chim(NtGi1L-Gs-CtGq)/β1/γ22.82024-07-24doi.org/10.1016/j.celrep.2024.114505
8ZSJ (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiens--2.82024-07-24doi.org/10.1016/j.celrep.2024.114505
8ZSPAAmineTrace Amine ReceptorsTA1Homo sapiensLSD-chim(NtGi1L-Gs-CtGq)/β1/γ23.142024-07-24doi.org/10.1016/j.celrep.2024.114505
8ZSP (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensLSD-3.142024-07-24doi.org/10.1016/j.celrep.2024.114505
8ZSSAAmineTrace Amine ReceptorsTA1Homo sapiensRO5263397-chim(NtGi1-Gs)/β1/γ23.072024-07-24doi.org/10.1016/j.celrep.2024.114505
8ZSS (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensRO5263397-3.072024-07-24doi.org/10.1016/j.celrep.2024.114505
8ZSVAAmineTrace Amine ReceptorsTA1Mus musculusRO5263397-chim(NtGi1-Gs)/β1/γ22.962024-07-24doi.org/10.1016/j.celrep.2024.114505
8ZSV (No Gprot) AAmineTrace Amine ReceptorsTA1Mus musculusRO5263397-2.962024-07-24doi.org/10.1016/j.celrep.2024.114505
8UHBAAmineTrace Amine ReceptorsTA1Homo sapiensRO5256390-Gs/β1/γ23.352024-01-10doi.org/10.1038/s41467-023-44601-4
8UHB (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensRO5256390-3.352024-01-10doi.org/10.1038/s41467-023-44601-4
8W87AAmineTrace Amine ReceptorsTA1Homo sapiensMETH-chim(NtGi1L-Gs)/β1/γ22.82023-11-22doi.org/10.1038/s41586-023-06775-1
8W87 (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensMETH-2.82023-11-22doi.org/10.1038/s41586-023-06775-1
8W88AAmineTrace Amine ReceptorsTA1Homo sapiensSEP-363856-Gs/β1/γ22.62023-11-22doi.org/10.1038/s41586-023-06775-1
8W88 (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensSEP-363856-2.62023-11-22doi.org/10.1038/s41586-023-06775-1
8W89AAmineTrace Amine ReceptorsTA1Homo sapiensPEA-chim(NtGi1L-Gs)/β1/γ232023-11-22doi.org/10.1038/s41586-023-06775-1
8W89 (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensPEA-32023-11-22doi.org/10.1038/s41586-023-06775-1
8W8AAAmineTrace Amine ReceptorsTA1Homo sapiensRO5256390-chim(NtGi1L-Gs)/β1/γ22.82023-11-22doi.org/10.1038/s41586-023-06775-1
8W8A (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensRO5256390-2.82023-11-22doi.org/10.1038/s41586-023-06775-1
8JLJAAmineTrace Amine ReceptorsTA1Mus musculusT1AM-chim(NtGi1-Gs)/β1/γ23.12023-11-15doi.org/10.1038/s41586-023-06804-z
8JLJ (No Gprot) AAmineTrace Amine ReceptorsTA1Mus musculusT1AM-3.12023-11-15doi.org/10.1038/s41586-023-06804-z
8JLKAAmineTrace Amine ReceptorsTA1Mus musculusUlotaront-chim(NtGi1-Gs)/β1/γ23.222023-11-15doi.org/10.1038/s41586-023-06804-z
8JLK (No Gprot) AAmineTrace Amine ReceptorsTA1Mus musculusUlotaront-3.222023-11-15doi.org/10.1038/s41586-023-06804-z
8JLNAAmineTrace Amine ReceptorsTA1Homo sapiensT1AM-Gs/β1/γ23.242023-11-15doi.org/10.1038/s41586-023-06804-z
8JLN (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensT1AM-3.242023-11-15doi.org/10.1038/s41586-023-06804-z
8JLOAAmineTrace Amine ReceptorsTA1Homo sapiensUlotaront-Gs/β1/γ23.522023-11-15doi.org/10.1038/s41586-023-06804-z
8JLO (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensUlotaront-3.522023-11-15doi.org/10.1038/s41586-023-06804-z
8JLPAAmineTrace Amine ReceptorsTA1Homo sapiensRalmitaront-Gs/β1/γ23.232023-11-15doi.org/10.1038/s41586-023-06804-z
8JLP (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensRalmitaront-3.232023-11-15doi.org/10.1038/s41586-023-06804-z
8JLQAAmineTrace Amine ReceptorsTA1Homo sapiensFenoldopam-Gs/β1/γ22.842023-11-15doi.org/10.1038/s41586-023-06804-z
8JLQ (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensFenoldopam-2.842023-11-15doi.org/10.1038/s41586-023-06804-z
8JLRAAmineTrace Amine ReceptorsTA1Homo sapiensA77636-chim(NtGi1-Gs)/β1/γ232023-11-15doi.org/10.1038/s41586-023-06804-z
8JLR (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensA77636-32023-11-15doi.org/10.1038/s41586-023-06804-z
8JSOAAmineTrace Amine ReceptorsTA1Homo sapiensAMPH-chim(NtGi1-Gs)/β1/γ23.42023-11-15doi.org/10.1038/s41586-023-06804-z
8JSO (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensAMPH-3.42023-11-15doi.org/10.1038/s41586-023-06804-z
9JKQAAmineTrace Amine ReceptorsTA1Homo sapiensMETH-Gs/β1/γ22.662024-10-16doi.org/10.1021/acs.jmedchem.4c01961
9JKQ (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensMETH-2.662024-10-16doi.org/10.1021/acs.jmedchem.4c01961
8PM2AAmineTrace Amine ReceptorsTA7Mus musculusDMCH-Gs/β1/γ22.922023-08-09doi.org/10.1101/2023.07.07.547762
8PM2 (No Gprot) AAmineTrace Amine ReceptorsTA7Mus musculusDMCH-2.922023-08-09doi.org/10.1101/2023.07.07.547762
7RKYAOtherUnclassifiedUS27Human betaherpesvirus 5-GDPGi1/β1/γ23.82022-01-26doi.org/10.1126/sciadv.abl5442
7RKY (No Gprot) AOtherUnclassifiedUS27Human betaherpesvirus 5-GDP3.82022-01-26doi.org/10.1126/sciadv.abl5442
7RKFAOtherUnclassifiedUS28Human betaherpesvirus 5FractalkineGDPchim(NtGi1-G11)/β1/γ242022-01-26doi.org/10.1126/sciadv.abl5442
7RKF (No Gprot) AOtherUnclassifiedUS28Human betaherpesvirus 5FractalkineGDP42022-01-26doi.org/10.1126/sciadv.abl5442
7JHJAOtherUnclassifiedBILF1Human gammaherpesvirus 4--Gi1/β1/γ23.22021-07-07doi.org/10.1016/j.immuni.2021.06.001
7JHJ (No Gprot) AOtherUnclassifiedBILF1Human gammaherpesvirus 4--3.22021-07-07doi.org/10.1016/j.immuni.2021.06.001
8K4OAOtherUnclassifiedKSHVHuman gammaherpesvirus 8CXCL1-Gi1/β1/γ13.012024-07-24doi.org/10.1073/pnas.2403217121
8K4O (No Gprot) AOtherUnclassifiedKSHVHuman gammaherpesvirus 8CXCL1-3.012024-07-24doi.org/10.1073/pnas.2403217121
8K4PAOtherUnclassifiedKSHVHuman gammaherpesvirus 8--Gi1/β1/γ12.812024-07-24doi.org/10.1073/pnas.2403217121
8K4P (No Gprot) AOtherUnclassifiedKSHVHuman gammaherpesvirus 8--2.812024-07-24doi.org/10.1073/pnas.2403217121
8Z1EAOtherUnclassifiedUL78Human herpesvirus 5---3.122024-05-15doi.org/10.1038/s41421-024-00684-x
7RKXAOtherUnclassifiedUS27Human betaherpesvirus 5--Gi1/β1/γ23.12022-01-26doi.org/10.1126/sciadv.abl5442
7RKX (No Gprot) AOtherUnclassifiedUS27Human betaherpesvirus 5--3.12022-01-26doi.org/10.1126/sciadv.abl5442
7RKMAOtherUnclassifiedUS28Human betaherpesvirus 5Fractalkine-Gi1/β1/γ23.52022-01-26doi.org/10.1126/sciadv.abl5442
7RKM (No Gprot) AOtherUnclassifiedUS28Human betaherpesvirus 5Fractalkine-3.52022-01-26doi.org/10.1126/sciadv.abl5442
7RKNAOtherUnclassifiedUS28Human betaherpesvirus 5Fractalkine-Gi1/β1/γ23.62022-01-26doi.org/10.1126/sciadv.abl5442
7RKN (No Gprot) AOtherUnclassifiedUS28Human betaherpesvirus 5Fractalkine-3.62022-01-26doi.org/10.1126/sciadv.abl5442
4XT1AOtherUnclassifiedUS28Human cytomegalovirus (strain ad169)Fractalkine--2.892015-03-04doi.org/10.1126/science.aaa5026
4XT3AOtherUnclassifiedUS28Human cytomegalovirus (strain ad169)Fractalkine--3.82015-03-04doi.org/10.1126/science.aaa5026
5WB1AOtherUnclassifiedUS28Human cytomegalovirus (strain towne)---3.512018-06-13doi.org/10.7554/eLife.35850
5WB2AOtherUnclassifiedUS28Human cytomegalovirus (strain towne)CX3CL1.35--3.52018-06-13doi.org/10.7554/eLife.35850
7QVMAPeptideVasopressin and OxytocinOTHomo sapiensOxytocin-chim(NtGi1-Go-CtGq)/β1/γ23.252022-08-10doi.org/10.1038/s41467-022-31325-0
7QVM (No Gprot) APeptideVasopressin and OxytocinOTHomo sapiensOxytocin-3.252022-08-10doi.org/10.1038/s41467-022-31325-0
7RYCAPeptideVasopressin and OxytocinOTHomo sapiensOxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ22.92022-03-09doi.org/10.1038/s41594-022-00728-4
7RYC (No Gprot) APeptideVasopressin and OxytocinOTHomo sapiensOxytocin-2.92022-03-09doi.org/10.1038/s41594-022-00728-4
6TPKAPeptideVasopressin and OxytocinOTHomo sapiensRetosiban--3.22020-08-05doi.org/10.1126/sciadv.abb5419
7DW9APeptideVasopressin and OxytocinV2Homo sapiensAVP-chim(NtGi1-Gs)/β1/γ22.62021-07-21doi.org/10.1038/s41422-021-00480-2
7DW9 (No Gprot) APeptideVasopressin and OxytocinV2Homo sapiensAVP-2.62021-07-21doi.org/10.1038/s41422-021-00480-2
7KH0APeptideVasopressin and OxytocinV2Homo sapiensAVP-chim(NtGi1-Gs)/β1/γ22.82021-05-26doi.org/10.1038/s41422-021-00483-z
7KH0 (No Gprot) APeptideVasopressin and OxytocinV2Homo sapiensAVP-2.82021-05-26doi.org/10.1038/s41422-021-00483-z
7BB6APeptideVasopressin and OxytocinV2Homo sapiensAVP-Gs/β1/γ24.22021-06-02doi.org/10.1126/sciadv.abg5628
7BB6 (No Gprot) APeptideVasopressin and OxytocinV2Homo sapiensAVP-4.22021-06-02doi.org/10.1126/sciadv.abg5628
7BB7APeptideVasopressin and OxytocinV2Homo sapiensAVP-Gs/β1/γ24.42021-06-02doi.org/10.1126/sciadv.abg5628
7BB7 (No Gprot) APeptideVasopressin and OxytocinV2Homo sapiensAVP-4.42021-06-02doi.org/10.1126/sciadv.abg5628
7R0CAPeptideVasopressin and OxytocinV2Homo sapiensAVP-Arrestin24.732022-09-14doi.org/10.1126/sciadv.abo7761
9HAPAPeptideVasopressin and OxytocinV2Homo sapiensTolvaptan--2.52025-06-04doi.org/10.1038/s41467-025-59114-5
9HB3APeptideVasopressin and OxytocinV2Homo sapiensMambaquaretin-1--2.52025-06-04doi.org/10.1038/s41467-025-59114-5
6P9YB1PeptideVIP and PACAPPAC1Homo sapiensPACAP-Gs/β1/γ23.012020-02-05doi.org/10.1016/j.molcel.2020.01.012
6P9Y (No Gprot) B1PeptideVIP and PACAPPAC1Homo sapiensPACAP-3.012020-02-05doi.org/10.1016/j.molcel.2020.01.012
6M1HB1PeptideVIP and PACAPPAC1Homo sapiensMaxadilan-Gs/β1/γ23.62020-03-11doi.org/10.1038/s41422-020-0280-2
6M1H (No Gprot) B1PeptideVIP and PACAPPAC1Homo sapiensMaxadilan-3.62020-03-11doi.org/10.1038/s41422-020-0280-2
6M1IB1PeptideVIP and PACAPPAC1Homo sapiensPACAP-Gs/β1/γ23.52020-03-11doi.org/10.1038/s41422-020-0280-2
6M1I (No Gprot) B1PeptideVIP and PACAPPAC1Homo sapiensPACAP-3.52020-03-11doi.org/10.1038/s41422-020-0280-2
8E3XB1PeptideVIP and PACAPPAC1Homo sapiensPACAP27-Gs/β1/γ22.32022-11-23doi.org/10.1038/s41467-022-34629-3
8E3X (No Gprot) B1PeptideVIP and PACAPPAC1Homo sapiensPACAP27-2.32022-11-23doi.org/10.1038/s41467-022-34629-3
6LPBB1PeptideVIP and PACAPPAC1Homo sapiensPACAP-Gs/β1/γ13.92020-03-11doi.org/10.1038/s41594-020-0386-8
6LPB (No Gprot) B1PeptideVIP and PACAPPAC1Homo sapiensPACAP-3.92020-03-11doi.org/10.1038/s41594-020-0386-8
6VN7B1PeptideVIP and PACAPVPAC1Homo sapiensPACAP-Gs/β1/γ23.22020-09-02doi.org/10.1038/s41467-020-17933-8
6VN7 (No Gprot) B1PeptideVIP and PACAPVPAC1Homo sapiensPACAP-3.22020-09-02doi.org/10.1038/s41467-020-17933-8
8E3YB1PeptideVIP and PACAPVPAC1Homo sapiensPACAP27-Gs/β1/γ22.32022-11-23doi.org/10.1038/s41467-022-34629-3
8E3Y (No Gprot) B1PeptideVIP and PACAPVPAC1Homo sapiensPACAP27-2.32022-11-23doi.org/10.1038/s41467-022-34629-3
8E3ZB1PeptideVIP and PACAPVPAC1Homo sapiensVIP-Gs/β1/γ22.72022-11-23doi.org/10.1038/s41467-022-34629-3
8E3Z (No Gprot) B1PeptideVIP and PACAPVPAC1Homo sapiensVIP-2.72022-11-23doi.org/10.1038/s41467-022-34629-3
7VQXB1PeptideVIP and PACAPVPAC1Homo sapiensPACAP27-Gs/β1/γ22.742022-05-18doi.org/10.1038/s41467-022-30041-z
7VQX (No Gprot) B1PeptideVIP and PACAPVPAC1Homo sapiensPACAP27-2.742022-05-18doi.org/10.1038/s41467-022-30041-z
7WBJB1PeptideVIP and PACAPVPAC1Homo sapiensPACAP27-Gs/β1/γ23.422022-05-18doi.org/10.1038/s41467-022-30041-z
7WBJ (No Gprot) B1PeptideVIP and PACAPVPAC1Homo sapiensPACAP27-3.422022-05-18doi.org/10.1038/s41467-022-30041-z
8W1AAOtherUclassifiedORF74Human gammaherpesvirus 8---2.892025-08-27To be published
9EHSANucleotideAdenosineA3AHomo sapiensLUF7602--3.22025-08-20doi.org/10.1038/s41467-025-62872-x
9IQRAAmineAdrenegicα2aHomo sapiens-Muscarinic toxin 3-3.42025-07-23To be published
9IQSAAmineAcetylcholine (muscarinic)M4Homo sapiens-Muscarinic toxin 3-3.62025-07-23To be published
9IQVAAmineAdrenegicAlpha1AHomo sapiens-Muscarinic toxin 3-3.32025-07-23To be published
9J05ANucleotideP2YP2Y14Homo sapiens---3.22025-08-06To be published
9JGKAAmine5-Hydroxytryptamine5-HT2BHomo sapiensBalovaptan--3.62025-07-16To be published
9KGKAOrphanOrphanLGR4Homo sapiens---2.632025-07-16To be published
9KHHAOrphanOrphanLGR4Homo sapiensNorrin--3.652025-07-16To be published
9OQ0CSensoryTaste1TAS1R2; TAS1R3Homo sapiens; mus musculus---3.672025-08-27To be published
9PLNAAmineAdrenegicα2aHomo sapiensN-(5-methylnaphthalen-1-yl)pyridin-4-amine--2.82025-08-20To be published
9PQDAAmineAdrenegicα2aHomo sapiens(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole--3.292025-08-20To be published
9S37AOrphanOrphanLGR4Homo sapiensNB21--3.942025-07-30To be published
9UT8CSensoryTaste1TAS1R2; TAS1R3Homo sapiens---3.412025-07-16doi.org/10.1038/s41586-025-09302-6
9UTACSensoryTaste1TAS1R2; TAS1R3Homo sapiens---3.772025-07-16doi.org/10.1038/s41586-025-09302-6
9UTBCSensoryTaste1TAS1R2; TAS1R3Homo sapiensSucralose--3.592025-07-16doi.org/10.1038/s41586-025-09302-6
9V0UB2AdhesionAdhesionADGRD1Homo sapiens--chim(NtGi1-G13)/β1/γ23.512025-07-30doi.org/10.1016/j.bbrc.2025.152165
9V0U (No Gprot) B2AdhesionAdhesionADGRD1Homo sapiens--3.512025-07-30doi.org/10.1016/j.bbrc.2025.152165
8YKDB2AdhesionAdhesionADGRG2Mus musculusDehydroepiandrosterone-chim(NtGi1-Gs)/β1/γ22.92025-08-13doi.org/10.1038/s41589-025-01896-2
8YKD (No Gprot) B2AdhesionAdhesionADGRG2Mus musculusDehydroepiandrosterone-2.92025-08-13doi.org/10.1038/s41589-025-01896-2
9IV6AOrphanOrphanGPR4Homo sapiens--chim(NtGi1-Gs)/β1/γ22.712025-07-30To be published
9IV6 (No Gprot) AOrphanOrphanGPR4Homo sapiens--2.712025-07-30To be published
9K3FAPeptideMelanocortinMC3Homo sapiens--chim(NtGi1-Gs)/β1/γ22.752025-08-06doi.org/10.1016/j.str.2025.03.004
9K3F (No Gprot) APeptideMelanocortinMC3Homo sapiens--2.752025-08-06doi.org/10.1016/j.str.2025.03.004
9K3HAPeptideMelanocortinMC5Homo sapiens--chim(NtGi1-Gs)/β1/γ22.862025-08-06doi.org/10.1016/j.str.2025.03.004
9K3H (No Gprot) APeptideMelanocortinMC5Homo sapiens--2.862025-08-06doi.org/10.1016/j.str.2025.03.004
9K3KAPeptideMelanocortinMC4Homo sapiens--chim(NtGi1-Gs)/β1/γ23.122025-08-06doi.org/10.1016/j.str.2025.03.004
9K3K (No Gprot) APeptideMelanocortinMC4Homo sapiens--3.122025-08-06doi.org/10.1016/j.str.2025.03.004
9K3LAPeptideMelanocortinMC2Homo sapiens--chim(NtGi1-Gs)/β1/γ23.012025-08-06doi.org/10.1016/j.str.2025.03.004
9K3L (No Gprot) APeptideMelanocortinMC2Homo sapiens--3.012025-08-06doi.org/10.1016/j.str.2025.03.004
9K3PAPeptideMelanocortinMC1Homo sapiens--chim(NtGi1-Gs)/β1/γ22.982025-08-06doi.org/10.1016/j.str.2025.03.004
9K3P (No Gprot) APeptideMelanocortinMC1Homo sapiens--2.982025-08-06doi.org/10.1016/j.str.2025.03.004
9EBIANucleotideAdenosineA3AHomo sapiensPiclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ23.62025-08-20doi.org/10.1038/s41467-025-62872-x
9EBI (No Gprot) ANucleotideAdenosineA3AHomo sapiensPiclidenoson-3.62025-08-20doi.org/10.1038/s41467-025-62872-x
9GG5ALipidProstanoidTXA2Homo sapiensU46619-chim(NtGi2L-Gs-CtGq)/β1/γ23.262025-08-27To be published
9GG5 (No Gprot) ALipidProstanoidTXA2Homo sapiensU46619-3.262025-08-27To be published
9GGGALipidProstanoidTXA2Homo sapiensI-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ23.252025-08-27To be published
9GGG (No Gprot) ALipidProstanoidTXA2Homo sapiensI-BOP-3.252025-08-27To be published
9K07APeptideBombesinBB3Homo sapiensDSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ22.872025-08-27/doi.org/10.1016/j.apsb.2025.06.025
9K07 (No Gprot) APeptideBombesinBB3Homo sapiensDSO-5a-2.872025-08-27/doi.org/10.1016/j.apsb.2025.06.025
9LWPAPeptideBombesinBB3Homo sapiens--chim(NtGi2L-Gs-CtGq)/β1/γ22.932025-07-16doi.org/10.1016/j.apsb.2025.06.025
9LWP (No Gprot) APeptideBombesinBB3Homo sapiens--2.932025-07-16doi.org/10.1016/j.apsb.2025.06.025
8Y73APeptideOpioidμHomo sapiensPeptideMPAM-15Gi1/β1/γ22.842025-08-06To be published
8Y73 (No Gprot) APeptideOpioidμHomo sapiensPeptideMPAM-152.842025-08-06To be published
9DYFAAmine5-Hydroxytryptamine5-HT1AHomo sapiensAsenapine-Gi1/β1/γ22.742025-08-13doi.org/10.1126/sciadv.adu9851
9DYF (No Gprot) AAmine5-Hydroxytryptamine5-HT1AHomo sapiensAsenapine-2.742025-08-13doi.org/10.1126/sciadv.adu9851
9EBHANucleotideAdenosineA3AHomo sapiensAdenosine-Gi1/β1/γ23.62025-08-20doi.org/10.1038/s41467-025-62872-x
9EBH (No Gprot) ANucleotideAdenosineA3AHomo sapiensAdenosine-3.62025-08-20doi.org/10.1038/s41467-025-62872-x
9M0RAPeptideNeuropeptide FFNPFF1Homo sapiensNeuropeptide VF-Gi1/β1/γ22.472025-07-23doi.org/10.1016/j.celrep.2025.116160
9M0R (No Gprot) APeptideNeuropeptide FFNPFF1Homo sapiensNeuropeptide VF-2.472025-07-23doi.org/10.1016/j.celrep.2025.116160
9M1OAPeptideNeuropeptide FFNPFF2Homo sapiensMorphine-Modulating Neuropeptide B-Gi1/β1/γ22.492025-07-23doi.org/10.1016/j.celrep.2025.116160
9M1O (No Gprot) APeptideNeuropeptide FFNPFF2Homo sapiensMorphine-Modulating Neuropeptide B-2.492025-07-23doi.org/10.1016/j.celrep.2025.116160
9M2FAPeptideNeuropeptide FFNPFF1Homo sapiensNeuropeptide FF-Gi1/β1/γ22.932025-07-23doi.org/10.1016/j.celrep.2025.116160
9M2F (No Gprot) APeptideNeuropeptide FFNPFF1Homo sapiensNeuropeptide FF-2.932025-07-23doi.org/10.1016/j.celrep.2025.116160
9M54APeptideNeuropeptide FFNPFF2Homo sapiensNeuropeptide VF-Gi1/β1/γ23.242025-07-23doi.org/10.1016/j.celrep.2025.116160
9M54 (No Gprot) APeptideNeuropeptide FFNPFF2Homo sapiensNeuropeptide VF-3.242025-07-23doi.org/10.1016/j.celrep.2025.116160
8Y72APeptideOpioidμHomo sapiensPeptideBMS-986122Gi1/β1/γ22.652025-08-06To be published
8Y72 (No Gprot) APeptideOpioidμHomo sapiensPeptideBMS-9861222.652025-08-06To be published
9KFIAPeptideRelaxinRXFP3Homo sapiensRelaxin-3-Gi2/β1/γ22.912025-08-13doi.org/10.1038/s42003-025-08220-7
9KFI (No Gprot) APeptideRelaxinRXFP3Homo sapiensRelaxin-3-2.912025-08-13doi.org/10.1038/s42003-025-08220-7
9KFJAPeptideRelaxinRXFP3Homo sapiensPubChem 138319674-Gi2/β1/γ23.12025-08-13doi.org/10.1038/s42003-025-08220-7
9KFJ (No Gprot) APeptideRelaxinRXFP3Homo sapiensPubChem 138319674-3.12025-08-13doi.org/10.1038/s42003-025-08220-7
9KFKAPeptideRelaxinRXFP4Homo sapiensRelaxin-3-Gi2/β1/γ22.952025-08-13doi.org/10.1038/s42003-025-08220-7
9KFK (No Gprot) APeptideRelaxinRXFP4Homo sapiensRelaxin-3-2.952025-08-13doi.org/10.1038/s42003-025-08220-7
9DYDAAmine5-Hydroxytryptamine5-HT1AHomo sapiensAsenapine-Go/β1/γ22.962025-08-13doi.org/10.1126/sciadv.adu9851
9DYD (No Gprot) AAmine5-Hydroxytryptamine5-HT1AHomo sapiensAsenapine-2.962025-08-13doi.org/10.1126/sciadv.adu9851
9DYEAAmine5-Hydroxytryptamine5-HT1AHomo sapiensBuspirone-Go/β1/γ22.92025-08-13doi.org/10.1126/sciadv.adu9851
9DYE (No Gprot) AAmine5-Hydroxytryptamine5-HT1AHomo sapiensBuspirone-2.92025-08-13doi.org/10.1126/sciadv.adu9851
9PLOAAmineAdrenegicα2aHomo sapiensN-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ22.742025-08-20To be published
9PLO (No Gprot) AAmineAdrenegicα2aHomo sapiensN-(5-methylnaphthalen-1-yl)pyridin-4-amine-2.742025-08-20To be published
8Z9OAOrphanOrphanGPR4Homo sapiens--Gs/β1/γ22.42025-07-16To be published
8Z9O (No Gprot) AOrphanOrphanGPR4Homo sapiens--2.42025-07-16To be published
9AU0ALipidProstaglandinDP1Homo sapiensBW245C-Gs/β1/γ22.452025-08-27To be published
9AU0 (No Gprot) ALipidProstaglandinDP1Homo sapiensBW245C-2.452025-08-27To be published
9I52AAmineDopamineD1Homo sapiensA1IZU-Gs/β1/γ22.82025-07-16doi.org/10.1021/acs.jmedchem.5c00294
9I52 (No Gprot) AAmineDopamineD1Homo sapiensA1IZU-2.82025-07-16doi.org/10.1021/acs.jmedchem.5c00294
9I54AAmineDopamineD1Homo sapiensA1IZV-Gs/β1/γ22.722025-07-16doi.org/10.1021/acs.jmedchem.5c00294
9I54 (No Gprot) AAmineDopamineD1Homo sapiensA1IZV-2.722025-07-16doi.org/10.1021/acs.jmedchem.5c00294
9IXJAAmineHistamineH2Homo sapiensHistamine-Gs/β1/γ22.922025-07-30To be published
9IXJ (No Gprot) AAmineHistamineH2Homo sapiensHistamine-2.922025-07-30To be published
9JFTAOrphanOrphanGPR65Homo sapiens--Gs/β1/γ23.272025-08-13doi.org/10.1038/s41422-025-01092-w
9JFT (No Gprot) AOrphanOrphanGPR65Homo sapiens--3.272025-08-13doi.org/10.1038/s41422-025-01092-w
9MD1AAmine5-Hydroxytryptamine5-HT1AHomo sapiensBuspirone-Gz/β1/γ23.032025-08-13doi.org/10.1126/sciadv.adu9851
9MD1 (No Gprot) AAmine5-Hydroxytryptamine5-HT1AHomo sapiensBuspirone-3.032025-08-13doi.org/10.1126/sciadv.adu9851