Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.33 2.05124404
2G.HN.37 2.66362403
3G.S1.02 4.8193446
4G.S2.08 4.94211446
5G.S3.03 5.5106608
6G.S3.04 9.129124117
7G.S3.06 8.547435117
8G.H2.06 5.58658629
9G.H2.07 4.54411609
10G.h2s4.01 9.10743409
11G.S4.04 4.29848409
12G.H3.01 2.04769809
13G.H3.09 5.17561609
14G.H3.13 9.18175406
15G.H3.17 8.7431555
16G.S5.05 3.609396169
17G.HG.03 2.10405406
18G.HG.16 2.10615404
19G.hgh4.05 7.07266506
20G.hgh4.08 7.27718406
21G.hgh4.11 3.46082405
22G.hgh4.20 3.89417503
23G.hgh4.21 3.91437404
24G.H4.03 2.73709404
25G.H4.08 5.0559493
26G.H4.10 8.63978507
27G.H4.12 5.10406594
28G.H4.15 6.96845408
29G.h4s6.12 4.15118402
30G.h4s6.20 4.51027444
31G.S6.02 7.9343408
32G.S6.05 6.06052595
33G.H5.03 3.517154169
34G.H5.05 4.6199445
35G.H5.08 5.40058648
36G.H5.17 4.44491745
37G.H5.20 3.89063408
38b.1x3 1.48184401
39b.1x4 1.80097508
40b.1x11 2.37079408
41b.lhb1x3 2.95929402
42b.lhb1x6 4.193885123
43b.b1x4 3.63966437
44b.l1x3 7.93623639
45b.l1x6 9.49037559
46b.b2x1 5.69208558
47b.b2x5 6.34902637
48b.b3x3 3.72671508
49b.l3x2 6.292235159
50b.b4x3 3.98146407
51b.b4x6 7.93934839
52b.b4x7 7.74985438
53b.l4x2 9.30091434
54b.b5x2 7.60945437
55b.b5x3 6.95712539
56b.b5x7 5.09457407
57b.l5x1 4.24315408
58b.l5x5 9.88464509
59b.b6x1 4.28937459
60b.b6x5 4.07511406
61b.b7x1 4.97571504
62b.l7x4 3.11243409
63b.b8x4 5.58008506
64b.l9x3 6.43694679
65b.l9x6 5.5451608
66b.b10x5 4.68378509
67b.b11x4 5.07954479
68b.l11x2 6.93165579
69b.b12x6 8.5203678
70b.b13x7 7.55863567
71b.l13x3 7.27828669
72b.l13x6 6.27547429
73b.l13x7 4.56886469
74b.b15x1 6.53338569
75b.l15x1 4.90814527
76b.l15x2 6.33537469
77b.b16x4 9.1194466
78b.b16x6 7.88727768
79b.b17x5 6.06951527
80b.b17x7 7.98411428
81b.l17x3 8.05611729
82b.l17x6 6.84998529
83b.b18x3 4.80267428
84b.l18x1 6.674097136
85b.l18x3 8.281324135
86b.b19x2 6.30006626
87b.b19x4 6.22133428
88b.l19x1 6.13997429
89b.l19x2 7.13008529
90b.b20x2 7.11865426
91b.b20x4 11.01528
92b.b20x6 6.05096726
93b.b21x1 5.92148627
94b.b21x5 5.39498404
95b.b21x7 5.57965605
96b.l21x2 5.19491404
97b.b22x5 6.00401407
98b.l22x5 7.300745129
99b.b23x6 7.12056147
100b.l23x1 6.19348556
101b.b24x4 7.48664146
102b.b24x6 6.950934148
103b.b25x3 5.397615145
104b.l25x3 8.680565109
105b.l25x6 11.8838558
106b.l27x1 9.85444759
107b.l27x2 7.459084109
108b.b28x3 4.99929437
109b.b28x4 6.874954106
110b.b28x6 8.425395109
111g.l1x4 3.92765528
112g.h2x11 8.634134136
113g.ctx3 7.13509409
114g.ctx6 3.249735126
115g.ctx14 5.37237439
116g.ctx15 6.76195439
117g.ctx16 5.20222838
118Lig 11.7463710
119NT 135.233715
1201x36 3.83047515
1211x39 4.49853617
1221x43 5.96113617
1231x50 4.26276409
1241x60 3.85051407
1252x39 6.6213409
1262x40 4.52101409
1272x50 6.80739608
1282x53 5.83849518
1292x57 6.27561417
1302x60 5.24727416
131E1 7.295271113
1323x32 5.72508516
1333x33 5.78772417
1343x34 4.5132689
1353x35 4.96351405
1363x36 5.91974416
1373x40 6.62709518
1383x42 7.81626689
1393x44 4.30443408
1403x46 8.45771409
1413x49 6.2513548
1423x54 3.591254178
143I2 5.196541647
1444x50 6.67371489
1454x53 4.04359589
1464x60 7.47781418
1474x64 9.10897408
148E2 9.09535915
149E2x51 10.3256518
1505x40 2.87462404
1515x41 6.39878416
1525x58 5.586564189
1535x68 5.56649449
1546x29 1.5183405
1556x44 4.725465189
1566x47 6.59144418
1576x48 7.51226518
1586x51 4.43479417
159E3 2.8421814
1607x38 5.60478417
1617x45 5.85929419
1628x58 1.98185405
163G.H1.07 1.03442500
164H.hahb.04 0.0354271400
165H.HB.05 0.0694625500
166H.hbhc.04 0.0808021600
167H.HC.06 0.079099400
168H.hchd.01 0.0384917500
169H.hdhe.01 0.0449583500
170H.HE.04 0.0986771400
171H.HE.05 0.0513292500
172G.hfs2.03 0.0484427400
173I3 2.85138540
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1G.HN.40 b.b5x3 10.19234.95312NoYes379
2b.b3x6 b.l1x3 26.643210.368NoYes099
3b.b3x6 b.l3x2 26.86878.29016NoYes099
4b.b4x6 b.l1x3 18.81524.85597YesYes399
5G.hns1.01 b.l3x2 28.65584.06365NoYes1549
6G.S1.03 G.hns1.01 29.795116.0228NoNo094
7G.S1.03 G.S3.06 30.01983.49665NoYes097
8G.S3.06 b.l5x5 32.263717.3344YesYes079
9b.l3x1 b.l5x5 31.78278.22616NoYes099
10b.l1x6 b.l3x1 15.99978.35066YesNo599
11b.l1x6 b.l27x1 16.1721.4929YesYes599
12G.H3.17 b.l27x1 49.96173.82614YesYes559
13G.H3.17 b.l23x1 49.96328.44321YesYes556
14b.l21x7 b.l23x1 1003.12931NoYes056
15b.l21x7 b.l23x2 99.98927.32193NoNo058
16b.b23x6 b.l23x2 99.90883.54679YesNo078
17b.b23x6 b.b24x6 99.27128.144YesYes1478
18b.b21x7 b.b24x6 99.60828.54093YesYes058
19b.b21x5 b.b21x7 99.495910.3266YesYes045
20b.b21x5 b.h2x1 99.43315.89324YesNo045
21b.h2x1 b.h2x5 99.40533.54669NoNo055
22b.h2x5 b.lhb1x3 49.81693.24457NoYes052
23b.l22x5 b.lhb1x3 49.614.06498YesYes092
24b.l22x5 g.ctx6 98.07914.61312YesYes1296
25g.ctx3 g.ctx6 97.92065.77714YesYes096
26b.l22x1 g.ctx3 97.54048.40955NoYes099
27b.l22x1 g.ctx5 97.44523.35952NoNo099
28b.lhb1x11 g.ctx5 94.06874.37272NoNo049
29b.b25x7 b.lhb1x11 93.97245.91861NoNo074
30b.b25x7 b.b28x6 91.407816.6775NoYes079
31b.b28x4 b.b28x6 89.03615.70527YesYes1069
32b.b1x5 b.b28x4 87.10815.91946NoYes036
33b.b1x5 b.l1x1 87.00919.5592NoNo037
34I1x48 b.l1x1 87.44787.7482NoNo087
35I1x48 I1x51 87.34823.72848NoNo087
362x41 I1x51 87.24823.49892NoNo067
372x41 4x43 87.14812.99146NoNo066
382x38 4x43 61.89175.0871NoNo076
392x38 I2 45.36436.34692NoYes477
40b.b2x1 b.l3x1 15.98999.50216YesNo589
41b.b2x1 b.l27x1 83.2645.30106YesYes589
42b.l25x6 b.l27x1 49.964719.9646YesYes589
43b.l23x1 b.l25x6 50.015314.3531YesYes568
44b.h2x5 b.l24x2 49.57974.35724NoNo056
45b.l22x5 b.l24x2 49.51078.50353YesNo096
46G.H3.01 G.s4h3.02 29.95281.5287YesNo099
47G.HG.03 G.s4h3.02 30.45832.7041YesNo069
48G.HG.03 G.s5hg.01 31.20753.90218YesNo069
49G.S5.07 G.s5hg.01 31.74132.98597NoNo099
50G.S5.07 G.s6h5.01 32.24644.12165NoNo099
51G.S5.05 G.s6h5.01 32.495.18762YesNo1699
52G.S5.03 G.S5.05 18.3643.35422NoYes099
53G.H5.10 G.S5.03 18.62347.81252NoNo079
54G.H5.10 G.S6.02 37.639611.3611NoYes078
55G.H5.13 G.S6.02 37.970410.4883NoYes088
565x68 G.H5.13 38.07457.01651YesNo498
575x68 G.H5.16 39.7187.7533YesNo496
58G.H5.16 I2 39.67194.5446NoYes467
59G.S5.05 G.S6.04 18.37263.66855YesNo099
60G.H5.10 G.S6.04 18.891410.3825NoNo079
61G.H3.01 G.s1h1.04 27.68696.5912YesNo099
62G.H2.07 b.l9x6 32.90023.46273YesYes098
63G.H2.06 b.l9x6 25.85853.59333YesYes098
64G.H2.06 b.l17x6 12.73357.62003YesYes299
65G.H2.04 G.H2.07 32.06276.98833NoYes099
66G.H2.04 G.H3.08 31.94916.78808NoNo098
67G.H2.06 b.l19x1 12.61223.10917YesYes299
68b.b2x1 b.b6x1 67.19025.65562YesYes589
69G.H3.08 G.S4.04 31.73816.62569NoYes089
70G.H3.09 G.S4.04 21.53144.51645YesYes099
71G.H4.10 G.H4.14 27.52339.96262YesNo075
72G.H3.06 G.H4.14 28.24253.0904NoNo065
73G.H3.06 G.H4.15 19.05379.14749NoYes068
74G.H4.10 G.hgh4.08 18.527711.2345YesYes076
75G.H4.07 G.S6.05 10.168812.17NoYes955
762x38 3x49 16.42527.58804NoYes478
772x42 3x46 15.54575.29668NoYes089
782x42 3x49 17.21495.30044NoYes088
79b.l17x5 b.l17x6 12.52843.45522NoYes269
80b.l17x5 b.l19x2 24.78593.24552NoYes269
81b.l17x3 b.l19x2 22.59594.38847YesYes299
82b.b20x6 b.l17x3 18.70163.33078YesYes269
83b.b17x7 b.b20x6 13.592410.4514YesYes286
84b.b17x7 b.b21x1 10.9194.16688YesYes287
85b.l17x5 b.l19x1 12.49844.16752NoYes269
86b.l11x1 b.l9x6 17.66666.38309NoYes098
87b.b11x6 b.l11x1 17.54673.49179NoNo099
88b.b11x6 b.l9x3 16.931314.0839NoYes799
89b.b11x4 b.l9x3 15.50174.99934YesYes799
90b.b10x3 b.b11x4 15.41293.21523NoYes089
91b.b10x3 b.b6x2 12.36774.81861NoNo088
92b.b10x2 b.b6x2 12.24513.06101NoNo068
93b.b10x2 b.b10x4 12.12254.39348NoNo066
944x43 4x47 25.20483.54746NoNo065
952x45 4x47 25.08025.25008NoNo095
962x45 3x42 20.343514.0627NoYes899
972x49 3x42 21.18163.26582NoYes099
982x49 3x39 21.04935.24092NoNo099
992x53 3x39 17.887610.6998YesNo089
1002x53 Lig 14.7723.16035YesYes180
101G.s1h1.04 H.hehf.07 27.20530.0808333NoNo090
102H.HF.03 H.hehf.07 26.96450.0674792NoNo000
103H.HF.03 H.hehf.04 22.39020.0527083NoNo000
104H.HE.12 H.hehf.04 19.26040.0553958NoNo000
105H.HC.04 H.HE.12 19.01960.0252083NoNo000
106H.HC.03 H.HC.04 17.81580.0730625NoNo000
107H.HC.03 H.hbhc.04 17.57510.100458NoYes000
108H.HB.12 H.hbhc.04 13.7230.0682708NoYes000
109H.HB.08 H.HB.12 13.24150.0762292NoNo000
110H.HB.08 H.HC.06 12.51920.0884792NoYes000
111H.HB.05 H.HC.06 11.55620.131646YesYes000
112H.HB.05 H.HC.10 10.11170.0784375YesNo000
113b.b6x1 b.l9x6 67.02865.34732YesYes098
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
3x33Lig5.773051YesYes7010
3x36Lig8.734571YesYes6010
5x41Lig5.98451YesYes6010
7x34Lig7.044031NoYes5010
7x37Lig7.735241NoYes8010
1x43Lig3.369451YesYes7010
2x53Lig3.160351YesYes8010
2x57Lig4.356311YesYes7010
3x32Lig7.903291YesYes6010
7x38Lig9.559911YesYes7010
7x41Lig3.350551NoYes6010
E2Lig16.73581YesYes5010
E3Lig4.30781YesYes4010
7x30Lig4.268791NoYes5010
1x32Lig14.98130NoYes5010
1x36Lig5.643851YesYes5010
1x39Lig4.581YesYes7010
2x60Lig6.079061YesYes6010
E2x52Lig10.4961NoYes5010
1x29Lig7.646691NoYes2010
LigNT77.52841YesYes0501
E1Lig19.76141YesYes3010
NTNT427.2781YesYes5511
E1NT8.276251YesYes3511
1x357x385.118830NoYes6721
1x361x393.958041YesYes5711
1x361x403.563081YesNo5712
1x362x614.65941YesNo5712
1x391x434.271411YesYes7711
1x392x614.153321YesNo7712
1x397x384.540951YesYes7711
1x397x425.487471YesNo7912
1x432x534.555241YesYes7811
1x432x545.552591YesNo7712
1x432x5711.00371YesYes7711
1x437x427.014411YesNo7912
2x533x367.21091YesYes8611
2x533x3910.69981YesNo8912
2x533x403.566211YesYes8812
2x563x323.596670NoYes6621
2x572x614.752631YesNo7712
2x603x283.136871YesNo6712
2x603x328.723321YesYes6611
E1E119.27011YesYes3311
3x26E26.46671NoYes8521
3x26E2x5123.75851NoYes8822
3x323x363.412351YesYes6611
3x334x606.528581YesYes7812
3x335x437.533171YesNo7712
3x363x404.321131YesYes6812
3x406x4810.65351YesYes8822
4x605x439.944911YesNo8722
4x68E211.06211NoYes6521
E2E2x514.962771YesYes5812
E2E212.38721YesYes5511
E2x50E2x523.174970NoNo9521
5x41E27.841911YesYes6511
5x415x434.104691YesNo6712
5x415x447.664041YesNo6611
5x425x446.75660NoNo7621
6x487x415.104731YesNo8621
6x517x336.266251YesNo7721
6x517x374.500751YesNo7821
E3E35.550991YesYes4411
7x307x343.036061NoNo5511
7x337x377.985961NoNo7811
E2NT3.491231YesYes5511
2x573x324.98981YesYes7611
2x602x643.049851YesNo6712
2x64E13.177651NoYes7321
E1E26.523191YesYes3511
3x293x333.316090NoYes5721
7x29E33.120930NoYes3421
7x347x383.199431NoYes5711
2x64E2x523.193951NoNo7521
1x291x334.083891NoNo2312
7x33Lig3.301811NoYes7010
5x44Lig9.523631NoYes6010
1x25Lig4.405870NoYes0010
1x28Lig2.912730NoYes0010
2x65Lig2.762990NoYes4010
6x54E32.439910NoYes5421
1x24NT2.34651NoYes0521
6x53Lig2.33950NoYes4010
5x486x522.116580NoNo4621
2x68Lig2.11650NoYes3010
1x21Lig2.10580NoYes0010
6x52Lig2.0681NoYes6010
3x24E12.026981NoYes3321
1x26Lig1.707830NoYes0010
2x67E11.534420NoYes3321
1x362x621.3281YesNo5312
1x22Lig1.094030NoYes0010
7x27E30.7683250NoYes4421
1x23Lig0.60640NoYes0010
6x55E30.5598540NoYes7421
6x56Lig0.4818330NoYes0010
7x28E30.4380NoYes2421
1x19NT0.4350NoYes0521
2x66E10.1688330NoYes3321
3x21E10.1643330NoYes0321
2x69E10.07481250NoYes4321

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
88.57Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
65.85Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
65.79Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
65.79Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
64.10Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
63.89Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
63.16Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
62.16Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
61.54Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
61.54Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
61.11Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
61.11Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
60.53Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
60.53Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
60.00Consensuspth_onOrthosteric Ligandpth1_on pth2_on
59.46Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
59.46Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
59.46Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
59.46Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
59.46Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
58.97Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
58.33Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
58.33Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
57.89Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
57.50Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
56.76Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
56.76Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
56.76Consensusglp_onOrthosteric Ligandglp1_on glp2_on
56.76Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
55.56Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
55.26Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
55.26Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
55.26Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
55.00Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
54.29Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
54.29Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
54.05Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
54.05Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
54.05Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
54.05Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
54.05Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
53.85Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
53.49Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
52.78Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
52.78Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
52.78Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
52.78Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
52.78Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
52.63Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
52.63Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
52.63Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
52.63Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
52.63Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
52.50Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
52.38Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
51.35Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
51.35Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
51.35Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
51.35Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
51.28Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
51.28Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
51.28Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
51.28Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
51.22Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
50.00Single6FJ3PTH6FJ3-PTH1-PTH
50.00Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
50.00Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
50.00Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
50.00Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
50.00Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
50.00Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
50.00Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
48.65Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
47.62Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
47.62Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
47.62Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
47.50Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
47.37Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
47.37Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
47.37Consensuspac_onOrthosteric Ligandpac1_on
47.22Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
46.51Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
46.15Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
46.15Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
45.95Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
45.95Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
45.24Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
45.00Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
45.00Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
44.74Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
44.74Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
44.74Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
44.74Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
44.44Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
43.90Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
43.90Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
43.59Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
43.59Consensuscalcitonin_onOrthosteric Ligandctlike_on
43.18Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
42.50Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
42.50Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
42.50Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
41.46Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
41.46Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
41.03Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
40.54Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
40.00Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
39.53Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
39.47Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
39.47Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
38.89Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
38.64Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
38.64Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
38.46Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
38.10Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
38.10Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
37.21Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
36.84Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
36.36Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
35.71Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
35.71Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
35.56Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
35.14Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
35.00Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
34.88Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
34.88Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
34.15Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
34.09Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
34.09Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
34.09Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
34.09Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
33.33Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
32.56Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
32.56Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
32.56Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
32.56Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
31.58Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
31.37Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
31.11Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
31.11Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
30.77Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
30.23Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
30.00Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
29.41Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
29.17Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
29.17Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
28.89Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
28.89Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
28.57Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
28.26Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
28.26Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
28.21Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
27.91Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
27.91Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
27.91Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
27.91Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
27.66Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
27.66Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
27.66Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
27.27Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
27.27Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
27.08Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
26.83Single4XT1Fractalkine4XT1-US28-Fractalkine
26.83Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
26.83Single7QA8Peptide7QA8-STE2-Peptide
26.83Single7QA8Peptide7QA8-STE2-Peptide
26.67Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
26.67Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
26.67Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
26.67Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
26.67Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
26.67Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
26.67Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
26.67Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
26.53Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
26.19Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
26.19Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
26.09Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
26.09Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
26.09Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
26.09Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
25.64Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
25.58Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
25.53Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
25.00Single6IGKEndothelin-36IGK-ETB-Endothelin-3
25.00Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
25.00Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
25.00Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
25.00Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
25.00Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
25.00Consensusbombesin_onOrthosteric Ligandbb2_on
25.00Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
25.00Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
25.00Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
25.00Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
25.00Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
25.00Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
24.44Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
24.44Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
24.44Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
24.44Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
24.39Single4UG2CGS216804UG2-A2A-CGS21680
24.39Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
24.39Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
24.39Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
24.39Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
23.91Single4XT3Fractalkine4XT3-US28-Fractalkine
23.91Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
23.81Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
23.81Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
23.81Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
23.68Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
23.40Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
23.40Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
23.40Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
23.40Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
23.40Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
23.40Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
23.40Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
23.26Single3QAKUK-4320973QAK-A2A-UK-432097
23.26Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
23.26Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
23.26Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
23.26Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
23.08Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
23.08Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
22.92Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
22.73Single5WF5UK-4320975WF5-A2A-UK-432097
22.73Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
22.73Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
22.73Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
22.73Consensusangiotensin_onOrthosteric Ligandat1_on
22.73Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
22.73Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
22.73Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
22.73Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
22.50Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
22.50Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
22.50Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
22.50Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
22.50Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
22.50Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
22.50Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
22.50Consensuslpl_offOrthosteric Ligands1p_off lpa_off
22.45Single5GLHEndothelin-15GLH-ETB-Endothelin-1
22.45Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
22.22Single5U09Taranabant5U09-CB1-Taranabant
22.22Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
22.22Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
22.22Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
22.22Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
22.22Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
21.95Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
21.95Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
21.95Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
21.95Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
21.74Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
21.74Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
21.74Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
21.74Single8ZRTET-18ZRT-ETB-ET-1
21.74Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
21.74Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
21.74Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
21.74Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
21.62Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
21.62Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
21.57Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
21.43Single3NY9ICI118-5513NY9-β2-ICI118-551
21.43Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
21.43Single7SK9CCX6627SK9-ACKR3-CCX662
21.43Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
21.43Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
21.43Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
21.28Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
21.28Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
21.05Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
21.05Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
21.05Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
21.05Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
20.93Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
20.93Single8WDTphotoNECA8WDT-A2A-photoNECA
20.93Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
20.93Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
20.93Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
20.93Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
20.93Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
20.93Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
20.93Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
20.83Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
20.83Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
20.83Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
20.51Single5C1MBU725C1M-μ-BU72
20.51Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
20.51Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
20.51Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
20.51Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
20.51Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
20.51Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
20.51Single9B9ZA1AKO9B9Z-CB1-A1AKO
20.51Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
20.51Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
20.51Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
20.45Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
20.45Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
20.45Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
20.45Single7XNACYN1548067XNA-SST2-CYN154806
20.45Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
20.45Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
20.45Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
20.45Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
20.45Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
20.41Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
20.41Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
20.41Single8IY6Endothelin-18IY6-ETB-Endothelin-1
20.41Consensusendothelin_onOrthosteric Ligandetb_on eta_on
20.37Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
20.37Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
20.00Single2YDVNECA2YDV-A2A-NECA
20.00Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
20.00Single4UHRCGS216804UHR-A2A-CGS21680
20.00Single5G53NECA5G53-A2A-NECA-Gs
20.00Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
20.00Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
20.00Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
20.00Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
20.00Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
20.00Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
20.00Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
20.00Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
20.00Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
20.00Single8E0GBU728E0G-μ-BU72
20.00Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
20.00Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
20.00Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
20.00Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
20.00Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
20.00Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
20.00Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
20.00Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
20.00Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
20.00Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
20.00Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
20.00Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
20.00Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
20.00Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
20.00Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
20.00Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
20.00Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
19.61Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
19.61Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
19.57Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
19.57Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
19.57Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
19.57Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
19.57Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
19.57Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
19.57Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
19.57Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
19.57Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
19.57Consensusvasop-oxy_onOrthosteric Ligandv2_on
19.57Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
19.51Single6OS2TRV0266OS2-AT1-TRV026
19.51Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
19.51Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
19.51Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
19.51Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
19.51Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
19.51Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
19.51Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
19.51Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
19.51Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
19.51Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
19.51Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
19.51Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
19.51Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
19.51Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
19.51Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
19.23Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
19.15Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
19.15Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
19.15Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
19.15Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
19.15Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
19.15Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
19.15Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
19.15Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
19.15Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
19.05Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
19.05Single7EZCUKA7EZC-A2A-UKA
19.05Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
19.05Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
19.05Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
19.05Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
19.05Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
19.05Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
19.05Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
19.05Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
19.05Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
19.05Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
19.05Consensuscck_onOrthosteric Ligandccka_on cckb_on
19.05Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
19.05Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
19.05Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
19.05Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
19.05Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
19.05Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
18.92Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
18.92Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
18.87Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
18.75Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
18.75Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
18.75Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
18.75Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
18.75Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
18.60Single5WF6UK-4320975WF6-A2A-UK-432097
18.60Single5ZTYAM102575ZTY-CB2-AM10257
18.60Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
18.60Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
18.60Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
18.60Single8QJ2pN1628QJ2-MC4-pN162-Gs
18.60Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
18.60Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
18.60Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
18.60Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
18.42Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
18.42Single7T32ZM-2413857T32-A2A-ZM-241385
18.42Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
18.42Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
18.42Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
18.42Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
18.42Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
18.42Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
18.42Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
18.37Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
18.37Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
18.37Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
18.37Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
18.37Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
18.33Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
18.18Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
18.18Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
18.18Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
18.18Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
18.18Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.18Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
18.18Consensuslpl_onOrthosteric Ligands1p_on lpa_on
18.18Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
18.18Consensussomatostatin_offOrthosteric Ligandsst2_off
18.00Single6IGLIRL16206IGL-ETB-IRL1620
18.00Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
18.00Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
18.00Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
18.00Consensusbradykinin_onOrthosteric Ligandbk2_on
18.00Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
18.00Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
18.00Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
17.95Single4DAJTiotropium4DAJ-M3-Tiotropium
17.95Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
17.95Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
17.95Single6PS1Timolol6PS1-β2-Timolol
17.95Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
17.95Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
17.95Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
17.95Single7V3ZCP559407V3Z-CB1-CP55940
17.95Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
17.95Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
17.95Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
17.95Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
17.95Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
17.95Single8T1WCVN4248T1W-GPR6-CVN424
17.95Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.95Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.95Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.95Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
17.95Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
17.95Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
17.95Single9AS1DMT9AS1-5-HT2A-DMT
17.95Single9CHXS-Carazolol9CHX-β2-S-Carazolol
17.95Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
17.95Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
17.95Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
17.95Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
17.95Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
17.95Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
17.95Consensushca_on_gpOrthosteric Ligandhca2_on_gp
17.78Single6HLOAprepitant6HLO-NK1-Aprepitant
17.78Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
17.78Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
17.78Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
17.78Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
17.78Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
17.78Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
17.78Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
17.78Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
17.78Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
17.78Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
17.78Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
17.78Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
17.78Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
17.78Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
17.50Single5JQHS-Carazolol5JQH-β2-S-Carazolol
17.50Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
17.50Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
17.50Single5TVNLSD5TVN-5-HT2B-LSD
17.50Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
17.50Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
17.50Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
17.50Single6PS6Timolol6PS6-β2-Timolol
17.50Single7C61Ergotamine7C61-5-HT1B-Ergotamine
17.50Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
17.50Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
17.50Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
17.50Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
17.50Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.50Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
17.50Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
17.50Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
17.50Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
17.50Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
17.50Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
17.50Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.50Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
17.50Single8JXSPF-61428JXS-D1-PF-6142
17.50Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
17.50Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
17.50Single8QOTNanobody-E8QOT-μ-Nanobody-E
17.50Single8S4DCMF-0198S4D-Apelin-CMF-019
17.50Single8TF5Oleic acid8TF5-GPR6-Oleic acid
17.50Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.50Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.50Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
17.50Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
17.50Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
17.50Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
17.50Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
17.50Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
17.50Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
17.50Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
17.50Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
17.50Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
17.50Consensusadenosine_offOrthosteric Liganda1_off a2_off
17.50Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
17.50Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
17.50Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
17.50Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
17.50Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
17.50Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
17.50Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
17.50Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.50Consensustrace-amine_onOrthosteric Ligandta1_on
17.39Single3OE0CVX153OE0-CXCR4-CVX15
17.39Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
17.39Single6PT2KGCHM076PT2-δ-KGCHM07
17.39Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
17.39Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
17.39Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
17.39Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.39Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.39Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
17.39Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
17.39Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
17.39Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
17.31Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
17.31Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
17.31Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
17.07Single3P0GBI1671073P0G-β2-BI167107
17.07Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
17.07Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
17.07Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
17.07Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
17.07Single5XR8AM8415XR8-CB1-AM841
17.07Single5XRAAM115425XRA-CB1-AM11542
17.07Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
17.07Single6WGTLSD6WGT-5-HT2A-LSD
17.07Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
17.07Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
17.07Single7PX4PSB-21137PX4-A2A-PSB-2113
17.07Single7TUYGSK682753A7TUY-GPR183-GSK682753A
17.07Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
17.07Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
17.07Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
17.07Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
17.07Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
17.07Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
17.07Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
17.07Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
17.07Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
17.07Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.07Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
17.07Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
17.07Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
17.07Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
17.07Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
17.07Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
17.07Single9AS9RS130-1809AS9-5-HT2A-RS130-180
17.07Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
17.07Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
17.07Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
17.07Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
17.07Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
17.07Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
17.07Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
17.07Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
17.07Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
17.07Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.07Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
17.07Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
17.07Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
17.07Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
17.07Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
17.07Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
17.07Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
17.07Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.07Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
17.02Single6JODAngiotensin II6JOD-AT2-Angiotensin II
17.02Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
17.02Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
17.02Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
17.02Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
17.02Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
17.02Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
17.02Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
17.02Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
17.02Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
17.02Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
17.02Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
16.67Single4XEENeurotensin4XEE-NTS1-Neurotensin
16.67Single4XESNeurotensin4XES-NTS1-Neurotensin
16.67Single5CXVTiotropium5CXV-M1-Tiotropium
16.67Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
16.67Single6A93Risperidone6A93-5-HT2A-Risperidone
16.67Single6IIURamatroban6IIU-TXA2-Ramatroban
16.67Single6KQICP559406KQI-CB1-CP55940-Org27569
16.67Single6MXTSalmeterol6MXT-β2-Salmeterol
16.67Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
16.67Single6YVRNTS8-136YVR-NTS1-NTS8-13
16.67Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
16.67Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
16.67Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
16.67Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
16.67Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
16.67Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
16.67Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
16.67Single7YITNalfurafine7YIT-κ-Nalfurafine
16.67Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
16.67Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
16.67Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
16.67Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8JJ8Formoterol8JJ8-β2-Formoterol
16.67Single8JJLOlodaterol8JJL-β2-Olodaterol
16.67Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
16.67Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
16.67Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
16.67Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
16.67Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
16.67Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
16.67Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
16.67Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
16.67Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
16.67Single9DGIZ85267113509DGI-CB1-Z8526711350
16.67Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
16.67Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
16.67Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
16.67Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
16.67Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
16.67Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
16.67Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
16.67Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
16.67Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
16.67Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
16.67Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
16.67Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
16.67Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
16.67Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
16.67Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
16.67Consensuslpa_offOrthosteric Ligandlpa1_off
16.67Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
16.67Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
16.67Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
16.67Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
16.67Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
16.67Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
16.67Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
16.67Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
16.67Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
16.33Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
16.33Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
16.33Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
16.33Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
16.33Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
16.33Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
16.28Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
16.28Single4BUONeurotensin4BUO-NTS1-Neurotensin
16.28Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
16.28Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
16.28Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
16.28Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
16.28Single5X93K-87945X93-ETB-K-8794
16.28Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
16.28Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
16.28Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
16.28Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
16.28Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
16.28Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.28Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
16.28Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
16.28Single7UM4AS26747237UM4-5-HT5A-AS2674723
16.28Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
16.28Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
16.28Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
16.28Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
16.28Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
16.28Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
16.28Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
16.28Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
16.28Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
16.28Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
16.28Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
16.28Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
16.28Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
16.28Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
16.28Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
16.28Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
16.28Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
16.28Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
16.28Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
16.28Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
16.28Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
16.28Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
16.28Consensuschemerin_onOrthosteric Ligandcml1_on
16.28Consensusendothelin_offOrthosteric Ligandetb_off
16.28Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
16.28Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
16.28Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
16.28Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.28Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.28Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
16.28Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
16.28Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
16.28Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
16.28Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
16.22Single6LI0C176LI0-GPR52-C17
16.22Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
16.22Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.22Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
16.22Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
16.22Single8K5BNiacin8K5B-HCA2-Niacin
16.22Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
16.22Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
15.91Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
15.91Single6PT3DPI-2876PT3-δ-DPI-287
15.91Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.91Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
15.91Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
15.91Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
15.91Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
15.91Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
15.91Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
15.91Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
15.91Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
15.91Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
15.91Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
15.91Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
15.91Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
15.91Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.91Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
15.91Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
15.91Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.91Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.91Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
15.91Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
15.79Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
15.79Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
15.79Single4BWBNeurotensin4BWB-NTS1-Neurotensin
15.79Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
15.79Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
15.79Single6AKXA4R6AKX-CCR5-A4R
15.79Single6AKYMaraviroc6AKY-CCR5-Maraviroc
15.79Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
15.79Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
15.79Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
15.79Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
15.79Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
15.79Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
15.79Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
15.79Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
15.79Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.79Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.79Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.79Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
15.79Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
15.79Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
15.79Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
15.79Single8IWESpermidine8IWE-TA9-Spermidine
15.79Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
15.79Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
15.79Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
15.79Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
15.79Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
15.79Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
15.79Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
15.79Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
15.79Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
15.79Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
15.79Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
15.79Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
15.79Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
15.79Consensusalpha2_offOrthosteric Ligandalpha2c_off
15.79Consensusangiotensin_offOrthosteric Ligandat1_off
15.79Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
15.79Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
15.79Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
15.79Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
15.79Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
15.79Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
15.69Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
15.56Single4IARErgotamine4IAR-5-HT1B-Ergotamine
15.56Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
15.56Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
15.56Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
15.56Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
15.56Single7F8XNN90567F8X-CCKA-NN9056
15.56Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
15.56Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
15.56Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
15.56Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
15.56Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
15.56Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
15.56Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
15.56Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
15.56Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
15.56Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
15.56Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
15.56Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
15.56Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
15.38Single2YDOAdenosine2YDO-A2A-Adenosine
15.38Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
15.38Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
15.38Single4MBSMaraviroc4MBS-CCR5-Maraviroc
15.38Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
15.38Single5IU7Q274563465IU7-A2A-Q27456346-Na
15.38Single5IUBQ274563445IUB-A2A-Q27456344-Na
15.38Single5JTBZM-2413855JTB-A2A-ZM-241385
15.38Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
15.38Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
15.38Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
15.38Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
15.38Single6PS0S-Carazolol6PS0-β2-S-Carazolol
15.38Single6PS4ICI118-5516PS4-β2-ICI118-551
15.38Single6PS5S-Propranolol6PS5-β2-S-Propranolol
15.38Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
15.38Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
15.38Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
15.38Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
15.38Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
15.38Single7F61PF-036547467F61-H3-PF-03654746
15.38Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
15.38Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
15.38Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
15.38Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
15.38Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
15.38Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
15.38Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
15.38Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
15.38Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
15.38Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
15.38Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
15.38Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
15.38Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
15.38Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
15.38Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
15.38Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
15.38Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
15.38Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
15.38Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
15.38Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
15.38Single8K5CAcipimox8K5C-HCA2-Acipimox
15.38Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
15.38Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
15.38Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
15.38Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
15.38Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
15.38Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
15.38Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
15.38Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
15.38Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
15.38Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
15.38Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
15.38Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
15.38Single9AS5Mescaline9AS5-5-HT2A-Mescaline
15.38Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
15.38Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
15.38Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
15.38Consensusa2_offOrthosteric Liganda2a_off
15.38Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
15.38Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
15.38Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
15.38Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
15.38Consensusgrh_offOrthosteric Ligandgnrh1_off
15.38Consensushca_onOrthosteric Ligandhca2_on
15.22Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
15.22Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
15.22Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
15.22Single7SK5CXCL127SK5-ACKR3-CXCL12
15.22Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
15.22Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.22Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
15.22Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
15.22Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
15.22Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
15.22Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
15.09Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
15.00Single2Y04Salbutamol2Y04-β1-Salbutamol
15.00Single3EMLZM-2413853EML-A2A-ZM-241385
15.00Single3NY8ICI118-5513NY8-β2-ICI118-551
15.00Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
15.00Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
15.00Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
15.00Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
15.00Single4GBRS-Carazolol4GBR-β2-S-Carazolol
15.00Single4MQSIperoxo4MQS-M2-Iperoxo
15.00Single4U14Tiotropium4U14-M3-Tiotropium
15.00Single4YAYZD-71554YAY-AT1-ZD-7155
15.00Single5DHHSB-6121115DHH-NOP-SB-612111
15.00Single5DSGTiotropium5DSG-M4-Tiotropium
15.00Single5IU8Q274563475IU8-A2A-Q27456347-Na
15.00Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
15.00Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
15.00Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
15.00Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
15.00Single5TGZAM65385TGZ-CB1-AM6538
15.00Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
15.00Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
15.00Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
15.00Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
15.00Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
15.00Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
15.00Single6H7MSalbutamol6H7M-β1-Salbutamol
15.00Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
15.00Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
15.00Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
15.00Single6S0LZM-2413856S0L-A2A-ZM-241385
15.00Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
15.00Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
15.00Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
15.00Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
15.00Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
15.00Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
15.00Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
15.00Single7PYRPSB-21157PYR-A2A-PSB-2115
15.00Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
15.00Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
15.00Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
15.00Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
15.00Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
15.00Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
15.00Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
15.00Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
15.00Single7WC7Lisuride7WC7-5-HT2A-Lisuride
15.00Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
15.00Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
15.00Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
15.00Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
15.00Single8CU6LJ-45178CU6-A2A-LJ-4517
15.00Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
15.00Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
15.00Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
15.00Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
15.00Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.00Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.00Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.00Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.00Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.00Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.00Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.00Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.00Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.00Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.00Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
15.00Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
15.00Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
15.00Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
15.00Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
15.00Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
15.00Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
15.00Single8JJOAlprenolol8JJO-β2-Alprenolol
15.00Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
15.00Single8JXRLSD8JXR-D1-LSD
15.00Single8K5DGSK2560738K5D-HCA2-GSK256073
15.00Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
15.00Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
15.00Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.00Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.00Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.00Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.00Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
15.00Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
15.00Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
15.00Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
15.00Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
15.00Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
15.00Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
15.00Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
15.00Single9H37A1IR09H37-A2A-A1IR0-Na
15.00Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
15.00Single9JEAAtropine9JEA-M1-Atropine
15.00Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
15.00Consensus5ht5_onOrthosteric Ligand5ht5a_on
15.00Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
15.00Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
15.00Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
15.00Consensusa3_onOrthosteric Liganda3a_on
15.00Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
15.00Consensusdopamine_offOrthosteric Ligandd2_off d3_off
15.00Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
15.00Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
15.00Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
15.00Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
15.00Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
15.00Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
15.00Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
14.89Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
14.89Single6W25SHU91196W25-MC4-SHU9119-Ca
14.89Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
14.89Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.89Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
14.89Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
14.89Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
14.63Single2RH1S-Carazolol2RH1-β2-S-Carazolol
14.63Single2Y03Isoprenaline2Y03-β1-Isoprenaline
14.63Single2YCWS-Carazolol2YCW-β1-S-Carazolol
14.63Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
14.63Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
14.63Single5D6LS-Carazolol5D6L-β2-S-Carazolol
14.63Single5IUAQ274563485IUA-A2A-Q27456348-Na
14.63Single5N2RPSB-365N2R-A2A-PSB-36-Na
14.63Single5N2SPSB365N2S-A1-PSB36
14.63Single5WIUNemonapride5WIU-D4-Nemonapride
14.63Single5WIVNemonapride5WIV-D4-Nemonapride-Na
14.63Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
14.63Single6D26Fevipiprant6D26-DP2-Fevipiprant
14.63Single6E67BI1671076E67-β2-BI167107-Gs(CT)
14.63Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
14.63Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
14.63Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
14.63Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
14.63Single6S0QZM-2413856S0Q-A2A-ZM-241385
14.63Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
14.63Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
14.63Single7C4SS1P7C4S-S1P3-S1P
14.63Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
14.63Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
14.63Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
14.63Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
14.63Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
14.63Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
14.63Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
14.63Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
14.63Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
14.63Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
14.63Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
14.63Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.63Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
14.63Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.63Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.63Single8GNEKW-63568GNE-A2A-KW-6356-Na
14.63Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
14.63Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
14.63Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
14.63Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
14.63Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
14.63Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
14.63Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
14.63Single9EHSLUF76029EHS-A3A-LUF7602
14.63Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
14.63Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
14.63Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
14.63Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.63Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
14.63Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
14.63Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
14.63Consensusa3_on_gpOrthosteric Liganda3a_on_gp
14.63Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
14.63Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
14.63Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
14.63Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
14.63Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
14.63Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
14.63Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
14.63Consensusamine_offonOrthosteric Ligandamine_off amine_on
14.63Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
14.63Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
14.63Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
14.63Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
14.63Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
14.63Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
14.63Consensusdp_offOrthosteric Liganddp2_off
14.63Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
14.63Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.63Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.63Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
14.63Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
14.58Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
14.58Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
14.58Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
14.58Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
14.58Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
14.58Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
14.58Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
14.29Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
14.29Single4BV0Neurotensin4BV0-NTS1-Neurotensin
14.29Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
14.29Single4U15Tiotropium4U15-M3-Tiotropium
14.29Single5D5AS-Carazolol5D5A-β2-S-Carazolol
14.29Single5D5BS-Carazolol5D5B-β2-S-Carazolol
14.29Single5V54Methiothepin5V54-5-HT1B-Methiothepin
14.29Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
14.29Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
14.29Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
14.29Single6H7JIsoprenaline6H7J-β1-Isoprenaline
14.29Single6J21Aprepitant6J21-NK1-Aprepitant
14.29Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
14.29Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
14.29Single6OL9Tiotropium6OL9-M5-Tiotropium
14.29Single6OS1TRV0266OS1-AT1-TRV026
14.29Single6TQ7SB-3348676TQ7-OX1-SB-334867
14.29Single7B6WCyclazosin7B6W-α1b-Cyclazosin
14.29Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
14.29Single7F1TMIP-1a7F1T-CCR5-MIP-1a
14.29Single7FEECP559407FEE-CB1-CP55940-ZCZ011
14.29Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
14.29Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
14.29Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
14.29Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
14.29Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
14.29Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
14.29Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
14.29Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
14.29Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
14.29Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
14.29Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
14.29Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
14.29Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
14.29Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
14.29Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
14.29Single8EA0Iperoxo8EA0-M3-Iperoxo
14.29Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
14.29Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
14.29Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
14.29Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
14.29Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
14.29Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
14.29Single8HS2Fab0468HS2-GPR20-Fab046
14.29Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
14.29Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
14.29Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
14.29Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
14.29Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
14.29Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
14.29Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
14.29Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
14.29Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
14.29Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
14.29Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
14.29Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
14.29Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
14.29Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
14.29Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
14.29Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
14.29Single8ZWFJR14a8ZWF-C3aB-JR14a
14.29Single9BJKNaloxone9BJK-μ-Naloxone-NAM
14.29Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
14.29Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
14.29Consensus5ht1_offOrthosteric Ligand5ht1b_off
14.29Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
14.29Consensusa2_onOrthosteric Liganda2b_on
14.29Consensusa2_on_gpOrthosteric Liganda2b_on_gp
14.29Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
14.29Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
14.29Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
14.29Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
14.29Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
14.29Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
14.29Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
14.29Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
14.29Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
14.29Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
14.29Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
14.29Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
14.29Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
14.29Consensuslpa_onOrthosteric Ligandlpa1_on
14.29Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
14.29Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
14.29Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
14.29Consensusneurotensin_onOrthosteric Ligandnts1_on
14.29Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
14.29Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
14.29Consensusrelaxin_onOrthosteric Ligandrxfp4_on
14.29Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
14.00Single7SK3CXCL127SK3-ACKR3-CXCL12
13.95Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
13.95Single3D4STimolol3D4S-β2-Timolol
13.95Single4AMIBucindolol4AMI-β1-Bucindolol
13.95Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
13.95Single4LDEBI1671074LDE-β2-BI167107
13.95Single4RWADIPP-NH24RWA-δ-DIPP-NH2
13.95Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
13.95Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
13.95Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
13.95Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
13.95Single6CM4Risperidone6CM4-D2-Risperidone
13.95Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
13.95Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
13.95Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
13.95Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
13.95Single7DFPSpiperone7DFP-D2-Spiperone
13.95Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
13.95Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
13.95Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
13.95Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
13.95Single7K15MKD0467K15-BLT1-MKD046-Na
13.95Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
13.95Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
13.95Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
13.95Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
13.95Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.95Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
13.95Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
13.95Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
13.95Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
13.95Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
13.95Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
13.95Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
13.95Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
13.95Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
13.95Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
13.95Single8JWY2-1188JWY-A2A-2-118
13.95Single8JWZAB9288JWZ-A2A-AB928-Na
13.95Single8XYIVUF106618XYI-CXCR3-VUF10661
13.95Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
13.95Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
13.95Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
13.95Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
13.95Consensusalpha1_offOrthosteric Ligandalpha1a_off
13.95Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
13.95Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
13.95Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
13.95Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
13.95Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
13.95Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
13.95Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
13.95Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
13.95Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
13.95Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
13.95Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
13.95Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
13.95Consensusorexin_onOrthosteric Ligandox2_on
13.89Single9CHUNoradrenaline9CHU-β2-Noradrenaline
13.73Single9KDFRES-701-39KDF-ETB-RES-701-3
13.64Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
13.64Single6H7LDobutamine6H7L-β1-Dobutamine
13.64Single6IBLArformoterol6IBL-β1-Arformoterol
13.64Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
13.64Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
13.64Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
13.64Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
13.64Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
13.64Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
13.64Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.64Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.64Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
13.64Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
13.64Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
13.64Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
13.64Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
13.64Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
13.64Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
13.64Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
13.64Single8XVUCXCL28XVU-CXCR2-CXCL2
13.64Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
13.64Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
13.64Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
13.64Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.64Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
13.64Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
13.64Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
13.64Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
13.64Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
13.64Consensusprostanoid_offOrthosteric Ligandep_off dp_off
13.51Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
13.51Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
13.51Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.51Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
13.51Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
13.51Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
13.51Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
13.51Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
13.51Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
13.51Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
13.51Single9LRCHistamine9LRC-H4-Histamine
13.51Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
13.51Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
13.51Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
13.33Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
13.33Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
13.33Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
13.33Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
13.33Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
13.33Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
13.33Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
13.33Single7XN9L-054,5227XN9-SST2-L-054,522
13.33Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
13.33Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
13.33Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
13.33Single8X5YAstemizole8X5Y-H1-Astemizole
13.33Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
13.33Single9IPYJR14a9IPY-C3aB-JR14a
13.33Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
13.33Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
13.33Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
13.33Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
13.16Single3OE9IT1t3OE9-CXCR4-IT1t
13.16Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
13.16Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
13.16Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
13.16Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
13.16Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
13.16Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
13.16Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
13.16Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
13.16Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
13.16Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
13.16Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
13.16Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
13.16Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
13.16Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
13.16Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
13.16Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
13.16Single8YKDDehydroepiandrosterone8YKD-ADGRG2-Dehydroepiandrosterone-chim(NtGi1-Gs)/β1/γ2
13.16Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
13.16Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
13.16Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
13.16Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
13.16Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
13.16Single9AS7Psilocin9AS7-5-HT2A-Psilocin
13.16Single9B9Y7DY9B9Y-CB1-7DY
13.16Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
13.16Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
13.16Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
13.16Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
13.16Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
13.16Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
13.04Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
13.04Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
13.04Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
13.04Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
13.04Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
13.04Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
13.04Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
13.04Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
13.04Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.04Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
13.04Single9M4TSilodosin9M4T-Alpha1A-Silodosin
13.04Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
13.04Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
13.04Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
13.04Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
13.04Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
12.82Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
12.82Single3ODUIT1t3ODU-CXCR4-IT1t
12.82Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
12.82Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
12.82Single5ZKQABT-4915ZKQ-PAF-ABT-491
12.82Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
12.82Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
12.82Single6ME2Ramelteon6ME2-MT1-Ramelteon
12.82Single7BR3Elagolix7BR3-GnRH1-Elagolix
12.82Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
12.82Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
12.82Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
12.82Single7F8ULintitript7F8U-CCKA-Lintitript
12.82Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
12.82Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
12.82Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
12.82Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
12.82Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
12.82Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
12.82Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
12.82Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
12.82Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
12.82Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
12.82Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
12.82Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
12.82Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
12.82Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
12.82Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
12.82Single8GNGIstradefylline8GNG-A2A-Istradefylline
12.82Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
12.82Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
12.82Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
12.82Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
12.82Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
12.82Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
12.82Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
12.82Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
12.82Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
12.82Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.82Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.82Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.82Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
12.82Single8Y0HVUF114188Y0H-CXCR3-VUF11418
12.82Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
12.82Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
12.82Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
12.82Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
12.82Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
12.82Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
12.82Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
12.82Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
12.82Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
12.82Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
12.82Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
12.82Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
12.82Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
12.82Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
12.77Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
12.77Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
12.77Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
12.77Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
12.77Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
12.77Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
12.77Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
12.77Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
12.50Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
12.50Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
12.50Single5UVIZM-2413855UVI-A2A-ZM-241385
12.50Single6A94Zotepine6A94-5-HT2A-Zotepine
12.50Single6AQFZM-2413856AQF-A2A-ZM-241385
12.50Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
12.50Single6KUXRS-799486KUX-α2a-RS-79948
12.50Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
12.50Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
12.50Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
12.50Single6TPGEMPA6TPG-OX2-EMPA
12.50Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
12.50Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
12.50Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
12.50Single7AROLUF58337ARO-A2A-LUF5833-Na
12.50Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
12.50Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
12.50Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
12.50Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
12.50Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
12.50Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
12.50Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.50Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
12.50Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
12.50Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
12.50Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
12.50Single7UL3Famotidine7UL3-H2-Famotidine
12.50Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
12.50Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
12.50Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
12.50Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
12.50Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
12.50Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
12.50Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.50Single8IHKAcifran8IHK-HCA3-Acifran
12.50Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
12.50Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
12.50Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
12.50Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
12.50Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.50Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.50Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
12.50Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
12.50Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
12.50Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
12.50Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
12.50Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
12.50Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
12.50Single8ZPMAMD0708ZPM-CXCR4-AMD070
12.50Single9ARXSerotonin9ARX-5-HT2A-Serotonin
12.50Single9AS3LSD9AS3-5-HT2A-LSD
12.50Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single9BA0A1AKN9BA0-CB1-A1AKN
12.50Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
12.50Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
12.50Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
12.50Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
12.50Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
12.50Consensusalpha1_onOrthosteric Ligandalpha1a_on
12.50Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
12.50Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
12.50Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
12.50Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
12.50Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
12.50Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
12.50Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
12.50Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
12.50Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
12.24Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
12.24Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
12.20Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
12.20Single2Y01Dobutamine2Y01-β1-Dobutamine
12.20Single2Y02Carmoterol2Y02-β1-Carmoterol
12.20Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
12.20Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
12.20Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
12.20Single4QKX35V4QKX-β2-35V
12.20Single5DHGC-355DHG-NOP-C-35
12.20Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
12.20Single5T04Neurotensin5T04-NTS1-Neurotensin
12.20Single5UENDU1725UEN-A1-DU172
12.20Single5UIGCmpd-15UIG-A2A-Cmpd-1
12.20Single6D27CAY104716D27-DP2-CAY10471
12.20Single6DRXLisuride6DRX-5-HT2B-Lisuride
12.20Single6IIVDaltroban6IIV-TXA2-Daltroban
12.20Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
12.20Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
12.20Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
12.20Single6TOTLemborexant6TOT-OX1-Lemborexant
12.20Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.20Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
12.20Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
12.20Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
12.20Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
12.20Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
12.20Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
12.20Single7UL4Alvimopan7UL4-μ-Alvimopan
12.20Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
12.20Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
12.20Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
12.20Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
12.20Single7YXAONO-54306087YXA-S1P5-ONO-5430608
12.20Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
12.20Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
12.20Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
12.20Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
12.20Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
12.20Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
12.20Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
12.20Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
12.20Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
12.20Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
12.20Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
12.20Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
12.20Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
12.20Single8X63Mepyramine8X63-H1-Mepyramine
12.20Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
12.20Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
12.20Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
12.20Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
12.20Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
12.20Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
12.20Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
12.20Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
12.20Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
12.20Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
12.20Consensusalpha2_onOrthosteric Ligandalpha2b_on
12.20Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
12.20Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
12.20Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
12.20Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
12.20Consensuscck_offOrthosteric Ligandccka_off
12.20Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
12.20Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
12.20Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
12.20Consensushistamine_offOrthosteric Ligandh1_off
12.20Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
12.20Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
12.00Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
11.90Single2Y00Dobutamine2Y00-β1-Dobutamine
11.90Single4JKVTaladegib4JKV-SMO-Taladegib
11.90Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
11.90Single5CGCHTL142425CGC-mGlu5-HTL14242
11.90Single5WQCEMPA5WQC-OX2-EMPA
11.90Single5XPRBosentan5XPR-ETB-Bosentan
11.90Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
11.90Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
11.90Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
11.90Single6LUQHaloperidol6LUQ-D2-Haloperidol
11.90Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
11.90Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
11.90Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
11.90Single6TP6Filorexant6TP6-OX1-Filorexant
11.90Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
11.90Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
11.90Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
11.90Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
11.90Single7W41PD1762527W41-BB2-PD176252
11.90Single7WC6LSD7WC6-5-HT2A-LSD
11.90Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
11.90Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
11.90Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
11.90Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
11.90Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
11.90Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
11.90Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
11.90Single8ZMFA1L108ZMF-5-HT2C-A1L10
11.90Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
11.90Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
11.90Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
11.90Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
11.90Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
11.90Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
11.90Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
11.90Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
11.90Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
11.90Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
11.90Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
11.90Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
11.90Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
11.90Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
11.90Consensusblt_offOrthosteric Ligandblt1_off
11.90Consensusbombesin_offOrthosteric Ligandbb2_off
11.90Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
11.90Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
11.90Consensusep_offOrthosteric Ligandep4_off
11.90Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
11.90Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
11.90Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
11.90Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
11.90Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
11.90Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
11.90Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
11.63Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
11.63Single4DJHJDTic4DJH-κ-JDTic
11.63Single5V56TC1145V56-SMO-TC114
11.63Single5V57TC1145V57-SMO-TC114
11.63Single6J20Aprepitant6J20-NK1-Aprepitant
11.63Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
11.63Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
11.63Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
11.63Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
11.63Single7P2L4YI7P2L-mGlu5-4YI
11.63Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.63Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
11.63Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
11.63Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
11.63Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
11.63Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.63Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
11.63Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
11.63Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
11.63Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
11.63Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
11.63Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
11.63Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
11.63Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
11.63Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
11.63Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
11.63Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
11.63Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
11.63Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
11.54Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
11.54Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
11.43Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
11.36Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
11.36Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
11.36Single6ZG4HTL00099366ZG4-M1-HTL0009936
11.36Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
11.36Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
11.36Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
11.36Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
11.36Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
11.36Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.36Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
11.36Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
11.36Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
11.36Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.36Single8XWMCXCL68XWM-CXCR2-CXCL6
11.36Single8XWSCXCL58XWS-CXCR2-CXCL5
11.36Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
11.36Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.36Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.32Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
11.11Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
11.11Single5CGDHTL142425CGD-mGlu5-HTL14242
11.11Single6K1QIRL25006K1Q-ETB-IRL2500
11.11Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
11.11Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
11.11Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
11.11Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
11.11Single8XVJMacitentan8XVJ-ETA-Macitentan
11.11Single8XWFCXCL38XWF-CXCR2-CXCL3
11.11Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
10.87Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
10.87Single8XQJJN2418XQJ-Apelin-JN241
10.87Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
10.87Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
10.87Single9JF4PD1683689JF4-BB1-PD168368
10.87Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
10.81Single8A2OTheophylline8A2O-A2A-Theophylline-Na
10.81Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.81Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
10.81Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
10.81Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
10.81Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
10.64Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
10.64Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
10.64Single8IEBA1LYA8IEB-GPR156-A1LYA
10.64Single8IEIA1LYA8IEI-GPR156-A1LYA
10.64Single8IEPA1LYA8IEP-GPR156-A1LYA
10.64Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
10.64Single8KIGSHU91198KIG-MC3-SHU9119-Ca
10.64Single8WKYPG-9348WKY-MC4-PG-934
10.64Single8XWNCXCL88XWN-CXCR2-CXCL8
10.64Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
10.64Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
10.53Single3OE6IT1t3OE6-CXCR4-IT1t
10.53Single4XNWMRS25004XNW-P2Y1-MRS2500
10.53Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
10.53Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
10.53Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
10.53Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
10.53Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
10.53Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
10.53Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
10.53Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
10.53Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
10.53Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
10.53Consensus5ht2_onOrthosteric Ligand5ht2b_on
10.53Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.53Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
10.53Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
10.42Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
10.42Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
10.42Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
10.26Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
10.26Single3PBLEticlopride3PBL-D3-Eticlopride
10.26Single4O9RCyclopamine4O9R-SMO-Cyclopamine
10.26Single5L7IVismodegib5L7I-SMO-Vismodegib
10.26Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
10.26Single7SRQLSD7SRQ-5-HT2B-LSD
10.26Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
10.26Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
10.26Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
10.26Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
10.26Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
10.26Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
10.26Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
10.26Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
10.26Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
10.26Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
10.26Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.26Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.26Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
10.26Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
10.26Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
10.26Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
10.26Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
10.26Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
10.26Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
10.20Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
10.20Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
10.20Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
10.20Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
10.20Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
10.20Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
10.00Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
10.00Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
10.00Single3PWHZM-2413853PWH-A2A-ZM-241385
10.00Single4QINSAG1.54QIN-SMO-SAG1.5
10.00Single4S0VSuvorexant4S0V-OX2-Suvorexant
10.00Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
10.00Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
10.00Single6B73MP11046B73-κ-MP1104
10.00Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
10.00Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
10.00Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
10.00Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
10.00Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
10.00Single6TPJSuvorexant6TPJ-OX2-Suvorexant
10.00Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
10.00Single7F8YDevazepide7F8Y-CCKA-Devazepide
10.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
10.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
10.00Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
10.00Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
10.00Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
10.00Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
10.00Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
10.00Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
10.00Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
10.00Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
10.00Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
10.00Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
10.00Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
10.00Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
10.00Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
10.00Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
10.00Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
10.00Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
10.00Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
10.00Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
10.00Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
10.00Single9H2XA1IR19H2X-A2A-A1IR1-Na
10.00Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
10.00Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
10.00Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
10.00Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
10.00Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
10.00Consensusorexin_offOrthosteric Ligandox2_off ox1_off
10.00Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
10.00Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
9.80Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
9.80Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
9.80Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
9.76Single3REYXAC3REY-A2A-XAC
9.76Single3RZECidoxepin3RZE-H1-Cidoxepin
9.76Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
9.76Single4ZJCSB-6740424ZJC-OX1-SB-674042
9.76Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
9.76Single6IQLL7458706IQL-D4-L745870
9.76Single6MH8ZM-2413856MH8-A2A-ZM-241385
9.76Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
9.76Single6TP3Nemorexant6TP3-OX1-Nemorexant
9.76Single6TPNHTL66416TPN-OX2-HTL6641
9.76Single6V9SGTPL114036V9S-OX1-GTPL11403
9.76Single6VI4JDTic6VI4-κ-JDTic
9.76Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
9.76Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
9.76Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
9.76Single6ZG9GSK10347026ZG9-M1-GSK1034702
9.76Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
9.76Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
9.76Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
9.76Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
9.76Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
9.76Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
9.76Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
9.76Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
9.76Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.76Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
9.76Single8JD6VU03647708JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
9.76Single8K2WAMG4878K2W-CXCR3-AMG487
9.76Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
9.76Single8RLNLUF58348RLN-A2A-LUF5834
9.76Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
9.76Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.76Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
9.76Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
9.76Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
9.76Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
9.76Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
9.76Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
9.76Single8ZPNAMD31008ZPN-CXCR4-AMD3100
9.76Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
9.76Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
9.76Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
9.76Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
9.76Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
9.76Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
9.76Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
9.76Consensusopsins_offOrthosteric Ligandrhodopsin_off
9.76Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
9.76Consensussensory_offOrthosteric Ligandopsins_off
9.52Single4EJ4Naltrindole4EJ4-δ-Naltrindole
9.52Single4QIMANTA XV4QIM-SMO-ANTA XV
9.52Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
9.52Single6GPSMK08126GPS-CCR2-MK0812
9.52Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
9.52Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
9.52Single7BU7BI1671077BU7-β1-BI167107
9.52Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
9.52Single7F83PF-051904577F83-Ghrelin-PF-05190457
9.52Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
9.52Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
9.52Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
9.52Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
9.52Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
9.52Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
9.52Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
9.52Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
9.52Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
9.52Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
9.52Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
9.52Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
9.52Single8X64Desloratadine8X64-H1-Desloratadine
9.52Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
9.52Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
9.52Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
9.52Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
9.52Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
9.52Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
9.52Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
9.52Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
9.52Consensusblt_onOrthosteric Ligandblt1_on
9.52Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
9.52Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
9.52Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
9.52Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
9.52Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
9.52Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
9.52Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
9.52Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
9.52Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
9.52Consensusleukotriene_onOrthosteric Ligandblt_on
9.52Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
9.52Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
9.30Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
9.30Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
9.30Single6GPXMK08126GPX-CCR2-MK0812
9.30Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
9.30Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
9.30Single7SINNPS-21437SIN-CaS-NPS-2143
9.30Single7SINNPS-21437SIN-CaS-NPS-2143
9.30Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
9.30Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
9.30Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.30Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
9.30Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
9.30Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
9.30Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
9.30Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
9.30Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
9.30Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
9.30Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
9.30Single9HC04YI9HC0-mGlu5-4YI
9.30Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
9.30Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
9.09Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
9.09Single6E59L-7607356E59-NK1-L-760735
9.09Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
9.09Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
9.09Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
9.09Single7R0CAVP7R0C-V2-AVP-Arrestin2
9.09Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
9.09Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single8XVLZibotentan8XVL-ETA-Zibotentan
9.09Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
9.09Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
9.09Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
9.09Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
9.09Consensustachykinin_offOrthosteric Ligandnk1_off
8.89Single4N4WSANT-14N4W-SMO-SANT-1
8.89Single5X33BIIL2605X33-BLT1-BIIL260
8.89Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
8.89Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
8.89Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.89Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
8.89Single8XQJJN2418XQJ-Apelin-JN241
8.89Single8XWACXCL18XWA-CXCR2-CXCL1
8.89Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
8.89Single9BJKNAM9BJK-μ-Naloxone-NAM
8.89Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
8.70Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
8.70Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
8.70Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
8.70Single8ZPLHF511168ZPL-CXCR4-HF51116
8.51Single6KNMJN241-96KNM-Apelin-JN241-9
8.51Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
8.51Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
8.51Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
8.51Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
8.51Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
8.51Consensuskisspeptin_onOrthosteric Ligandkiss1_on
8.33Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
8.33Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Single8IEIA1LYA8IEI-GPR156-A1LYA
8.33Single8IEPA1LYA8IEP-GPR156-A1LYA
8.33Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
8.33Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
8.33Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
8.33Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
8.33Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
8.33Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
8.33Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
8.33Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
8.33Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
8.33Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
8.16Single8IEBA1LYA8IEB-GPR156-A1LYA
8.16Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
8.16Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
8.16Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
8.11Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
8.11Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
8.11Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
8.11Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
8.11Single8PWNTheophylline8PWN-A2A-Theophylline
8.11Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
7.89Single3OE8IT1t3OE8-CXCR4-IT1t
7.89Single3RFMCaffeine3RFM-A2A-Caffeine
7.89Single6TQ9SB-4081246TQ9-OX1-SB-408124
7.89Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
7.89Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
7.89Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
7.89Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
7.89Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
7.89Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
7.89Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
7.89Consensusp2y_offOrthosteric Ligandp2y1_off
7.84Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
7.69Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
7.69Single3UZAGTPL92363UZA-A2A-GTPL9236
7.69Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
7.69Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
7.69Single6ME5Agomelatine6ME5-MT1-Agomelatine
7.69Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
7.69Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
7.69Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
7.69Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
7.50Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
7.50Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
7.50Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
7.50Single6HLLCP999946HLL-NK1-CP99994
7.50Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
7.50Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
7.50Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
7.50Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
7.50Single7UL2SR486927UL2-NTS1-SR48692-Na
7.50Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
7.50Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
7.50Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.50Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
7.50Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
7.50Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.50Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
7.50Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
7.50Consensusneurotensin_offOrthosteric Ligandnts1_off
7.50Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
7.32Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
7.32Single5WS3EMPA5WS3-OX2-EMPA
7.32Single6DS0Ly2660976DS0-5-HT2B-Ly266097
7.32Single6ME9Ramelteon6ME9-MT2-Ramelteon
7.32Single6TODEMPA6TOD-OX1-EMPA-Na
7.32Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
7.32Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
7.32Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
7.32Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
7.32Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
7.32Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
7.32Single7XRRLemborexant7XRR-OX2-Lemborexant
7.32Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
7.32Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
7.32Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
7.32Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
7.32Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
7.32Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
7.32Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
7.32Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
7.14Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
7.14Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
7.14Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
7.14Single7VODCariprazine7VOD-5-HT2A-Cariprazine
7.14Single7VV6C48/807VV6-MRGPRX2-C48/80
7.14Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
7.14Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
7.14Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
7.14Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.14Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
6.98Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
6.98Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
6.98Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
6.98Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
6.98Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
6.98Single9IYAONO-97105319IYA-GPR55-ONO-9710531
6.82Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
6.82Single6HLPNetupitant6HLP-NK1-Netupitant
6.82Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
6.82Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
6.82Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
6.82Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
6.82Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
6.82Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
6.82Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
6.82Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
6.82Single9HAPTolvaptan9HAP-V2-Tolvaptan
6.82Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
6.67Single5TZRMK86665TZR-FFA1-MK8666
6.67Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
6.67Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
6.67Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
6.67Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
6.67Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
6.67Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
6.67Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
6.67Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
6.67Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
6.52Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
6.52Single4PY02MeSATP4PY0-P2Y12-2MeSATP
6.52Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
6.52Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
6.52Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
6.38Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
6.38Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
6.25Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
6.25Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
5.41Single5MZPCaffeine5MZP-A2A-Caffeine-Na
5.26Single6VCBLSN31604406VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
5.26Single7WC4Serotonin7WC4-5-HT2A-Serotonin
5.13Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
5.13Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
5.13Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
5.13Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
5.13Single9IVMLSN33188399IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
5.13Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
5.13Consensussensory_onOrthosteric Ligandopsins_on
5.00Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
5.00Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
5.00Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
5.00Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
5.00Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
5.00Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
5.00Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
5.00Single7WC5Psilocin7WC5-5-HT2A-Psilocin
5.00Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.00Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
5.00Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
5.00Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
5.00Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
5.00Single8JPSCCL78JPS-ACKR1-CCL7
5.00Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
5.00Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
5.00Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
5.00Consensusgi_sensoryOrthosteric Ligandgi_opsins
5.00Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
5.00Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
5.00Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
5.00Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
5.00Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
4.88Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
4.88Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
4.88Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
4.88Single6TP4ACT-4622066TP4-OX1-ACT-462206
4.88Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
4.88Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
4.88Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
4.88Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
4.88Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
4.88Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.88Consensusgq_nucleotideOrthosteric Ligandgq_p2y
4.88Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
4.76Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
4.76Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
4.76Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
4.76Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
4.76Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
4.76Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.76Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
4.76Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.76Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.65Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
4.65Single6FFIMMPEP6FFI-mGlu5-MMPEP
4.65Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
4.65Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
4.65Single6TPKRetosiban6TPK-OT-Retosiban
4.65Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
4.65Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
4.65Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
4.65Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.65Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
4.65Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
4.65Consensusvasop-oxy_offOrthosteric Ligandot_off
4.55Single6FFHFenobam6FFH-mGlu5-Fenobam
4.55Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
4.55Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
4.55Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
4.44Single4NTJAZD12834NTJ-P2Y12-AZD1283
4.44Single6Z4SSR486926Z4S-NTS1-SR48692
4.44Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
4.44Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
4.35Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
4.26Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
4.26Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
4.26Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
4.26Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
4.26Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
4.17Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
4.17Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
4.08Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
4.08Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
4.00Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
2.86Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
2.86Single6D35Cholesterol6D35-SMO-Cholesterol
2.86Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
2.86Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
2.86Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
2.86Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
2.86Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042
2.86Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
2.86Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
2.86Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-BHFF
2.86Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
2.86Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626
2.86Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
2.86Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
2.86Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
2.86Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
2.86Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
2.86Single7DTTCa7DTT-CaS-Ca-Ca
2.86Single7DTTCa7DTT-CaS-Ca-Ca
2.86Single7DTUTryptophan7DTU-CaS-Tryptophan
2.86Single7DTUTryptophan7DTU-CaS-Tryptophan
2.86Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
2.86Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
2.86Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
2.86Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
2.86Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
2.86Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
2.86Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
2.86Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
2.86Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
2.86Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
2.86Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
2.86Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
2.86Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
2.86Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
2.86Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
2.86Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
2.86Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
2.86Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
2.86Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
2.86Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
2.86Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
2.86Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
2.86Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
2.86Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
2.86Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
2.86Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
2.86Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
2.86Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
2.86Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
2.86Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
2.86Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
2.86Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
2.86Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
2.86Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
2.86Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
2.86Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
2.86Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
2.86Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
2.86Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
2.86Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
2.86Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
2.86Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
2.86Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
2.86Single7T9NM22 Fab7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
2.86Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
2.86Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
2.86Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
2.86Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
2.86Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
2.86Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
2.86Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
2.86Single7XW7K1-707XW7-TSH-K1-70
2.86Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
2.86Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
2.86Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
2.86Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
2.86Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
2.86Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
2.86Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
2.86Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
2.86Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
2.86Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
2.86Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
2.86Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
2.86Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
2.86Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
2.86Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
2.86Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
2.86Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
2.86Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
2.86Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
2.86Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
2.86Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
2.86Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
2.86Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
2.86Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
2.86Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
2.86Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
2.86Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
2.86Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
2.86Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
2.86Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
2.86Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
2.86Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
2.86Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
2.86Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
2.86Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
2.86Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
2.86Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
2.86Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
2.86Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
2.86Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
2.86Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
2.86Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
2.86Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
2.86Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
2.86Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
2.86Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
2.86Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
2.86Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
2.86Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
2.86Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
2.86Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
2.86Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
2.86Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
2.86Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
2.86Single8WVXNorrin8WVX-LGR4-Norrin
2.86Single8WVYNorrin8WVY-LGR4-Norrin
2.86Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
2.86Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
2.86Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
2.86Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
2.86Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
2.86Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
2.86Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
2.86Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
2.86Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
2.86Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
2.86Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
2.86Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
2.86Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
2.86Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
2.86Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
2.86Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
2.86Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
2.86Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
2.86Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
2.86Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
2.86Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
2.86Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
2.86Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
2.86Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
2.86Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
2.86Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
2.86Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
2.86Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
2.86Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
2.86Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
2.86Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
2.86Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
2.86Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
2.86Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
2.86Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
2.86Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
2.86Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
2.86Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
2.86Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
2.86Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
2.86Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
2.86Single9KHHNorrin9KHH-LGR4-Norrin
2.86Single9S37NB219S37-LGR4-NB21
2.86Single9UTBSucralose9UTB-TAS1R2; TAS1R3-Sucralose
2.78Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
2.78Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
2.78Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
2.78Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
2.78Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
2.78Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
2.78Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
2.78Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
2.78Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
2.78Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
2.78Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
2.78Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
2.78Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
2.78Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
2.78Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
2.78Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
2.78Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
2.78Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
2.70Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
2.70Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
2.70Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
2.63Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
2.63Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
2.63Single7UTZTR14027UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
2.63Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
2.63Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
2.56Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
2.56Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
2.56Single5L7DCholesterol5L7D-SMO-Cholesterol
2.56Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
2.56Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
2.50Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
2.50Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
2.44Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
2.44Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
2.38Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
2.38Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
2.38Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
2.38Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
2.38Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
2.33Single4XNVBPTU4XNV-P2Y1-BPTU
2.33Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
2.33Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
2.33Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
2.27Single6ZINSR486926ZIN-NTS1-SR48692
2.27Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
2.27Single8IYXYL-3658IYX-GPR34-YL-365
2.13Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
2.04Single9JH5C16:0 Ceramide9JH5-CysLT2-C16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
1.96Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
1.96Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
1.89Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
1.89Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
1.85Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
1.75Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
glucagon_on_gp glp_on_gp
gluc_on_gp
secretin_on_gp
gip_on_gp
vip-pacap_on_gp vpac_on_gp
pac_on_gp
pth_on_gp pth1_on_gp
pth2_on_gp
crf_on_gp crf2_on_gp
crf1_on_gp
calcitonin_on_gp ctlike_on_gp
Net Summary
Imin 3.01003
Number of Linked Nodes 1041
Number of Links 1216
Number of Hubs 173
Number of Links mediated by Hubs 704
Number of Communities 18
Number of Nodes involved in Communities 204
Number of Links involved in Communities 314
Path Summary
Number Of Nodes in MetaPath 114
Number Of Links MetaPath 113
Number of Shortest Paths 4197493
Length Of Smallest Path 3
Average Path Length 46.9357
Length of Longest Path 95
Minimum Path Strength 0.28
Average Path Strength 6.07515
Maximum Path Strength 31.2695
Minimum Path Correlation 0.700283
Average Path Correlation 0.977851
Maximum Path Correlation 0.999771
Minimum % Of Corr. Nodes 1.16279
Average % Of Corr. Nodes 30.8872
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 47.6072
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following differences:
Id1st Network2nd Network
class-a_class-b1_diff_on_gpclass-a_on_gpclass-b1_on_gp
class-b1_class-b2_diff_on_gpclass-b1_on_gpclass-b2_on_gp
This network is also present in following consensuses:
IdComponents
class-a_class-b1_cons_on_gpclass-a_on_gp
class-b1_on_gp
class-b1_class-b2_cons_on_gpclass-b1_on_gp
class-b2_on_gp



You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

Download class-b1_on_gp.zip



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