Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.11 2.28165603
2G.HN.37 2.95422402
3G.HN.52 1.23811404
4G.S1.02 6.05614454
5G.S1.03 3.78748419
6G.S1.05 5.56626409
7G.S1.06 3.53317458
8G.S2.08 7.32056455
9G.S3.01 4.81531454
10G.S3.03 7.8729557
11G.S3.04 8.43308416
12G.S3.05 3.45992556
13G.S3.06 7.81044516
14G.S3.07 3.39567459
15G.s3h2.03 5.1518519
16G.H2.04 4.23458409
17G.H2.06 5.78742719
18G.H2.07 5.36425619
19G.h2s4.01 7.80026419
20G.s4h3.02 4.86191409
21G.s4h3.03 5.611074138
22G.s4h3.04 5.18892788
23G.H3.09 6.27501679
24G.H3.17 7.24198614
25G.H3.18 6.37058419
26G.S5.04 4.86428479
27G.S5.05 3.889177119
28G.S5.06 5.51951408
29G.HG.04 5.44203588
30G.hgh4.02 4.659068148
31G.hgh4.05 8.66209406
32G.H4.03 7.05836403
33G.H4.12 7.07058475
34G.H4.15 4.9595478
35G.h4s6.02 5.21735477
36G.h4s6.11 4.38404478
37G.S6.02 7.79068408
38G.s6h5.01 5.889324119
39G.H5.08 5.54094458
40G.H5.26 6.95075405
41b.1x4 1.88527408
42b.h2x1 3.4493405
43b.lhb1x6 3.93108403
44b.lhb1x9 3.58366403
45b.b1x4 4.86891447
46b.b1x6 8.18906449
47b.l1x3 8.67694649
48b.b2x1 8.72974518
49b.b2x5 7.02346507
50b.b3x3 4.35017468
51b.l3x2 5.48692549
52b.b4x2 5.37869408
53b.b4x3 5.78847467
54b.b4x4 8.95848448
55b.b4x5 4.5737467
56b.b4x6 8.94526749
57b.b5x2 6.08562407
58b.b5x3 6.93217649
59b.b5x5 5.72234465
60b.b5x7 5.77101407
61b.l5x1 4.41496568
62b.l5x5 7.86934719
63b.b6x5 4.03442866
64b.l6x5 6.487684124
65b.b7x1 5.743055124
66b.l7x2 4.61325419
67b.l7x4 3.58501409
68b.b8x3 4.25692406
69b.b8x4 5.67149406
70b.l8x1 3.98219465
71b.l8x3 3.61582403
72b.l9x3 7.47392519
73b.l9x6 5.73833818
74b.b10x5 4.88817609
75b.b11x2 4.67203407
76b.l11x2 8.43137419
77b.b12x3 3.57666438
78b.b12x6 7.96459718
79b.b12x7 5.55402439
80b.b13x7 8.17875537
81b.l13x3 8.91032539
82b.l13x6 5.68428419
83b.l13x7 4.71748439
84b.b14x3 4.74645405
85b.b15x1 7.3762539
86b.b15x3 4.72674439
87b.l15x2 6.58763439
88b.b16x4 9.03407536
89b.b16x5 4.43306405
90b.b16x6 9.81845538
91b.b17x5 7.07225417
92b.b17x7 9.06852418
93b.l17x3 8.27057719
94b.l17x6 7.43562519
95b.b18x3 5.31053418
96b.b18x5 5.62854405
97b.l18x1 5.267588106
98b.l18x3 5.984354105
99b.b19x2 8.2791516
100b.b19x4 6.13852418
101b.l19x2 6.21839519
102b.b20x2 6.08099416
103b.b20x4 10.5518
104b.b20x6 7.76393516
105b.b20x7 4.43203409
106b.l20x2 4.96868509
107b.b21x1 6.85052517
108b.b21x2 3.32963406
109b.b21x5 6.22267404
110b.b21x7 5.52754605
111b.l22x5 6.02414509
112b.b23x1 4.4632405
113b.b23x6 6.79512717
114b.l23x1 7.84953416
115b.b24x4 7.47153416
116b.b24x6 6.05861418
117b.l24x2 4.13196406
118b.l24x3 3.90251405
119b.l25x3 8.76407599
120b.l25x4 3.59162405
121b.l25x6 11.8946418
122b.b27x1 2.92244406
123b.l27x1 10.9381719
124b.l27x2 8.07243499
125b.b28x3 4.84207447
126b.b28x4 8.53542496
127b.b28x6 8.81066599
128g.h1x8 3.2252407
129g.h1x11 2.64636409
130g.l1x4 4.00303508
131g.h2x11 9.434364106
132g.ctx3 6.59716409
133g.ctx4 4.01507407
134g.ctx6 3.77316606
135g.ctx15 7.10602449
136g.ctx16 5.42022748
137Lig 21.50212420
138NT 10.8617423
1391x35 3.66037405
1401x39 4.65408
1411x59 2.69512404
1422x42 5.55705607
1432x46 5.20472429
1442x50 6.0648529
1452x53 5.33442506
146E1x50 7.75391628
147E1x52 6.22794507
1483x33 4.16242425
1493x50 6.23645529
1503x54 3.55833408
1514x54 2.9296404
152E2 13.46941524
1535x50 3.28644409
1545x58 7.49086629
1555x64 2.9785405
1566x44 5.6794429
1576x48 7.21417529
1586x51 5.34509527
1596x59 4.16682405
160E3 4.56915504
1617x26 2.00436401
1627x42 4.68253507
1637x49 5.50167629
1647x53 5.28757629
1657x55 2.20283406
1668x50 3.40073408
167G.H1.08 4.11178450
168I2x57 7.605154170
169g.ntx4 0.836833400
170I1 5.67400
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1b.l2x3 b.l2x5 20.33193.71131NoNo085
2b.b3x1 b.l2x3 20.26196.04175NoNo058
3b.b3x1 b.b6x5 20.25194.20769NoYes056
4b.b3x2 b.b4x6 83.7436.139NoYes059
5b.b2x5 b.b3x2 83.81898.54169YesNo075
6b.b2x3 b.b2x5 96.91845.20492NoYes067
7b.b26x2 b.b2x3 96.97415.69025NoNo076
8b.b26x1 b.b26x2 97.0053.225NoNo097
9b.b26x1 b.l27x1 97.03895.04862NoYes099
10b.b2x1 b.l27x1 55.67558.72106YesYes189
11b.b2x1 b.l3x1 55.690916.5158YesNo189
12b.l3x1 b.l5x5 55.79626.52123NoYes199
13b.l1x3 b.l3x2 86.82375.64375YesYes499
14b.l1x4 b.l3x2 1003.70519NoYes069
15I1 b.l1x4 99.7454.23YesNo006
168x48 I1 97.01318.155NoYes050
177x56 8x48 96.89894.11575NoNo075
187x56 8x47 96.63883.06617NoNo078
198x47 8x50 96.50853.01NoYes088
207x54 8x50 94.68223.51271NoYes068
212x43 7x54 94.28093.7016NoNo086
222x43 7x53 94.14672.67244NoYes089
233x46 7x53 39.53545.67754NoYes299
242x42 3x46 40.63624.54025YesNo079
252x42 3x49 19.43948.90323YesNo078
263x49 I2x57 19.0159.77246NoYes1780
273x53 I2x57 37.61434.479NoYes080
283x53 G.H5.19 36.7645.655NoNo088
29G.H5.15 G.H5.19 36.33852.65454NoNo088
30G.H5.11 G.H5.15 35.48682.69937NoNo088
31b.b4x6 b.l1x3 85.42313.58481YesYes499
322x38 2x42 19.22253.88108NoYes067
332x38 I2x57 19.015110.1841NoYes060
34G.H5.11 G.S3.03 29.84214.17563NoYes587
35G.S1.04 G.S3.03 17.40475.21108NoYes077
36G.S1.04 G.S4.03 11.84535.54602NoNo077
37G.h2s4.01 b.l5x5 18.178111.2605YesYes199
38G.H3.17 b.l27x1 34.75573.28317YesYes149
39G.H3.15 G.H3.17 42.41227.14348NoYes184
40G.S4.03 G.S5.05 11.40933.45458NoYes079
41b.l5x5 b.l7x2 36.31146.27131YesYes199
42G.s3h2.03 b.l7x2 18.53484.02929YesYes199
433x50 7x53 11.02876.71477YesYes299
443x50 5x58 10.4288.65385YesYes299
453x47 5x58 14.377412.1694NoYes299
463x47 5x57 14.61473.11646NoNo097
473x51 5x57 13.77796.90271NoNo087
483x51 3x55 12.10196.42688NoNo087
496x40 7x53 10.40725.74108NoYes079
50G.H2.04 G.H2.07 26.5225.75625YesYes099
51G.H2.04 G.H2.08 41.63583.63983YesNo098
52G.H2.08 G.H3.15 41.59293.25283NoNo188
53G.H2.07 b.l7x2 17.79324.36483YesYes199
54G.H2.07 G.h2s4.01 18.66943.75869YesYes199
55G.H2.07 b.l9x6 60.68053.57963YesYes198
56G.s3h2.03 b.l9x6 17.63156.5045YesYes198
57G.H2.06 b.l9x6 57.59373.34137YesYes198
58G.H2.04 G.H3.08 24.90994.79231YesNo099
59G.H2.06 b.l17x6 55.23829.14317YesYes199
60G.H3.08 G.S4.04 24.79655.76625NoNo099
61G.H3.09 G.S4.04 24.680713.8067YesNo099
62G.H3.06 G.hgh4.02 14.71934.81308NoYes078
63b.b2x4 b.b6x5 32.29323.1065NoYes066
64b.b10x4 b.b2x4 32.029116.7545NoNo066
65b.b10x2 b.b10x4 31.76644.33902NoNo066
66b.b10x2 b.b14x3 31.50365.37738NoYes065
67b.b14x3 b.b15x1 27.95094.35325YesYes059
68b.b15x1 b.b16x6 22.465914.5744YesYes398
69b.b16x4 b.b16x6 11.19657.8445YesYes368
70b.b16x4 b.b17x6 10.688811.7853YesNo067
71b.b17x6 g.h1x14 10.41336.2015NoNo079
72g.h1x11 g.h1x14 20.21241.35923YesNo099
73b.1x11 g.h1x11 18.54935.23958NoYes089
74b.1x11 g.h1x12 14.1053.149NoNo086
75g.h1x12 g.h1x8 11.32031.83921NoYes067
76b.b16x6 b.b17x3 10.9025.96108YesNo385
77b.b17x3 g.h1x10 10.62895.40471NoNo059
78g.h1x10 g.h1x14 10.35318.78785NoNo099
79b.l17x5 b.l17x6 54.55544.38752NoYes169
80b.l17x5 b.l19x2 54.19442.434NoYes169
81b.l17x3 b.l19x2 36.55345.46313YesYes199
82b.b19x4 b.l17x3 19.30667.95467YesYes189
83b.b19x4 b.b20x6 14.45667.34325YesYes186
84b.b17x7 b.b20x6 39.709610.7519YesYes186
85b.b17x7 b.b21x1 19.19844.50694YesYes187
86b.b20x4 b.l17x3 15.659817.6019YesYes189
87b.b20x4 b.b20x6 28.89474.39173YesYes186
88b.b20x2 b.l19x2 16.45577.31021YesYes169
89b.b20x2 b.b20x4 15.65587.68517YesYes168
90b.l2x5 b.l4x2 20.749128.1418NoNo054
91b.l26x5 g.ctx15 11.20017.90913NoYes059
92b.l26x5 g.ctx4 18.4716.80825NoYes057
93g.ctx3 g.ctx4 16.87433.75667YesYes097
94g.ctx3 g.ctx6 12.65647.5146YesYes096
95b.l4x2 g.ctx16 16.14116.75592NoYes448
96b.b2x5 b.l4x1 17.49066.27317YesNo075
97b.l4x1 g.ctx16 17.3353.69129NoYes058
98b.b4x2 b.b5x8 23.17033.57175YesNo085
99b.b5x7 b.b5x8 22.84653.39YesNo075
100b.l11x1 b.l9x6 19.02387.92521NoYes198
101b.b11x6 b.l11x1 18.63423.46719NoNo199
102b.b11x6 b.l9x3 15.739615.1755NoYes199
103b.b12x6 b.l9x3 14.52684.12875YesYes189
104b.b17x5 b.b17x7 19.33629.7895YesYes178
105b.b16x5 b.b17x5 17.06665.67013YesYes057
106b.b16x5 b.b17x4 13.4132.49175YesNo055
1077x49 7x53 39.2333.66533YesYes299
1087x45 7x49 25.68283.39352NoYes099
1096x48 7x45 25.30112.3805YesNo099
1103x36 6x48 24.29525.77423NoYes279
1113x36 Lig 24.03713.62312NoYes270
1122x53 7x46 10.51114.5061YesNo068
1132x50 7x46 11.06783.54567YesNo098
1142x50 7x49 11.31478.41181YesYes299
115b.b4x2 b.l3x2 20.27697.04213YesYes089
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
7x34Lig4.478272NoYes5010
LigNT22.57922YesYes0301
7x31Lig3.207212NoYes5010
E2Lig24.27652YesYes4010
E2x51Lig18.39042NoYes3010
NTNT8.991152YesYes3311
2x533x327.843830YesNo6721
2x533x363.408630YesNo6721
2x537x425.421460YesYes6722
2x603x323.864192NoNo6711
2x63E1x508.844292NoYes5822
E1x49E25.466790NoYes4421
E1x50E23.572882YesYes8421
3x22E24.514060NoYes4421
3x334x574.529212YesNo5612
3x334x613.552542YesNo5411
4x614x653.401122NoNo4512
4x64E215.17172NoYes4421
4x645x353.479792NoNo4222
4x65E2x527.16760NoNo5521
E2E248.52292YesYes4411
E2E2x519.897542YesNo4311
E2E2x528.484232YesNo4511
5x35E26.480192NoYes2421
5x36E210.7282NoYes4411
5x39E26.314192NoYes5421
5x32E23.583350NoYes2421
6x516x524.94242YesNo7812
6x517x373.425252YesNo7612
6x517x384.280062YesNo7611
6x547x346.504060NoNo5521
6x61E35.12942NoYes4412
7x387x423.94762NoYes6712
2x602x633.297812NoNo6512
2x60Lig7.744422NoYes6010
2x63E23.741212NoYes5421
3x32Lig7.173522NoYes7010
3x33Lig4.837672YesYes5010
3x366x485.774232NoYes7912
5x366x593.667252NoYes4512
6x516x559.3432YesNo7612
6x51Lig4.734752YesYes7010
6x587x304.800212NoNo4411
6x58Lig9.546692NoYes4010
6x61Lig8.10652NoYes4010
7x27Lig4.254060NoYes4010
7x38Lig5.497632NoYes6010
5x43Lig5.470812NoYes5010
E2x52Lig4.530752NoYes5010
3x335x433.730252YesNo5511
3x375x435.352770NoNo7521
5x36Lig3.696192NoYes4010
4x61Lig3.331582NoYes4010
3x36Lig3.623122NoYes7010
7x30Lig6.765942NoYes4010
E1Lig4.642NoYes0010
7x24NT2.885460NoYes7321
2x67E22.7652NoYes4421
2x64E120NoNo5021
6x62Lig1.742270NoYes5010
1x28Lig1.704252NoYes4010
1x247x311.298750NoNo0521
1x251x280.3710NoNo4421
6x657x300.36550NoNo1421

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
100.00Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
90.91Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
75.00Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
75.00Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
69.57Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
69.57Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
69.57Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
69.23Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
65.38Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
64.29Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
64.29Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
64.29Consensusbradykinin_onOrthosteric Ligandbk2_on
64.29Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
64.29Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
64.00Consensusangiotensin_onOrthosteric Ligandat1_on
64.00Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
62.50Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
61.54Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
61.54Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
61.54Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
61.54Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
60.87Consensuschemerin_onOrthosteric Ligandcml1_on
60.71Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
60.71Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
60.71Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
60.00Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
60.00Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
57.14Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
56.52Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
56.52Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
55.56Single6JODAngiotensin II6JOD-AT2-Angiotensin II
55.56Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
55.56Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
55.17Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
55.17Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
53.85Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
53.85Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
53.85Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
53.57Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
53.57Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
53.57Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
53.57Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
53.33Single8IY6Endothelin-18IY6-ETB-Endothelin-1
53.33Consensusendothelin_onOrthosteric Ligandetb_on eta_on
52.00Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
52.00Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
51.85Single3OE0CVX153OE0-CXCR4-CVX15
51.85Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
51.61Single5GLHEndothelin-15GLH-ETB-Endothelin-1
51.61Single6IGKEndothelin-36IGK-ETB-Endothelin-3
51.61Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
51.61Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
51.61Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
50.00Single6OS2TRV0266OS2-AT1-TRV026
50.00Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
50.00Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
50.00Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
50.00Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
50.00Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
50.00Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
48.48Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
48.39Single6IGLIRL16206IGL-ETB-IRL1620
48.39Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
48.28Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
48.28Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
48.28Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
48.28Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
48.28Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
48.28Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
48.28Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
48.15Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
48.15Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
48.15Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
48.15Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
48.00Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
48.00Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
47.06Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
46.88Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
46.67Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
46.67Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
46.67Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
46.67Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
46.43Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
46.43Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
46.43Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
46.43Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
46.43Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
46.43Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
46.43Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
46.43Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
45.83Single6OS1TRV0266OS1-AT1-TRV026
45.16Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
45.16Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
45.16Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
45.16Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
45.16Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
44.83Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
44.83Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
44.83Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
44.44Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
44.44Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
44.44Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
44.00Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
44.00Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
44.00Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
44.00Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
44.00Single8XWSCXCL58XWS-CXCR2-CXCL5
43.48Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
43.48Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
43.33Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
43.33Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
43.33Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
43.33Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
43.33Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
43.33Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
43.33Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
42.86Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
42.86Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
42.86Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
42.86Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
42.86Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
42.86Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
42.42Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
42.31Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
42.31Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
42.31Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
41.94Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
41.94Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
41.67Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
41.67Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
41.67Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
41.67Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
41.67Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
41.38Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
41.38Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
41.38Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
41.38Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
41.38Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
41.38Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
41.18Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
40.74Single6KNMJN241-96KNM-Apelin-JN241-9
40.74Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
40.74Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
40.74Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
40.74Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
40.74Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
40.74Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
40.74Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
40.74Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
40.74Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
40.74Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
40.74Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
40.74Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
40.62Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
40.62Single9KDFRES-701-39KDF-ETB-RES-701-3
40.00Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
40.00Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
40.00Single7F1TMIP-1a7F1T-CCR5-MIP-1a
40.00Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
40.00Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
40.00Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
40.00Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
40.00Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
40.00Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
40.00Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
40.00Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
40.00Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
40.00Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
40.00Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
40.00Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
40.00Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
40.00Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
40.00Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
40.00Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
40.00Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
40.00Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
40.00Consensusvasop-oxy_onOrthosteric Ligandv2_on
40.00Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
39.39Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
39.39Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
39.29Single4IARErgotamine4IAR-5-HT1B-Ergotamine
39.29Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
39.29Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
39.29Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
39.29Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
39.29Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
39.29Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
39.29Single8WDTphotoNECA8WDT-A2A-photoNECA
39.29Single8XWNCXCL88XWN-CXCR2-CXCL8
39.29Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
39.29Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
39.29Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
39.13Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
39.13Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
38.89Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
38.71Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
38.71Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
38.71Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
38.71Single8ZRTET-18ZRT-ETB-ET-1
38.71Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
38.71Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
38.46Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
38.46Single6MXTSalmeterol6MXT-β2-Salmeterol
38.46Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
38.46Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
38.46Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
38.46Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
38.46Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
38.46Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
38.46Single8XWACXCL18XWA-CXCR2-CXCL1
38.46Single8XWMCXCL68XWM-CXCR2-CXCL6
38.46Consensusorexin_onOrthosteric Ligandox2_on
38.24Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
38.24Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
37.93Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
37.93Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
37.93Single7XNACYN1548067XNA-SST2-CYN154806
37.93Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
37.93Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
37.93Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
37.93Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
37.93Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
37.93Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
37.93Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
37.93Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
37.93Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
37.50Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
37.50Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
37.50Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
37.50Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
37.50Single7SK3CXCL127SK3-ACKR3-CXCL12
37.50Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
37.50Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
37.50Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
37.50Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
37.50Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
37.50Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
37.50Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
37.50Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
37.50Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
37.50Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
37.50Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
37.14Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
37.14Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
37.04Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
37.04Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
37.04Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
37.04Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
37.04Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
37.04Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
37.04Single8XVUCXCL28XVU-CXCR2-CXCL2
37.04Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
37.04Single8ZPLHF511168ZPL-CXCR4-HF51116
37.04Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
37.04Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
36.67Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
36.67Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
36.67Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
36.67Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
36.67Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
36.67Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
36.67Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
36.36Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
36.00Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
36.00Single5C1MBU725C1M-μ-BU72
36.00Single6D26Fevipiprant6D26-DP2-Fevipiprant
36.00Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
36.00Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
36.00Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
36.00Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
36.00Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
36.00Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
36.00Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
36.00Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
36.00Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
36.00Consensusdp_offOrthosteric Liganddp2_off
35.71Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
35.71Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
35.71Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
35.71Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
35.71Single7XN9L-054,5227XN9-SST2-L-054,522
35.71Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
35.71Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
35.71Single8XQJJN2418XQJ-Apelin-JN241
35.71Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
35.71Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
35.71Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
35.71Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
35.48Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
35.48Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
35.48Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
35.48Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
35.48Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
35.48Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
35.48Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
35.29Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
35.29Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
34.78Single6AKYMaraviroc6AKY-CCR5-Maraviroc
34.78Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
34.78Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
34.78Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
34.78Single8GNGIstradefylline8GNG-A2A-Istradefylline
34.78Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
34.78Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
34.62Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
34.62Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
34.62Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
34.62Single8E0GBU728E0G-μ-BU72
34.62Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
34.62Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
34.62Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
34.62Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
34.62Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
34.62Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
34.62Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
34.62Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
34.62Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
34.62Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
34.62Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
34.62Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
34.48Single4XT1Fractalkine4XT1-US28-Fractalkine
34.48Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
34.48Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
34.48Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
34.48Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
34.48Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
34.48Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
34.48Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
34.48Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
34.48Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
34.48Consensuslpl_onOrthosteric Ligands1p_on lpa_on
34.48Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
34.48Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
34.48Consensussomatostatin_offOrthosteric Ligandsst2_off
34.38Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
34.38Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
34.38Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
34.38Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
34.38Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
34.38Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
34.38Consensuspac_onOrthosteric Ligandpac1_on
34.29Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
34.29Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
34.29Consensusbombesin_onOrthosteric Ligandbb2_on
34.29Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
34.29Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
33.33Single3QAKUK-4320973QAK-A2A-UK-432097
33.33Single4MBSMaraviroc4MBS-CCR5-Maraviroc
33.33Single4RWADIPP-NH24RWA-δ-DIPP-NH2
33.33Single4XEENeurotensin4XEE-NTS1-Neurotensin
33.33Single4XESNeurotensin4XES-NTS1-Neurotensin
33.33Single4XT3Fractalkine4XT3-US28-Fractalkine
33.33Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
33.33Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
33.33Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
33.33Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
33.33Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
33.33Single6YVRNTS8-136YVR-NTS1-NTS8-13
33.33Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
33.33Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
33.33Single7F61PF-036547467F61-H3-PF-03654746
33.33Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
33.33Single7SK5CXCL127SK5-ACKR3-CXCL12
33.33Single7UL3Famotidine7UL3-H2-Famotidine
33.33Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
33.33Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
33.33Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
33.33Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
33.33Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
33.33Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8JJLOlodaterol8JJL-β2-Olodaterol
33.33Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
33.33Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
33.33Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
33.33Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
33.33Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8XQJJN2418XQJ-Apelin-JN241
33.33Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
33.33Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
33.33Single8ZPNAMD31008ZPN-CXCR4-AMD3100
33.33Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
33.33Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
33.33Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
33.33Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
33.33Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
33.33Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
33.33Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
33.33Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
33.33Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
33.33Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
33.33Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
33.33Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
33.33Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
33.33Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
33.33Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
33.33Consensuslpa_offOrthosteric Ligandlpa1_off
33.33Consensuslpl_offOrthosteric Ligands1p_off lpa_off
33.33Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
33.33Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
33.33Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
32.50Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
32.35Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
32.35Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
32.35Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
32.35Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
32.35Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
32.35Consensusglp_onOrthosteric Ligandglp1_on glp2_on
32.35Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
32.26Single5WF5UK-4320975WF5-A2A-UK-432097
32.26Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
32.26Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
32.26Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
32.26Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
32.26Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
32.26Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
32.26Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
32.26Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
32.26Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
32.26Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
32.14Single4BUONeurotensin4BUO-NTS1-Neurotensin
32.14Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
32.14Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
32.14Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
32.14Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
32.14Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
32.14Single6IBLArformoterol6IBL-β1-Arformoterol
32.14Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
32.14Single7EZCUKA7EZC-A2A-UKA
32.14Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
32.14Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
32.14Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
32.14Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
32.14Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
32.14Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
32.14Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
32.14Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
32.14Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
32.14Single8XWFCXCL38XWF-CXCR2-CXCL3
32.14Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
32.14Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
32.14Consensuscck_onOrthosteric Ligandccka_on cckb_on
32.14Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
32.14Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
32.14Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
32.14Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
32.14Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
32.14Consensusprostanoid_offOrthosteric Ligandep_off dp_off
32.00Single6D27CAY104716D27-DP2-CAY10471
32.00Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
32.00Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
32.00Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
32.00Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
32.00Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
32.00Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
32.00Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
32.00Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
32.00Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
32.00Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
32.00Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
32.00Single9CHXS-Carazolol9CHX-β2-S-Carazolol
32.00Consensusa3_onOrthosteric Liganda3a_on
32.00Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
32.00Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
32.00Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
32.00Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
32.00Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
32.00Consensushca_on_gpOrthosteric Ligandhca2_on_gp
31.82Single6ME5Agomelatine6ME5-MT1-Agomelatine
31.82Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.43Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
31.43Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
31.43Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
31.43Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
31.43Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
31.43Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
31.25Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
31.25Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
31.25Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
31.25Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
31.03Single3NY9ICI118-5513NY9-β2-ICI118-551
31.03Single4UG2CGS216804UG2-A2A-CGS21680
31.03Single5WF6UK-4320975WF6-A2A-UK-432097
31.03Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
31.03Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
31.03Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
31.03Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
31.03Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
31.03Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
31.03Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
31.03Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
31.03Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
31.03Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
31.03Single8QJ2pN1628QJ2-MC4-pN162-Gs
31.03Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
31.03Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
31.03Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
31.03Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
31.03Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
31.03Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
30.77Single7C61Ergotamine7C61-5-HT1B-Ergotamine
30.77Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
30.77Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
30.77Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
30.77Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
30.77Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
30.77Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
30.77Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
30.77Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
30.77Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
30.77Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
30.77Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
30.77Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
30.77Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
30.77Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
30.77Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
30.77Single8JXSPF-61428JXS-D1-PF-6142
30.77Single8S4DCMF-0198S4D-Apelin-CMF-019
30.77Single8TF5Oleic acid8TF5-GPR6-Oleic acid
30.77Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
30.77Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
30.77Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
30.77Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
30.77Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
30.77Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
30.77Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
30.77Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
30.77Consensusa3_on_gpOrthosteric Liganda3a_on_gp
30.77Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
30.77Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
30.77Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
30.77Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
30.77Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
30.77Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
30.77Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
30.77Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
30.77Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
30.77Consensuspth_onOrthosteric Ligandpth1_on pth2_on
30.77Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
30.77Consensustrace-amine_onOrthosteric Ligandta1_on
30.56Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
30.43Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
30.43Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
30.30Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
30.30Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
30.30Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
30.30Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
30.30Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
30.30Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
30.30Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
30.00Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
30.00Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
30.00Single7F8XNN90567F8X-CCKA-NN9056
30.00Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
30.00Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
30.00Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
30.00Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
30.00Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
30.00Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
30.00Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
30.00Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
30.00Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
30.00Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
30.00Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
30.00Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
30.00Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
30.00Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
30.00Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
29.73Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
29.73Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
29.73Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
29.63Single2YDVNECA2YDV-A2A-NECA
29.63Single3P0GBI1671073P0G-β2-BI167107
29.63Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
29.63Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
29.63Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
29.63Single4UHRCGS216804UHR-A2A-CGS21680
29.63Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
29.63Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
29.63Single5G53NECA5G53-A2A-NECA-Gs
29.63Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
29.63Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
29.63Single6J21Aprepitant6J21-NK1-Aprepitant
29.63Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
29.63Single6WGTLSD6WGT-5-HT2A-LSD
29.63Single7B6WCyclazosin7B6W-α1b-Cyclazosin
29.63Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
29.63Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
29.63Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
29.63Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
29.63Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
29.63Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
29.63Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
29.63Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
29.63Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
29.63Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
29.63Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
29.63Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
29.63Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
29.63Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
29.63Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
29.63Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
29.63Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
29.63Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
29.63Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
29.63Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
29.63Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
29.63Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
29.63Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
29.63Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
29.63Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Consensusneurotensin_onOrthosteric Ligandnts1_on
29.63Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
29.63Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
29.63Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
29.41Single6FJ3PTH6FJ3-PTH1-PTH
29.41Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
29.41Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
29.41Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
29.41Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
29.41Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
29.41Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
29.27Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
29.17Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
29.17Single4BWBNeurotensin4BWB-NTS1-Neurotensin
29.17Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
29.17Single6AKXA4R6AKX-CCR5-A4R
29.17Single6ME2Ramelteon6ME2-MT1-Ramelteon
29.17Single6ME9Ramelteon6ME9-MT2-Ramelteon
29.17Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
29.17Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
29.17Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
29.17Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
29.17Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.17Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
29.17Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
29.17Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
29.17Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
29.17Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
29.17Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
29.17Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
29.17Single8IWESpermidine8IWE-TA9-Spermidine
29.17Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
29.17Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
29.17Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
29.17Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
29.17Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
29.17Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
29.17Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
29.17Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
29.17Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
29.17Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
29.17Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
29.17Consensusorexin_offOrthosteric Ligandox2_off ox1_off
29.17Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
29.03Single6HLOAprepitant6HLO-NK1-Aprepitant
29.03Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
29.03Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
29.03Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
29.03Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
29.03Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
29.03Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
29.03Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
29.03Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
29.03Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
29.03Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
29.03Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
29.03Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
29.03Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
28.95Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
28.95Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
28.57Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
28.57Single4AMIBucindolol4AMI-β1-Bucindolol
28.57Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
28.57Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
28.57Single6A93Risperidone6A93-5-HT2A-Risperidone
28.57Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
28.57Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
28.57Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
28.57Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
28.57Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
28.57Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
28.57Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
28.57Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
28.57Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
28.57Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
28.57Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.57Single7YITNalfurafine7YIT-κ-Nalfurafine
28.57Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
28.57Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
28.57Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
28.57Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
28.57Single8JJ8Formoterol8JJ8-β2-Formoterol
28.57Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
28.57Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
28.57Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
28.57Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
28.57Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
28.57Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
28.57Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
28.57Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
28.57Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
28.57Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
28.57Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
28.57Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
28.57Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
28.57Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
28.57Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
28.57Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
28.57Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
28.57Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
28.57Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
28.57Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
28.57Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
28.57Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
28.57Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
28.57Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
28.57Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
28.21Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
28.21Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
28.21Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
28.12Single6PT2KGCHM076PT2-δ-KGCHM07
28.12Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
28.12Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.12Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
28.12Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
28.12Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
28.12Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
28.12Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
28.12Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
28.00Single4ZJCSB-6740424ZJC-OX1-SB-674042
28.00Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
28.00Single6KUXRS-799486KUX-α2a-RS-79948
28.00Single6MH8ZM-2413856MH8-A2A-ZM-241385
28.00Single6PS0S-Carazolol6PS0-β2-S-Carazolol
28.00Single6PS4ICI118-5516PS4-β2-ICI118-551
28.00Single6PS5S-Propranolol6PS5-β2-S-Propranolol
28.00Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
28.00Single7AROLUF58337ARO-A2A-LUF5833-Na
28.00Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
28.00Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
28.00Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
28.00Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
28.00Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
28.00Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
28.00Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
28.00Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
28.00Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
28.00Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
28.00Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
28.00Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
28.00Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
28.00Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
28.00Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.00Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.00Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
28.00Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
28.00Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
28.00Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
28.00Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
28.00Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
28.00Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
28.00Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
28.00Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
28.00Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
28.00Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
28.00Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
28.00Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
28.00Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
28.00Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.00Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.00Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
28.00Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
28.00Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
28.00Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
28.00Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
28.00Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
28.00Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
28.00Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
28.00Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
28.00Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
28.00Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
28.00Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
28.00Consensushca_onOrthosteric Ligandhca2_on
28.00Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
27.91Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
27.78Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
27.78Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
27.78Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
27.78Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
27.78Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
27.78Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
27.78Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
27.78Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
27.59Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
27.59Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
27.59Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
27.59Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
27.59Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
27.59Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
27.59Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.59Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
27.59Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
27.59Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
27.59Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.59Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
27.59Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
27.59Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
27.59Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
27.59Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.59Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
27.59Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
27.59Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
27.59Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
27.59Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
27.59Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
27.59Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
27.59Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
27.59Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
27.50Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
27.27Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
27.27Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
27.27Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
27.27Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
27.27Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
27.27Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
27.27Consensusp2y_offOrthosteric Ligandp2y1_off
27.27Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
27.03Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
26.92Single2Y02Carmoterol2Y02-β1-Carmoterol
26.92Single2Y04Salbutamol2Y04-β1-Salbutamol
26.92Single3NY8ICI118-5513NY8-β2-ICI118-551
26.92Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
26.92Single4EJ4Naltrindole4EJ4-δ-Naltrindole
26.92Single4GBRS-Carazolol4GBR-β2-S-Carazolol
26.92Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
26.92Single4QKX35V4QKX-β2-35V
26.92Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
26.92Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
26.92Single6H7MSalbutamol6H7M-β1-Salbutamol
26.92Single6PS1Timolol6PS1-β2-Timolol
26.92Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
26.92Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
26.92Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
26.92Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
26.92Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
26.92Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
26.92Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
26.92Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
26.92Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
26.92Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
26.92Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
26.92Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
26.92Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
26.92Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
26.92Single7UL4Alvimopan7UL4-μ-Alvimopan
26.92Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
26.92Single7V3ZCP559407V3Z-CB1-CP55940
26.92Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
26.92Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
26.92Single7WC7Lisuride7WC7-5-HT2A-Lisuride
26.92Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
26.92Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
26.92Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
26.92Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
26.92Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
26.92Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
26.92Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
26.92Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
26.92Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
26.92Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
26.92Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
26.92Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
26.92Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
26.92Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
26.92Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
26.92Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
26.92Single8JXRLSD8JXR-D1-LSD
26.92Single8K5DGSK2560738K5D-HCA2-GSK256073
26.92Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
26.92Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
26.92Single8T1WCVN4248T1W-GPR6-CVN424
26.92Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
26.92Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
26.92Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
26.92Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
26.92Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
26.92Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
26.92Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
26.92Consensus5ht5_onOrthosteric Ligand5ht5a_on
26.92Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
26.92Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
26.92Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
26.92Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
26.92Consensusdopamine_offOrthosteric Ligandd2_off d3_off
26.92Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
26.92Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
26.92Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
26.92Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
26.92Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
26.92Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
26.67Single5ZTYAM102575ZTY-CB2-AM10257
26.67Single6PT3DPI-2876PT3-δ-DPI-287
26.67Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
26.67Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
26.67Single7SK9CCX6627SK9-ACKR3-CCX662
26.67Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
26.67Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
26.67Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
26.67Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
26.67Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
26.67Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
26.67Single9IPYJR14a9IPY-C3aB-JR14a
26.67Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
26.67Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
26.67Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
26.47Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
26.47Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
26.47Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
26.47Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
26.47Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
26.32Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
26.09Single4XNWMRS25004XNW-P2Y1-MRS2500
26.09Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
26.09Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
26.09Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.09Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
26.09Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
26.09Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
26.09Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
26.09Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
25.93Single2RH1S-Carazolol2RH1-β2-S-Carazolol
25.93Single2Y03Isoprenaline2Y03-β1-Isoprenaline
25.93Single2YCWS-Carazolol2YCW-β1-S-Carazolol
25.93Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
25.93Single5D6LS-Carazolol5D6L-β2-S-Carazolol
25.93Single5JQHS-Carazolol5JQH-β2-S-Carazolol
25.93Single5N2RPSB-365N2R-A2A-PSB-36-Na
25.93Single5N2SPSB365N2S-A1-PSB36
25.93Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
25.93Single5TVNLSD5TVN-5-HT2B-LSD
25.93Single5WIUNemonapride5WIU-D4-Nemonapride
25.93Single5WIVNemonapride5WIV-D4-Nemonapride-Na
25.93Single5WQCEMPA5WQC-OX2-EMPA
25.93Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
25.93Single6E67BI1671076E67-β2-BI167107-Gs(CT)
25.93Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
25.93Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
25.93Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
25.93Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
25.93Single6TP6Filorexant6TP6-OX1-Filorexant
25.93Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
25.93Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
25.93Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
25.93Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
25.93Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
25.93Single7W41PD1762527W41-BB2-PD176252
25.93Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
25.93Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
25.93Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
25.93Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.93Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.93Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
25.93Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
25.93Single8QOTNanobody-E8QOT-μ-Nanobody-E
25.93Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
25.93Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
25.93Single8ZMFA1L108ZMF-5-HT2C-A1L10
25.93Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
25.93Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
25.93Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
25.93Single9EHSLUF76029EHS-A3A-LUF7602
25.93Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
25.93Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
25.93Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
25.93Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.93Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
25.93Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
25.93Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
25.93Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
25.93Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
25.93Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
25.93Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
25.93Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
25.93Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
25.93Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
25.93Consensusamine_offonOrthosteric Ligandamine_off amine_on
25.93Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
25.93Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
25.93Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
25.93Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
25.93Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
25.93Consensusbombesin_offOrthosteric Ligandbb2_off
25.93Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
25.93Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
25.93Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
25.93Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
25.93Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
25.93Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
25.81Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
25.81Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
25.81Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
25.81Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
25.81Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
25.81Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
25.81Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
25.81Single8WKYPG-9348WKY-MC4-PG-934
25.81Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
25.81Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
25.71Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
25.71Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
25.71Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
25.71Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
25.64Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
25.64Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
25.64Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.64Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
25.00Single3OE9IT1t3OE9-CXCR4-IT1t
25.00Single4BV0Neurotensin4BV0-NTS1-Neurotensin
25.00Single5D5AS-Carazolol5D5A-β2-S-Carazolol
25.00Single5D5BS-Carazolol5D5B-β2-S-Carazolol
25.00Single5XR8AM8415XR8-CB1-AM841
25.00Single6H7JIsoprenaline6H7J-β1-Isoprenaline
25.00Single6HLLCP999946HLL-NK1-CP99994
25.00Single6J20Aprepitant6J20-NK1-Aprepitant
25.00Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
25.00Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
25.00Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
25.00Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
25.00Single6TQ7SB-3348676TQ7-OX1-SB-334867
25.00Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
25.00Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
25.00Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
25.00Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
25.00Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
25.00Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
25.00Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
25.00Single7PX4PSB-21137PX4-A2A-PSB-2113
25.00Single7R0CAVP7R0C-V2-AVP-Arrestin2
25.00Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
25.00Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
25.00Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
25.00Single7TUYGSK682753A7TUY-GPR183-GSK682753A
25.00Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
25.00Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
25.00Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
25.00Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
25.00Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
25.00Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
25.00Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
25.00Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
25.00Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
25.00Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
25.00Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
25.00Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
25.00Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
25.00Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
25.00Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
25.00Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
25.00Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
25.00Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
25.00Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
25.00Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
25.00Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
25.00Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
25.00Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
25.00Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
25.00Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
25.00Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
25.00Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
25.00Single8K5BNiacin8K5B-HCA2-Niacin
25.00Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
25.00Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
25.00Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
25.00Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
25.00Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
25.00Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
25.00Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
25.00Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
25.00Single8ZWFJR14a8ZWF-C3aB-JR14a
25.00Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
25.00Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
25.00Single9BJKNaloxone9BJK-μ-Naloxone-NAM
25.00Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
25.00Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
25.00Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
25.00Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
25.00Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
25.00Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
25.00Consensusa2_onOrthosteric Liganda2b_on
25.00Consensusa2_on_gpOrthosteric Liganda2b_on_gp
25.00Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
25.00Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
25.00Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
25.00Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
25.00Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
25.00Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
25.00Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
25.00Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
25.00Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
25.00Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
25.00Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
25.00Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
25.00Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
25.00Consensuslpa_onOrthosteric Ligandlpa1_on
25.00Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
25.00Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
25.00Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
25.00Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
25.00Consensusrelaxin_onOrthosteric Ligandrxfp4_on
25.00Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
25.00Consensustachykinin_offOrthosteric Ligandnk1_off
24.39Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
24.32Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
24.32Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
24.24Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
24.24Single6W25SHU91196W25-MC4-SHU9119-Ca
24.24Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
24.24Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
24.24Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
24.24Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
24.24Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
24.24Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
24.14Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
24.14Single3D4STimolol3D4S-β2-Timolol
24.14Single4LDEBI1671074LDE-β2-BI167107
24.14Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
24.14Single4PY02MeSATP4PY0-P2Y12-2MeSATP
24.14Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
24.14Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
24.14Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
24.14Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
24.14Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
24.14Single7DFPSpiperone7DFP-D2-Spiperone
24.14Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
24.14Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
24.14Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
24.14Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
24.14Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
24.14Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
24.14Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
24.14Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
24.14Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
24.14Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
24.14Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
24.14Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
24.14Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
24.14Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
24.14Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
24.14Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
24.14Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
24.14Single8XYIVUF106618XYI-CXCR3-VUF10661
24.14Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
24.14Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
24.14Single9DGIZ85267113509DGI-CB1-Z8526711350
24.14Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
24.14Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
24.14Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
24.14Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
24.14Consensusalpha1_offOrthosteric Ligandalpha1a_off
24.14Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
24.14Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
24.14Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
24.14Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
24.00Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
24.00Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
24.00Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
24.00Single5WS3EMPA5WS3-OX2-EMPA
24.00Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
24.00Single6TODEMPA6TOD-OX1-EMPA-Na
24.00Single7BR3Elagolix7BR3-GnRH1-Elagolix
24.00Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
24.00Single7F8ULintitript7F8U-CCKA-Lintitript
24.00Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
24.00Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
24.00Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
24.00Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
24.00Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
24.00Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
24.00Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
24.00Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
24.00Single7XRRLemborexant7XRR-OX2-Lemborexant
24.00Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
24.00Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
24.00Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
24.00Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
24.00Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
24.00Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
24.00Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
24.00Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
24.00Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
24.00Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
24.00Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
24.00Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
24.00Consensusalpha2_offOrthosteric Ligandalpha2c_off
24.00Consensusangiotensin_offOrthosteric Ligandat1_off
24.00Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
24.00Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
24.00Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
24.00Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
24.00Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
23.68Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
23.68Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
23.53Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
23.53Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
23.53Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
23.53Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
23.53Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
23.33Single5X93K-87945X93-ETB-K-8794
23.33Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
23.33Single6H7LDobutamine6H7L-β1-Dobutamine
23.33Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
23.33Single7UM4AS26747237UM4-5-HT5A-AS2674723
23.33Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
23.33Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
23.33Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
23.33Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
23.33Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
23.33Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
23.33Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
23.33Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
23.33Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
23.33Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
23.33Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
23.33Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
23.33Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
23.33Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
23.33Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
23.33Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
23.33Consensusendothelin_offOrthosteric Ligandetb_off
23.33Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
23.33Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
23.26Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
23.08Single2YDOAdenosine2YDO-A2A-Adenosine
23.08Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
23.08Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
23.08Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
23.08Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
23.08Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
23.08Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
23.08Single6A94Zotepine6A94-5-HT2A-Zotepine
23.08Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
23.08Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
23.08Single6TPGEMPA6TPG-OX2-EMPA
23.08Single6TPNHTL66416TPN-OX2-HTL6641
23.08Single6V9SGTPL114036V9S-OX1-GTPL11403
23.08Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
23.08Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
23.08Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
23.08Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
23.08Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
23.08Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
23.08Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
23.08Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
23.08Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.08Single7T32ZM-2413857T32-A2A-ZM-241385
23.08Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
23.08Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
23.08Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
23.08Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
23.08Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
23.08Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
23.08Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Single8IHKAcifran8IHK-HCA3-Acifran
23.08Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
23.08Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
23.08Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
23.08Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
23.08Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
23.08Single8K5CAcipimox8K5C-HCA2-Acipimox
23.08Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
23.08Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.08Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.08Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
23.08Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
23.08Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
23.08Single8ZPMAMD0708ZPM-CXCR4-AMD070
23.08Single9AS5Mescaline9AS5-5-HT2A-Mescaline
23.08Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
23.08Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
23.08Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
23.08Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
23.08Consensusalpha1_onOrthosteric Ligandalpha1a_on
23.08Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
23.08Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
23.08Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
23.08Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
23.08Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
23.08Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
23.08Consensusgrh_offOrthosteric Ligandgnrh1_off
22.86Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
22.86Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
22.86Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
22.73Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
22.73Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
22.58Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
22.58Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
22.58Single8X5YAstemizole8X5Y-H1-Astemizole
22.58Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
22.58Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
22.58Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
22.58Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
22.50Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
22.50Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
22.22Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
22.22Single2Y01Dobutamine2Y01-β1-Dobutamine
22.22Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
22.22Single3EMLZM-2413853EML-A2A-ZM-241385
22.22Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
22.22Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
22.22Single4QIMANTA XV4QIM-SMO-ANTA XV
22.22Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
22.22Single4YAYZD-71554YAY-AT1-ZD-7155
22.22Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
22.22Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
22.22Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
22.22Single5T04Neurotensin5T04-NTS1-Neurotensin
22.22Single5UENDU1725UEN-A1-DU172
22.22Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
22.22Single6DRXLisuride6DRX-5-HT2B-Lisuride
22.22Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
22.22Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
22.22Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
22.22Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
22.22Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
22.22Single6S0LZM-2413856S0L-A2A-ZM-241385
22.22Single6TOTLemborexant6TOT-OX1-Lemborexant
22.22Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
22.22Single7BU7BI1671077BU7-β1-BI167107
22.22Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
22.22Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
22.22Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
22.22Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
22.22Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
22.22Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
22.22Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
22.22Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
22.22Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
22.22Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
22.22Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
22.22Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
22.22Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
22.22Single8CU6LJ-45178CU6-A2A-LJ-4517
22.22Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
22.22Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
22.22Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
22.22Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
22.22Single8JJOAlprenolol8JJO-β2-Alprenolol
22.22Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
22.22Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
22.22Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
22.22Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
22.22Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
22.22Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
22.22Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
22.22Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
22.22Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
22.22Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
22.22Single9AS1DMT9AS1-5-HT2A-DMT
22.22Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
22.22Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
22.22Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
22.22Single9H37A1IR09H37-A2A-A1IR0-Na
22.22Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
22.22Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
22.22Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
22.22Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
22.22Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
22.22Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
22.22Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
22.22Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
22.22Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
22.22Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
22.22Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
22.22Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
22.22Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
22.22Consensusblt_onOrthosteric Ligandblt1_on
22.22Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
22.22Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
22.22Consensuscck_offOrthosteric Ligandccka_off
22.22Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
22.22Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
22.22Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
22.22Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
22.22Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
22.22Consensusleukotriene_onOrthosteric Ligandblt_on
22.22Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
22.22Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
22.22Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
22.22Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
21.95Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.95Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
21.88Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
21.88Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
21.88Single8IEBA1LYA8IEB-GPR156-A1LYA
21.88Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
21.74Single6TQ9SB-4081246TQ9-OX1-SB-408124
21.74Single8A2OTheophylline8A2O-A2A-Theophylline-Na
21.74Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.74Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
21.74Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
21.74Single9CHUNoradrenaline9CHU-β2-Noradrenaline
21.74Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
21.74Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
21.74Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
21.62Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
21.62Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
21.62Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
21.62Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
21.43Single2Y00Dobutamine2Y00-β1-Dobutamine
21.43Single5IUAQ274563485IUA-A2A-Q27456348-Na
21.43Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
21.43Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
21.43Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
21.43Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
21.43Single6PS6Timolol6PS6-β2-Timolol
21.43Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
21.43Single6S0QZM-2413856S0Q-A2A-ZM-241385
21.43Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
21.43Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
21.43Single6Z4SSR486926Z4S-NTS1-SR48692
21.43Single7C4SS1P7C4S-S1P3-S1P
21.43Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
21.43Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
21.43Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
21.43Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
21.43Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
21.43Single7WC6LSD7WC6-5-HT2A-LSD
21.43Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
21.43Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
21.43Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
21.43Single8GNEKW-63568GNE-A2A-KW-6356-Na
21.43Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
21.43Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
21.43Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
21.43Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
21.43Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
21.43Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
21.43Single9HAPTolvaptan9HAP-V2-Tolvaptan
21.43Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
21.43Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
21.43Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
21.43Consensusadenosine_offOrthosteric Liganda1_off a2_off
21.43Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
21.43Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
21.43Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
21.43Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
21.43Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
21.43Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
21.21Single8IEBA1LYA8IEB-GPR156-A1LYA
21.21Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
21.21Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
21.05Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
21.05Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
21.05Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
20.83Single3OE6IT1t3OE6-CXCR4-IT1t
20.83Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
20.83Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
20.83Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
20.83Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
20.83Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
20.83Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.83Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
20.83Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
20.83Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
20.83Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
20.83Single8JPSCCL78JPS-ACKR1-CCL7
20.83Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
20.83Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
20.83Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
20.83Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
20.83Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
20.83Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
20.83Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
20.83Single9LRCHistamine9LRC-H4-Histamine
20.83Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
20.83Consensus5ht2_onOrthosteric Ligand5ht2b_on
20.83Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.83Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
20.83Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
20.83Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
20.69Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
20.69Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
20.69Single4DJHJDTic4DJH-κ-JDTic
20.69Single4U15Tiotropium4U15-M3-Tiotropium
20.69Single5TZRMK86665TZR-FFA1-MK8666
20.69Single5V54Methiothepin5V54-5-HT1B-Methiothepin
20.69Single5XRAAM115425XRA-CB1-AM11542
20.69Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
20.69Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
20.69Single6E59L-7607356E59-NK1-L-760735
20.69Single6OL9Tiotropium6OL9-M5-Tiotropium
20.69Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
20.69Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
20.69Single7FEECP559407FEE-CB1-CP55940-ZCZ011
20.69Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
20.69Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
20.69Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
20.69Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
20.69Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
20.69Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
20.69Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
20.69Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.69Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
20.69Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
20.69Consensus5ht1_offOrthosteric Ligand5ht1b_off
20.69Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
20.69Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
20.69Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
20.69Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
20.69Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
20.69Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
20.69Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
20.69Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
20.69Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
20.69Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
20.59Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
20.59Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
20.59Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
20.59Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
20.51Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
20.51Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
20.00Single3PBLEticlopride3PBL-D3-Eticlopride
20.00Single4O9RCyclopamine4O9R-SMO-Cyclopamine
20.00Single5CXVTiotropium5CXV-M1-Tiotropium
20.00Single6CM4Risperidone6CM4-D2-Risperidone
20.00Single6KQICP559406KQI-CB1-CP55940-Org27569
20.00Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
20.00Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
20.00Single6ZG4HTL00099366ZG4-M1-HTL0009936
20.00Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
20.00Single7K15MKD0467K15-BLT1-MKD046-Na
20.00Single7SRQLSD7SRQ-5-HT2B-LSD
20.00Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
20.00Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
20.00Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
20.00Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
20.00Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
20.00Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
20.00Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
20.00Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
20.00Single8JWY2-1188JWY-A2A-2-118
20.00Single8JWZAB9288JWZ-A2A-AB928-Na
20.00Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
20.00Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
20.00Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
20.00Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
20.00Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
20.00Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
20.00Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
20.00Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
20.00Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
20.00Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
20.00Single9B9Y7DY9B9Y-CB1-7DY
20.00Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
20.00Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
20.00Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
20.00Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
20.00Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
20.00Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
20.00Consensusgq_nucleotideOrthosteric Ligandgq_p2y
20.00Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
20.00Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
20.00Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
20.00Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
20.00Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
19.57Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
19.51Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
19.51Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
19.44Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
19.44Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
19.44Consensuscalcitonin_onOrthosteric Ligandctlike_on
19.44Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
19.35Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
19.35Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
19.35Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
19.35Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.35Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
19.35Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
19.23Single3ODUIT1t3ODU-CXCR4-IT1t
19.23Single3PWHZM-2413853PWH-A2A-ZM-241385
19.23Single4QINSAG1.54QIN-SMO-SAG1.5
19.23Single4S0VSuvorexant4S0V-OX2-Suvorexant
19.23Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
19.23Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
19.23Single5ZKQABT-4915ZKQ-PAF-ABT-491
19.23Single6B73MP11046B73-κ-MP1104
19.23Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
19.23Single6DS0Ly2660976DS0-5-HT2B-Ly266097
19.23Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
19.23Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
19.23Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
19.23Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
19.23Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
19.23Single6TPJSuvorexant6TPJ-OX2-Suvorexant
19.23Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
19.23Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
19.23Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
19.23Single7F8YDevazepide7F8Y-CCKA-Devazepide
19.23Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
19.23Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
19.23Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
19.23Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
19.23Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
19.23Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
19.23Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
19.23Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
19.23Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
19.23Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
19.23Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
19.23Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
19.23Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
19.23Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
19.23Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
19.23Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
19.23Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
19.23Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
19.23Single8Y0HVUF114188Y0H-CXCR3-VUF11418
19.23Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
19.23Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
19.23Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
19.23Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
19.23Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
19.23Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
19.23Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
19.23Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
19.23Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
19.23Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
19.23Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
19.23Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
19.23Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
19.23Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
19.23Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
19.23Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
19.23Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
19.23Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
19.23Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
19.23Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
19.05Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
19.05Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
18.92Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
18.92Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
18.92Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
18.92Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
18.75Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
18.75Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
18.75Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.75Single9JF4PD1683689JF4-BB1-PD168368
18.75Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
18.75Consensuskisspeptin_onOrthosteric Ligandkiss1_on
18.60Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
18.52Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
18.52Single3REYXAC3REY-A2A-XAC
18.52Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
18.52Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
18.52Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
18.52Single5IU7Q274563465IU7-A2A-Q27456346-Na
18.52Single5IUBQ274563445IUB-A2A-Q27456344-Na
18.52Single5JTBZM-2413855JTB-A2A-ZM-241385
18.52Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
18.52Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
18.52Single5UVIZM-2413855UVI-A2A-ZM-241385
18.52Single6AQFZM-2413856AQF-A2A-ZM-241385
18.52Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
18.52Single6TP3Nemorexant6TP3-OX1-Nemorexant
18.52Single6VI4JDTic6VI4-κ-JDTic
18.52Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
18.52Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
18.52Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
18.52Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
18.52Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
18.52Single6ZINSR486926ZIN-NTS1-SR48692
18.52Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
18.52Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
18.52Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
18.52Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
18.52Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
18.52Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
18.52Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
18.52Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
18.52Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
18.52Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
18.52Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.52Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
18.52Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
18.52Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
18.52Single8RLNLUF58348RLN-A2A-LUF5834
18.52Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
18.52Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
18.52Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
18.52Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
18.52Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
18.52Single9ARXSerotonin9ARX-5-HT2A-Serotonin
18.52Single9AS3LSD9AS3-5-HT2A-LSD
18.52Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single9BA0A1AKN9BA0-CB1-A1AKN
18.52Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
18.52Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
18.52Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
18.52Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
18.52Consensusa2_offOrthosteric Liganda2a_off
18.52Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
18.52Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
18.42Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
18.42Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
18.42Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
18.42Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
18.18Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
18.18Single7QA8Peptide7QA8-STE2-Peptide
18.18Single7QA8Peptide7QA8-STE2-Peptide
18.18Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
18.18Single8IEIA1LYA8IEI-GPR156-A1LYA
18.18Single8IEIA1LYA8IEI-GPR156-A1LYA
18.18Single8IEPA1LYA8IEP-GPR156-A1LYA
18.18Single8IEPA1LYA8IEP-GPR156-A1LYA
18.18Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
18.18Single8KIGSHU91198KIG-MC3-SHU9119-Ca
18.18Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
18.18Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
18.18Single9M4TSilodosin9M4T-Alpha1A-Silodosin
18.18Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
18.18Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
18.18Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
18.18Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
17.95Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
17.95Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
17.95Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
17.95Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
17.95Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
17.86Single4DAJTiotropium4DAJ-M3-Tiotropium
17.86Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
17.86Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
17.86Single4MQSIperoxo4MQS-M2-Iperoxo
17.86Single4U14Tiotropium4U14-M3-Tiotropium
17.86Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
17.86Single5DHHSB-6121115DHH-NOP-SB-612111
17.86Single5IU8Q274563475IU8-A2A-Q27456347-Na
17.86Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
17.86Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
17.86Single5TGZAM65385TGZ-CB1-AM6538
17.86Single5UIGCmpd-15UIG-A2A-Cmpd-1
17.86Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
17.86Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
17.86Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
17.86Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
17.86Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
17.86Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
17.86Single7PYRPSB-21157PYR-A2A-PSB-2115
17.86Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
17.86Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
17.86Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
17.86Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
17.86Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.86Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
17.86Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
17.86Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
17.86Single8X63Mepyramine8X63-H1-Mepyramine
17.86Single8X64Desloratadine8X64-H1-Desloratadine
17.86Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
17.86Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
17.86Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
17.86Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
17.86Single9IYAONO-97105319IYA-GPR55-ONO-9710531
17.86Single9JEAAtropine9JEA-M1-Atropine
17.86Consensusalpha2_onOrthosteric Ligandalpha2b_on
17.86Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
17.86Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
17.86Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
17.86Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
17.86Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
17.86Consensushistamine_offOrthosteric Ligandh1_off
17.86Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
17.86Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
17.65Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
17.65Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
17.65Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
17.50Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
17.50Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
17.39Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
17.39Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
17.39Single7WC4Serotonin7WC4-5-HT2A-Serotonin
17.39Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
17.39Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
17.39Single8PWNTheophylline8PWN-A2A-Theophylline
17.24Single4JKVTaladegib4JKV-SMO-Taladegib
17.24Single4NTJAZD12834NTJ-P2Y12-AZD1283
17.24Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
17.24Single5XPRBosentan5XPR-ETB-Bosentan
17.24Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
17.24Single6HLPNetupitant6HLP-NK1-Netupitant
17.24Single6LUQHaloperidol6LUQ-D2-Haloperidol
17.24Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
17.24Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.24Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.24Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
17.24Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
17.24Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
17.24Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
17.24Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
17.24Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single9B9ZA1AKO9B9Z-CB1-A1AKO
17.24Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
17.24Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
17.24Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
17.24Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
17.24Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.24Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.24Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
16.67Single3RFMCaffeine3RFM-A2A-Caffeine
16.67Single5V56TC1145V56-SMO-TC114
16.67Single5V57TC1145V57-SMO-TC114
16.67Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
16.67Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
16.67Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
16.67Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
16.67Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
16.67Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
16.67Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
16.67Single8EA0Iperoxo8EA0-M3-Iperoxo
16.67Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
16.67Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
16.67Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
16.67Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
16.67Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8XVLZibotentan8XVL-ETA-Zibotentan
16.67Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
16.67Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
16.67Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
16.67Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
16.67Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
16.67Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
16.67Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
16.67Consensussensory_onOrthosteric Ligandopsins_on
16.28Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
16.22Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
16.13Single4N4WSANT-14N4W-SMO-SANT-1
16.13Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
16.13Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
16.13Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
16.13Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
16.13Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
16.13Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
16.13Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
16.13Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
16.13Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
16.00Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
16.00Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
16.00Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
16.00Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
16.00Single7WC5Psilocin7WC5-5-HT2A-Psilocin
16.00Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.00Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
16.00Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
16.00Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
16.00Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
16.00Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
16.00Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
16.00Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
16.00Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
16.00Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
15.79Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
15.79Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
15.79Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
15.79Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
15.62Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
15.62Single6K1QIRL25006K1Q-ETB-IRL2500
15.62Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
15.62Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
15.62Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single8XVJMacitentan8XVJ-ETA-Macitentan
15.62Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
15.62Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single5L7IVismodegib5L7I-SMO-Vismodegib
15.38Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
15.38Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
15.38Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
15.38Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
15.38Single6TP4ACT-4622066TP4-OX1-ACT-462206
15.38Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
15.38Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
15.38Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
15.38Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
15.38Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
15.38Single7UL2SR486927UL2-NTS1-SR48692-Na
15.38Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
15.38Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
15.38Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
15.38Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
15.38Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
15.38Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
15.38Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.38Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
15.38Single9AS7Psilocin9AS7-5-HT2A-Psilocin
15.38Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
15.38Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
15.38Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
15.38Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
15.38Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
15.38Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
15.38Consensusneurotensin_offOrthosteric Ligandnts1_off
15.38Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
15.15Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
15.15Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
15.15Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
15.15Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
15.00Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
15.00Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
15.00Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
15.00Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
14.81Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
14.81Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
14.81Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
14.81Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
14.81Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
14.81Single5U09Taranabant5U09-CB1-Taranabant
14.81Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
14.81Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
14.81Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
14.81Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
14.81Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
14.81Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.81Single9H2XA1IR19H2X-A2A-A1IR1-Na
14.81Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
14.81Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
14.81Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
14.81Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
14.81Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
14.71Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
14.71Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
14.71Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.71Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
14.71Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
14.71Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
14.29Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
14.29Single3RZECidoxepin3RZE-H1-Cidoxepin
14.29Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
14.29Single6IQLL7458706IQL-D4-L745870
14.29Single6TPKRetosiban6TPK-OT-Retosiban
14.29Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
14.29Single6ZG9GSK10347026ZG9-M1-GSK1034702
14.29Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
14.29Single7VODCariprazine7VOD-5-HT2A-Cariprazine
14.29Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
14.29Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
14.29Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
14.29Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
14.29Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
14.29Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
14.29Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
14.29Consensusopsins_offOrthosteric Ligandrhodopsin_off
14.29Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
14.29Consensussensory_offOrthosteric Ligandopsins_off
14.29Consensusvasop-oxy_offOrthosteric Ligandot_off
13.79Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
13.79Single5DHGC-355DHG-NOP-C-35
13.79Single5DSGTiotropium5DSG-M4-Tiotropium
13.79Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
13.79Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
13.79Single6GPSMK08126GPS-CCR2-MK0812
13.79Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
13.79Single7YXAONO-54306087YXA-S1P5-ONO-5430608
13.79Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
13.79Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
13.79Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
13.79Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
13.51Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
13.51Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
13.51Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
13.33Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
13.33Single5CGCHTL142425CGC-mGlu5-HTL14242
13.33Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
13.33Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
13.33Single6GPXMK08126GPX-CCR2-MK0812
13.33Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
13.33Single7SINNPS-21437SIN-CaS-NPS-2143
13.33Single7SINNPS-21437SIN-CaS-NPS-2143
13.33Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
13.33Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
13.33Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
13.33Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
13.33Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
13.33Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
13.33Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
13.33Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
13.33Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
13.33Consensusblt_offOrthosteric Ligandblt1_off
13.33Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
13.33Consensusep_offOrthosteric Ligandep4_off
13.16Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
13.04Single5MZPCaffeine5MZP-A2A-Caffeine-Na
13.04Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
12.90Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
12.90Single9AS9RS130-1809AS9-5-HT2A-RS130-180
12.90Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
12.50Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
12.50Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
12.50Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
12.50Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
12.50Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
12.50Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single5CGDHTL142425CGD-mGlu5-HTL14242
12.12Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
12.12Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.12Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
12.12Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
12.12Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single3OE8IT1t3OE8-CXCR4-IT1t
12.00Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
12.00Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
12.00Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
12.00Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
11.76Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
11.76Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
11.54Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
11.54Single3UZAGTPL92363UZA-A2A-GTPL9236
11.54Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
11.54Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
11.54Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
11.54Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
11.54Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
11.54Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
11.54Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
11.54Consensusgi_sensoryOrthosteric Ligandgi_opsins
11.54Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
11.54Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
11.43Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
11.11Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
11.11Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
11.11Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
11.11Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
11.11Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
11.11Single6LI0C176LI0-GPR52-C17
11.11Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
11.11Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
11.11Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
11.11Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
11.11Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
11.11Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
11.11Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
11.11Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
11.11Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
10.71Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
10.71Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
10.71Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
10.71Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
10.71Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
10.71Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
10.71Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
10.71Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
10.71Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
10.71Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
10.71Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
10.71Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
10.71Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
10.71Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
10.71Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
10.71Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
10.71Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
10.71Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
10.53Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
10.34Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
10.34Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
10.34Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
10.34Single7VV6C48/807VV6-MRGPRX2-C48/80
10.34Single8K2WAMG4878K2W-CXCR3-AMG487
10.34Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.34Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
10.34Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
10.34Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
10.34Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
10.00Single6IIVDaltroban6IIV-TXA2-Daltroban
10.00Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
10.00Single7F83PF-051904577F83-Ghrelin-PF-05190457
10.00Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
10.00Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
10.00Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
10.00Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
10.00Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
10.00Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
10.00Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
10.00Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
9.68Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
9.68Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
9.68Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
9.68Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
9.68Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
9.68Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
9.68Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
9.68Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
9.68Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
9.68Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
9.68Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
9.38Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
9.38Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
9.38Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
9.38Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
9.09Single5X33BIIL2605X33-BLT1-BIIL260
9.09Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
9.09Single6IIURamatroban6IIU-TXA2-Ramatroban
9.09Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
9.09Single9BJKNAM9BJK-μ-Naloxone-NAM
8.82Single9JH5C16:0 Ceramide9JH5-CysLT2-C16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
8.33Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
8.00Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
8.00Single8HS2Fab0468HS2-GPR20-Fab046
8.00Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
7.69Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
7.69Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
7.69Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
7.69Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
7.69Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
7.41Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
7.41Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
7.14Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
7.14Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
7.14Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
7.14Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
7.14Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
7.14Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
7.14Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
7.14Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
7.14Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
6.90Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
6.90Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
6.90Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
6.67Single6FFIMMPEP6FFI-mGlu5-MMPEP
6.67Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
6.67Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
6.45Single6FFHFenobam6FFH-mGlu5-Fenobam
6.25Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
6.25Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
6.25Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single9HC04YI9HC0-mGlu5-4YI
6.06Single7P2L4YI7P2L-mGlu5-4YI
6.06Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
6.06Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
6.06Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
6.06Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
5.71Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
5.56Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
5.41Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
4.55Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
4.55Single6D35Cholesterol6D35-SMO-Cholesterol
4.55Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.55Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.55Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
4.55Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
4.55Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042
4.55Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
4.55Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
4.55Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-BHFF
4.55Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
4.55Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626
4.55Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
4.55Single7DTTCa7DTT-CaS-Ca-Ca
4.55Single7DTTCa7DTT-CaS-Ca-Ca
4.55Single7DTUTryptophan7DTU-CaS-Tryptophan
4.55Single7DTUTryptophan7DTU-CaS-Tryptophan
4.55Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.55Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.55Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.55Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.55Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
4.55Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.55Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.55Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.55Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.55Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.55Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.55Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
4.55Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
4.55Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.55Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.55Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.55Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.55Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.55Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.55Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.55Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.55Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.55Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7T9NM22 Fab7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
4.55Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.55Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.55Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.55Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.55Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.55Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.55Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
4.55Single7XW7K1-707XW7-TSH-K1-70
4.55Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.55Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.55Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.55Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.55Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.55Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.55Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.55Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.55Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.55Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.55Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.55Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.55Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
4.55Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.55Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.55Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.55Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.55Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
4.55Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
4.55Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.55Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.55Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
4.55Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
4.55Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
4.55Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
4.55Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.55Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.55Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
4.55Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.55Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.55Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.55Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.55Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.55Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.55Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.55Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.55Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.55Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.55Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.55Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.55Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.55Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.55Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.55Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.55Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
4.55Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
4.55Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
4.55Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
4.55Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
4.55Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
4.55Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.55Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.55Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.55Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.55Single8WVXNorrin8WVX-LGR4-Norrin
4.55Single8WVYNorrin8WVY-LGR4-Norrin
4.55Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.55Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.55Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.55Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.55Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.55Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.55Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
4.55Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.55Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.55Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.55Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.55Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.55Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.55Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.55Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.55Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single9KHHNorrin9KHH-LGR4-Norrin
4.55Single9S37NB219S37-LGR4-NB21
4.55Single9UTBSucralose9UTB-TAS1R2; TAS1R3-Sucralose
4.35Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.35Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.35Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.35Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.35Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.35Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.35Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
4.35Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
4.17Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
4.17Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
4.17Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
4.17Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
4.00Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
4.00Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
4.00Single7UTZTR14027UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
4.00Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
4.00Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
3.85Single5L7DCholesterol5L7D-SMO-Cholesterol
3.85Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
3.85Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
3.57Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
3.57Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.45Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
3.45Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.33Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
3.33Single8G94CD698G94-S1P1-CD69-Gi1/β1/γ2
3.23Single8IYXYL-3658IYX-GPR34-YL-365
3.12Single8Y73MPAM-158Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
3.03Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
3.03Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
2.94Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
2.63Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.63Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.50Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.50Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.44Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.27Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
chemokine_on_gp ccr_on_gp
cxcr_on_gp
chemerin_on_gp cml1_on_gp
Net Summary
Imin 3.11613
Number of Linked Nodes 949
Number of Links 1127
Number of Hubs 170
Number of Links mediated by Hubs 671
Number of Communities 18
Number of Nodes involved in Communities 218
Number of Links involved in Communities 316
Path Summary
Number Of Nodes in MetaPath 116
Number Of Links MetaPath 115
Number of Shortest Paths 1610165
Length Of Smallest Path 3
Average Path Length 31.3089
Length of Longest Path 58
Minimum Path Strength 0.139
Average Path Strength 5.71479
Maximum Path Strength 22.8182
Minimum Path Correlation 0.701604
Average Path Correlation 0.971441
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 2.08333
Average % Of Corr. Nodes 39.4473
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 49.7618
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following differences:
Id1st Network2nd Network
protein_off_on_gpprotein_on_gpprotein_off
This network is also present in following consensuses:
IdComponents
protein_offon_gpprotein_on_gp
protein_off
class-a_on_gpsensory_on_gp
alicarboxylic_on_gp
amine_on_gp
lipid_on_gp
nucleotide_on_gp
peptide_on_gp
protein_on_gp



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Download protein_on_gp.zip



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