Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.hns1.01 8.1275414
2G.S1.03 5.7475419
3G.S1.06 5.5725438
4G.S3.03 5.7956208
5G.S3.06 10.4075417
6G.s3h2.03 4.9775419
7G.H2.06 6.072519
8G.H2.07 6.816519
9G.h2s4.01 6.498519
10G.S4.02 4.088518
11G.S4.03 3.495437
12G.S4.04 6409
13G.s4h3.04 6.792508
14G.H3.09 3.1125409
15G.H3.17 7.84615
16G.S5.03 4.23539
17G.S5.05 4.186539
18G.S5.06 3.66254128
19G.hgh4.05 12.7475406
20G.hgh4.11 5.9075405
21G.H4.04 3.30754244
22G.S6.01 4.1925405
23G.S6.02 6.4425408
24G.S6.05 9.24254125
25G.s6h5.01 6.48439
26G.s6h5.05 9.4475439
27G.H5.20 2.765478
28G.H5.23 5.86404
29b.1x4 2.765408
30b.1x11 3.13408
31b.1x15 4.24254177
32b.h2x5 5.078595
33b.lhb1x3 3.98492
34b.lhb1x11 6.15454
35b.l1x3 10.116589
36b.b2x3 3.66754136
37b.b2x5 8.5425137
38b.b4x6 12.54589
39b.b5x2 4.33754197
40b.b5x3 6.21571789
41b.b5x7 7.4075447
42b.l5x1 6.3508
43b.l5x5 7.0525819
44b.b6x5 4.365646
45b.b7x1 6.7075404
46b.l7x2 4.016519
47b.l7x4 5.67409
48b.b8x3 3.352566
49b.b8x4 6.65546
50b.l8x1 3.0825445
51b.b9x4 5.9175469
52b.l9x3 7.15569
53b.l9x6 4.732518
54b.b10x5 5.386509
55b.l10x1 3.9525403
56b.l11x2 8.105469
57b.b12x6 10.085468
58b.l12x3 3.66754275
59b.b13x7 7.7545107
60b.l13x3 8.635109
61b.l13x6 6.87409
62b.l13x7 4.1475409
63b.b15x2 7.5325416
64b.l15x1 5.58407
65b.l15x2 6.0254109
66b.b16x6 8.536108
67b.l17x3 10.4917619
68b.l17x6 6.7625419
69b.b18x1 6.505419
70b.b18x3 4.3225418
71b.b18x5 6.864515
72b.l18x1 6.2056286
73b.l18x3 7.7085285
74b.b19x2 7.90833616
75b.b19x4 6.24418
76b.b19x6 7.7475419
77b.l19x1 6419
78b.l19x2 7.2625419
79b.b20x4 8.57418
80b.b20x6 8.18333616
81b.b20x7 4.8175409
82b.l20x2 6.37409
83b.b21x1 10.6054177
84b.b21x2 3.3525406
85b.b21x7 4.4145265
86b.l21x2 4.8254144
87b.l21x5 4.90754144
88b.b22x5 6.1025407
89b.l22x5 7.655409
90b.b23x2 3.835406
91b.b23x3 3.73254297
92b.b23x6 6.216676147
93b.l23x1 6.57416
94b.b24x4 6.444146
95b.b24x5 3.475405
96b.b24x6 6.61254148
97b.b24x7 8.4875499
98b.l24x3 5.692595
99b.b25x7 5.4025457
100b.l25x3 10.6925459
101b.l25x6 12.374518
102b.b26x3 3.385406
103b.l26x1 6.77754137
104b.b27x3 4.06408
105b.l27x1 11.02619
106b.l27x2 9.3775459
107b.b28x4 8.0325456
108b.b28x6 5.75167659
109g.ntx4 3.0854164
110g.h1x1 3.0965162
111g.h1x14 4.7754179
112g.l1x4 4.705408
113g.ctx3 7.79509
114Lig 7.374291420
115NT.F33 6.118526
1161x36 3.38754306
1171x56 4.4385118
1181x60 12.014115
1192x40 6.6625408
1202x42 9.3765318
1212x50 4.551676159
1222x57 6.45408
1232x63 5.5775426
1243x30 7.255406
1253x33 10.0225426
1263x37 5.97286727
1273x39 4.194159
1283x42 7.06408
1293x51 8.616577
1303x54 3.414578
1314x64 3.56405
1325x40 4.8225426
1335x41 4.384525
1345x50 4.49754339
1355x57 6.31407
1365x58 9.0954348
1375x61 3.2825478
1386x48 9.0675408
1396x53 4.3254186
1406x55 8.594527
1416x57 4.34754186
1426x59 2.9975406
1437x41 4.954509
1447x49 7.2225159
1457x52 2.97408
1468x50 7.8945119
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1b.b5x7 b.b5x8 11.02533.39YesNo075
2b.b4x2 b.b5x8 11.23495.02NoNo085
3b.b4x2 b.l3x2 11.86224.15NoNo089
4G.hns1.01 b.l3x2 12.042611.49YesNo149
5G.S1.03 G.hns1.01 13.317211.32YesYes194
6G.S1.03 b.l5x5 13.66593YesYes199
7b.l3x1 b.l5x5 18.84136.57NoYes199
8b.b2x1 b.l3x1 33.666514.65NoNo189
9b.b2x1 b.l27x1 33.345519.29NoYes189
10b.b26x1 b.l27x1 54.77844.94NoYes099
11b.b26x1 b.b26x2 54.63143.44NoNo097
12b.b26x2 b.b2x3 54.37234.86NoYes076
13b.b2x3 b.b3x2 11.44112.83YesNo1365
14b.b28x3 b.b3x2 16.5872.77NoNo075
15b.b4x6 b.b5x3 10.053911.6YesYes899
16G.H2.07 G.h2s4.01 12.26234.01YesYes199
17G.H2.04 G.H2.07 52.333911NoYes099
18G.H2.04 G.H3.08 52.245510.72NoNo098
19G.H3.08 G.S4.04 52.07325.97NoYes089
20G.S4.04 G.s1h1.01 54.45743.01YesNo099
21G.s1h1.01 G.s1h1.05 54.36793.71NoNo099
22G.H1.01 G.s1h1.05 53.64626.12NoNo099
23G.H1.01 G.S1.06 53.41062.82NoYes398
24G.S1.06 G.S4.03 52.92182.85YesYes387
25G.H5.07 G.S4.03 38.19224.42NoYes397
26G.H1.08 G.H5.07 44.78822.92NoNo099
27G.H1.08 G.S2.06 44.50777.46NoNo099
28G.S2.06 G.S3.03 44.369510.72NoYes098
29G.S1.02 G.S3.03 41.82268.53NoYes068
30G.S1.02 I2x54 41.58474.86NoNo066
31b.l5x5 b.l7x2 21.91025.69YesYes199
32b.l7x2 b.l9x6 44.43043.52YesYes198
33G.H2.06 b.l9x6 1002.39YesYes198
34G.H2.06 b.l17x6 49.66449.68YesYes199
35G.H2.06 b.b18x1 49.25835.6YesYes199
36G.H2.08 G.h2s4.01 13.97523.77NoYes199
37G.H2.08 G.H3.15 13.56194.25NoNo198
38G.H3.15 G.H3.17 20.29883.39NoYes185
39G.H3.17 b.l27x1 12.22133.75YesYes159
40G.S4.03 G.S5.03 19.41382.94YesYes379
41G.H3.09 G.S6.01 12.58362.79YesYes095
42G.S5.04 G.S6.01 10.89713.17NoYes095
43G.H4.15 G.S5.04 10.71316.09NoNo089
44G.H4.15 G.S5.06 10.16043.65NoYes088
45G.H3.17 b.l23x1 20.363.35YesYes156
46G.H5.14 G.S5.03 11.73972.94NoYes069
47G.H5.10 G.S5.03 11.51827NoYes079
48G.H5.10 G.S6.02 13.33924.6NoYes078
49G.H5.14 G.S6.02 11.30934.84NoYes068
50G.H5.13 G.S6.02 23.693411.49NoYes088
51G.H5.13 G.H5.17 23.21593.92NoNo085
52G.H5.15 I2x51 41.20914.28NoNo086
53I2x51 I2x54 41.33336.07NoNo066
54G.H5.15 G.H5.19 41.0862.83NoNo088
556x30 G.H5.20 17.9472.57NoYes078
566x30 G.H5.17 22.73823.71NoNo075
573x54 G.H5.20 15.53792.85YesYes788
58G.H5.19 G.H5.23 40.96386.98NoYes084
59G.H5.22 G.H5.23 40.52163.37NoYes044
602x37 G.H5.22 40.416714.11NoNo084
612x37 2x39 32.91553.14NoNo088
62b.l17x6 b.l19x1 49.44343.99YesYes199
63b.l17x5 b.l19x1 98.20425.89NoYes169
64b.b19x6 b.l17x5 96.88513.26YesNo196
65b.b19x6 b.l17x3 95.194511.16YesYes199
66b.b20x6 b.l17x3 92.03894.53YesYes169
67b.b17x7 b.b20x6 86.605216.08NoYes186
68b.b17x5 b.b17x7 87.16357.03NoNo078
69b.b17x5 b.b21x1 86.925418.27NoYes077
70b.1x14 b.1x15 22.43381.37NoYes047
71b.1x14 g.h1x15 21.57411.52NoNo048
72b.1x11 g.h1x15 19.8541.58YesNo088
73b.1x11 g.h1x11 16.41075.54YesNo089
74b.1x12 g.h1x11 14.68762.82NoNo069
75b.1x12 b.1x9 13.82564.05NoNo064
76b.1x5 b.1x9 12.96344.65NoNo034
77b.1x1 b.1x5 12.10092.43NoNo043
78b.b18x1 b.l19x1 49.214710.77YesYes199
79b.b21x1 g.h1x14 70.65823.9YesYes1779
80b.l21x7 b.l23x1 26.44713.11NoYes056
81b.l21x7 b.l23x2 25.97486.22NoNo058
82b.b23x6 b.l23x2 31.84874.6YesNo078
83b.b23x6 b.l21x9 24.69988.46YesNo076
84b.b20x3 b.l21x9 23.50483.27NoNo086
85b.b20x3 b.b21x7 22.90694.03NoYes085
86b.b21x7 b.b23x2 18.71464.69YesYes056
87b.b22x5 b.b23x2 16.31346.09YesYes076
88b.b22x5 b.l18x1 14.50998.57YesYes076
89b.l18x1 b.l18x3 10.28649.67YesYes2865
90b.b2x3 b.b2x5 42.67183.49YesYes1367
91b.b2x5 b.l26x1 47.77839.7YesYes1377
92b.l26x1 b.l26x4 45.63983.64YesNo079
93b.l26x4 g.ctx4 45.49944.06NoNo097
94g.ctx3 g.ctx4 46.35374.83YesNo097
95g.ctx3 g.ctx6 10.612312.21YesNo096
96b.l22x1 g.ctx3 38.42718.83NoYes099
97b.l22x1 g.ctx5 38.27846.01NoNo099
98b.lhb1x11 g.ctx5 36.67184.24YesNo049
99b.b28x6 b.lhb1x11 35.06163.49YesYes594
100b.b28x4 b.b28x6 18.99223.48YesYes569
101b.b27x3 b.b28x6 19.79354.85YesYes089
102b.b27x3 b.l25x3 19.34866.85YesYes089
103b.l25x3 b.l27x2 37.33347.56YesYes599
104b.b28x4 b.l25x3 18.90914.41YesYes569
105g.h1x10 g.h1x14 63.7922.55NoYes099
106b.b17x3 g.h1x10 63.53826.1NoNo059
107b.b16x6 b.b17x3 63.284113.06YesNo085
108b.b13x7 b.b16x6 30.832814.03YesYes1078
109b.b12x3 b.b13x7 15.01445.59NoYes087
110b.b12x3 b.l13x7 14.73735.12NoYes089
111b.b11x5 b.l13x7 43.37184.85NoYes069
112b.b11x5 b.b14x3 41.68359.01NoNo065
113b.b10x2 b.b14x3 40.83944.76NoNo065
114b.b10x2 b.b10x4 38.30696.96NoNo066
115b.b10x4 b.b2x4 49.96224.51NoNo066
116b.b16x6 b.l13x3 31.11338.46YesYes1089
117b.b15x3 b.l13x3 15.0096.97NoYes099
118b.b15x3 b.l13x7 14.73253.23NoYes099
119b.b15x5 b.l13x3 15.00864.39NoYes1089
120b.b15x5 b.l13x7 14.7533.39NoYes089
121b.b13x5 b.b13x7 15.30526.49NoYes047
122b.b12x5 b.b13x5 14.74824.42NoNo064
123b.b11x3 b.b12x5 14.19132.98NoNo056
124b.b11x3 b.l10x1 13.91282.98NoYes053
125b.b14x5 b.l10x1 13.07776.92NoYes053
126b.b10x4 b.b14x5 12.80074.86NoNo065
127b.b2x4 b.b6x4 48.83212.93NoNo067
128b.b10x5 b.b6x4 47.70182.77YesNo097
129b.b10x5 b.b7x3 43.1782.77YesNo099
130b.b7x3 b.b8x3 42.04643.25NoYes096
131b.b8x1 b.b8x3 10.24113.27NoYes686
132b.b8x3 b.b9x4 18.20642.85YesYes669
133b.b12x6 b.b9x4 10.251515.94YesYes689
134b.l25x4 b.l27x2 35.78977.98NoYes059
135I1x48 b.l25x4 35.37897.15NoNo065
1362x39 3x46 33.11345.9NoNo088
1372x42 3x46 32.89523.52YesNo088
1382x42 4x46 30.24356.04YesNo3188
1392x45 4x46 30.43683.1NoNo098
1402x45 3x42 30.36559.76NoYes098
1413x42 4x50 52.32914.23YesNo089
1424x50 4x54 51.38763.42NoNo094
1433x30 4x54 51.07329.38YesNo064
1443x30 4x59 49.81332.9YesNo065
1454x59 4x60 49.49764.06NoNo059
1464x60 5x40 49.18183.35NoYes096
1475x40 5x41 39.49795.65YesYes265
1485x41 Lig 31.40282.84YesYes250
1497x41 Lig 14.4633.34YesYes090
1502x57 7x42 13.845312.89YesNo088
1512x50 7x49 17.56326.73YesYes1599
1521x50 2x50 33.23314.04NoYes099
1531x50 2x47 33.64733.13NoNo099
1542x44 2x47 33.40331.95NoNo079
1551x57 2x44 33.77941.76NoNo087
1561x57 1x58 34.15821.76NoNo084
1571x58 I1x51 34.56483NoNo048
158I1x48 I1x51 34.972613.86NoNo068
1592x46 3x39 14.60573.01NoYes099
1602x50 3x39 14.74884.34YesYes1599
1612x46 7x49 16.50458.41NoYes099
1622x46 3x42 31.0825.25NoYes098
163G.H3.09 G.S4.04 16.18753.22YesYes099
164G.H2.10 b.l3x1 14.94974.58NoNo189
165G.H2.10 b.l7x2 15.1043.17NoYes189
166G.H2.07 b.l9x6 55.36349.65YesYes198
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
LigNT.F334.172YesYes0601
2x60Lig10.222NoYes7010
2x63Lig12.482YesYes6010
2x64Lig2.840NoYes6010
3x29Lig5.692NoYes5010
E2.E234Lig5.440NoYes4010
E2x51Lig6.650NoYes5010
5x41Lig2.842YesYes5010
6x55Lig7.492YesYes7010
6x58Lig16.052NoYes5010
7x31Lig11.852NoYes5010
7x34Lig3.762NoYes6010
7x38Lig10.420NoYes6010
7x41Lig3.340YesYes9010
7x31NT.F337.032NoYes5611
7x32NT.F334.130NoYes4621
7x35NT.F3313.820NoYes6621
2x537x416.280NoYes7921
2x602x633.572NoYes7611
2x633x293.642YesNo6511
2x67E2.E2348.620NoNo5421
3x283x294.50NoNo6521
3x333x364.232YesNo6822
3x333x376.732YesYes6722
3x336x5510.472YesYes6721
3x363x373.752NoYes8722
3x367x413.892NoYes8921
3x375x446.242YesNo7722
3x376x554.122YesYes7721
5x375x402.832NoYes4622
5x375x414.152NoYes4521
5x405x415.652YesYes6521
5x415x444.422YesNo5712
5x416x554.862YesYes5711
6x487x413.010YesYes8921
6x516x5516.030NoYes6721
6x587x343.492NoNo5611
7x387x425.860NoNo6812
7x417x428.250YesNo9812
2x63E1x512.622YesNo6512
6x587x302.542NoNo5712
7x31NT.P321.582NoNo5312
1x28NT.F331.440NoYes8621

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
100.00Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
92.86Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
57.14Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
56.25Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
56.25Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
56.25Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
56.25Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
56.25Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
55.00Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
54.55Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
53.33Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
50.00Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
50.00Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
50.00Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
50.00Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
50.00Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
50.00Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
50.00Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
50.00Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
50.00Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
48.00Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
48.00Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
48.00Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
47.62Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
47.62Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
47.37Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
47.37Single6OS2TRV0266OS2-AT1-TRV026
47.37Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
47.37Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
47.37Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
47.37Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
47.37Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
47.37Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
47.37Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
47.37Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
47.06Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
47.06Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
46.67Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
45.83Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
45.83Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
45.45Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
45.45Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
45.45Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
45.00Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
45.00Single8ZPLHF511168ZPL-CXCR4-HF51116
45.00Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
43.75Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
43.75Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
43.75Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
43.48Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
43.48Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
43.48Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
43.48Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
43.48Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
42.86Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
42.86Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
42.86Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
42.86Single8QJ2pN1628QJ2-MC4-pN162-Gs
42.86Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
42.86Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
42.86Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
42.31Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
42.31Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
42.31Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
42.11Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
42.11Single6OS1TRV0266OS1-AT1-TRV026
42.11Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
42.11Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
42.11Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
42.11Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
42.11Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
42.11Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
42.11Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
42.11Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
42.11Consensusneurotensin_onOrthosteric Ligandnts1_on
42.11Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
41.67Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
41.67Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
41.67Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
41.67Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
41.67Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
41.18Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
41.18Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
41.18Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
41.18Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
40.91Single4XT1Fractalkine4XT1-US28-Fractalkine
40.91Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
40.91Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
40.91Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
40.91Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
40.91Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
40.91Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Single3OE6IT1t3OE6-CXCR4-IT1t
40.00Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
40.00Single4XEENeurotensin4XEE-NTS1-Neurotensin
40.00Single4XESNeurotensin4XES-NTS1-Neurotensin
40.00Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
40.00Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
40.00Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
40.00Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
40.00Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
40.00Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
40.00Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
40.00Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
40.00Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
40.00Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
40.00Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
40.00Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
40.00Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
40.00Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
39.29Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
39.29Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
39.29Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
39.29Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
39.13Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
39.13Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
39.13Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
39.13Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
39.13Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
39.13Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
39.13Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
39.13Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
39.13Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
39.13Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
39.13Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
38.89Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
38.89Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
38.89Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
38.46Single4XT3Fractalkine4XT3-US28-Fractalkine
38.46Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
38.46Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
38.46Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
38.46Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
38.46Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
38.46Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
38.46Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
38.46Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
38.10Single4BUONeurotensin4BUO-NTS1-Neurotensin
38.10Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
38.10Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
38.10Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
38.10Consensuscck_onOrthosteric Ligandccka_on cckb_on
38.10Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
38.10Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
38.10Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
38.10Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
37.50Single3OE9IT1t3OE9-CXCR4-IT1t
37.50Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
37.50Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
37.50Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
37.50Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
37.50Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
37.50Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
37.50Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
37.50Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
37.50Consensusangiotensin_onOrthosteric Ligandat1_on
37.50Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
37.50Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
37.50Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
37.50Consensusgq_nucleotideOrthosteric Ligandgq_p2y
37.50Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
37.50Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
37.04Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
37.04Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
37.04Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
36.84Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
36.84Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
36.36Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
36.36Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
36.36Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
36.36Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
36.36Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
36.36Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
36.36Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
36.36Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
36.36Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
36.36Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
36.36Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
36.36Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
36.36Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
36.36Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
36.00Single6JODAngiotensin II6JOD-AT2-Angiotensin II
36.00Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
36.00Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
36.00Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
36.00Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
36.00Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
36.00Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
36.00Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
36.00Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
36.00Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
36.00Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
35.71Single6IGLIRL16206IGL-ETB-IRL1620
35.71Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
35.29Single3ODUIT1t3ODU-CXCR4-IT1t
35.29Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
35.29Single8GNGIstradefylline8GNG-A2A-Istradefylline
35.29Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
35.29Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
35.29Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
35.29Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
35.29Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
35.29Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
35.00Single4BV0Neurotensin4BV0-NTS1-Neurotensin
35.00Single5XRAAM115425XRA-CB1-AM11542
35.00Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
35.00Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
35.00Single7FEECP559407FEE-CB1-CP55940-ZCZ011
35.00Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
35.00Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
35.00Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
35.00Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
35.00Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
35.00Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
35.00Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
35.00Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
35.00Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
35.00Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
34.78Single7F8XNN90567F8X-CCKA-NN9056
34.78Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
34.78Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
34.78Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
34.78Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
34.78Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
34.78Single8XWNCXCL88XWN-CXCR2-CXCL8
34.78Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
34.78Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
34.78Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
34.78Consensuslpl_onOrthosteric Ligands1p_on lpa_on
34.78Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
34.78Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
34.78Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
34.78Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
34.78Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
34.62Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
34.62Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
34.62Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
34.62Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
34.62Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
34.62Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
34.62Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
34.62Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
34.62Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Single8ZRTET-18ZRT-ETB-ET-1
34.62Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
34.62Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
34.62Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
34.62Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
34.62Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
34.62Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
34.48Single5GLHEndothelin-15GLH-ETB-Endothelin-1
34.48Single6IGKEndothelin-36IGK-ETB-Endothelin-3
33.33Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
33.33Single6KQICP559406KQI-CB1-CP55940-Org27569
33.33Single6MH8ZM-2413856MH8-A2A-ZM-241385
33.33Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
33.33Single6YVRNTS8-136YVR-NTS1-NTS8-13
33.33Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
33.33Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
33.33Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
33.33Single7SK3CXCL127SK3-ACKR3-CXCL12
33.33Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
33.33Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
33.33Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
33.33Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
33.33Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
33.33Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
33.33Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
33.33Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
33.33Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
33.33Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
33.33Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
33.33Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
33.33Single8IHKAcifran8IHK-HCA3-Acifran
33.33Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
33.33Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
33.33Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
33.33Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
33.33Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
33.33Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
33.33Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
33.33Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
33.33Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
33.33Single8XQJJN2418XQJ-Apelin-JN241
33.33Single8ZPMAMD0708ZPM-CXCR4-AMD070
33.33Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
33.33Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
33.33Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
33.33Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
33.33Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
33.33Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
33.33Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
33.33Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
33.33Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
33.33Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
33.33Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
33.33Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
33.33Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
33.33Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
33.33Consensushca_onOrthosteric Ligandhca2_on
33.33Consensuslpl_offOrthosteric Ligands1p_off lpa_off
33.33Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
33.33Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
33.33Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
33.33Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
33.33Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
33.33Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
33.33Consensusp2y_offOrthosteric Ligandp2y1_off
33.33Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
33.33Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
33.33Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
32.26Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
32.14Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
32.14Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
32.14Single9KDFRES-701-39KDF-ETB-RES-701-3
32.00Single3OE0CVX153OE0-CXCR4-CVX15
32.00Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
32.00Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
32.00Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
32.00Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
32.00Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
32.00Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
32.00Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
32.00Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
32.00Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
32.00Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
32.00Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
32.00Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
32.00Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
32.00Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
32.00Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
32.00Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
31.82Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
31.82Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
31.82Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
31.82Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
31.82Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
31.82Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
31.82Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
31.82Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
31.82Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
31.82Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
31.82Single8XVUCXCL28XVU-CXCR2-CXCL2
31.82Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
31.82Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
31.82Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
31.82Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
31.82Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
31.82Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
31.82Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
31.82Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
31.82Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
31.82Consensusprostanoid_offOrthosteric Ligandep_off dp_off
31.58Single4QIMANTA XV4QIM-SMO-ANTA XV
31.58Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
31.58Single6D27CAY104716D27-DP2-CAY10471
31.58Single6TOTLemborexant6TOT-OX1-Lemborexant
31.58Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
31.58Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
31.58Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
31.58Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
31.58Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
31.58Single7V3ZCP559407V3Z-CB1-CP55940
31.58Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
31.58Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
31.58Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
31.58Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
31.58Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
31.58Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
31.58Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
31.58Single8K5DGSK2560738K5D-HCA2-GSK256073
31.58Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
31.58Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
31.58Single9H37A1IR09H37-A2A-A1IR0-Na
31.58Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
31.58Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
31.58Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
31.58Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
31.58Consensushca_on_gpOrthosteric Ligandhca2_on_gp
31.25Single4XNWMRS25004XNW-P2Y1-MRS2500
31.25Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
31.25Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
31.25Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
31.03Single8IY6Endothelin-18IY6-ETB-Endothelin-1
31.03Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
31.03Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
31.03Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
31.03Consensusbradykinin_onOrthosteric Ligandbk2_on
31.03Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
31.03Consensusendothelin_onOrthosteric Ligandetb_on eta_on
31.03Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
30.77Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
30.77Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
30.77Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
30.77Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
30.77Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
30.77Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
30.77Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
30.77Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
30.43Single5WF6UK-4320975WF6-A2A-UK-432097
30.43Single5ZTYAM102575ZTY-CB2-AM10257
30.43Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
30.43Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
30.43Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
30.43Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
30.43Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
30.43Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Single8XQJJN2418XQJ-Apelin-JN241
30.43Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
30.43Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
30.43Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
30.43Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
30.43Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
30.43Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
30.00Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
30.00Single5N2SPSB365N2S-A1-PSB36
30.00Single6D26Fevipiprant6D26-DP2-Fevipiprant
30.00Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
30.00Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
30.00Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
30.00Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
30.00Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
30.00Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.00Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
30.00Single8GNEKW-63568GNE-A2A-KW-6356-Na
30.00Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
30.00Single8S4DCMF-0198S4D-Apelin-CMF-019
30.00Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
30.00Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
30.00Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
30.00Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
30.00Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
30.00Single9EHSLUF76029EHS-A3A-LUF7602
30.00Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
30.00Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
30.00Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
30.00Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
30.00Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
30.00Consensusdp_offOrthosteric Liganddp2_off
30.00Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
30.00Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
30.00Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
30.00Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
30.00Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
29.63Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
29.63Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.63Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
29.63Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
29.63Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
29.63Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
29.63Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
29.41Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
29.41Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
29.41Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
29.17Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
29.17Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
29.17Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
29.17Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
29.17Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
29.17Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
29.17Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
29.17Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
29.17Single8WDTphotoNECA8WDT-A2A-photoNECA
29.17Single8WKYPG-9348WKY-MC4-PG-934
29.17Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
29.17Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
29.17Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
29.17Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
29.17Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
29.17Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
29.17Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
29.17Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
29.17Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
29.03Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
29.03Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
28.57Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
28.57Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
28.57Single6FJ3PTH6FJ3-PTH1-PTH
28.57Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
28.57Single7R0CAVP7R0C-V2-AVP-Arrestin2
28.57Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
28.57Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
28.57Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
28.57Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.57Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
28.57Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
28.57Single8E0GBU728E0G-μ-BU72
28.57Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
28.57Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
28.57Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
28.57Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
28.57Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
28.57Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
28.57Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
28.57Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
28.57Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
28.57Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
28.57Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
28.57Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
28.57Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
28.57Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
28.57Consensuslpa_onOrthosteric Ligandlpa1_on
28.57Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
28.57Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
28.57Consensusrelaxin_onOrthosteric Ligandrxfp4_on
28.57Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
28.21Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
28.12Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
28.00Single3QAKUK-4320973QAK-A2A-UK-432097
28.00Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
28.00Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
28.00Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
28.00Single7SK5CXCL127SK5-ACKR3-CXCL12
28.00Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
28.00Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
28.00Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
28.00Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
28.00Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
28.00Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
28.00Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
28.00Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
28.00Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
28.00Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
28.00Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
28.00Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
28.00Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
27.78Single3PWHZM-2413853PWH-A2A-ZM-241385
27.78Single4BWBNeurotensin4BWB-NTS1-Neurotensin
27.78Single4S0VSuvorexant4S0V-OX2-Suvorexant
27.78Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
27.78Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
27.78Single5ZKQABT-4915ZKQ-PAF-ABT-491
27.78Single6TPJSuvorexant6TPJ-OX2-Suvorexant
27.78Single7BR3Elagolix7BR3-GnRH1-Elagolix
27.78Single7F8YDevazepide7F8Y-CCKA-Devazepide
27.78Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
27.78Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
27.78Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
27.78Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
27.78Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
27.78Single7XRRLemborexant7XRR-OX2-Lemborexant
27.78Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
27.78Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
27.78Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
27.78Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
27.78Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
27.78Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
27.78Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
27.78Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
27.78Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
27.78Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
27.59Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
27.59Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
27.59Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
27.59Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
27.27Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
27.27Single4RWADIPP-NH24RWA-δ-DIPP-NH2
27.27Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
27.27Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
27.27Single7K15MKD0467K15-BLT1-MKD046-Na
27.27Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
27.27Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
27.27Single8XWACXCL18XWA-CXCR2-CXCL1
27.27Single8XWMCXCL68XWM-CXCR2-CXCL6
27.27Single8XWSCXCL58XWS-CXCR2-CXCL5
27.27Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
27.27Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.27Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
27.27Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
27.27Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
27.27Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
27.27Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
27.27Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
27.27Consensuslpa_offOrthosteric Ligandlpa1_off
27.27Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
27.27Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
27.27Consensusorexin_onOrthosteric Ligandox2_on
27.27Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
26.92Single5WF5UK-4320975WF5-A2A-UK-432097
26.92Single6W25SHU91196W25-MC4-SHU9119-Ca
26.92Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
26.92Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.92Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
26.92Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
26.92Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
26.92Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
26.92Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
26.92Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
26.67Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
26.67Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
26.67Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
26.67Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
26.67Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
26.32Single3REYXAC3REY-A2A-XAC
26.32Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
26.32Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
26.32Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
26.32Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
26.32Single6TP3Nemorexant6TP3-OX1-Nemorexant
26.32Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
26.32Single6ZINSR486926ZIN-NTS1-SR48692
26.32Single7AROLUF58337ARO-A2A-LUF5833-Na
26.32Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
26.32Single7F61PF-036547467F61-H3-PF-03654746
26.32Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
26.32Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
26.32Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
26.32Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
26.32Single8K5CAcipimox8K5C-HCA2-Acipimox
26.32Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
26.32Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
26.32Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
26.32Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
26.32Single8ZPNAMD31008ZPN-CXCR4-AMD3100
26.32Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
26.32Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
26.32Consensusgrh_offOrthosteric Ligandgnrh1_off
26.09Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
26.09Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
26.09Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
26.09Single7EZCUKA7EZC-A2A-UKA
26.09Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
26.09Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
26.09Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.09Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
26.09Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
26.09Single8XWFCXCL38XWF-CXCR2-CXCL3
26.09Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
26.09Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
26.09Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
26.09Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
26.09Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
26.09Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
26.09Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
25.93Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
25.93Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
25.93Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
25.93Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
25.93Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
25.93Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
25.81Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
25.81Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
25.81Consensusbombesin_onOrthosteric Ligandbb2_on
25.81Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
25.81Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
25.00Single3EMLZM-2413853EML-A2A-ZM-241385
25.00Single3OE8IT1t3OE8-CXCR4-IT1t
25.00Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
25.00Single4UG2CGS216804UG2-A2A-CGS21680
25.00Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
25.00Single5T04Neurotensin5T04-NTS1-Neurotensin
25.00Single5TGZAM65385TGZ-CB1-AM6538
25.00Single5UIGCmpd-15UIG-A2A-Cmpd-1
25.00Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
25.00Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
25.00Single6KNMJN241-96KNM-Apelin-JN241-9
25.00Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
25.00Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
25.00Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
25.00Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
25.00Single6S0LZM-2413856S0L-A2A-ZM-241385
25.00Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
25.00Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
25.00Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
25.00Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
25.00Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
25.00Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
25.00Single7XN9L-054,5227XN9-SST2-L-054,522
25.00Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
25.00Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
25.00Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
25.00Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
25.00Single8A2OTheophylline8A2O-A2A-Theophylline-Na
25.00Single8CU6LJ-45178CU6-A2A-LJ-4517
25.00Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
25.00Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
25.00Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
25.00Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
25.00Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
25.00Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
25.00Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
25.00Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
25.00Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
25.00Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
25.00Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
25.00Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
25.00Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
25.00Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
25.00Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
25.00Single9IPYJR14a9IPY-C3aB-JR14a
25.00Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
25.00Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
25.00Consensusa3_onOrthosteric Liganda3a_on
25.00Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
25.00Consensuscck_offOrthosteric Ligandccka_off
25.00Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
25.00Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
25.00Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
25.00Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
25.00Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
25.00Consensuspac_onOrthosteric Ligandpac1_on
24.14Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
24.14Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
24.14Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
24.14Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
24.14Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
24.14Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
24.14Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
24.00Single4IARErgotamine4IAR-5-HT1B-Ergotamine
24.00Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
24.00Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
24.00Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
24.00Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
24.00Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
24.00Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
24.00Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
24.00Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
24.00Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
24.00Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
23.81Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
23.81Single5C1MBU725C1M-μ-BU72
23.81Single5IUAQ274563485IUA-A2A-Q27456348-Na
23.81Single5N2RPSB-365N2R-A2A-PSB-36-Na
23.81Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
23.81Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
23.81Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
23.81Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
23.81Single6S0QZM-2413856S0Q-A2A-ZM-241385
23.81Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
23.81Single6TP6Filorexant6TP6-OX1-Filorexant
23.81Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
23.81Single6Z4SSR486926Z4S-NTS1-SR48692
23.81Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
23.81Single7C4SS1P7C4S-S1P3-S1P
23.81Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
23.81Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
23.81Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
23.81Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
23.81Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
23.81Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.81Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
23.81Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
23.81Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
23.81Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
23.81Single8TF5Oleic acid8TF5-GPR6-Oleic acid
23.81Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
23.81Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
23.81Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
23.81Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
23.81Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
23.81Consensusa3_on_gpOrthosteric Liganda3a_on_gp
23.81Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
23.81Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
23.81Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
23.81Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
23.81Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
23.81Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
23.68Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
23.53Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
23.53Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
23.33Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
23.33Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
23.33Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
23.33Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
23.33Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
23.33Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
23.33Consensusglp_onOrthosteric Ligandglp1_on glp2_on
23.33Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
23.33Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
23.08Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
23.08Single7XNACYN1548067XNA-SST2-CYN154806
23.08Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
23.08Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
23.08Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
22.86Consensuspth_onOrthosteric Ligandpth1_on pth2_on
22.73Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
22.73Single5V56TC1145V56-SMO-TC114
22.73Single5XR8AM8415XR8-CB1-AM841
22.73Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
22.73Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
22.73Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
22.73Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
22.73Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
22.73Single7F1TMIP-1a7F1T-CCR5-MIP-1a
22.73Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
22.73Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
22.73Single7PX4PSB-21137PX4-A2A-PSB-2113
22.73Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
22.73Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
22.73Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
22.73Single7TUYGSK682753A7TUY-GPR183-GSK682753A
22.73Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
22.73Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
22.73Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
22.73Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
22.73Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
22.73Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
22.73Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
22.73Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
22.73Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
22.73Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
22.73Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
22.73Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
22.73Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
22.73Single8ZWFJR14a8ZWF-C3aB-JR14a
22.73Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
22.73Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
22.73Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
22.73Consensusa2_onOrthosteric Liganda2b_on
22.73Consensusa2_on_gpOrthosteric Liganda2b_on_gp
22.73Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
22.73Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
22.73Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
22.73Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
22.73Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
22.73Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
22.73Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
22.73Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
22.73Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
22.58Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
22.58Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
22.58Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
22.58Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
22.58Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
22.58Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
22.58Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
22.58Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
22.58Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
22.58Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
22.22Single6PT2KGCHM076PT2-δ-KGCHM07
22.22Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
22.22Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
22.22Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
22.22Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
22.22Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
22.22Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
22.22Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
22.22Single8K5BNiacin8K5B-HCA2-Niacin
22.22Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
22.22Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
22.22Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
22.22Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
22.22Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
22.22Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
22.22Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
22.22Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
21.88Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
21.88Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
21.88Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
21.88Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
21.88Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
21.74Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
21.74Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
21.74Single6MXTSalmeterol6MXT-β2-Salmeterol
21.74Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
21.74Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
21.74Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
21.74Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
21.74Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
21.74Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
21.74Single7YITNalfurafine7YIT-κ-Nalfurafine
21.74Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
21.74Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
21.74Single8JJLOlodaterol8JJL-β2-Olodaterol
21.74Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
21.74Single8JWY2-1188JWY-A2A-2-118
21.74Single8JWZAB9288JWZ-A2A-AB928-Na
21.74Single9BJKNAM9BJK-μ-Naloxone-NAM
21.74Single9DGIZ85267113509DGI-CB1-Z8526711350
21.74Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
21.74Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
21.74Consensusalpha1_offOrthosteric Ligandalpha1a_off
21.74Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
21.74Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
21.74Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
21.74Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
21.74Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
21.74Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
21.62Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
21.43Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
21.43Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
21.43Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
21.43Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
21.43Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
21.43Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
21.43Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
21.43Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
21.43Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
21.43Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
21.43Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
21.21Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
21.21Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
21.21Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
21.05Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
21.05Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
21.05Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
21.05Single5U09Taranabant5U09-CB1-Taranabant
21.05Single5WS3EMPA5WS3-OX2-EMPA
21.05Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
21.05Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
21.05Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
21.05Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
21.05Single7F8ULintitript7F8U-CCKA-Lintitript
21.05Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
21.05Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
21.05Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
21.05Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
21.05Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.05Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
21.05Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
21.05Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
21.05Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
21.05Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
21.05Single8Y0HVUF114188Y0H-CXCR3-VUF11418
21.05Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
21.05Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
21.05Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
21.05Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
21.05Single9H2XA1IR19H2X-A2A-A1IR1-Na
21.05Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
21.05Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
21.05Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
21.05Consensusorexin_offOrthosteric Ligandox2_off ox1_off
21.05Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
21.05Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
21.05Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
21.05Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
21.05Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
20.83Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
20.83Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
20.83Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
20.83Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
20.83Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
20.83Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
20.83Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
20.83Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
20.83Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
20.83Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
20.83Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
20.83Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
20.83Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
20.83Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
20.83Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
20.83Consensusendothelin_offOrthosteric Ligandetb_off
20.83Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
20.83Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
20.69Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
20.69Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
20.69Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
20.69Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
20.69Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
20.59Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
20.59Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.59Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
20.00Single2YDOAdenosine2YDO-A2A-Adenosine
20.00Single4ZJCSB-6740424ZJC-OX1-SB-674042
20.00Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
20.00Single5IU7Q274563465IU7-A2A-Q27456346-Na
20.00Single5IUBQ274563445IUB-A2A-Q27456344-Na
20.00Single5JTBZM-2413855JTB-A2A-ZM-241385
20.00Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
20.00Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
20.00Single5UVIZM-2413855UVI-A2A-ZM-241385
20.00Single6AQFZM-2413856AQF-A2A-ZM-241385
20.00Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
20.00Single6IQLL7458706IQL-D4-L745870
20.00Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
20.00Single6TPGEMPA6TPG-OX2-EMPA
20.00Single6V9SGTPL114036V9S-OX1-GTPL11403
20.00Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
20.00Single6ZG9GSK10347026ZG9-M1-GSK1034702
20.00Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
20.00Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
20.00Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
20.00Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
20.00Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
20.00Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
20.00Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
20.00Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
20.00Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
20.00Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
20.00Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
20.00Single8K2WAMG4878K2W-CXCR3-AMG487
20.00Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
20.00Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
20.00Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
20.00Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
20.00Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
20.00Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
20.00Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
20.00Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
20.00Consensusa2_offOrthosteric Liganda2a_off
20.00Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
20.00Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
20.00Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
20.00Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
20.00Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
20.00Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
20.00Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
20.00Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
20.00Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
20.00Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
20.00Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
20.00Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
19.44Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
19.35Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
19.35Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
19.35Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
19.35Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
19.35Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
19.35Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
19.35Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
19.35Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
19.23Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
19.23Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
19.23Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
19.23Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
19.23Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
19.23Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
19.23Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
19.23Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
19.23Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
19.23Single8KIGSHU91198KIG-MC3-SHU9119-Ca
19.23Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
19.23Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
19.23Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
19.23Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
19.23Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
19.23Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
19.23Consensussomatostatin_offOrthosteric Ligandsst2_off
19.05Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
19.05Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
19.05Single4YAYZD-71554YAY-AT1-ZD-7155
19.05Single5DHGC-355DHG-NOP-C-35
19.05Single5DHHSB-6121115DHH-NOP-SB-612111
19.05Single5IU8Q274563475IU8-A2A-Q27456347-Na
19.05Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
19.05Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
19.05Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
19.05Single5UENDU1725UEN-A1-DU172
19.05Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
19.05Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
19.05Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
19.05Single7F83PF-051904577F83-Ghrelin-PF-05190457
19.05Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
19.05Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
19.05Single7PYRPSB-21157PYR-A2A-PSB-2115
19.05Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
19.05Single7UL4Alvimopan7UL4-μ-Alvimopan
19.05Single7YXAONO-54306087YXA-S1P5-ONO-5430608
19.05Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
19.05Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
19.05Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
19.05Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
19.05Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
19.05Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
19.05Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
19.05Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
19.05Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
18.75Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
18.75Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
18.75Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
18.75Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
18.75Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
18.75Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
18.75Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
18.75Single8PWNTheophylline8PWN-A2A-Theophylline
18.75Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
18.75Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
18.75Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
18.75Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
18.52Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
18.52Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
18.52Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
18.52Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
18.52Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
18.52Single8IEBA1LYA8IEB-GPR156-A1LYA
18.52Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
18.52Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
18.42Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
18.18Single4JKVTaladegib4JKV-SMO-Taladegib
18.18Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
18.18Single5WQCEMPA5WQC-OX2-EMPA
18.18Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
18.18Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
18.18Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
18.18Single7C61Ergotamine7C61-5-HT1B-Ergotamine
18.18Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
18.18Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
18.18Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
18.18Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
18.18Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
18.18Single7W41PD1762527W41-BB2-PD176252
18.18Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
18.18Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
18.18Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
18.18Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
18.18Single8JXSPF-61428JXS-D1-PF-6142
18.18Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
18.18Single8QOTNanobody-E8QOT-μ-Nanobody-E
18.18Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
18.18Single9B9ZA1AKO9B9Z-CB1-A1AKO
18.18Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
18.18Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
18.18Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
18.18Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
18.18Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
18.18Consensusadenosine_offOrthosteric Liganda1_off a2_off
18.18Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
18.18Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
18.18Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
18.18Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
18.18Consensusblt_offOrthosteric Ligandblt1_off
18.18Consensusbombesin_offOrthosteric Ligandbb2_off
18.18Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
18.18Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
18.18Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
18.18Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
18.18Consensusep_offOrthosteric Ligandep4_off
18.18Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
18.18Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
18.18Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
17.86Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
17.86Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
17.86Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
17.86Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
17.86Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
17.86Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
17.65Single3RFMCaffeine3RFM-A2A-Caffeine
17.65Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
17.65Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
17.65Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
17.65Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
17.65Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
17.39Single2YDVNECA2YDV-A2A-NECA
17.39Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
17.39Single4DJHJDTic4DJH-κ-JDTic
17.39Single4UHRCGS216804UHR-A2A-CGS21680
17.39Single5G53NECA5G53-A2A-NECA-Gs
17.39Single5TZRMK86665TZR-FFA1-MK8666
17.39Single5V57TC1145V57-SMO-TC114
17.39Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
17.39Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
17.39Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
17.39Single6TQ7SB-3348676TQ7-OX1-SB-334867
17.39Single7B6WCyclazosin7B6W-α1b-Cyclazosin
17.39Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
17.39Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
17.39Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
17.39Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
17.39Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
17.39Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
17.39Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.39Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
17.39Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
17.39Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
17.39Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
17.39Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
17.39Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
17.39Single8XVLZibotentan8XVL-ETA-Zibotentan
17.39Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
17.39Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
17.39Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.39Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
17.39Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
17.39Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
17.39Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
17.39Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
17.24Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
17.24Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
17.24Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
17.24Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
17.24Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
17.24Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
17.24Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
17.24Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
17.24Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
17.24Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
17.24Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
17.24Consensusvasop-oxy_onOrthosteric Ligandv2_on
17.24Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
17.14Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
17.14Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
17.14Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
17.14Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
17.14Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
17.14Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
16.67Single4N4WSANT-14N4W-SMO-SANT-1
16.67Single4PY02MeSATP4PY0-P2Y12-2MeSATP
16.67Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
16.67Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
16.67Single5X33BIIL2605X33-BLT1-BIIL260
16.67Single6A93Risperidone6A93-5-HT2A-Risperidone
16.67Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
16.67Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
16.67Single6ZG4HTL00099366ZG4-M1-HTL0009936
16.67Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
16.67Single7DFPSpiperone7DFP-D2-Spiperone
16.67Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
16.67Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
16.67Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
16.67Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
16.67Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
16.67Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
16.67Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
16.67Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
16.67Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
16.67Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
16.67Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
16.67Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
16.67Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
16.67Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
16.67Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
16.67Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
16.67Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
16.67Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
16.67Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
16.67Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
16.67Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
16.67Single8XYIVUF106618XYI-CXCR3-VUF10661
16.67Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
16.67Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
16.67Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
16.67Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
16.67Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
16.67Consensuscalcitonin_onOrthosteric Ligandctlike_on
16.67Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
16.67Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
16.67Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
16.67Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
16.67Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
16.67Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
16.67Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
16.22Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
16.22Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
16.13Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
16.13Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
16.13Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
16.13Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
16.13Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
16.13Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
16.13Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
16.13Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
16.00Single5X93K-87945X93-ETB-K-8794
16.00Single6IBLArformoterol6IBL-β1-Arformoterol
16.00Single6K1QIRL25006K1Q-ETB-IRL2500
16.00Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
16.00Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
16.00Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
16.00Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
16.00Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
16.00Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
16.00Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
16.00Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
16.00Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
16.00Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
16.00Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
16.00Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
16.00Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
16.00Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
16.00Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
16.00Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
16.00Consensuschemerin_onOrthosteric Ligandcml1_on
16.00Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
15.79Single4O9RCyclopamine4O9R-SMO-Cyclopamine
15.79Single5L7IVismodegib5L7I-SMO-Vismodegib
15.79Single6LI0C176LI0-GPR52-C17
15.79Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
15.79Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
15.79Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.79Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
15.79Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
15.79Single9B9Y7DY9B9Y-CB1-7DY
15.79Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
15.79Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
15.79Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
15.79Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
15.79Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
15.62Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
15.62Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
15.62Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
15.62Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
15.62Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
15.38Single3NY9ICI118-5513NY9-β2-ICI118-551
15.38Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
15.38Single6PT3DPI-2876PT3-δ-DPI-287
15.38Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
15.38Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
15.38Single7SK9CCX6627SK9-ACKR3-CCX662
15.38Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
15.38Single8X5YAstemizole8X5Y-H1-Astemizole
15.38Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
15.38Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
15.38Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
15.38Consensuskisspeptin_onOrthosteric Ligandkiss1_on
15.15Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
15.15Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
15.15Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
15.00Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
15.00Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
15.00Single4QINSAG1.54QIN-SMO-SAG1.5
15.00Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
15.00Single6AKXA4R6AKX-CCR5-A4R
15.00Single6B73MP11046B73-κ-MP1104
15.00Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
15.00Single6DS0Ly2660976DS0-5-HT2B-Ly266097
15.00Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
15.00Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
15.00Single6TODEMPA6TOD-OX1-EMPA-Na
15.00Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
15.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
15.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
15.00Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
15.00Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
15.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
15.00Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
15.00Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
15.00Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.00Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
15.00Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
15.00Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
15.00Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
15.00Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
15.00Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
15.00Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
15.00Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
15.00Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
15.00Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
15.00Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
15.00Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
14.81Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
14.81Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
14.81Single7QA8Peptide7QA8-STE2-Peptide
14.81Single7QA8Peptide7QA8-STE2-Peptide
14.81Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
14.81Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.81Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
14.81Single8IEBA1LYA8IEB-GPR156-A1LYA
14.81Single8IEIA1LYA8IEI-GPR156-A1LYA
14.81Single8IEIA1LYA8IEI-GPR156-A1LYA
14.81Single8IEPA1LYA8IEP-GPR156-A1LYA
14.81Single8IEPA1LYA8IEP-GPR156-A1LYA
14.81Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
14.81Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
14.81Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
14.81Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
14.81Single9M4TSilodosin9M4T-Alpha1A-Silodosin
14.71Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
14.71Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
14.29Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
14.29Single4MBSMaraviroc4MBS-CCR5-Maraviroc
14.29Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
14.29Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
14.29Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
14.29Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
14.29Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
14.29Single7T32ZM-2413857T32-A2A-ZM-241385
14.29Single7VV6C48/807VV6-MRGPRX2-C48/80
14.29Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
14.29Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.29Single8RLNLUF58348RLN-A2A-LUF5834
14.29Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
14.29Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
14.29Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
14.29Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
14.29Single9BA0A1AKN9BA0-CB1-A1AKN
14.29Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
14.29Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
14.29Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
14.29Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
13.89Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
13.79Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
13.79Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
13.79Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
13.79Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
13.64Single2Y02Carmoterol2Y02-β1-Carmoterol
13.64Single4EJ4Naltrindole4EJ4-δ-Naltrindole
13.64Single6DRXLisuride6DRX-5-HT2B-Lisuride
13.64Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
13.64Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
13.64Single6GPSMK08126GPS-CCR2-MK0812
13.64Single6PS1Timolol6PS1-β2-Timolol
13.64Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
13.64Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
13.64Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
13.64Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
13.64Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
13.64Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
13.64Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
13.64Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
13.64Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
13.64Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.64Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
13.64Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
13.64Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
13.64Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
13.64Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
13.64Single8T1WCVN4248T1W-GPR6-CVN424
13.64Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
13.64Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
13.64Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.64Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.64Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.64Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.64Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.64Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
13.64Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
13.64Single9CHXS-Carazolol9CHX-β2-S-Carazolol
13.64Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
13.64Single9IYAONO-97105319IYA-GPR55-ONO-9710531
13.64Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
13.64Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
13.64Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
13.64Consensusblt_onOrthosteric Ligandblt1_on
13.64Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
13.64Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
13.64Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
13.64Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
13.64Consensusleukotriene_onOrthosteric Ligandblt_on
13.64Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
13.51Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
13.51Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
13.51Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
13.33Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
13.33Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
13.33Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
13.33Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
13.33Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
13.33Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
13.33Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
13.04Single4NTJAZD12834NTJ-P2Y12-AZD1283
13.04Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
13.04Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
13.04Single5XPRBosentan5XPR-ETB-Bosentan
13.04Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
13.04Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
13.04Single6GPXMK08126GPX-CCR2-MK0812
13.04Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
13.04Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
13.04Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
13.04Single7SINNPS-21437SIN-CaS-NPS-2143
13.04Single7SINNPS-21437SIN-CaS-NPS-2143
13.04Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
13.04Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
13.04Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
13.04Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.04Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
13.04Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
13.04Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
13.04Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.04Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
13.04Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
13.04Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
13.04Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
13.04Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
13.04Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.04Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.04Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
13.04Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
13.04Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
13.04Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
13.04Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
13.04Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
13.04Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
13.04Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
13.04Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
13.04Single9HAPTolvaptan9HAP-V2-Tolvaptan
13.04Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
13.04Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
13.04Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
13.04Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
12.90Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
12.50Single3P0GBI1671073P0G-β2-BI167107
12.50Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
12.50Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
12.50Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
12.50Single5MZPCaffeine5MZP-A2A-Caffeine-Na
12.50Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
12.50Single6H7JIsoprenaline6H7J-β1-Isoprenaline
12.50Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
12.50Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
12.50Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
12.50Single6WGTLSD6WGT-5-HT2A-LSD
12.50Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
12.50Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
12.50Single7P2L4YI7P2L-mGlu5-4YI
12.50Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
12.50Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
12.50Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
12.50Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
12.50Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
12.50Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
12.50Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
12.50Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
12.50Single9BJKNaloxone9BJK-μ-Naloxone-NAM
12.50Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
12.50Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
12.50Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
12.50Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
12.50Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
12.50Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
12.50Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
12.50Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
12.50Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
12.50Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
12.50Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
12.12Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
12.12Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
12.12Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
12.12Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
12.12Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
12.00Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
12.00Single4AMIBucindolol4AMI-β1-Bucindolol
12.00Single4LDEBI1671074LDE-β2-BI167107
12.00Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
12.00Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
12.00Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
12.00Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
12.00Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
12.00Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.00Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.00Single8JJ8Formoterol8JJ8-β2-Formoterol
12.00Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.00Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
12.00Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
12.00Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.00Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
12.00Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
12.00Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
12.00Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
12.00Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
11.76Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
11.76Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
11.76Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
11.76Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
11.76Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
11.76Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
11.76Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
11.76Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
11.76Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
11.76Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
11.54Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
11.54Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
11.54Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
11.54Single6H7LDobutamine6H7L-β1-Dobutamine
11.54Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
11.54Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
11.54Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
11.54Single7UM4AS26747237UM4-5-HT5A-AS2674723
11.54Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
11.54Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
11.54Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
11.54Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
11.54Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
11.54Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
11.43Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
11.11Single6TQ9SB-4081246TQ9-OX1-SB-408124
11.11Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
11.11Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
11.11Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
11.11Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
11.11Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
11.11Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
11.11Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
11.11Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single9JF4PD1683689JF4-BB1-PD168368
11.11Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
11.11Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
10.53Single3UZAGTPL92363UZA-A2A-GTPL9236
10.53Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
10.53Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
10.53Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
10.53Single6ME5Agomelatine6ME5-MT1-Agomelatine
10.53Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
10.53Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
10.53Single7WC5Psilocin7WC5-5-HT2A-Psilocin
10.53Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.53Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.53Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
10.53Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
10.53Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
10.53Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
10.53Single8JPSCCL78JPS-ACKR1-CCL7
10.53Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
10.53Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
10.53Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
10.53Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
10.53Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
10.53Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
10.53Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
10.53Single9LRCHistamine9LRC-H4-Histamine
10.53Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
10.53Consensus5ht2_onOrthosteric Ligand5ht2b_on
10.53Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.53Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
10.53Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
10.53Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
10.53Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
10.34Single6HLOAprepitant6HLO-NK1-Aprepitant
10.00Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
10.00Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
10.00Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
10.00Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
10.00Single6TP4ACT-4622066TP4-OX1-ACT-462206
10.00Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
10.00Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
10.00Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
10.00Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
10.00Single7SRQLSD7SRQ-5-HT2B-LSD
10.00Single7UL2SR486927UL2-NTS1-SR48692-Na
10.00Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
10.00Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
10.00Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
10.00Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
10.00Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
10.00Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
10.00Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
10.00Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
10.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
10.00Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
10.00Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
10.00Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
10.00Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
10.00Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
10.00Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
10.00Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
10.00Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
10.00Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
10.00Consensusneurotensin_offOrthosteric Ligandnts1_off
10.00Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
9.68Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
9.52Single6AKYMaraviroc6AKY-CCR5-Maraviroc
9.52Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
9.52Single6ME9Ramelteon6ME9-MT2-Ramelteon
9.52Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
9.52Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
9.52Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
9.52Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
9.52Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.52Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
9.52Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
9.52Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
9.52Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
9.52Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
9.52Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
9.52Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
9.52Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.52Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
9.52Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
9.52Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
9.52Single8IWESpermidine8IWE-TA9-Spermidine
9.52Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
9.52Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
9.52Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.52Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.52Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.52Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.52Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.52Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
9.52Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
9.52Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
9.52Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
9.52Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
9.52Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
9.52Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
9.52Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.52Consensusalpha2_offOrthosteric Ligandalpha2c_off
9.52Consensusangiotensin_offOrthosteric Ligandat1_off
9.52Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
9.52Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
9.52Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
9.52Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
9.38Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
9.38Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
9.30Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
9.09Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
9.09Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
9.09Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
9.09Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
9.09Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
9.09Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
9.09Single6KUXRS-799486KUX-α2a-RS-79948
9.09Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
9.09Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
9.09Single6PS0S-Carazolol6PS0-β2-S-Carazolol
9.09Single6PS4ICI118-5516PS4-β2-ICI118-551
9.09Single6PS5S-Propranolol6PS5-β2-S-Propranolol
9.09Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
9.09Single6TPKRetosiban6TPK-OT-Retosiban
9.09Single6TPNHTL66416TPN-OX2-HTL6641
9.09Single6VI4JDTic6VI4-κ-JDTic
9.09Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
9.09Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
9.09Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
9.09Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
9.09Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
9.09Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
9.09Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
9.09Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
9.09Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
9.09Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
9.09Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.09Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
9.09Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
9.09Single7UL3Famotidine7UL3-H2-Famotidine
9.09Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
9.09Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
9.09Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
9.09Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
9.09Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.09Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.09Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.09Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
9.09Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
9.09Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
9.09Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
9.09Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
9.09Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
9.09Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
9.09Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
9.09Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
9.09Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
9.09Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.09Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.09Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.09Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.09Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.09Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
9.09Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
9.09Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
9.09Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
9.09Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
9.09Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
9.09Single9AS5Mescaline9AS5-5-HT2A-Mescaline
9.09Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
9.09Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
9.09Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
9.09Consensusalpha1_onOrthosteric Ligandalpha1a_on
9.09Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
9.09Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
9.09Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
9.09Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
9.09Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
9.09Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
9.09Consensusvasop-oxy_offOrthosteric Ligandot_off
8.70Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
8.70Single2Y04Salbutamol2Y04-β1-Salbutamol
8.70Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
8.70Single3NY8ICI118-5513NY8-β2-ICI118-551
8.70Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
8.70Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
8.70Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
8.70Single4DAJTiotropium4DAJ-M3-Tiotropium
8.70Single4GBRS-Carazolol4GBR-β2-S-Carazolol
8.70Single4MQSIperoxo4MQS-M2-Iperoxo
8.70Single4QKX35V4QKX-β2-35V
8.70Single4U14Tiotropium4U14-M3-Tiotropium
8.70Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
8.70Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
8.70Single5DSGTiotropium5DSG-M4-Tiotropium
8.70Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
8.70Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
8.70Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
8.70Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
8.70Single6IIVDaltroban6IIV-TXA2-Daltroban
8.70Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
8.70Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
8.70Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
8.70Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.70Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
8.70Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
8.70Single7BU7BI1671077BU7-β1-BI167107
8.70Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
8.70Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
8.70Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
8.70Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
8.70Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
8.70Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
8.70Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
8.70Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
8.70Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
8.70Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
8.70Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
8.70Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
8.70Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
8.70Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.70Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.70Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.70Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.70Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.70Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.70Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.70Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.70Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.70Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.70Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
8.70Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
8.70Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
8.70Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
8.70Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
8.70Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
8.70Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
8.70Single8JJOAlprenolol8JJO-β2-Alprenolol
8.70Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
8.70Single8JXRLSD8JXR-D1-LSD
8.70Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
8.70Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
8.70Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.70Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.70Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
8.70Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
8.70Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
8.70Single8X63Mepyramine8X63-H1-Mepyramine
8.70Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
8.70Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
8.70Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
8.70Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
8.70Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
8.70Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
8.70Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
8.70Single9JEAAtropine9JEA-M1-Atropine
8.70Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
8.70Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
8.70Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
8.70Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
8.70Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
8.70Consensus5ht5_onOrthosteric Ligand5ht5a_on
8.70Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
8.70Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
8.70Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
8.70Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
8.70Consensusalpha2_onOrthosteric Ligandalpha2b_on
8.70Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
8.70Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
8.70Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
8.70Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
8.70Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
8.70Consensusdopamine_offOrthosteric Ligandd2_off d3_off
8.70Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
8.70Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
8.70Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
8.70Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
8.70Consensushistamine_offOrthosteric Ligandh1_off
8.70Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
8.70Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
8.70Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
8.33Single2RH1S-Carazolol2RH1-β2-S-Carazolol
8.33Single2Y00Dobutamine2Y00-β1-Dobutamine
8.33Single2Y03Isoprenaline2Y03-β1-Isoprenaline
8.33Single2YCWS-Carazolol2YCW-β1-S-Carazolol
8.33Single5D6LS-Carazolol5D6L-β2-S-Carazolol
8.33Single5JQHS-Carazolol5JQH-β2-S-Carazolol
8.33Single5TVNLSD5TVN-5-HT2B-LSD
8.33Single5WIUNemonapride5WIU-D4-Nemonapride
8.33Single5WIVNemonapride5WIV-D4-Nemonapride-Na
8.33Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
8.33Single6E67BI1671076E67-β2-BI167107-Gs(CT)
8.33Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
8.33Single6LUQHaloperidol6LUQ-D2-Haloperidol
8.33Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
8.33Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
8.33Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
8.33Single6PS6Timolol6PS6-β2-Timolol
8.33Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
8.33Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
8.33Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
8.33Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
8.33Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
8.33Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
8.33Single7WC6LSD7WC6-5-HT2A-LSD
8.33Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
8.33Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
8.33Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
8.33Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.33Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.33Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
8.33Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
8.33Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
8.33Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
8.33Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
8.33Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
8.33Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
8.33Single9HC04YI9HC0-mGlu5-4YI
8.33Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
8.33Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
8.33Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
8.33Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
8.33Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
8.33Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
8.33Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
8.33Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
8.33Consensusamine_offonOrthosteric Ligandamine_off amine_on
8.33Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
8.33Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
8.33Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
8.33Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
8.33Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
8.33Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
8.33Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
8.33Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
8.33Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
8.33Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.33Consensustrace-amine_onOrthosteric Ligandta1_on
8.00Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
8.00Single4U15Tiotropium4U15-M3-Tiotropium
8.00Single5D5AS-Carazolol5D5A-β2-S-Carazolol
8.00Single5D5BS-Carazolol5D5B-β2-S-Carazolol
8.00Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
8.00Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
8.00Single6E59L-7607356E59-NK1-L-760735
8.00Single6J20Aprepitant6J20-NK1-Aprepitant
8.00Single6J21Aprepitant6J21-NK1-Aprepitant
8.00Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
8.00Single6OL9Tiotropium6OL9-M5-Tiotropium
8.00Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
8.00Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
8.00Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
8.00Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
8.00Single8EA0Iperoxo8EA0-M3-Iperoxo
8.00Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
8.00Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
8.00Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
8.00Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
8.00Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
8.00Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
8.00Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
8.00Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
8.00Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
8.00Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
8.00Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
8.00Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
8.00Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
8.00Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
8.00Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
8.00Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.00Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
7.69Single3D4STimolol3D4S-β2-Timolol
7.69Single5CXVTiotropium5CXV-M1-Tiotropium
7.69Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
7.69Single6CM4Risperidone6CM4-D2-Risperidone
7.69Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
7.69Single6IIURamatroban6IIU-TXA2-Ramatroban
7.69Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
7.69Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
7.69Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
7.69Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
7.69Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
7.69Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.69Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
7.69Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
7.69Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
7.69Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
7.41Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
7.41Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
7.41Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Single8XVJMacitentan8XVJ-ETA-Macitentan
7.41Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
7.41Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.41Single9JH5C16:0 Ceramide9JH5-CysLT2-C16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
7.41Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
7.41Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
7.41Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
7.14Single6D35Cholesterol6D35-SMO-Cholesterol
7.14Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
7.14Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
7.14Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
7.14Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
7.14Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042
7.14Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
7.14Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
7.14Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-BHFF
7.14Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
7.14Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626
7.14Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
7.14Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
7.14Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
7.14Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
7.14Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
7.14Single7DTTCa7DTT-CaS-Ca-Ca
7.14Single7DTTCa7DTT-CaS-Ca-Ca
7.14Single7DTUTryptophan7DTU-CaS-Tryptophan
7.14Single7DTUTryptophan7DTU-CaS-Tryptophan
7.14Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
7.14Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
7.14Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
7.14Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
7.14Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
7.14Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
7.14Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
7.14Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
7.14Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
7.14Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
7.14Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
7.14Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
7.14Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
7.14Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
7.14Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
7.14Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
7.14Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
7.14Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
7.14Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
7.14Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
7.14Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
7.14Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
7.14Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
7.14Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
7.14Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
7.14Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
7.14Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
7.14Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
7.14Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
7.14Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
7.14Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
7.14Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
7.14Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
7.14Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
7.14Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
7.14Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
7.14Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
7.14Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
7.14Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
7.14Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
7.14Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
7.14Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
7.14Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
7.14Single7T9NM22 Fab7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
7.14Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
7.14Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
7.14Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
7.14Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
7.14Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
7.14Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
7.14Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
7.14Single7XW7K1-707XW7-TSH-K1-70
7.14Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
7.14Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
7.14Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
7.14Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
7.14Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
7.14Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
7.14Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
7.14Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
7.14Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
7.14Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
7.14Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
7.14Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
7.14Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
7.14Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
7.14Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
7.14Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
7.14Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
7.14Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
7.14Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
7.14Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
7.14Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
7.14Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
7.14Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
7.14Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
7.14Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
7.14Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
7.14Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
7.14Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
7.14Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
7.14Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
7.14Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
7.14Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
7.14Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
7.14Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
7.14Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
7.14Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
7.14Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
7.14Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
7.14Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
7.14Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
7.14Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
7.14Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
7.14Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
7.14Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
7.14Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
7.14Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
7.14Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
7.14Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
7.14Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
7.14Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
7.14Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
7.14Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
7.14Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
7.14Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
7.14Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single8WVXNorrin8WVX-LGR4-Norrin
7.14Single8WVYNorrin8WVY-LGR4-Norrin
7.14Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
7.14Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
7.14Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
7.14Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
7.14Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
7.14Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
7.14Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
7.14Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
7.14Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
7.14Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
7.14Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
7.14Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
7.14Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
7.14Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
7.14Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
7.14Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
7.14Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
7.14Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
7.14Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
7.14Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
7.14Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
7.14Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
7.14Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
7.14Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
7.14Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
7.14Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
7.14Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
7.14Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
7.14Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
7.14Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
7.14Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
7.14Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
7.14Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
7.14Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
7.14Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
7.14Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
7.14Single9KHHNorrin9KHH-LGR4-Norrin
7.14Single9S37NB219S37-LGR4-NB21
7.14Single9UTBSucralose9UTB-TAS1R2; TAS1R3-Sucralose
6.67Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
6.67Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
6.67Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
6.67Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
6.67Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
6.67Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
6.67Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
6.67Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
6.67Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
6.67Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
6.67Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
6.67Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
6.67Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
6.67Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
6.67Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
6.67Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
6.25Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
6.25Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
6.25Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
6.25Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
5.88Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
5.88Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
5.88Single7UTZTR14027UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
5.88Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
5.88Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
5.88Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
5.88Single8JGBConorfamide-Tx28JGB-MRGPRX1-Conorfamide-Tx2-Gi1/β1/γ2
5.88Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
5.56Single5L7DCholesterol5L7D-SMO-Cholesterol
5.56Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
5.56Single7WC4Serotonin7WC4-5-HT2A-Serotonin
5.56Single8HS2Fab0468HS2-GPR20-Fab046
5.56Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
5.26Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
5.26Single7Y14Beta-Alanine7Y14-MRGPRD-β-Alanine
5.26Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.26Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
5.26Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
5.26Single9CHUNoradrenaline9CHU-β2-Noradrenaline
5.26Single9IVMLSN33188399IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
5.00Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
5.00Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
5.00Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
5.00Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
5.00Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
5.00Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
5.00Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
5.00Single7Y12Beta-Alanine7Y12-MRGPRD-β-Alanine-Gi1/β1/γ2
5.00Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.00Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
5.00Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
5.00Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
5.00Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
4.76Single3PBLEticlopride3PBL-D3-Eticlopride
4.76Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
4.76Single6HLLCP999946HLL-NK1-CP99994
4.76Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
4.76Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
4.76Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
4.76Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
4.76Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
4.76Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.76Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
4.76Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
4.76Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
4.76Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
4.76Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
4.76Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
4.76Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
4.76Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
4.55Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
4.55Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
4.55Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
4.55Single6ME2Ramelteon6ME2-MT1-Ramelteon
4.55Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
4.55Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
4.55Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
4.55Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.55Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
4.55Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
4.55Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
4.55Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
4.55Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
4.55Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
4.55Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.55Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
4.55Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
4.55Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
4.55Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
4.55Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
4.55Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
4.55Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
4.55Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
4.55Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
4.55Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
4.55Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
4.55Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
4.55Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
4.55Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
4.35Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
4.35Single3RZECidoxepin3RZE-H1-Cidoxepin
4.35Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
4.35Single6FFIMMPEP6FFI-mGlu5-MMPEP
4.35Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
4.35Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
4.35Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
4.35Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
4.35Single7VODCariprazine7VOD-5-HT2A-Cariprazine
4.35Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
4.35Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
4.35Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
4.35Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
4.35Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
4.35Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
4.35Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
4.35Single8JD6VU03647708JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
4.35Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
4.35Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.35Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
4.35Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
4.35Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
4.35Single9ARXSerotonin9ARX-5-HT2A-Serotonin
4.35Single9AS3LSD9AS3-5-HT2A-LSD
4.35Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
4.35Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
4.35Consensusopsins_offOrthosteric Ligandrhodopsin_off
4.35Consensussensory_offOrthosteric Ligandopsins_off
4.17Single2Y01Dobutamine2Y01-β1-Dobutamine
4.17Single6FFHFenobam6FFH-mGlu5-Fenobam
4.17Single6H7MSalbutamol6H7M-β1-Salbutamol
4.17Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
4.17Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
4.17Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
4.17Single7WC7Lisuride7WC7-5-HT2A-Lisuride
4.17Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
4.17Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
4.17Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
4.17Single8X64Desloratadine8X64-H1-Desloratadine
4.17Single9AS1DMT9AS1-5-HT2A-DMT
4.17Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
4.17Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
4.17Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
4.17Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
4.17Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
4.00Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
4.00Single5CGCHTL142425CGC-mGlu5-HTL14242
4.00Single6HLPNetupitant6HLP-NK1-Netupitant
4.00Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
4.00Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
4.00Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
4.00Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
4.00Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
4.00Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
4.00Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
3.85Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
3.85Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
3.85Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
3.85Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
3.85Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
3.85Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
3.85Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
3.85Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
3.85Single9AS9RS130-1809AS9-5-HT2A-RS130-180
3.85Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
3.85Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.85Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
3.85Consensustachykinin_offOrthosteric Ligandnk1_off
3.70Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
3.70Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
3.70Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
3.57Single5CGDHTL142425CGD-mGlu5-HTL14242
3.57Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
3.45Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
3.33Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
3.33Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
3.33Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
3.12Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
3.12Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
3.03Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.78Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
8IBU 8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
Net Summary
Imin 2.79
Number of Linked Nodes 837
Number of Links 979
Number of Hubs 146
Number of Links mediated by Hubs 549
Number of Communities 34
Number of Nodes involved in Communities 233
Number of Links involved in Communities 309
Path Summary
Number Of Nodes in MetaPath 167
Number Of Links MetaPath 166
Number of Shortest Paths 1448677
Length Of Smallest Path 3
Average Path Length 37.3339
Length of Longest Path 79
Minimum Path Strength 1.21
Average Path Strength 6.07233
Maximum Path Strength 19.33
Minimum Path Correlation 0.7
Average Path Correlation 0.984452
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 1.78571
Average % Of Corr. Nodes 42.953
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 45.3305
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
peptide_on_gpcck_on_gp
angiotensin_on_gp
apelin_on_gp
bombesin_on_gp
bradykinin_on_gp
compl-peptide_on_gp
endothelin_on_gp
formylpeptide_on_gp
galanin_on_gp
ghrelin_on_gp
kisspeptin_on_gp
melanocortin_on_gp
motilin_on_gp
neuromedin-u_on_gp
npy_on_gp
neurotensin_on_gp
opioid_on_gp
orexin_on_gp
relaxin_on_gp
somatostatin_on_gp
tachykinin_on_gp
trh_on_gp
vasop-oxy_on_gp



You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

Download motilin_on_gp.zip



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