Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.11 0.361605602
2G.H1.01 1.60313509
3G.S2.04 0.953723406
4G.S2.06 2.2252509
5G.S3.03 3.30147507
6G.S3.07 1.48738409
7G.H2.07 3.19369409
8G.h2s4.01 3.66321409
9G.s4h3.04 2.79912508
10G.H3.01 2.34461509
11G.H3.09 2.75589509
12G.H3.17 3.72123505
13G.H3.18 2.79279409
14G.S5.05 1.68563509
15G.S5.07 1.93699509
16G.HG.14 1.40756405
17G.hgh4.05 3.12101607
18G.hgh4.08 1.00916403
19G.H4.10 3.76988406
20G.H4.12 2.52721405
21G.H4.15 2.69381408
22G.h4s6.02 1.66858408
23G.h4s6.12 1.48277404
24G.S6.02 2.65462607
25G.S6.05 2.66831504
26G.H5.03 1.93971408
27b.1x4 0.782595408
28b.1x11 0.98854408
29b.lhb1x3 0.89688502
30b.l1x3 5.1903409
31b.b2x1 4.24088428
32b.b2x5 3.23746607
33b.l3x2 2.82183409
34b.b4x6 6.00026409
35b.b5x2 2.86054407
36b.b5x3 3.72503409
37b.b5x5 2.61619405
38b.b5x7 2.96577407
39b.l5x5 3.81219609
40b.b6x5 1.98144606
41b.b7x1 2.94693404
42b.l7x4 1.61093409
43b.b8x4 2.91845406
44b.l8x5 1.32177403
45b.b9x3 1.74383406
46b.l9x6 2.59144608
47b.b10x5 2.30737509
48b.l11x2 3.83778439
49b.b12x6 5.06022408
50b.b13x7 3.88081547
51b.l13x3 4.34308409
52b.b15x1 3.60405449
53b.l15x2 2.7266409
54b.b16x6 4.02926648
55b.l17x3 4.8345509
56b.l17x6 3.5339409
57b.l18x1 2.72115706
58b.l18x3 3.21168405
59b.b19x2 3.94987456
60b.l19x2 3.25848409
61b.b20x4 5.73343408
62b.b20x7 1.79089409
63b.l20x2 3.00811409
64b.b21x1 3.16595507
65b.b21x5 2.55689404
66b.b21x7 2.86434505
67b.b22x5 2.87819407
68b.l22x5 2.8733509
69b.b23x6 3.32309607
70b.l24x2 2.09518406
71b.l25x3 4.19006569
72b.l25x6 6.1401408
73b.l27x1 6.3008529
74b.l27x2 3.91344469
75b.b28x6 4.43688409
76g.l1x4 2.04002408
77g.ctx3 3.29139409
78g.ctx6 1.59693406
79NT 4.39046413
801x31 1.79782401
811x39 4.23726407
821x50 5.75703409
831x60 2.5901506
842x40 3.39829409
852x41 2.32699405
862x42 4.32817608
872x50 4.78461509
88E1x50 6.05592618
89E1x52 5.36459506
903x37 3.75857407
913x49 4.01639409
923x50 2.99992709
933x51 4.94831678
943x56 2.75781476
954x41 1.35045407
96E2 9.612231913
975x39 3.86024418
985x58 4.92559509
996x30 2.02092408
1006x48 6.785508
1016x51 4.97779417
1026x52 5.98116407
1036x60 2.11387405
104E3 3.094711213
1057x42 4.54264407
1067x49 4.3238409
1077x53 4.61187409
1088x50 3.83913409
109Lig 7.482442210
110E1 0.685113410
111H.HA.16 0.22513500
112H.hahb.06 0.279848500
113H.HB.02 0.309212400
114H.HB.10 0.248342400
115H.hchd.01 0.272446400
116H.HD.07 0.320174500
117H.hehf.04 0.351277400
118H.HF.03 0.425027400
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
13x50 5x58 97.66563.63821YesYes099
25x58 5x61 98.98872.82361YesNo099
33x54 5x61 1005.15652NoNo099
43x54 G.H5.20 98.95761.84963NoNo099
5G.H5.20 G.H5.26 98.83651.74983NoNo095
6G.H5.21 G.H5.26 98.58971.60626NoNo055
7G.H5.21 G.h4s6.12 98.46861.03694NoYes054
8G.S6.02 G.h4s6.12 97.74192.60019YesYes074
9G.H5.10 G.S6.02 96.65193.65196NoYes067
10G.H5.10 G.S5.03 96.53082.73159NoNo068
11G.S5.03 G.S5.05 96.28861.84621NoYes089
12G.S5.05 G.s6h5.01 77.02782.35794YesNo099
13G.S5.07 G.s6h5.01 74.96883.01628YesNo099
14G.S5.07 G.s5hg.01 73.99991.84396YesNo099
15G.HG.03 G.s5hg.01 72.06211.90916NoNo069
16G.HG.03 G.s4h3.02 71.81992.79232NoNo069
17G.HG.07 G.s4h3.02 71.69881.67465NoNo099
18G.HG.07 G.s4h3.04 71.33553.63751NoYes098
19G.HG.04 G.s4h3.04 67.09652.1578NoYes098
20G.HG.04 G.s4h3.01 66.85433.4813NoNo097
21G.S5.06 G.s4h3.01 66.61213.02482NoNo087
22G.S5.06 G.S6.05 66.4913.32162NoYes084
23G.H4.12 G.S6.05 64.55312.58544YesYes054
24G.H4.12 G.S6.03 63.58425.10359YesNo055
25G.S5.04 G.S6.03 63.46311.81032NoNo095
26G.H4.15 G.S5.04 63.3422.19766YesNo089
27G.H3.09 G.H4.15 62.49422.51743YesYes098
28G.H3.09 G.S4.04 61.04094.76532YesNo099
29G.H3.08 G.S4.04 60.91982.52283NoNo099
30G.H2.04 G.H3.08 60.79862.49986NoNo099
31G.H2.04 G.H2.07 60.55643.28229NoYes099
32G.H2.07 G.h2s4.01 40.93611.93324YesYes099
33G.h2s4.01 b.l5x5 40.33065.24173YesYes099
34b.l3x1 b.l5x5 38.51393.3578NoYes099
35b.b2x1 b.l3x1 38.39286.69907YesNo089
36b.b2x1 b.l27x1 38.02944.49383YesYes289
37b.l25x6 b.l27x1 37.54510.0995YesYes089
38b.l23x1 b.l25x6 36.09169.07618NoYes068
39b.l21x7 b.l23x1 35.84942.05102NoNo056
40b.l21x7 b.l23x2 35.72833.23456NoNo058
41b.b23x6 b.l23x2 35.36491.94963YesNo078
42b.b23x6 b.b24x6 33.79053.32106YesNo078
43b.b21x7 b.b24x6 33.66944.24637YesNo058
44b.b21x5 b.b21x7 28.34044.21769YesYes045
45b.b21x5 b.h2x1 27.61373.42YesNo045
46b.h2x1 b.h2x5 27.25041.67898NoNo055
47b.h2x5 b.l24x2 27.12932.53588NoYes056
48b.l22x5 b.l24x2 26.76593.76465YesYes096
49b.l22x5 g.ctx6 24.34372.00799YesYes096
50g.ctx3 g.ctx6 23.85923.16693YesYes096
51g.ctx3 g.ctx4 19.49921.97384YesNo097
52b.l26x5 g.ctx4 19.13582.66574NoNo057
53b.l26x5 g.ctx15 14.41242.43054NoNo059
54b.l4x2 g.ctx15 12.59574.5646NoNo049
55b.l2x5 b.l4x2 11.869111.4302NoNo054
562x57 7x42 10.80397.35163NoYes077
572x53 7x42 11.13853.67687NoYes087
582x53 7x46 11.86523.59183NoNo089
592x50 7x46 14.486.85096YesNo099
602x50 7x49 18.07215.2148YesYes099
612x46 7x49 57.83283.73523NoYes099
622x46 3x42 92.13473.81993NoNo098
632x45 3x42 93.99695.27156NoNo098
642x45 4x46 96.2289.02172NoNo097
652x42 4x46 96.39013.34893YesNo087
662x42 3x49 97.56065.19704YesYes089
673x49 3x50 97.51613.10685YesYes099
682x46 3x43 34.33833.46521NoNo098
693x36 Lig 48.9114.11995NoYes170
703x36 6x48 49.54365.90292NoYes078
716x44 6x48 33.031310.4317NoYes098
723x43 6x44 34.0523.6277NoNo089
736x48 7x45 35.06397.11965YesNo089
747x45 7x49 35.63664.96652NoYes099
75E2 Lig 20.19299.6219YesYes130
764x60 5x39 11.13964.16416NoYes088
776x48 6x52 14.37783.90255YesYes087
78G.H5.07 G.S5.05 18.77631.6697NoYes089
79G.H5.07 G.S4.03 18.65521.40399NoNo087
80G.S1.04 G.S4.03 18.53411.97948NoNo077
81G.S1.04 G.S3.03 18.4131.99546NoYes077
82G.S2.06 G.S3.03 16.22915.69756YesYes097
83G.S2.06 G.S3.05 15.74471.85972YesNo097
84G.S1.06 G.S3.05 13.44352.54262NoNo087
85G.H1.01 G.S1.06 13.32242.70126YesNo098
86G.H2.07 G.s3h2.03 19.37813.36686YesNo099
87G.s3h2.03 b.l9x6 18.77251.95234NoYes098
88b.b14x1 b.l9x6 12.47462.13925NoYes088
89G.H2.06 b.b14x1 12.35354.44602NoNo098
90G.H2.06 b.l17x6 12.23244.01245NoYes099
91b.l17x6 b.l19x1 11.74792.80366YesNo099
92b.l17x5 b.l19x1 11.50571.81794NoNo069
93b.l17x5 b.l19x2 11.38462.28079NoYes069
94b.b19x6 b.l19x2 10.53683.50333NoYes099
95b.b19x6 b.l17x3 10.41576.47495NoYes099
96G.H1.01 G.hfs2.02 12.35350.353696YesNo090
97G.hfs2.02 H.hdhe.04 12.23240.188261NoNo000
98H.HE.01 H.hdhe.04 11.62680.212609NoNo000
99H.HE.01 H.HF.06 11.50570.45837NoNo000
100H.HE.04 H.HF.06 11.14241.10717NoNo000
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
2x563x323.847380NoNo7721
2x607x423.457291NoYes7712
2x60Lig6.606461NoYes7010
2x63E1x505.713421NoYes5812
2x63Lig3.937221NoYes5010
E1x49E26.663961NoYes4321
E1x50E23.400151YesYes8321
3x22E27.74941NoYes4321
3x294x658.716721NoNo6612
3x29Lig5.652591NoYes6010
3x32Lig9.118951NoYes7010
3x334x573.551851NoNo6812
3x334x615.779381NoNo6711
3x33Lig5.231171NoYes6010
3x366x485.902921NoYes7812
3x36Lig4.119951NoYes7010
4x61Lig4.342471NoYes7010
4x64E29.096491NoYes5321
4x65E2x524.664270NoNo6521
E2E251.74971YesYes3311
E2E2x518.704571YesNo3411
E2Lig9.62191YesYes3010
E2x51Lig3.355241NoYes4010
E2E2x525.28281YesNo3511
E2x52Lig3.98431NoYes5010
5x35E27.641091NoYes4321
5x39E23.323061YesYes8321
5x395x433.805111YesNo8721
6x486x523.902550YesYes8722
6x487x416.568240YesNo8722
6x516x523.714951YesYes7712
6x516x556.433081YesNo7711
6x517x413.465681YesNo7712
6x51Lig6.297451YesYes7010
6x547x346.076990NoNo5521
6x55Lig9.949791NoYes7010
6x57E33.266670NoYes5321
6x58Lig7.159771NoYes4010
6x61E34.036870NoYes4321
E3E37.520051YesYes3311
E3Lig5.683051YesYes3010
7x347x383.561221NoNo5611
7x34Lig7.846881NoYes5010
7x387x423.684771NoYes6712
4x615x394.148631NoYes7812
5x36E27.919110NoYes5321
7x38Lig5.226941NoYes6010
5x43Lig3.859691NoYes7010
7x31Lig4.317911NoYes3010
E2NT5.149131YesYes3312
NTNT5.644591YesYes3322
7x30E33.186520NoYes0321
5x406x552.795420NoNo6721
E1Lig2.538961YesYes0010
7x26E31.840691NoYes0321
5x34E21.668391NoYes2321
2x67E21.643620NoYes4321
7x27E31.633241NoYes0321
5x33E31.297210NoYes2321
6x586x621.203531NoNo4012
5x31E20.6739520NoYes0321
6x63E30.5894330NoYes0321
7x25E30.5151330NoYes0321
2x68E20.2701270NoYes0321
1x277x310.2284480NoNo0321
5x27E20.1963041NoYes0321
5x28E20.1288771NoYes0321
3x29Ca50.1247611NoNo6012
2x69E10.1120510NoYes0021
1x25Lig0.09690220NoYes0010
3x20E10.08661590NoYes0021
6x65E30.04760870NoYes0321
2x70E10.002826090NoYes0021

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
95.00Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
86.96Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
86.96Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
82.61Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
79.17Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
66.67Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
66.67Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
65.38Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
65.22Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
64.00Single8ZRTET-18ZRT-ETB-ET-1
63.64Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
63.64Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
62.96Single6IGLIRL16206IGL-ETB-IRL1620
62.50Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
62.50Consensusangiotensin_onOrthosteric Ligandat1_on
62.50Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
62.50Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
61.90Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
61.90Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
61.90Consensusorexin_onOrthosteric Ligandox2_on
61.54Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
60.87Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
60.87Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
60.87Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
60.87Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
60.71Single5GLHEndothelin-15GLH-ETB-Endothelin-1
60.71Single6IGKEndothelin-36IGK-ETB-Endothelin-3
60.00Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
60.00Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
60.00Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
60.00Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
60.00Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
60.00Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
60.00Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
59.09Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
58.33Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
58.33Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
58.33Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
58.33Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
58.33Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
58.33Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
58.33Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
57.69Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
57.69Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
56.67Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
56.52Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
56.52Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
56.52Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
56.52Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
56.00Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
56.00Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
56.00Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
56.00Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
56.00Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
56.00Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
55.56Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
55.56Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
55.56Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
55.56Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
55.56Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
55.56Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
55.17Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
54.55Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
54.55Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
54.55Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
54.55Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
54.55Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
54.55Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
54.55Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
54.55Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
54.17Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
54.17Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
54.17Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
54.17Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
54.17Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
53.85Single6JODAngiotensin II6JOD-AT2-Angiotensin II
53.85Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
53.57Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
53.57Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
53.57Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
53.57Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
53.57Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
53.33Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
53.33Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
53.33Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
52.38Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
52.38Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
52.17Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
52.17Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
52.17Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
52.17Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
52.17Consensuscck_onOrthosteric Ligandccka_on cckb_on
52.17Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
52.17Consensuschemerin_onOrthosteric Ligandcml1_on
52.17Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
52.17Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
52.00Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
52.00Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
52.00Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
52.00Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
52.00Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
52.00Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
51.85Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
51.85Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
51.85Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
51.85Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
51.85Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
51.72Single8IY6Endothelin-18IY6-ETB-Endothelin-1
51.72Consensusendothelin_onOrthosteric Ligandetb_on eta_on
51.72Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
51.61Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
50.00Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
50.00Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
50.00Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
50.00Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
50.00Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
50.00Single7XN9L-054,5227XN9-SST2-L-054,522
50.00Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
50.00Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
50.00Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
50.00Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
50.00Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
50.00Single8QJ2pN1628QJ2-MC4-pN162-Gs
50.00Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
50.00Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
50.00Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
50.00Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
50.00Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
50.00Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
50.00Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
50.00Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
50.00Consensusbombesin_onOrthosteric Ligandbb2_on
50.00Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
50.00Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
50.00Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
50.00Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
50.00Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
50.00Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
50.00Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
50.00Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
50.00Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
50.00Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
50.00Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
48.28Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
48.28Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
48.28Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
48.28Single9KDFRES-701-39KDF-ETB-RES-701-3
48.15Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
48.15Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
48.15Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
48.15Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
48.15Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
48.15Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
48.00Single4IARErgotamine4IAR-5-HT1B-Ergotamine
48.00Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
48.00Single7F8XNN90567F8X-CCKA-NN9056
48.00Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
48.00Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
48.00Single8WDTphotoNECA8WDT-A2A-photoNECA
48.00Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
48.00Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
48.00Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
48.00Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
48.00Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
48.00Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
48.00Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
47.83Single4RWADIPP-NH24RWA-δ-DIPP-NH2
47.83Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
47.83Single6MXTSalmeterol6MXT-β2-Salmeterol
47.83Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
47.83Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
47.83Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
47.83Single8JJLOlodaterol8JJL-β2-Olodaterol
47.62Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
47.62Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
47.62Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
46.67Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
46.67Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
46.67Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
46.67Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
46.67Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
46.67Consensusbradykinin_onOrthosteric Ligandbk2_on
46.67Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
46.67Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
46.43Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
46.43Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
46.43Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
46.43Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
46.43Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
46.43Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
46.43Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
46.43Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
46.43Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
46.43Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
46.43Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
46.15Single3QAKUK-4320973QAK-A2A-UK-432097
46.15Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
46.15Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
46.15Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
46.15Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
46.15Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
46.15Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
46.15Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
46.15Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
46.15Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
46.15Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
46.15Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
46.15Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
45.83Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
45.83Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
45.83Single7EZCUKA7EZC-A2A-UKA
45.83Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
45.83Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
45.83Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
45.83Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
45.83Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
45.45Single5N2SPSB365N2S-A1-PSB36
45.45Single6D26Fevipiprant6D26-DP2-Fevipiprant
45.45Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
45.45Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
45.45Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
45.45Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
45.45Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
45.45Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
45.45Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
45.45Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
45.45Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
45.45Consensusdp_offOrthosteric Liganddp2_off
45.00Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
45.00Single7XRRLemborexant7XRR-OX2-Lemborexant
45.00Single8GNGIstradefylline8GNG-A2A-Istradefylline
45.00Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
45.00Consensusorexin_offOrthosteric Ligandox2_off ox1_off
45.00Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
44.83Single4XT3Fractalkine4XT3-US28-Fractalkine
44.83Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
44.83Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
44.83Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
44.83Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
44.44Single5WF5UK-4320975WF5-A2A-UK-432097
44.44Single6PT2KGCHM076PT2-δ-KGCHM07
44.44Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
44.44Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
44.44Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
44.44Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
44.44Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
44.44Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
44.44Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
44.44Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
44.00Single4UG2CGS216804UG2-A2A-CGS21680
44.00Single5WF6UK-4320975WF6-A2A-UK-432097
44.00Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
44.00Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
44.00Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
44.00Single9IPYJR14a9IPY-C3aB-JR14a
44.00Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
43.75Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
43.75Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
43.75Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
43.48Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
43.48Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
43.48Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
43.48Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
43.48Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
43.48Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
43.48Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
43.48Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
43.48Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
43.48Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
43.48Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
43.48Single8E0GBU728E0G-μ-BU72
43.48Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
43.48Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
43.48Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
43.48Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
43.48Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
43.48Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
43.48Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
43.48Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
43.48Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
43.48Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
43.48Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
43.48Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
43.48Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
43.48Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
43.48Consensusrelaxin_onOrthosteric Ligandrxfp4_on
43.48Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
43.33Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
43.33Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
42.86Single4ZJCSB-6740424ZJC-OX1-SB-674042
42.86Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
42.86Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
42.86Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
42.86Single7F61PF-036547467F61-H3-PF-03654746
42.86Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
42.86Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
42.86Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
42.86Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
42.86Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
42.86Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
42.86Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
42.86Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
42.86Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
42.86Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.86Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
42.86Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
42.86Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
42.86Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
42.86Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
42.86Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
42.86Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
42.86Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
42.86Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
42.86Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
42.31Single4XT1Fractalkine4XT1-US28-Fractalkine
42.31Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
42.31Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
42.31Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
42.31Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
42.31Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
42.31Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
42.31Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
42.31Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
42.31Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
42.31Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
42.31Consensuslpl_onOrthosteric Ligands1p_on lpa_on
42.31Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
42.31Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
42.31Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
41.94Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
41.94Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
41.67Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
41.67Single6OS2TRV0266OS2-AT1-TRV026
41.67Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
41.67Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
41.67Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
41.67Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
41.67Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
41.67Single7YITNalfurafine7YIT-κ-Nalfurafine
41.67Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
41.67Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
41.67Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
41.67Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
41.67Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
41.67Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
41.67Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
41.67Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
41.67Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
41.67Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
41.67Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
41.67Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
41.67Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
41.67Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
41.67Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
41.67Consensuslpa_offOrthosteric Ligandlpa1_off
41.67Consensuslpl_offOrthosteric Ligands1p_off lpa_off
41.67Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
41.67Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
41.67Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
41.67Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
41.38Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
41.38Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
41.38Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
41.38Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
41.38Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
41.38Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
41.38Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
41.38Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
41.38Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
41.38Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
41.38Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
41.18Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
40.91Single6TOTLemborexant6TOT-OX1-Lemborexant
40.91Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
40.91Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
40.91Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
40.91Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
40.91Single7UL4Alvimopan7UL4-μ-Alvimopan
40.91Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
40.91Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
40.91Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
40.91Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
40.91Single8K5DGSK2560738K5D-HCA2-GSK256073
40.91Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
40.91Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
40.91Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
40.91Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
40.91Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
40.91Single9CHXS-Carazolol9CHX-β2-S-Carazolol
40.91Consensusa3_onOrthosteric Liganda3a_on
40.91Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
40.91Consensuscck_offOrthosteric Ligandccka_off
40.91Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
40.91Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
40.91Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
40.91Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
40.91Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
40.91Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
40.91Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
40.91Consensushca_on_gpOrthosteric Ligandhca2_on_gp
40.91Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
40.91Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
40.74Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
40.74Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
40.74Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
40.74Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
40.74Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
40.74Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
40.74Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
40.62Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
40.62Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
40.00Single3OE9IT1t3OE9-CXCR4-IT1t
40.00Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
40.00Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
40.00Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
40.00Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
40.00Single6IBLArformoterol6IBL-β1-Arformoterol
40.00Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
40.00Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
40.00Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
40.00Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
40.00Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
40.00Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
40.00Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
40.00Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
40.00Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
40.00Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
40.00Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
40.00Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
40.00Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
40.00Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
40.00Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
40.00Consensusendothelin_offOrthosteric Ligandetb_off
40.00Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
40.00Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
40.00Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
40.00Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
40.00Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
40.00Consensusprostanoid_offOrthosteric Ligandep_off dp_off
39.29Single3OE0CVX153OE0-CXCR4-CVX15
39.29Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
39.29Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
39.29Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
39.29Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
39.29Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
39.29Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
39.29Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
39.29Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
39.29Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
39.29Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
39.13Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
39.13Single5C1MBU725C1M-μ-BU72
39.13Single5N2RPSB-365N2R-A2A-PSB-36-Na
39.13Single5WQCEMPA5WQC-OX2-EMPA
39.13Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
39.13Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
39.13Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
39.13Single6TP6Filorexant6TP6-OX1-Filorexant
39.13Single7C61Ergotamine7C61-5-HT1B-Ergotamine
39.13Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
39.13Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
39.13Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
39.13Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
39.13Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
39.13Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
39.13Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
39.13Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
39.13Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
39.13Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
39.13Single8GNEKW-63568GNE-A2A-KW-6356-Na
39.13Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
39.13Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
39.13Single8JXSPF-61428JXS-D1-PF-6142
39.13Single8S4DCMF-0198S4D-Apelin-CMF-019
39.13Single8TF5Oleic acid8TF5-GPR6-Oleic acid
39.13Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
39.13Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
39.13Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
39.13Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
39.13Single9EHSLUF76029EHS-A3A-LUF7602
39.13Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
39.13Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
39.13Consensusa3_on_gpOrthosteric Liganda3a_on_gp
39.13Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
39.13Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
39.13Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
39.13Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
39.13Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
39.13Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
39.13Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
39.13Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
39.13Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
39.13Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
39.13Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
39.13Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
38.71Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
38.71Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
38.71Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
38.46Single3NY9ICI118-5513NY9-β2-ICI118-551
38.46Single5ZTYAM102575ZTY-CB2-AM10257
38.46Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
38.46Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
38.46Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
38.46Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
38.46Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
38.46Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
38.46Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
38.46Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
38.46Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
38.46Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
38.46Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
38.46Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
38.46Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
38.46Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
38.46Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
38.10Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
38.10Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
38.10Single5WS3EMPA5WS3-OX2-EMPA
38.10Single6AKXA4R6AKX-CCR5-A4R
38.10Single6TODEMPA6TOD-OX1-EMPA-Na
38.10Single7F8ULintitript7F8U-CCKA-Lintitript
38.10Single7F8YDevazepide7F8Y-CCKA-Devazepide
38.10Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
38.10Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
38.10Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
38.10Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
38.10Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
38.10Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.10Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
38.10Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
38.10Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
38.10Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
38.10Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
38.10Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
38.10Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
38.10Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
38.10Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
38.10Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
38.10Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
37.93Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
37.93Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
37.93Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
37.93Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
37.93Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
37.93Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
37.93Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
37.93Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
37.93Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
37.93Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
37.93Consensusvasop-oxy_onOrthosteric Ligandv2_on
37.93Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
37.50Single2YDVNECA2YDV-A2A-NECA
37.50Single3P0GBI1671073P0G-β2-BI167107
37.50Single4UHRCGS216804UHR-A2A-CGS21680
37.50Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
37.50Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
37.50Single5G53NECA5G53-A2A-NECA-Gs
37.50Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
37.50Single6H7JIsoprenaline6H7J-β1-Isoprenaline
37.50Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
37.50Single6OS1TRV0266OS1-AT1-TRV026
37.50Single6TQ7SB-3348676TQ7-OX1-SB-334867
37.50Single6WGTLSD6WGT-5-HT2A-LSD
37.50Single7B6WCyclazosin7B6W-α1b-Cyclazosin
37.50Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
37.50Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
37.50Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
37.50Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
37.50Single7TUYGSK682753A7TUY-GPR183-GSK682753A
37.50Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
37.50Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
37.50Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
37.50Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
37.50Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
37.50Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
37.50Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
37.50Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
37.50Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
37.50Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
37.50Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
37.50Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
37.50Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
37.50Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
37.50Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
37.50Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
37.50Single8ZWFJR14a8ZWF-C3aB-JR14a
37.50Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
37.50Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
37.50Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
37.50Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
37.50Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
37.50Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
37.50Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
37.50Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
37.50Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
37.50Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
37.50Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
37.50Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
37.04Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
37.04Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
37.04Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
37.04Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
37.04Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
37.04Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
37.04Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
37.04Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
37.04Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
37.04Single8WKYPG-9348WKY-MC4-PG-934
37.04Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
37.04Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
37.04Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
37.04Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
37.04Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
37.04Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
37.04Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
37.04Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
37.04Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
36.67Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
36.67Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
36.67Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
36.67Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
36.67Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
36.59Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
36.36Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
36.36Single4MBSMaraviroc4MBS-CCR5-Maraviroc
36.36Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
36.36Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
36.36Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
36.36Single6MH8ZM-2413856MH8-A2A-ZM-241385
36.36Single6PS0S-Carazolol6PS0-β2-S-Carazolol
36.36Single6PS4ICI118-5516PS4-β2-ICI118-551
36.36Single6PS5S-Propranolol6PS5-β2-S-Propranolol
36.36Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
36.36Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
36.36Single6TPGEMPA6TPG-OX2-EMPA
36.36Single6TPNHTL66416TPN-OX2-HTL6641
36.36Single6V9SGTPL114036V9S-OX1-GTPL11403
36.36Single7AROLUF58337ARO-A2A-LUF5833-Na
36.36Single7UL3Famotidine7UL3-H2-Famotidine
36.36Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.36Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
36.36Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
36.36Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
36.36Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
36.36Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
36.36Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
36.36Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
36.36Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
36.36Single8IHKAcifran8IHK-HCA3-Acifran
36.36Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
36.36Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
36.36Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
36.36Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
36.36Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
36.36Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
36.36Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.36Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.36Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
36.36Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
36.36Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
36.36Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
36.36Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
36.36Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
36.36Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
36.36Consensushca_onOrthosteric Ligandhca2_on
36.36Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
36.00Single4AMIBucindolol4AMI-β1-Bucindolol
36.00Single4LDEBI1671074LDE-β2-BI167107
36.00Single4XEENeurotensin4XEE-NTS1-Neurotensin
36.00Single4XESNeurotensin4XES-NTS1-Neurotensin
36.00Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
36.00Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
36.00Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
36.00Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
36.00Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
36.00Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
36.00Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
36.00Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
36.00Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
36.00Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
36.00Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
36.00Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
36.00Single8JJ8Formoterol8JJ8-β2-Formoterol
36.00Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
36.00Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
36.00Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
36.00Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
36.00Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
36.00Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
36.00Consensusalpha1_offOrthosteric Ligandalpha1a_off
36.00Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
36.00Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
36.00Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
36.00Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
36.00Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
36.00Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
36.00Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
36.00Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
36.00Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
36.00Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
36.00Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
36.00Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
36.00Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
36.00Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
36.00Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
36.00Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
36.00Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
36.00Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
36.00Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
36.00Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
35.71Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
35.71Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
35.71Single7SK5CXCL127SK5-ACKR3-CXCL12
35.71Single7XNACYN1548067XNA-SST2-CYN154806
35.71Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
35.71Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
35.71Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
35.71Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
35.71Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
35.71Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
35.48Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
35.48Single7SK3CXCL127SK3-ACKR3-CXCL12
35.48Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
35.00Single3OE6IT1t3OE6-CXCR4-IT1t
35.00Single6ME5Agomelatine6ME5-MT1-Agomelatine
35.00Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
35.00Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
35.00Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
34.78Single2Y02Carmoterol2Y02-β1-Carmoterol
34.78Single2Y04Salbutamol2Y04-β1-Salbutamol
34.78Single3EMLZM-2413853EML-A2A-ZM-241385
34.78Single3NY8ICI118-5513NY8-β2-ICI118-551
34.78Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
34.78Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
34.78Single4EJ4Naltrindole4EJ4-δ-Naltrindole
34.78Single4GBRS-Carazolol4GBR-β2-S-Carazolol
34.78Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
34.78Single4QKX35V4QKX-β2-35V
34.78Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
34.78Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
34.78Single6D27CAY104716D27-DP2-CAY10471
34.78Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
34.78Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
34.78Single6PS1Timolol6PS1-β2-Timolol
34.78Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
34.78Single6S0LZM-2413856S0L-A2A-ZM-241385
34.78Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
34.78Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
34.78Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
34.78Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
34.78Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
34.78Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
34.78Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
34.78Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
34.78Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
34.78Single7V3ZCP559407V3Z-CB1-CP55940
34.78Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
34.78Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
34.78Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
34.78Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
34.78Single8CU6LJ-45178CU6-A2A-LJ-4517
34.78Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
34.78Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
34.78Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
34.78Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
34.78Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
34.78Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
34.78Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
34.78Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
34.78Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
34.78Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
34.78Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
34.78Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
34.78Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
34.78Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
34.78Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
34.78Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
34.78Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
34.78Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
34.78Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
34.78Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
34.78Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
34.78Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
34.78Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
34.78Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
34.78Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
34.78Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
34.78Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
34.78Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
34.78Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
34.78Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
34.78Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
34.78Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
34.78Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
34.78Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
34.78Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
34.78Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
34.78Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
34.78Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
34.78Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
34.78Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
34.78Single9H37A1IR09H37-A2A-A1IR0-Na
34.78Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
34.78Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
34.78Consensus5ht5_onOrthosteric Ligand5ht5a_on
34.78Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
34.78Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
34.78Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
34.78Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
34.78Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
34.78Consensusdopamine_offOrthosteric Ligandd2_off d3_off
34.78Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
34.78Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
34.78Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
34.78Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
34.62Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
34.62Single4BUONeurotensin4BUO-NTS1-Neurotensin
34.62Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
34.62Single5X93K-87945X93-ETB-K-8794
34.62Single6H7LDobutamine6H7L-β1-Dobutamine
34.62Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
34.62Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
34.62Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
34.62Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
34.62Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
34.62Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
34.62Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
34.62Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
34.62Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
34.62Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
34.62Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
34.62Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
34.62Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
34.62Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
34.62Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
34.62Single8ZPLHF511168ZPL-CXCR4-HF51116
34.62Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
34.62Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
34.62Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
34.62Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
34.62Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
34.62Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
34.48Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
34.48Single6W25SHU91196W25-MC4-SHU9119-Ca
34.48Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
34.48Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
34.48Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
34.48Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
34.48Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
34.48Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
34.48Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
34.48Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
34.48Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
34.48Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
34.48Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
34.48Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
34.38Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
34.38Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
33.33Single2RH1S-Carazolol2RH1-β2-S-Carazolol
33.33Single2Y03Isoprenaline2Y03-β1-Isoprenaline
33.33Single2YCWS-Carazolol2YCW-β1-S-Carazolol
33.33Single5D6LS-Carazolol5D6L-β2-S-Carazolol
33.33Single5IUAQ274563485IUA-A2A-Q27456348-Na
33.33Single5JQHS-Carazolol5JQH-β2-S-Carazolol
33.33Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
33.33Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
33.33Single5TVNLSD5TVN-5-HT2B-LSD
33.33Single5WIUNemonapride5WIU-D4-Nemonapride
33.33Single5WIVNemonapride5WIV-D4-Nemonapride-Na
33.33Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
33.33Single6E67BI1671076E67-β2-BI167107-Gs(CT)
33.33Single6HLLCP999946HLL-NK1-CP99994
33.33Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
33.33Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
33.33Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
33.33Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
33.33Single6PT3DPI-2876PT3-δ-DPI-287
33.33Single6S0QZM-2413856S0Q-A2A-ZM-241385
33.33Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
33.33Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
33.33Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
33.33Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
33.33Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
33.33Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
33.33Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
33.33Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
33.33Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
33.33Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
33.33Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
33.33Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
33.33Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
33.33Single7W41PD1762527W41-BB2-PD176252
33.33Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
33.33Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
33.33Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
33.33Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
33.33Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
33.33Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
33.33Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
33.33Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
33.33Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
33.33Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
33.33Single8QOTNanobody-E8QOT-μ-Nanobody-E
33.33Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
33.33Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
33.33Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
33.33Single8X5YAstemizole8X5Y-H1-Astemizole
33.33Single8XQJJN2418XQJ-Apelin-JN241
33.33Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
33.33Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
33.33Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
33.33Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
33.33Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
33.33Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
33.33Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
33.33Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
33.33Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
33.33Single9HAPTolvaptan9HAP-V2-Tolvaptan
33.33Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
33.33Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
33.33Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
33.33Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
33.33Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
33.33Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
33.33Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
33.33Consensusadenosine_offOrthosteric Liganda1_off a2_off
33.33Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
33.33Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
33.33Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
33.33Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
33.33Consensusamine_offonOrthosteric Ligandamine_off amine_on
33.33Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
33.33Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
33.33Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
33.33Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
33.33Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
33.33Consensusbombesin_offOrthosteric Ligandbb2_off
33.33Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
33.33Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
33.33Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
33.33Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
33.33Consensuskisspeptin_onOrthosteric Ligandkiss1_on
33.33Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
33.33Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
33.33Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
33.33Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
33.33Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
33.33Consensustrace-amine_onOrthosteric Ligandta1_on
33.33Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
33.33Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
32.43Consensuspth_onOrthosteric Ligandpth1_on pth2_on
32.26Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
32.26Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
32.26Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
32.26Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
32.26Consensuspac_onOrthosteric Ligandpac1_on
32.14Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
32.14Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
32.14Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
32.14Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
32.14Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
32.14Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
32.14Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
32.14Consensussomatostatin_offOrthosteric Ligandsst2_off
32.00Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
32.00Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
32.00Single4DJHJDTic4DJH-κ-JDTic
32.00Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
32.00Single5D5AS-Carazolol5D5A-β2-S-Carazolol
32.00Single5D5BS-Carazolol5D5B-β2-S-Carazolol
32.00Single5XR8AM8415XR8-CB1-AM841
32.00Single5XRAAM115425XRA-CB1-AM11542
32.00Single6J20Aprepitant6J20-NK1-Aprepitant
32.00Single6J21Aprepitant6J21-NK1-Aprepitant
32.00Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
32.00Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
32.00Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
32.00Single7FEECP559407FEE-CB1-CP55940-ZCZ011
32.00Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
32.00Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
32.00Single7PX4PSB-21137PX4-A2A-PSB-2113
32.00Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
32.00Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
32.00Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
32.00Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
32.00Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
32.00Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
32.00Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
32.00Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
32.00Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
32.00Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
32.00Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
32.00Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
32.00Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
32.00Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
32.00Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
32.00Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
32.00Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
32.00Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
32.00Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
32.00Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
32.00Single8XVLZibotentan8XVL-ETA-Zibotentan
32.00Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
32.00Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
32.00Single9BJKNaloxone9BJK-μ-Naloxone-NAM
32.00Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
32.00Consensusa2_onOrthosteric Liganda2b_on
32.00Consensusa2_on_gpOrthosteric Liganda2b_on_gp
32.00Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
32.00Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
32.00Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
32.00Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
32.00Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
32.00Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
32.00Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
32.00Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
32.00Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
32.00Consensuslpa_onOrthosteric Ligandlpa1_on
32.00Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
32.00Consensusneurotensin_onOrthosteric Ligandnts1_on
32.00Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
32.00Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
32.00Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
32.00Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
32.00Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
31.82Single3ODUIT1t3ODU-CXCR4-IT1t
31.82Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
31.82Single4S0VSuvorexant4S0V-OX2-Suvorexant
31.82Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
31.82Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
31.82Single6AKYMaraviroc6AKY-CCR5-Maraviroc
31.82Single6B73MP11046B73-κ-MP1104
31.82Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
31.82Single6ME2Ramelteon6ME2-MT1-Ramelteon
31.82Single6ME9Ramelteon6ME9-MT2-Ramelteon
31.82Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
31.82Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
31.82Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
31.82Single6TPJSuvorexant6TPJ-OX2-Suvorexant
31.82Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
31.82Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
31.82Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
31.82Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
31.82Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
31.82Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.82Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
31.82Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
31.82Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
31.82Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
31.82Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
31.82Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
31.82Single8IWESpermidine8IWE-TA9-Spermidine
31.82Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
31.82Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.82Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.82Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.82Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
31.82Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
31.82Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
31.82Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
31.82Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
31.82Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
31.82Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
31.82Consensusalpha2_offOrthosteric Ligandalpha2c_off
31.82Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
31.25Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
31.25Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
31.25Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
31.03Single6HLOAprepitant6HLO-NK1-Aprepitant
31.03Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
31.03Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
31.03Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
31.03Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
31.03Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
31.03Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
31.03Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
30.77Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
30.77Single3D4STimolol3D4S-β2-Timolol
30.77Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
30.77Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
30.77Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
30.77Single6A93Risperidone6A93-5-HT2A-Risperidone
30.77Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
30.77Single6KQICP559406KQI-CB1-CP55940-Org27569
30.77Single6YVRNTS8-136YVR-NTS1-NTS8-13
30.77Single6ZG4HTL00099366ZG4-M1-HTL0009936
30.77Single7DFPSpiperone7DFP-D2-Spiperone
30.77Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
30.77Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
30.77Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
30.77Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
30.77Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
30.77Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
30.77Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
30.77Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
30.77Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
30.77Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
30.77Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
30.77Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
30.77Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
30.77Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
30.77Single8JWY2-1188JWY-A2A-2-118
30.77Single8JWZAB9288JWZ-A2A-AB928-Na
30.77Single8XYIVUF106618XYI-CXCR3-VUF10661
30.77Single9DGIZ85267113509DGI-CB1-Z8526711350
30.77Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
30.77Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
30.77Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
30.77Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
30.77Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
30.77Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
30.77Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
30.77Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
30.56Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
30.43Single2YDOAdenosine2YDO-A2A-Adenosine
30.43Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
30.43Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
30.43Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
30.43Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
30.43Single5IU7Q274563465IU7-A2A-Q27456346-Na
30.43Single5IUBQ274563445IUB-A2A-Q27456344-Na
30.43Single5JTBZM-2413855JTB-A2A-ZM-241385
30.43Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
30.43Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
30.43Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
30.43Single5UVIZM-2413855UVI-A2A-ZM-241385
30.43Single6IQLL7458706IQL-D4-L745870
30.43Single6KUXRS-799486KUX-α2a-RS-79948
30.43Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
30.43Single6TP3Nemorexant6TP3-OX1-Nemorexant
30.43Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
30.43Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
30.43Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
30.43Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
30.43Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
30.43Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
30.43Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
30.43Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
30.43Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
30.43Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
30.43Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
30.43Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.43Single7T32ZM-2413857T32-A2A-ZM-241385
30.43Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
30.43Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
30.43Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
30.43Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
30.43Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
30.43Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
30.43Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
30.43Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
30.43Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
30.43Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
30.43Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
30.43Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
30.43Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
30.43Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
30.43Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
30.43Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
30.43Single8K5CAcipimox8K5C-HCA2-Acipimox
30.43Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
30.43Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.43Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
30.43Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
30.43Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
30.43Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
30.43Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
30.43Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
30.43Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
30.43Single8ZPMAMD0708ZPM-CXCR4-AMD070
30.43Single9AS5Mescaline9AS5-5-HT2A-Mescaline
30.43Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
30.43Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
30.43Consensusa2_offOrthosteric Liganda2a_off
30.43Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
30.43Consensusalpha1_onOrthosteric Ligandalpha1a_on
30.43Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
30.43Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
30.43Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
30.43Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
30.43Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
30.43Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
30.43Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
30.43Consensusgrh_offOrthosteric Ligandgnrh1_off
30.43Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
30.43Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
30.30Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
30.30Consensusglp_onOrthosteric Ligandglp1_on glp2_on
30.30Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
30.00Single6TQ9SB-4081246TQ9-OX1-SB-408124
30.00Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
30.00Single8A2OTheophylline8A2O-A2A-Theophylline-Na
30.00Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
29.63Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
29.63Single6K1QIRL25006K1Q-ETB-IRL2500
29.63Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
29.63Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
29.63Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
29.63Single7UM4AS26747237UM4-5-HT5A-AS2674723
29.63Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
29.63Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
29.63Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
29.63Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
29.63Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
29.63Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
29.63Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
29.63Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
29.63Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
29.63Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
29.63Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
29.63Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
29.41Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
29.41Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
29.41Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
29.41Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
29.41Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
29.27Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
29.17Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
29.17Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
29.17Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
29.17Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
29.17Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
29.17Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
29.17Single4YAYZD-71554YAY-AT1-ZD-7155
29.17Single5DHGC-355DHG-NOP-C-35
29.17Single5DHHSB-6121115DHH-NOP-SB-612111
29.17Single5IU8Q274563475IU8-A2A-Q27456347-Na
29.17Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
29.17Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
29.17Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
29.17Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
29.17Single5UENDU1725UEN-A1-DU172
29.17Single5UIGCmpd-15UIG-A2A-Cmpd-1
29.17Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
29.17Single6DRXLisuride6DRX-5-HT2B-Lisuride
29.17Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
29.17Single6H7MSalbutamol6H7M-β1-Salbutamol
29.17Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
29.17Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
29.17Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
29.17Single7BU7BI1671077BU7-β1-BI167107
29.17Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
29.17Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
29.17Single7PYRPSB-21157PYR-A2A-PSB-2115
29.17Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
29.17Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
29.17Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
29.17Single7WC7Lisuride7WC7-5-HT2A-Lisuride
29.17Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
29.17Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
29.17Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
29.17Single8JJOAlprenolol8JJO-β2-Alprenolol
29.17Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
29.17Single8JXRLSD8JXR-D1-LSD
29.17Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
29.17Single8T1WCVN4248T1W-GPR6-CVN424
29.17Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
29.17Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
29.17Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
29.17Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
29.17Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
29.17Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
29.17Single9IYAONO-97105319IYA-GPR55-ONO-9710531
29.17Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
29.17Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
29.17Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
29.17Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
29.17Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
29.17Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
29.17Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
29.17Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
29.17Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
29.17Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
29.17Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
29.17Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
29.03Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
29.03Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
29.03Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
29.03Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
29.03Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
29.03Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
29.03Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
28.57Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
28.57Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
28.57Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
28.57Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
28.57Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
28.57Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
28.57Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
28.57Single7SK9CCX6627SK9-ACKR3-CCX662
28.57Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.57Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
28.57Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
28.57Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
28.57Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
28.57Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
28.57Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
28.57Consensus5ht2_onOrthosteric Ligand5ht2b_on
28.57Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.12Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
28.12Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
28.00Single2Y00Dobutamine2Y00-β1-Dobutamine
28.00Single5XPRBosentan5XPR-ETB-Bosentan
28.00Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
28.00Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
28.00Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
28.00Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
28.00Single6PS6Timolol6PS6-β2-Timolol
28.00Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
28.00Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
28.00Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
28.00Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
28.00Single7WC6LSD7WC6-5-HT2A-LSD
28.00Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
28.00Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
28.00Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
28.00Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
28.00Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
28.00Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
28.00Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
28.00Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
28.00Single8ZMFA1L108ZMF-5-HT2C-A1L10
28.00Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
28.00Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
28.00Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
28.00Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
28.00Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
28.00Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
28.00Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
28.00Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
28.00Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
28.00Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
28.00Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
28.00Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
28.00Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
28.00Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
27.78Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
27.78Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
27.59Single7QA8Peptide7QA8-STE2-Peptide
27.59Single7QA8Peptide7QA8-STE2-Peptide
27.59Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
27.59Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
27.59Single8IEBA1LYA8IEB-GPR156-A1LYA
27.59Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
27.59Single9M4TSilodosin9M4T-Alpha1A-Silodosin
27.50Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
27.27Single3PBLEticlopride3PBL-D3-Eticlopride
27.27Single6FJ3PTH6FJ3-PTH1-PTH
27.27Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
27.27Single6TP4ACT-4622066TP4-OX1-ACT-462206
27.27Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
27.27Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
27.27Single7SRQLSD7SRQ-5-HT2B-LSD
27.27Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
27.27Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
27.27Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
27.27Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
27.27Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
27.27Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
27.27Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
27.27Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
27.27Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
27.27Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
27.27Single8K5BNiacin8K5B-HCA2-Niacin
27.27Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
27.27Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
27.27Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
27.27Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.27Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
27.27Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
27.27Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
27.27Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
27.27Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
27.27Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
27.27Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
27.27Consensusgq_nucleotideOrthosteric Ligandgq_p2y
27.27Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
27.27Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
26.92Single4BV0Neurotensin4BV0-NTS1-Neurotensin
26.92Single5TZRMK86665TZR-FFA1-MK8666
26.92Single6E59L-7607356E59-NK1-L-760735
26.92Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
26.92Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
26.92Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
26.92Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
26.92Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
26.92Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.92Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
26.92Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
26.92Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
26.92Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
26.92Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
26.92Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
26.92Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
26.92Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
26.92Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
26.92Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
26.92Consensustachykinin_offOrthosteric Ligandnk1_off
26.67Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
26.67Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
26.67Single8IEBA1LYA8IEB-GPR156-A1LYA
26.67Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
26.47Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
26.47Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
26.47Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
26.47Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
26.32Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
26.32Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
26.32Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
26.32Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
26.09Single3PWHZM-2413853PWH-A2A-ZM-241385
26.09Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
26.09Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
26.09Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
26.09Single6DS0Ly2660976DS0-5-HT2B-Ly266097
26.09Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
26.09Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
26.09Single7BR3Elagolix7BR3-GnRH1-Elagolix
26.09Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
26.09Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
26.09Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.09Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
26.09Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
26.09Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
26.09Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
26.09Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
26.09Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
26.09Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
26.09Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
26.09Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.09Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
26.09Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
26.09Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
26.09Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
26.09Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
26.09Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
26.09Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
26.09Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
26.09Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
26.09Single8Y0HVUF114188Y0H-CXCR3-VUF11418
26.09Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
26.09Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
26.09Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
26.09Single9H2XA1IR19H2X-A2A-A1IR1-Na
26.09Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
26.09Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
26.09Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
26.09Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.09Consensusangiotensin_offOrthosteric Ligandat1_off
26.09Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
26.09Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
26.09Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
26.09Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
26.09Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
26.09Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
25.93Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
25.93Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
25.93Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
25.93Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
25.93Single7K15MKD0467K15-BLT1-MKD046-Na
25.93Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
25.93Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
25.93Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
25.93Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
25.93Single8XQJJN2418XQJ-Apelin-JN241
25.93Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
25.93Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
25.93Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
25.81Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.81Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
25.81Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
25.81Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
25.81Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
25.71Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
25.71Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
25.71Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
25.71Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
25.71Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
25.71Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
25.71Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
25.71Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
25.64Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
25.64Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
25.00Single3REYXAC3REY-A2A-XAC
25.00Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
25.00Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
25.00Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
25.00Single6A94Zotepine6A94-5-HT2A-Zotepine
25.00Single6AQFZM-2413856AQF-A2A-ZM-241385
25.00Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
25.00Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
25.00Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
25.00Single6TPKRetosiban6TPK-OT-Retosiban
25.00Single6VI4JDTic6VI4-κ-JDTic
25.00Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
25.00Single6ZG9GSK10347026ZG9-M1-GSK1034702
25.00Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
25.00Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
25.00Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
25.00Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
25.00Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
25.00Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
25.00Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
25.00Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
25.00Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
25.00Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
25.00Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
25.00Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
25.00Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
25.00Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
25.00Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
25.00Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
25.00Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Single8PWNTheophylline8PWN-A2A-Theophylline
25.00Single8RLNLUF58348RLN-A2A-LUF5834
25.00Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
25.00Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
25.00Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
25.00Single8XVUCXCL28XVU-CXCR2-CXCL2
25.00Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
25.00Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
25.00Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
25.00Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
25.00Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
25.00Single8ZPNAMD31008ZPN-CXCR4-AMD3100
25.00Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
25.00Single9ARXSerotonin9ARX-5-HT2A-Serotonin
25.00Single9AS3LSD9AS3-5-HT2A-LSD
25.00Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
25.00Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
25.00Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
25.00Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
25.00Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
25.00Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
25.00Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
25.00Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
25.00Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
25.00Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
25.00Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
25.00Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
25.00Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
25.00Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
25.00Consensusvasop-oxy_offOrthosteric Ligandot_off
24.39Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
24.32Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
24.24Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
24.24Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
24.24Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
24.24Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
24.24Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
24.24Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
24.14Single6KNMJN241-96KNM-Apelin-JN241-9
24.14Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
24.14Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
24.14Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
24.14Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
24.14Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
24.14Single9JF4PD1683689JF4-BB1-PD168368
24.14Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
24.00Single2Y01Dobutamine2Y01-β1-Dobutamine
24.00Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
24.00Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
24.00Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
24.00Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
24.00Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
24.00Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
24.00Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
24.00Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
24.00Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
24.00Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
24.00Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
24.00Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
24.00Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
24.00Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
24.00Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
24.00Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
24.00Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
24.00Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
24.00Single8X63Mepyramine8X63-H1-Mepyramine
24.00Single8X64Desloratadine8X64-H1-Desloratadine
24.00Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
24.00Single9AS1DMT9AS1-5-HT2A-DMT
24.00Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
24.00Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
24.00Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
24.00Consensusalpha2_onOrthosteric Ligandalpha2b_on
24.00Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
24.00Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
24.00Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
24.00Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
24.00Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
24.00Consensusblt_onOrthosteric Ligandblt1_on
24.00Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
24.00Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
24.00Consensushistamine_offOrthosteric Ligandh1_off
24.00Consensusleukotriene_onOrthosteric Ligandblt_on
24.00Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
23.81Single3OE8IT1t3OE8-CXCR4-IT1t
23.81Single3RFMCaffeine3RFM-A2A-Caffeine
23.81Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.81Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
23.81Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
23.81Single9CHUNoradrenaline9CHU-β2-Noradrenaline
23.81Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
23.81Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
23.81Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
23.68Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
23.68Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
23.68Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
23.68Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
23.53Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
23.53Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
23.53Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
23.53Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
23.53Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
23.53Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
23.53Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
23.53Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
23.33Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
23.33Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
23.33Single8IEIA1LYA8IEI-GPR156-A1LYA
23.33Single8IEIA1LYA8IEI-GPR156-A1LYA
23.33Single8IEPA1LYA8IEP-GPR156-A1LYA
23.33Single8IEPA1LYA8IEP-GPR156-A1LYA
23.33Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
23.33Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
23.33Single8KIGSHU91198KIG-MC3-SHU9119-Ca
23.33Single8XWNCXCL88XWN-CXCR2-CXCL8
23.33Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
23.08Single4NTJAZD12834NTJ-P2Y12-AZD1283
23.08Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
23.08Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
23.08Single6HLPNetupitant6HLP-NK1-Netupitant
23.08Single6LUQHaloperidol6LUQ-D2-Haloperidol
23.08Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
23.08Single7C4SS1P7C4S-S1P3-S1P
23.08Single7SINNPS-21437SIN-CaS-NPS-2143
23.08Single7SINNPS-21437SIN-CaS-NPS-2143
23.08Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
23.08Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
23.08Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.08Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
23.08Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
23.08Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
23.08Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
23.08Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
23.08Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
23.08Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
23.08Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
23.08Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
23.08Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
23.08Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
22.86Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
22.86Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
22.86Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
22.86Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
22.86Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
22.86Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
22.86Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
22.86Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
22.86Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
22.73Single4XNWMRS25004XNW-P2Y1-MRS2500
22.73Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
22.73Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
22.73Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
22.73Single7WC5Psilocin7WC5-5-HT2A-Psilocin
22.73Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
22.73Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
22.73Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
22.73Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
22.73Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
22.73Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
22.73Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
22.73Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
22.73Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
22.73Single9LRCHistamine9LRC-H4-Histamine
22.73Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
22.73Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
22.73Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
22.73Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
22.73Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
22.73Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
22.73Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
22.22Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
22.22Single4U15Tiotropium4U15-M3-Tiotropium
22.22Single5V54Methiothepin5V54-5-HT1B-Methiothepin
22.22Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
22.22Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
22.22Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
22.22Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
22.22Single6OL9Tiotropium6OL9-M5-Tiotropium
22.22Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
22.22Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
22.22Single7F1TMIP-1a7F1T-CCR5-MIP-1a
22.22Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
22.22Single7R0CAVP7R0C-V2-AVP-Arrestin2
22.22Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
22.22Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
22.22Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
22.22Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
22.22Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
22.22Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
22.22Consensus5ht1_offOrthosteric Ligand5ht1b_off
22.22Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
22.22Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
22.22Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
22.22Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
22.22Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
22.22Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
22.22Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
22.22Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
22.22Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
22.22Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
22.22Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
21.88Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
21.88Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
21.88Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
21.74Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
21.74Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
21.74Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
21.74Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
21.74Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.74Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
21.74Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
21.74Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
21.74Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
21.74Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
21.74Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
21.74Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
21.74Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.74Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
21.74Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
21.62Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
21.62Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
21.62Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
21.43Single4N4WSANT-14N4W-SMO-SANT-1
21.43Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
21.43Single4PY02MeSATP4PY0-P2Y12-2MeSATP
21.43Single5CXVTiotropium5CXV-M1-Tiotropium
21.43Single6CM4Risperidone6CM4-D2-Risperidone
21.43Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
21.43Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
21.43Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.43Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
21.43Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
21.43Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
21.43Single8XWACXCL18XWA-CXCR2-CXCL1
21.43Single8XWMCXCL68XWM-CXCR2-CXCL6
21.43Single8XWSCXCL58XWS-CXCR2-CXCL5
21.43Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
21.43Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.43Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
21.21Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
21.21Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
21.05Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
21.05Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
21.05Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
20.83Single4BWBNeurotensin4BWB-NTS1-Neurotensin
20.83Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
20.83Single5ZKQABT-4915ZKQ-PAF-ABT-491
20.83Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
20.83Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
20.83Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
20.83Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
20.83Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
20.83Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
20.83Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
20.83Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
20.83Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.83Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
20.83Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
20.83Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
20.83Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
20.83Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
20.83Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
20.83Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
20.83Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.83Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
20.83Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
20.83Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
20.83Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
20.83Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
20.83Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
20.83Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
20.83Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
20.83Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
20.83Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
20.83Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
20.83Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
20.83Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
20.83Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
20.83Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
20.83Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
20.83Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
20.83Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
20.83Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
20.69Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
20.69Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Single8XVJMacitentan8XVJ-ETA-Macitentan
20.69Single8XWFCXCL38XWF-CXCR2-CXCL3
20.69Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
20.59Consensuscalcitonin_onOrthosteric Ligandctlike_on
20.59Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
20.51Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
20.51Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
20.51Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.51Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
20.51Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
20.00Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
20.00Single3RZECidoxepin3RZE-H1-Cidoxepin
20.00Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
20.00Single5MZPCaffeine5MZP-A2A-Caffeine-Na
20.00Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
20.00Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
20.00Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
20.00Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
20.00Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
20.00Single6ZINSR486926ZIN-NTS1-SR48692
20.00Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
20.00Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
20.00Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
20.00Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
20.00Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
20.00Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
20.00Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
20.00Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
20.00Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
20.00Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
20.00Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
20.00Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
20.00Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
20.00Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
20.00Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
20.00Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
20.00Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
20.00Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
20.00Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
19.44Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
19.44Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
19.44Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
19.44Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
19.35Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
19.35Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single4DAJTiotropium4DAJ-M3-Tiotropium
19.23Single4MQSIperoxo4MQS-M2-Iperoxo
19.23Single4QIMANTA XV4QIM-SMO-ANTA XV
19.23Single4U14Tiotropium4U14-M3-Tiotropium
19.23Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
19.23Single5T04Neurotensin5T04-NTS1-Neurotensin
19.23Single5TGZAM65385TGZ-CB1-AM6538
19.23Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
19.23Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
19.23Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
19.23Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
19.23Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
19.23Single6GPSMK08126GPS-CCR2-MK0812
19.23Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
19.23Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
19.23Single7F83PF-051904577F83-Ghrelin-PF-05190457
19.23Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
19.23Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
19.23Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
19.23Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
19.23Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
19.23Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
19.23Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
19.23Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
19.23Single9JEAAtropine9JEA-M1-Atropine
19.23Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
19.23Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
19.23Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
19.23Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
19.23Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
19.23Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
19.05Single7WC4Serotonin7WC4-5-HT2A-Serotonin
19.05Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
19.05Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
19.05Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
18.92Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
18.92Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
18.92Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
18.75Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
18.75Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
18.75Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
18.52Single6GPXMK08126GPX-CCR2-MK0812
18.52Single6Z4SSR486926Z4S-NTS1-SR48692
18.52Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
18.52Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
18.52Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
18.52Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.52Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
18.52Consensusblt_offOrthosteric Ligandblt1_off
18.52Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
18.52Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
18.52Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
18.52Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.52Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.52Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
18.18Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
18.18Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
18.18Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
18.18Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
18.18Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
18.18Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
18.18Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
18.18Consensusp2y_offOrthosteric Ligandp2y1_off
18.18Consensussensory_onOrthosteric Ligandopsins_on
17.95Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
17.86Single5V56TC1145V56-SMO-TC114
17.86Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
17.86Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
17.86Single8EA0Iperoxo8EA0-M3-Iperoxo
17.86Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
17.86Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
17.86Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.86Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
17.86Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
17.78Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
17.65Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
17.65Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
17.65Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
17.65Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
17.65Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
17.39Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
17.39Single3UZAGTPL92363UZA-A2A-GTPL9236
17.39Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
17.39Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
17.39Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
17.39Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
17.39Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
17.39Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.39Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
17.39Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
17.39Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
17.39Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
17.39Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
17.39Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
17.39Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
17.24Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
17.24Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
17.24Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
17.24Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
17.24Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.24Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
17.24Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
17.24Single9BJKNAM9BJK-μ-Naloxone-NAM
17.24Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.24Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
17.24Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
17.14Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
17.07Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
16.67Single4O9RCyclopamine4O9R-SMO-Cyclopamine
16.67Single5L7IVismodegib5L7I-SMO-Vismodegib
16.67Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
16.67Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
16.67Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
16.67Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
16.67Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
16.67Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
16.67Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
16.67Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
16.67Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
16.67Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
16.67Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
16.67Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
16.67Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
16.67Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
16.67Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Single9AS7Psilocin9AS7-5-HT2A-Psilocin
16.67Single9B9Y7DY9B9Y-CB1-7DY
16.67Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
16.67Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
16.67Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
16.67Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
16.67Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
16.67Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
16.67Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
16.67Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
16.67Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
16.13Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
16.00Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
16.00Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
16.00Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
16.00Single4QINSAG1.54QIN-SMO-SAG1.5
16.00Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
16.00Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
16.00Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
16.00Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
16.00Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
16.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
16.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
16.00Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.00Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
16.00Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
16.00Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
16.00Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
15.79Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
15.79Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
15.79Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
15.79Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
15.79Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
15.62Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
15.62Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
15.62Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
15.62Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
15.62Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
15.38Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
15.38Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
15.38Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
15.38Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
15.38Single7VODCariprazine7VOD-5-HT2A-Cariprazine
15.38Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
15.38Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
15.38Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
15.38Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
15.38Single8K2WAMG4878K2W-CXCR3-AMG487
15.38Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
15.38Single9BA0A1AKN9BA0-CB1-A1AKN
15.38Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
15.38Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
15.38Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
15.38Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
15.38Consensusopsins_offOrthosteric Ligandrhodopsin_off
15.38Consensussensory_offOrthosteric Ligandopsins_off
15.15Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
15.00Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
14.81Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
14.81Single5DSGTiotropium5DSG-M4-Tiotropium
14.81Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.81Single7YXAONO-54306087YXA-S1P5-ONO-5430608
14.81Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
14.81Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
14.81Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
14.81Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
14.81Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
14.81Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
14.81Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
14.29Single4JKVTaladegib4JKV-SMO-Taladegib
14.29Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
14.29Single5CGCHTL142425CGC-mGlu5-HTL14242
14.29Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
14.29Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
14.29Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
14.29Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
14.29Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
14.29Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
14.29Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
14.29Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
14.29Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
14.29Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
14.29Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
14.29Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
14.29Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
14.29Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
14.29Single9B9ZA1AKO9B9Z-CB1-A1AKO
14.29Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
14.29Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
14.29Consensusep_offOrthosteric Ligandep4_off
13.95Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
13.89Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
13.89Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
13.79Single5V57TC1145V57-SMO-TC114
13.79Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
13.79Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
13.79Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
13.79Single9AS9RS130-1809AS9-5-HT2A-RS130-180
13.79Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
13.64Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
13.64Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
13.64Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
13.51Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
13.33Single5X33BIIL2605X33-BLT1-BIIL260
13.33Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
13.33Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
13.16Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
13.16Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
13.16Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
13.16Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
13.04Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
12.90Single5CGDHTL142425CGD-mGlu5-HTL14242
12.90Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
12.90Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
12.90Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.90Single9JH5C16:0 Ceramide9JH5-CysLT2-C16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
12.90Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
12.90Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
12.50Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
12.50Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
12.50Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
12.50Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
12.50Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.50Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
12.50Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.50Consensusgi_sensoryOrthosteric Ligandgi_opsins
12.50Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.50Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.12Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
12.00Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
12.00Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
12.00Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
12.00Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
12.00Single7UL2SR486927UL2-NTS1-SR48692-Na
12.00Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
12.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
12.00Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
12.00Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
12.00Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
12.00Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
12.00Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
12.00Consensusneurotensin_offOrthosteric Ligandnts1_off
12.00Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
11.54Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
11.54Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
11.54Single5U09Taranabant5U09-CB1-Taranabant
11.54Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
11.54Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
11.54Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
11.54Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
11.54Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
11.54Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
11.54Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
11.54Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
11.11Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
11.11Single7VV6C48/807VV6-MRGPRX2-C48/80
11.11Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
10.71Single6IIVDaltroban6IIV-TXA2-Daltroban
10.71Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
10.71Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
10.34Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
10.34Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
10.34Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
10.34Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
10.34Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
10.34Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
10.34Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single9HC04YI9HC0-mGlu5-4YI
10.34Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
10.34Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
10.00Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
10.00Single7P2L4YI7P2L-mGlu5-4YI
10.00Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
10.00Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
10.00Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
10.00Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
9.68Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
9.68Single6IIURamatroban6IIU-TXA2-Ramatroban
9.68Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
9.52Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
9.09Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
9.09Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
8.70Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
8.33Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
8.33Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
8.33Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
8.33Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
8.33Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
8.00Single8JPSCCL78JPS-ACKR1-CCL7
8.00Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
7.69Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
7.69Single6LI0C176LI0-GPR52-C17
7.69Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
7.41Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
7.14Single6FFIMMPEP6FFI-mGlu5-MMPEP
7.14Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
6.90Single6FFHFenobam6FFH-mGlu5-Fenobam
6.90Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
6.67Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
6.45Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
6.45Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
6.45Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
6.06Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
5.88Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
5.71Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
4.76Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
4.76Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
4.55Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
4.35Single8JGBConorfamide-Tx28JGB-MRGPRX1-Conorfamide-Tx2-Gi1/β1/γ2
4.17Single8HS2Fab0468HS2-GPR20-Fab046
4.17Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
4.00Single7Y14Beta-Alanine7Y14-MRGPRD-β-Alanine
3.85Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
3.85Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
3.85Single7Y12Beta-Alanine7Y12-MRGPRD-β-Alanine-Gi1/β1/γ2
3.85Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
3.70Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
3.70Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
3.70Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
3.70Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
3.70Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
3.57Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
3.57Single8G94CD698G94-S1P1-CD69-Gi1/β1/γ2
3.45Single8IYXYL-3658IYX-GPR34-YL-365
3.33Single8Y73MPAM-158Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
3.23Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
3.23Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB

Consensus Members
Id Members
peptide_on_gp cck_on_gp
angiotensin_on_gp
apelin_on_gp
bombesin_on_gp
bradykinin_on_gp
compl-peptide_on_gp
endothelin_on_gp
formylpeptide_on_gp
galanin_on_gp
ghrelin_on_gp
kisspeptin_on_gp
melanocortin_on_gp
motilin_on_gp
neuromedin-u_on_gp
npy_on_gp
neurotensin_on_gp
opioid_on_gp
orexin_on_gp
relaxin_on_gp
somatostatin_on_gp
tachykinin_on_gp
trh_on_gp
vasop-oxy_on_gp
peptide_off cck_off
angiotensin_off
bombesin_off
endothelin_off
ghrelin_off
npy_off
opioid_off
orexin_off
somatostatin_off
tachykinin_off
vasop-oxy_off
neurotensin_off
Net Summary
Imin 3.26482
Number of Linked Nodes 1154
Number of Links 1181
Number of Hubs 118
Number of Links mediated by Hubs 517
Number of Communities 7
Number of Nodes involved in Communities 52
Number of Links involved in Communities 64
Path Summary
Number Of Nodes in MetaPath 101
Number Of Links MetaPath 100
Number of Shortest Paths 365640
Length Of Smallest Path 3
Average Path Length 44.2027
Length of Longest Path 94
Minimum Path Strength 0.261749
Average Path Strength 3.54194
Maximum Path Strength 10.1876
Minimum Path Correlation 0.70125
Average Path Correlation 0.891672
Maximum Path Correlation 0.986143
Minimum % Of Corr. Nodes 1.11111
Average % Of Corr. Nodes 14.5191
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 37.5168
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .




You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

Download peptide_offon_gp.zip



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You can also  read or  download a guide explaining the meaning of all files and numerical data.