Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.11 3.08333402
2G.HN.47 3.30583466
3G.S1.02 4.74067595
4G.H1.01 4.07417409
5G.H1.07 5.83409
6G.S2.03 4.075419
7G.S2.05 4.39413
8G.S2.08 6.26417495
9G.S3.03 7.61267597
10G.S3.04 6.5025416
11G.S3.05 3.49833407
12G.S3.06 7.746515
13G.s3h2.03 6.0475419
14G.H2.06 5.21952719
15G.H2.07 6.3025419
16G.H2.10 3.0775417
17G.h2s4.01 6.26917419
18G.S4.04 5.49333589
19G.S4.06 3.6125407
20G.s4h3.04 6.65444658
21G.s4h3.05 7.1125459
22G.H3.02 2.60667458
23G.H3.04 3.79417409
24G.H3.09 6.28111689
25G.H3.13 3.595485
26G.H3.17 6.485615
27G.H3.18 7.83833419
28G.S5.02 3.36083486
29G.S5.03 2.7875408
30G.S5.05 3.5445149
31G.S5.06 4.19167408
32G.HG.01 3.285405
33G.HG.04 4.97733559
34G.HG.07 4.35917459
35G.HG.15 4.54917457
36G.hgh4.01 4.78133556
37G.hgh4.02 5.94067557
38G.hgh4.05 10.4992407
39G.H4.03 5.52667404
40G.H4.10 12.5933456
41G.H4.15 4.23458
42G.h4s6.02 3.94133588
43G.h4s6.12 6.838534
44G.S6.01 4.35485
45G.S6.02 5.30778637
46G.S6.05 3.93333404
47G.H5.03 4.335834148
48G.H5.05 3.90833495
49G.H5.08 4.66222698
50G.H5.13 7.50667438
51G.H5.16 3.0075406
52G.H5.20 4.08867539
53G.H5.25 3.67833437
54b.1x1 2.01833404
55b.1x4 2.54667508
56b.1x11 4.078508
57b.1x19 4.72083446
58b.lh12x2 5.24833408
59b.h2x1 4.30583405
60b.lhb1x3 4.134162
61b.b1x6 7.33333569
62b.l1x3 7.978509
63b.b2x1 5.84933518
64b.b2x3 4.0075466
65b.b2x5 6.12056667
66b.b3x2 5.69417465
67b.l3x2 4.301674179
68b.b4x4 7.27083468
69b.b4x6 10.2422669
70b.l4x2 10.8767464
71b.b5x2 4.79917407
72b.b5x3 6.16556669
73b.b5x5 4.7554195
74b.b5x7 4.68167407
75b.l5x1 3.934158
76b.l5x5 6.47905719
77b.b6x5 3.7506
78b.b7x1 6.0285204
79b.b7x4 2.850834158
80b.l7x2 3.1875419
81b.b8x3 3.484174206
82b.b8x4 4.319335156
83b.l8x5 2.44917403
84b.b9x2 2.59083405
85b.l9x3 5.83048719
86b.l9x6 4.477671018
87b.b10x4 3.24186
88b.b10x5 3.65222609
89b.b11x2 2.8725417
90b.b11x4 4.47467519
91b.b11x6 7.015419
92b.l11x2 7.49867519
93b.b12x6 8.5881718
94b.b13x7 8.44867577
95b.l13x3 6.99389679
96b.l13x6 4.9075419
97b.l13x7 3.85917479
98b.b14x3 3.558334185
99b.b15x1 6.36167479
100b.b15x2 7.08083446
101b.b15x3 3.80083479
102b.l15x2 5.56579
103b.b16x4 7.62667576
104b.b16x5 4.61467545
105b.b16x6 8.92867578
106b.b17x4 3.99333445
107b.b17x5 6.45133547
108b.b17x7 5.725448
109b.l17x3 7.76611649
110b.l17x6 6.79733519
111b.b18x3 4.4775448
112b.b18x5 6.14417405
113b.l18x1 5.395717126
114b.l18x2 6.730834127
115b.b19x2 5.44095746
116b.b19x4 4.65083448
117b.l19x1 6.28083419
118b.l19x2 7.70833449
119b.b20x4 10.0267548
120b.b20x6 5.51546
121b.l20x2 6.76333409
122b.b21x1 6.46333547
123b.b21x2 3.39733506
124b.b21x7 4.79933505
125b.b22x5 4.812786127
126b.l22x5 7.761674169
127b.b23x6 6.601116117
128b.l23x1 7.36583406
129b.b24x4 6.849174116
130b.b24x6 6.57754118
131b.l24x2 5.214174166
132b.l24x3 4.982505
133b.l25x3 7.3485109
134b.l26x1 6.115467
135b.l26x5 4.96833405
136b.l27x1 12.3153519
137b.b28x3 4.2975467
138b.b28x4 5.560834106
139b.b28x6 8.450556109
140g.h1x1 2.38833402
141g.h1x11 2.82167409
142g.l1x4 4.84333548
143g.h2x11 7.074174126
144g.ctx3 5.368336229
145g.ctx6 3.25833406
146g.ctx14 2.398509
147g.ctx16 4.39611668
148Lig 4.642981920
149NT.H21 4.64467527
150NT.Y22 5.04733529
1511x39 3.345407
1521x50 5.40333409
1531x60 2.86333407
154I1x49 4.76667406
1552x39 4.3975438
1562x40 6.141674239
1572x41 4.215404
1582x42 6.06267508
1592x45 3.755335139
1602x46 4.38333439
1612x50 6.42917409
1622x57 4.59267526
1632x60 5.112526
1642x64 4.5625425
165E1x501 5.29944627
166E1x52 2.92333526
1673x25 9.98583429
1683x26 6.995426
1693x28 4.62857726
1703x29 6.71267525
1713x33 4.85425
1723x43 4.97583439
1733x46 4.4425439
1743x49 7.07409
1753x50 4.14133539
176I2x52 3.92917405
177I2x53 4.33083407
1784x42 5.225407
1794x46 2.493334137
1804x50 3.901116139
181E2.L179 3.33583423
182E2.I188 4.3425424
183E2.L189 4.56917425
184E2.Y192 6.1375423
1855x39 6.83762726
1865x58 3.26143739
1875x62 5.42867536
1886x26 7.41556634
1896x29 5.25667634
1906x33 3.20167438
1916x48 5.14458828
1926x52 9.64333426
1936x58 7.12833424
1947x31 5.17933522
1957x53 4.29389639
1968x50 3.555834238
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1b.b2x5 b.l4x1 19.28014.94YesNo675
2b.b2x3 b.b2x5 32.21493.1YesYes667
3b.b26x2 b.b2x3 41.07016.48NoYes076
4b.b26x1 b.b26x2 41.40262.29333NoNo097
5b.b26x1 b.l27x1 41.56914.94NoYes099
6b.b2x1 b.l27x1 56.35436.11YesYes189
7G.H2.10 b.b2x1 23.51623.58333YesYes178
8G.H2.10 G.h2s4.01 31.01793.72667YesYes179
9G.S3.06 G.h2s4.01 36.33975.71667YesYes159
10G.S1.03 G.S3.06 1007.03NoYes095
11G.S1.03 I2x53 99.9727.56333NoYes097
12I2x52 I2x53 93.18945.09667YesYes057
13I2x51 I2x52 87.92781.44NoYes065
143x56 I2x51 87.84674.12667NoNo056
153x56 4x38 87.76661.44NoNo057
16b.b2x1 b.l3x1 33.928710.5233YesNo189
17b.l3x1 b.l5x5 34.48336.57333NoYes199
18G.S3.06 b.l5x5 63.254510.69YesYes159
19G.S1.05 G.h2s4.01 13.0735.27667NoYes099
20G.S1.05 G.S1.07 12.83592.30667NoNo099
21G.S1.07 G.S4.04 12.48932.43667NoYes899
22G.S4.04 G.S4.06 12.34692.62YesYes097
23b.l5x5 b.l7x2 56.72494.56YesYes199
24b.l7x2 b.l9x6 56.08852.73333YesYes198
25b.l11x1 b.l9x6 12.14145.31NoYes198
26b.b11x6 b.l11x1 12.05313.71YesNo199
27b.l25x6 b.l27x1 14.984618.99NoYes089
282x39 3x50 22.2914.13333YesYes389
292x39 3x49 40.97145.86333YesYes089
302x38 3x49 60.46476.97667NoYes059
312x38 4x41 87.36449.59667NoNo055
324x38 4x41 87.44488.25NoNo075
33b.b10x1 b.l9x6 49.27443.39333NoYes098
34b.b10x1 b.b11x5 49.2033.26NoNo096
35b.b11x5 b.l13x7 44.02175.38667NoYes069
36b.l13x3 b.l13x7 22.25025.07667YesYes799
37b.b16x4 b.l13x3 21.45415.72YesYes769
38b.b16x4 b.b17x3 21.0644.31333YesNo765
39b.b17x3 g.h1x10 43.77857.12NoNo059
40g.h1x10 g.h1x13 43.60662.26667NoNo091
41b.b17x2 g.h1x13 43.41812.88667NoNo031
42b.b17x2 b.b17x4 42.63832.89333NoYes035
43b.b17x4 b.b17x5 31.60374.28333YesYes457
44b.b17x5 b.b21x1 17.020310.4433YesYes477
45b.1x15 g.h1x15 19.69792.70667NoNo078
46b.1x11 g.h1x15 19.08692.10333YesNo088
47b.1x11 b.1x7 10.48071.33YesNo088
48b.b15x3 b.l13x7 21.12212.69333YesYes799
49b.b15x3 b.b16x6 21.05475.35333YesYes798
50b.b16x6 b.b17x3 22.90265.22YesNo785
51b.1x15 g.l1x4 13.48722.50667NoYes478
52b.l26x5 g.ctx4 24.28485.03YesNo057
53g.ctx3 g.ctx4 23.93212.68333YesNo097
54b.l26x5 g.ctx16 12.48232.49YesYes058
55g.ctx3 g.ctx5 12.37932.71333YesNo2299
56b.b27x1 g.ctx5 12.0192.48333NoNo069
57b.b23x3 b.b27x1 10.92863.97333NoNo076
58b.b2x5 b.l26x1 12.698110.92YesYes677
59b.l26x3 b.l26x5 12.00725.08333NoYes075
60b.b16x5 b.b17x4 10.46733.23667YesYes455
61b.l23x1 b.l25x6 20.728617.47YesNo068
62b.l21x7 b.l23x1 19.71715.18667NoYes056
63b.l21x7 b.l23x2 19.46676.22333NoNo058
64b.b23x6 b.l23x2 18.47474.21667YesNo078
65b.b23x6 b.l21x9 16.016212.4933YesNo1176
66b.b20x3 b.b21x7 14.80063.58333NoYes085
672x38 4x42 26.89385.23NoYes057
682x39 3x46 18.4142.91667YesYes389
693x46 7x53 55.25355.24YesYes399
703x43 7x53 70.0487.81667YesYes399
713x43 6x44 68.55682.44YesNo099
726x44 6x48 67.45275.68NoYes098
736x48 Lig 62.71482.33333YesYes280
742x42 3x49 19.41659.32667YesYes089
752x42 3x46 37.43824.60333YesYes089
762x42 4x42 20.00128.74333YesYes087
773x50 7x53 19.51053.09YesYes399
78Lig NT.Y22 10.82572.54333YesYes209
793x28 Lig 13.78563.03667YesYes260
803x29 Lig 10.23555.32YesYes250
81E2.L189 Lig 10.35162.30333YesYes250
823x25 E2.L191 11.863412.1467YesNo294
83E2.L191 NT.H21 11.07549.85667NoYes247
84b.l26x1 b.l26x3 12.16815.78333YesNo677
85b.b20x3 b.l21x9 15.01196.55NoNo1186
86b.l4x1 g.ctx16 14.28285.28NoYes658
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
LigNT.Y222.543332YesYes0001
LigNT.R316.286672YesNo0001
2x60Lig9.152YesYes6010
2x64Lig7.883332YesYes5010
E1x50Lig2.826672NoYes5010
3x28Lig3.036672YesYes6010
3x29Lig5.322YesYes5010
3x32Lig5.422NoYes6010
3x33Lig6.316672YesYes5010
3x36Lig10.83332NoYes6010
E2.L189Lig2.303332YesYes0010
5x47Lig3.982NoYes7010
6x51Lig2.493332NoYes6010
6x52Lig3.563332YesYes6010
6x55Lig5.963332NoYes6010
7x38Lig3.352NoYes5010
NT.K27NT.Y224.376670NoYes0021
E1x50NT.Y223.746672NoYes5011
E2.P190NT.Y2211.130NoYes0021
E1x501NT.R312.852YesNo7021
2x573x328.382YesNo6621
2x577x383.626672YesNo6521
2x602x642.982YesYes6511
2x603x286.432YesYes6611
2x63E1x522.353332NoYes4622
2x633x282.482NoYes4621
2x643x286.152YesYes5611
3x28E1x522.426672YesYes6612
3x253x2882YesYes9621
3x253x2913.452YesYes9521
3x283x293.876672YesYes6511
3x29E2.L1895.303332YesYes5011
3x29E2.Y1925.613332YesYes5012
3x335x399.283332YesYes5612
3x335x432.793332YesNo5611
3x366x483.416672NoYes6811
3x406x484.850NoYes7821
E2.I188E2.L1892.853332YesYes0021
E2.L189E2.Y1927.816672YesYes0012
5x39E2.Y1922.313332YesYes6022
5x395x435.376672YesNo6621
5x446x524.186670NoYes4621
5x446x552.510NoNo4621
5x476x486.013332NoYes7811
5x476x5227.152NoYes7611
6x446x485.680NoYes9821
6x486x523.673332YesYes8611
6x487x413.892YesNo8712
6x487x4511.32YesNo8912
6x516x557.713332NoNo6611
6x517x382.382NoNo6511
E1x501NT.Y223.442YesYes7021
2x572x602.326672YesYes6621
2x603x324.673332YesNo6611
E1x50E1x5015.622NoYes5712
5x43Lig2.393332NoYes6010
6x48Lig2.333332YesYes8010
3x37Lig2.220NoYes5010
2x533x361.580NoNo8621
3x374x531.30NoNo5812
2x64E1x471.236672YesNo5612
3x303x331.006670NoYes6521

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
83.33Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
78.95Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
78.95Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
77.78Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
77.78Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
77.78Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
77.78Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
75.00Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
72.22Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
66.67Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
66.67Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
66.67Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
66.67Consensuslpl_onOrthosteric Ligands1p_on lpa_on
66.67Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
65.00Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
65.00Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
65.00Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
63.16Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
61.11Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
61.11Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
60.87Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
60.00Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
60.00Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
60.00Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
60.00Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
60.00Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
59.09Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
57.89Single7C4SS1P7C4S-S1P3-S1P
57.89Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
57.14Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
57.14Single5X93K-87945X93-ETB-K-8794
57.14Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
57.14Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
55.56Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
55.00Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
55.00Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
55.00Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
55.00Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
55.00Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
55.00Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
55.00Single8E0GBU728E0G-μ-BU72
55.00Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
55.00Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
55.00Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
54.55Single5ZTYAM102575ZTY-CB2-AM10257
54.55Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
54.55Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
54.17Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
54.17Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
53.85Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
52.63Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
52.63Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
52.63Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
52.63Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
52.63Single9CHXS-Carazolol9CHX-β2-S-Carazolol
52.63Consensus5ht5_onOrthosteric Ligand5ht5a_on
52.63Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
52.38Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
52.38Single7YITNalfurafine7YIT-κ-Nalfurafine
52.38Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
52.38Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
52.38Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
52.38Consensusalpha1_offOrthosteric Ligandalpha1a_off
52.38Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
52.38Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
52.38Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
52.17Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
52.17Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
50.00Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
50.00Single5C1MBU725C1M-μ-BU72
50.00Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
50.00Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
50.00Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
50.00Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
50.00Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
50.00Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
50.00Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
50.00Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
50.00Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
50.00Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
50.00Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
50.00Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
50.00Single8JXSPF-61428JXS-D1-PF-6142
50.00Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
50.00Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
50.00Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
50.00Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
50.00Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
50.00Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
50.00Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
50.00Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
50.00Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
50.00Consensusendothelin_offOrthosteric Ligandetb_off
50.00Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
50.00Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
50.00Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
47.83Single4UG2CGS216804UG2-A2A-CGS21680
47.83Single7SK9CCX6627SK9-ACKR3-CCX662
47.83Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
47.83Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
47.83Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
47.83Single8X5YAstemizole8X5Y-H1-Astemizole
47.62Single2YDVNECA2YDV-A2A-NECA
47.62Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
47.62Single4DJHJDTic4DJH-κ-JDTic
47.62Single4UHRCGS216804UHR-A2A-CGS21680
47.62Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
47.62Single5G53NECA5G53-A2A-NECA-Gs
47.62Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
47.62Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
47.62Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
47.62Single6H7JIsoprenaline6H7J-β1-Isoprenaline
47.62Single6TQ7SB-3348676TQ7-OX1-SB-334867
47.62Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
47.62Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
47.62Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
47.62Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
47.62Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
47.62Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
47.62Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
47.62Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
47.62Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
47.62Single8XVLZibotentan8XVL-ETA-Zibotentan
47.62Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
47.62Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
47.62Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
47.62Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
47.62Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
47.62Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
47.62Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
47.62Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
47.62Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
47.62Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
47.37Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
47.37Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
47.37Single6TPGEMPA6TPG-OX2-EMPA
47.37Single6TPNHTL66416TPN-OX2-HTL6641
47.37Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
47.37Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
47.37Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
47.37Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
47.37Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
47.37Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
47.37Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
47.37Consensusalpha1_onOrthosteric Ligandalpha1a_on
47.37Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
47.37Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
47.37Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
47.37Consensusopsins_offOrthosteric Ligandrhodopsin_off
47.37Consensussensory_offOrthosteric Ligandopsins_off
46.43Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
46.15Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
45.83Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
45.83Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
45.83Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
45.83Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
45.83Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
45.45Single3D4STimolol3D4S-β2-Timolol
45.45Single4AMIBucindolol4AMI-β1-Bucindolol
45.45Single4LDEBI1671074LDE-β2-BI167107
45.45Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
45.45Single6ZG4HTL00099366ZG4-M1-HTL0009936
45.45Single7DFPSpiperone7DFP-D2-Spiperone
45.45Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
45.45Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
45.45Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
45.45Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
45.45Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
45.45Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
45.45Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
45.45Single9DGIZ85267113509DGI-CB1-Z8526711350
45.45Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
45.45Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
45.45Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
45.45Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
45.45Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
45.45Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
45.45Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
45.45Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
45.45Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
45.45Consensuslpa_offOrthosteric Ligandlpa1_off
45.45Consensuslpl_offOrthosteric Ligands1p_off lpa_off
45.00Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
45.00Single2Y04Salbutamol2Y04-β1-Salbutamol
45.00Single3NY8ICI118-5513NY8-β2-ICI118-551
45.00Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
45.00Single4GBRS-Carazolol4GBR-β2-S-Carazolol
45.00Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
45.00Single6DRXLisuride6DRX-5-HT2B-Lisuride
45.00Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
45.00Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
45.00Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
45.00Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
45.00Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
45.00Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
45.00Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
45.00Single7UL4Alvimopan7UL4-μ-Alvimopan
45.00Single7WC7Lisuride7WC7-5-HT2A-Lisuride
45.00Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
45.00Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
45.00Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
45.00Single8JXRLSD8JXR-D1-LSD
45.00Single8T1WCVN4248T1W-GPR6-CVN424
45.00Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
45.00Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
45.00Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
45.00Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
45.00Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
45.00Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
45.00Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
45.00Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
45.00Consensusalpha2_onOrthosteric Ligandalpha2b_on
45.00Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
45.00Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
45.00Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
45.00Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
45.00Consensusdopamine_offOrthosteric Ligandd2_off d3_off
45.00Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
45.00Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
44.44Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
44.44Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
44.44Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
44.44Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
44.44Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
44.00Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
44.00Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
43.48Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
43.48Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
43.48Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
43.48Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
43.48Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
43.48Single7UM4AS26747237UM4-5-HT5A-AS2674723
43.48Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
43.48Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
43.48Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
43.48Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
43.48Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
43.48Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
43.48Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
43.48Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
43.48Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
43.48Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
43.48Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
43.33Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
43.33Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
43.33Consensusbombesin_onOrthosteric Ligandbb2_on
43.33Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
43.33Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
42.86Single2RH1S-Carazolol2RH1-β2-S-Carazolol
42.86Single2Y03Isoprenaline2Y03-β1-Isoprenaline
42.86Single2YCWS-Carazolol2YCW-β1-S-Carazolol
42.86Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
42.86Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
42.86Single5D6LS-Carazolol5D6L-β2-S-Carazolol
42.86Single5JQHS-Carazolol5JQH-β2-S-Carazolol
42.86Single5TVNLSD5TVN-5-HT2B-LSD
42.86Single5WQCEMPA5WQC-OX2-EMPA
42.86Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
42.86Single5XPRBosentan5XPR-ETB-Bosentan
42.86Single6E67BI1671076E67-β2-BI167107-Gs(CT)
42.86Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
42.86Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
42.86Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
42.86Single6TP6Filorexant6TP6-OX1-Filorexant
42.86Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
42.86Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
42.86Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
42.86Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
42.86Single7WC6LSD7WC6-5-HT2A-LSD
42.86Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
42.86Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
42.86Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
42.86Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
42.86Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.86Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.86Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
42.86Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
42.86Single8TF5Oleic acid8TF5-GPR6-Oleic acid
42.86Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
42.86Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
42.86Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
42.86Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
42.86Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
42.86Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
42.86Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
42.86Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
42.86Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
42.86Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
42.86Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
42.86Consensusamine_offonOrthosteric Ligandamine_off amine_on
42.86Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
42.86Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
42.86Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
42.86Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
42.86Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
42.86Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
42.86Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
42.86Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
42.86Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
42.86Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
42.86Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
42.86Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
42.86Consensustrace-amine_onOrthosteric Ligandta1_on
42.31Single6PT2KGCHM076PT2-δ-KGCHM07
42.31Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
42.31Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
42.31Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
42.31Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
42.11Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
42.11Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
42.11Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
42.11Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
42.11Single6AKXA4R6AKX-CCR5-A4R
42.11Single6B73MP11046B73-κ-MP1104
42.11Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
42.11Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
42.11Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
42.11Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
42.11Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
42.11Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
42.11Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
42.11Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
42.11Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
42.11Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
42.11Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
42.11Consensusorexin_offOrthosteric Ligandox2_off ox1_off
42.11Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
42.11Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
42.11Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
41.67Single3NY9ICI118-5513NY9-β2-ICI118-551
41.67Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
41.67Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
41.67Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
41.67Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
41.67Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
41.67Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
41.38Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
41.38Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
41.38Single9KDFRES-701-39KDF-ETB-RES-701-3
41.38Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
41.38Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
41.38Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
40.91Single3P0GBI1671073P0G-β2-BI167107
40.91Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
40.91Single4U15Tiotropium4U15-M3-Tiotropium
40.91Single5D5AS-Carazolol5D5A-β2-S-Carazolol
40.91Single5D5BS-Carazolol5D5B-β2-S-Carazolol
40.91Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
40.91Single6J21Aprepitant6J21-NK1-Aprepitant
40.91Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
40.91Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
40.91Single6OL9Tiotropium6OL9-M5-Tiotropium
40.91Single6WGTLSD6WGT-5-HT2A-LSD
40.91Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
40.91Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
40.91Single7FEECP559407FEE-CB1-CP55940-ZCZ011
40.91Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
40.91Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
40.91Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
40.91Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
40.91Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
40.91Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
40.91Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
40.91Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
40.91Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
40.91Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
40.91Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
40.91Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
40.91Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
40.91Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
40.91Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
40.91Single9BJKNaloxone9BJK-μ-Naloxone-NAM
40.91Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
40.91Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
40.91Consensusa2_onOrthosteric Liganda2b_on
40.91Consensusa2_on_gpOrthosteric Liganda2b_on_gp
40.91Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
40.91Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
40.91Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
40.91Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
40.91Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
40.91Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
40.91Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
40.91Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
40.91Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
40.91Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
40.91Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
40.91Consensuslpa_onOrthosteric Ligandlpa1_on
40.91Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
40.91Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
40.91Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
40.74Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
40.74Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
40.74Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
40.74Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
40.00Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
40.00Single3RZECidoxepin3RZE-H1-Cidoxepin
40.00Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
40.00Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
40.00Single4MBSMaraviroc4MBS-CCR5-Maraviroc
40.00Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
40.00Single4ZJCSB-6740424ZJC-OX1-SB-674042
40.00Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
40.00Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
40.00Single6IQLL7458706IQL-D4-L745870
40.00Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
40.00Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
40.00Single6PS0S-Carazolol6PS0-β2-S-Carazolol
40.00Single6PS4ICI118-5516PS4-β2-ICI118-551
40.00Single6PS5S-Propranolol6PS5-β2-S-Propranolol
40.00Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
40.00Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
40.00Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
40.00Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
40.00Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
40.00Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
40.00Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
40.00Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
40.00Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
40.00Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
40.00Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
40.00Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
40.00Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
40.00Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
40.00Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
40.00Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
40.00Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
40.00Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
40.00Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
40.00Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
40.00Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
40.00Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
40.00Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
40.00Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
40.00Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
40.00Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
40.00Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
40.00Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
40.00Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
40.00Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
40.00Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
40.00Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
40.00Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
40.00Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
40.00Single8WDTphotoNECA8WDT-A2A-photoNECA
40.00Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
40.00Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
40.00Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
40.00Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
40.00Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
40.00Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
40.00Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
40.00Single9M4TSilodosin9M4T-Alpha1A-Silodosin
40.00Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
40.00Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
40.00Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
40.00Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
40.00Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
40.00Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
39.29Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
39.29Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
39.29Single8ZRTET-18ZRT-ETB-ET-1
39.13Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
39.13Single4RWADIPP-NH24RWA-δ-DIPP-NH2
39.13Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
39.13Single5CXVTiotropium5CXV-M1-Tiotropium
39.13Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
39.13Single6CM4Risperidone6CM4-D2-Risperidone
39.13Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
39.13Single6KQICP559406KQI-CB1-CP55940-Org27569
39.13Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
39.13Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
39.13Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
39.13Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
39.13Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
39.13Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
39.13Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
39.13Single8JJ8Formoterol8JJ8-β2-Formoterol
39.13Single8JJLOlodaterol8JJL-β2-Olodaterol
39.13Single8JWY2-1188JWY-A2A-2-118
39.13Single8JWZAB9288JWZ-A2A-AB928-Na
39.13Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
39.13Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
39.13Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
39.13Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
39.13Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
39.13Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
39.13Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
39.13Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
39.13Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
39.13Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
39.13Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
39.13Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
39.13Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
39.13Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
39.13Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
39.13Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
39.13Consensusorexin_onOrthosteric Ligandox2_on
38.89Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
38.89Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
38.46Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
38.46Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
38.46Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
38.46Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
38.46Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
38.46Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
38.10Single2Y02Carmoterol2Y02-β1-Carmoterol
38.10Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
38.10Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
38.10Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
38.10Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
38.10Single4EJ4Naltrindole4EJ4-δ-Naltrindole
38.10Single4MQSIperoxo4MQS-M2-Iperoxo
38.10Single4U14Tiotropium4U14-M3-Tiotropium
38.10Single5DHGC-355DHG-NOP-C-35
38.10Single5DHHSB-6121115DHH-NOP-SB-612111
38.10Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
38.10Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
38.10Single6H7MSalbutamol6H7M-β1-Salbutamol
38.10Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
38.10Single6TOTLemborexant6TOT-OX1-Lemborexant
38.10Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
38.10Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
38.10Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
38.10Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
38.10Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
38.10Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
38.10Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
38.10Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
38.10Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
38.10Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
38.10Single7V3ZCP559407V3Z-CB1-CP55940
38.10Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
38.10Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
38.10Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
38.10Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
38.10Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
38.10Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
38.10Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
38.10Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
38.10Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
38.10Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
38.10Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
38.10Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.10Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.10Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.10Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.10Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.10Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.10Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.10Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.10Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.10Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.10Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
38.10Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
38.10Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
38.10Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
38.10Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
38.10Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
38.10Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
38.10Single8JJOAlprenolol8JJO-β2-Alprenolol
38.10Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
38.10Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
38.10Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
38.10Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.10Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.10Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.10Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.10Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.10Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
38.10Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
38.10Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
38.10Single8X63Mepyramine8X63-H1-Mepyramine
38.10Single8X64Desloratadine8X64-H1-Desloratadine
38.10Single9AS1DMT9AS1-5-HT2A-DMT
38.10Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
38.10Single9JEAAtropine9JEA-M1-Atropine
38.10Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
38.10Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
38.10Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
38.10Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
38.10Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
38.10Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
38.10Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
38.10Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
38.10Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
38.10Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
38.10Consensusblt_onOrthosteric Ligandblt1_on
38.10Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
38.10Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
38.10Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
38.10Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
38.10Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
38.10Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
38.10Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
38.10Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
38.10Consensushistamine_offOrthosteric Ligandh1_off
38.10Consensusleukotriene_onOrthosteric Ligandblt_on
38.10Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
37.50Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
37.50Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
37.50Single6H7LDobutamine6H7L-β1-Dobutamine
37.50Single6IBLArformoterol6IBL-β1-Arformoterol
37.50Single6K1QIRL25006K1Q-ETB-IRL2500
37.50Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
37.50Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
37.50Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
37.50Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
37.50Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
37.50Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
37.50Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
37.50Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
37.50Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
37.50Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
37.50Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
37.50Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
37.50Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
37.50Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
37.50Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
37.50Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
37.50Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
37.04Single5WF5UK-4320975WF5-A2A-UK-432097
37.04Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
37.04Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
37.04Consensusangiotensin_onOrthosteric Ligandat1_on
37.04Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
37.04Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
36.84Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
36.84Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
36.84Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
36.84Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
36.84Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
36.84Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
36.84Single6TP4ACT-4622066TP4-OX1-ACT-462206
36.84Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
36.84Single7SRQLSD7SRQ-5-HT2B-LSD
36.84Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
36.84Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
36.84Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
36.84Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
36.84Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
36.84Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
36.84Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
36.84Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
36.84Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
36.67Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
36.36Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
36.36Single5WIUNemonapride5WIU-D4-Nemonapride
36.36Single5WIVNemonapride5WIV-D4-Nemonapride-Na
36.36Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
36.36Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
36.36Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
36.36Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
36.36Single6PS6Timolol6PS6-β2-Timolol
36.36Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
36.36Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
36.36Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
36.36Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
36.36Single7W41PD1762527W41-BB2-PD176252
36.36Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
36.36Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
36.36Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
36.36Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
36.36Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
36.36Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
36.36Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.36Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
36.36Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
36.36Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.36Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.36Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
36.36Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
36.36Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
36.36Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
36.36Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
36.36Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
36.36Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
36.36Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
36.36Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
36.36Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
36.36Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
36.36Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
36.36Consensusbombesin_offOrthosteric Ligandbb2_off
36.36Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
36.36Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
36.36Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
36.36Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
36.36Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
36.36Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
36.36Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
36.36Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
36.00Single6PT3DPI-2876PT3-δ-DPI-287
36.00Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
36.00Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
36.00Single8QJ2pN1628QJ2-MC4-pN162-Gs
36.00Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
36.00Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
36.00Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
36.00Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
36.00Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
35.71Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
35.71Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
35.71Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
35.71Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
35.71Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
35.71Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
35.71Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
35.71Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
35.71Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
35.71Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
35.48Single6IGLIRL16206IGL-ETB-IRL1620
35.48Consensusendothelin_onOrthosteric Ligandetb_on eta_on
35.00Single5WS3EMPA5WS3-OX2-EMPA
35.00Single6AKYMaraviroc6AKY-CCR5-Maraviroc
35.00Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
35.00Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
35.00Single6TODEMPA6TOD-OX1-EMPA-Na
35.00Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
35.00Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
35.00Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
35.00Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
35.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
35.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
35.00Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
35.00Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
35.00Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
35.00Single7XRRLemborexant7XRR-OX2-Lemborexant
35.00Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
35.00Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
35.00Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
35.00Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
35.00Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
35.00Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
35.00Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
35.00Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
35.00Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
35.00Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
35.00Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
35.00Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
35.00Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
35.00Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
35.00Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
35.00Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
35.00Single8Y0HVUF114188Y0H-CXCR3-VUF11418
35.00Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
35.00Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
35.00Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
35.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
35.00Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
35.00Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
35.00Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
35.00Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
35.00Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
35.00Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
35.00Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
35.00Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
35.00Consensusalpha2_offOrthosteric Ligandalpha2c_off
35.00Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
35.00Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
35.00Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
35.00Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
35.00Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
35.00Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
34.78Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
34.78Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
34.78Single5V54Methiothepin5V54-5-HT1B-Methiothepin
34.78Single5XR8AM8415XR8-CB1-AM841
34.78Single5XRAAM115425XRA-CB1-AM11542
34.78Single6E59L-7607356E59-NK1-L-760735
34.78Single6J20Aprepitant6J20-NK1-Aprepitant
34.78Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
34.78Single7B6WCyclazosin7B6W-α1b-Cyclazosin
34.78Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
34.78Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
34.78Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
34.78Single8EA0Iperoxo8EA0-M3-Iperoxo
34.78Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
34.78Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
34.78Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
34.78Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
34.78Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
34.78Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
34.78Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
34.78Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
34.78Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
34.78Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
34.78Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
34.78Consensus5ht1_offOrthosteric Ligand5ht1b_off
34.78Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
34.78Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
34.78Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
34.78Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
34.78Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
34.78Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
34.62Single4IARErgotamine4IAR-5-HT1B-Ergotamine
34.62Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
34.62Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
34.62Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
34.62Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
34.62Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
34.62Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
34.62Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
34.62Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
34.62Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
34.62Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
34.48Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
34.48Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
34.48Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
34.48Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
34.48Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
34.38Single5GLHEndothelin-15GLH-ETB-Endothelin-1
34.38Single6IGKEndothelin-36IGK-ETB-Endothelin-3
34.38Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
33.33Single2YDOAdenosine2YDO-A2A-Adenosine
33.33Single3QAKUK-4320973QAK-A2A-UK-432097
33.33Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
33.33Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
33.33Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
33.33Single6A93Risperidone6A93-5-HT2A-Risperidone
33.33Single6A94Zotepine6A94-5-HT2A-Zotepine
33.33Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
33.33Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
33.33Single6HLOAprepitant6HLO-NK1-Aprepitant
33.33Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
33.33Single6KUXRS-799486KUX-α2a-RS-79948
33.33Single6MXTSalmeterol6MXT-β2-Salmeterol
33.33Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
33.33Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
33.33Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
33.33Single6TP3Nemorexant6TP3-OX1-Nemorexant
33.33Single6V9SGTPL114036V9S-OX1-GTPL11403
33.33Single6VI4JDTic6VI4-κ-JDTic
33.33Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
33.33Single6ZG9GSK10347026ZG9-M1-GSK1034702
33.33Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
33.33Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
33.33Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
33.33Single7F61PF-036547467F61-H3-PF-03654746
33.33Single7UL3Famotidine7UL3-H2-Famotidine
33.33Single7VODCariprazine7VOD-5-HT2A-Cariprazine
33.33Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
33.33Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
33.33Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
33.33Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
33.33Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
33.33Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
33.33Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
33.33Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
33.33Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
33.33Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
33.33Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
33.33Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
33.33Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
33.33Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
33.33Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
33.33Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
33.33Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
33.33Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
33.33Single8IHKAcifran8IHK-HCA3-Acifran
33.33Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
33.33Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
33.33Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
33.33Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
33.33Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
33.33Single8K5CAcipimox8K5C-HCA2-Acipimox
33.33Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
33.33Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
33.33Single8RLNLUF58348RLN-A2A-LUF5834
33.33Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
33.33Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
33.33Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
33.33Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
33.33Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
33.33Single8XYIVUF106618XYI-CXCR3-VUF10661
33.33Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
33.33Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
33.33Single9ARXSerotonin9ARX-5-HT2A-Serotonin
33.33Single9AS3LSD9AS3-5-HT2A-LSD
33.33Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single9AS5Mescaline9AS5-5-HT2A-Mescaline
33.33Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single9CHUNoradrenaline9CHU-β2-Noradrenaline
33.33Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
33.33Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
33.33Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
33.33Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
33.33Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
33.33Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
33.33Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
33.33Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
33.33Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
33.33Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
33.33Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
33.33Consensushca_onOrthosteric Ligandhca2_on
33.33Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
33.33Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
33.33Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
33.33Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
32.35Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
32.26Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
32.26Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
32.26Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
32.14Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
32.14Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
32.14Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
32.14Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
32.14Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
32.14Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
32.00Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
32.00Single7EZCUKA7EZC-A2A-UKA
32.00Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
32.00Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
32.00Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
32.00Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
32.00Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
32.00Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
32.00Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
31.82Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
31.82Single2Y01Dobutamine2Y01-β1-Dobutamine
31.82Single4DAJTiotropium4DAJ-M3-Tiotropium
31.82Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
31.82Single4QKX35V4QKX-β2-35V
31.82Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
31.82Single5TGZAM65385TGZ-CB1-AM6538
31.82Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
31.82Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
31.82Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
31.82Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
31.82Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
31.82Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
31.82Single6PS1Timolol6PS1-β2-Timolol
31.82Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.82Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
31.82Single7BU7BI1671077BU7-β1-BI167107
31.82Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
31.82Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
31.82Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
31.82Single8CU6LJ-45178CU6-A2A-LJ-4517
31.82Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
31.82Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
31.82Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
31.82Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
31.82Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
31.82Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
31.82Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
31.82Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
31.82Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.82Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.82Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
31.82Single9H37A1IR09H37-A2A-A1IR0-Na
31.82Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
31.82Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
31.82Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
31.82Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
31.82Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
31.82Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
31.82Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
31.82Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
31.82Consensushca_on_gpOrthosteric Ligandhca2_on_gp
31.82Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
31.82Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
31.58Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
31.58Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
31.58Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
31.58Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
31.58Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
31.58Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
31.58Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
31.58Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
31.58Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
31.58Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
31.58Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
31.58Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
31.58Consensus5ht2_onOrthosteric Ligand5ht2b_on
31.58Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.25Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
31.25Single8IY6Endothelin-18IY6-ETB-Endothelin-1
31.25Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
31.25Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
31.03Single6JODAngiotensin II6JOD-AT2-Angiotensin II
31.03Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
31.03Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
31.03Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
31.03Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
31.03Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
31.03Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
31.03Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
31.03Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
31.03Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
31.03Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
31.03Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
31.03Consensusvasop-oxy_onOrthosteric Ligandv2_on
31.03Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
30.77Single5WF6UK-4320975WF6-A2A-UK-432097
30.77Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
30.77Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
30.77Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
30.77Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
30.77Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
30.77Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
30.77Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
30.77Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
30.77Single9IPYJR14a9IPY-C3aB-JR14a
30.77Single9JF4PD1683689JF4-BB1-PD168368
30.77Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
30.77Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
30.77Consensuskisspeptin_onOrthosteric Ligandkiss1_on
30.56Consensuspth_onOrthosteric Ligandpth1_on pth2_on
30.43Single2Y00Dobutamine2Y00-β1-Dobutamine
30.43Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
30.43Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
30.43Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
30.43Single6HLPNetupitant6HLP-NK1-Netupitant
30.43Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
30.43Single6LUQHaloperidol6LUQ-D2-Haloperidol
30.43Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
30.43Single7C61Ergotamine7C61-5-HT1B-Ergotamine
30.43Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
30.43Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
30.43Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
30.43Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
30.43Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.43Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
30.43Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
30.43Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
30.43Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
30.43Single8S4DCMF-0198S4D-Apelin-CMF-019
30.43Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
30.43Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
30.43Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
30.43Single8ZMFA1L108ZMF-5-HT2C-A1L10
30.43Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
30.43Single9EHSLUF76029EHS-A3A-LUF7602
30.43Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
30.43Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
30.43Single9HAPTolvaptan9HAP-V2-Tolvaptan
30.43Consensusa3_on_gpOrthosteric Liganda3a_on_gp
30.43Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
30.43Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
30.43Consensusadenosine_offOrthosteric Liganda1_off a2_off
30.43Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
30.43Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
30.43Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
30.43Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
30.30Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
30.00Single3PBLEticlopride3PBL-D3-Eticlopride
30.00Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
30.00Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
30.00Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
30.00Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
30.00Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
30.00Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.00Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
30.00Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
30.00Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.00Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
30.00Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
30.00Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
30.00Single8K5BNiacin8K5B-HCA2-Niacin
30.00Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
30.00Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
30.00Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.00Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
30.00Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
30.00Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
30.00Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
30.00Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
30.00Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
30.00Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
30.00Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
30.00Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
29.73Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
29.73Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
29.63Single4XT1Fractalkine4XT1-US28-Fractalkine
29.63Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
29.63Single7F8XNN90567F8X-CCKA-NN9056
29.63Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
29.63Single8IEBA1LYA8IEB-GPR156-A1LYA
29.63Single8WKYPG-9348WKY-MC4-PG-934
29.63Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
29.63Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
29.63Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
29.63Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
29.63Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
29.63Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
29.17Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
29.17Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
29.17Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
29.17Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
29.17Single7TUYGSK682753A7TUY-GPR183-GSK682753A
29.17Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
29.17Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
29.17Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
29.17Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
29.17Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
29.17Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
29.17Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
29.17Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
29.17Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
29.17Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
29.17Single8ZWFJR14a8ZWF-C3aB-JR14a
29.17Single9AS9RS130-1809AS9-5-HT2A-RS130-180
29.17Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
29.17Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
29.17Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
29.17Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
29.17Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
29.17Consensustachykinin_offOrthosteric Ligandnk1_off
29.03Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
29.03Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
29.03Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
29.03Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
29.03Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
29.03Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
29.03Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
29.03Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
29.03Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
28.95Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
28.57Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
28.57Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
28.57Single4S0VSuvorexant4S0V-OX2-Suvorexant
28.57Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
28.57Single6DS0Ly2660976DS0-5-HT2B-Ly266097
28.57Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
28.57Single6ME2Ramelteon6ME2-MT1-Ramelteon
28.57Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
28.57Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
28.57Single6TPJSuvorexant6TPJ-OX2-Suvorexant
28.57Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
28.57Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
28.57Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
28.57Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
28.57Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
28.57Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
28.57Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
28.57Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
28.57Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
28.57Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
28.57Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
28.57Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
28.57Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
28.57Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
28.57Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
28.57Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.57Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
28.57Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
28.57Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
28.57Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
28.57Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
28.57Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
28.57Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
28.57Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
28.57Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
28.57Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
28.57Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
28.57Single9H2XA1IR19H2X-A2A-A1IR1-Na
28.57Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
28.57Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
28.57Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
28.57Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
28.57Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
28.57Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
28.57Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
28.57Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
28.57Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
28.57Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
28.57Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
28.57Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
28.57Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
28.57Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
28.57Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
28.57Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
28.57Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
28.57Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
28.12Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
28.12Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
28.12Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
28.12Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
28.12Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
28.12Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
28.00Single7K15MKD0467K15-BLT1-MKD046-Na
28.00Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
28.00Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
28.00Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
28.00Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
28.00Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
28.00Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
28.00Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
28.00Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
28.00Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
28.00Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
27.78Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
27.78Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.78Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
27.59Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
27.59Single6W25SHU91196W25-MC4-SHU9119-Ca
27.59Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
27.59Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
27.59Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
27.59Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
27.59Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
27.59Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
27.59Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
27.59Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
27.59Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
27.59Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
27.59Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
27.50Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
27.27Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
27.27Single5IU7Q274563465IU7-A2A-Q27456346-Na
27.27Single5JTBZM-2413855JTB-A2A-ZM-241385
27.27Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
27.27Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
27.27Single6AQFZM-2413856AQF-A2A-ZM-241385
27.27Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
27.27Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
27.27Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
27.27Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
27.27Single6TPKRetosiban6TPK-OT-Retosiban
27.27Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
27.27Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
27.27Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
27.27Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
27.27Single7T32ZM-2413857T32-A2A-ZM-241385
27.27Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
27.27Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
27.27Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
27.27Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
27.27Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
27.27Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.27Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
27.27Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
27.27Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
27.27Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
27.27Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
27.27Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
27.27Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
27.27Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
27.27Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
27.27Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
27.27Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
27.27Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
27.27Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
27.27Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
27.27Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
27.27Consensusa2_offOrthosteric Liganda2a_off
27.27Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
27.27Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
27.27Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
27.27Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
27.27Consensusbradykinin_onOrthosteric Ligandbk2_on
27.27Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
27.27Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
27.27Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
27.27Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
27.27Consensusvasop-oxy_offOrthosteric Ligandot_off
26.92Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
26.92Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
26.92Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
26.92Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.92Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
26.92Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
26.92Single8XVJMacitentan8XVJ-ETA-Macitentan
26.92Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
26.92Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
26.92Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
26.92Consensuscck_onOrthosteric Ligandccka_on cckb_on
26.92Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
26.92Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
26.92Consensusprostanoid_offOrthosteric Ligandep_off dp_off
26.67Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
26.67Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
26.67Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
26.67Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
26.67Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
26.67Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
26.67Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
26.67Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
26.67Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
26.67Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
26.47Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
26.47Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
26.47Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
26.47Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
26.47Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
26.47Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
26.47Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
26.47Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
26.32Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
26.32Single3OE8IT1t3OE8-CXCR4-IT1t
26.32Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
26.32Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
26.32Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.32Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
26.32Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
26.32Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
26.09Single3EMLZM-2413853EML-A2A-ZM-241385
26.09Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
26.09Single4YAYZD-71554YAY-AT1-ZD-7155
26.09Single5DSGTiotropium5DSG-M4-Tiotropium
26.09Single5IU8Q274563475IU8-A2A-Q27456347-Na
26.09Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
26.09Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
26.09Single5UIGCmpd-15UIG-A2A-Cmpd-1
26.09Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
26.09Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
26.09Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
26.09Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
26.09Single6S0LZM-2413856S0L-A2A-ZM-241385
26.09Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
26.09Single7F83PF-051904577F83-Ghrelin-PF-05190457
26.09Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
26.09Single7PYRPSB-21157PYR-A2A-PSB-2115
26.09Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
26.09Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
26.09Single7YXAONO-54306087YXA-S1P5-ONO-5430608
26.09Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
26.09Single8K5DGSK2560738K5D-HCA2-GSK256073
26.09Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
26.09Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
26.09Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
26.09Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
26.09Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
26.09Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
26.09Single9IYAONO-97105319IYA-GPR55-ONO-9710531
26.09Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
26.09Consensusa3_onOrthosteric Liganda3a_on
26.09Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
26.09Consensuscck_offOrthosteric Ligandccka_off
26.09Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
26.09Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
26.09Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
26.09Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
26.09Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
25.93Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
25.93Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.93Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
25.93Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
25.93Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
25.81Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
25.81Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
25.81Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
25.81Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
25.81Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
25.81Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
25.81Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
25.81Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
25.81Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
25.81Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
25.71Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
25.58Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
25.00Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
25.00Single3OE6IT1t3OE6-CXCR4-IT1t
25.00Single4XT3Fractalkine4XT3-US28-Fractalkine
25.00Single5IUAQ274563485IUA-A2A-Q27456348-Na
25.00Single5N2RPSB-365N2R-A2A-PSB-36-Na
25.00Single5N2SPSB365N2S-A1-PSB36
25.00Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
25.00Single6D26Fevipiprant6D26-DP2-Fevipiprant
25.00Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
25.00Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
25.00Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
25.00Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
25.00Single6S0QZM-2413856S0Q-A2A-ZM-241385
25.00Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
25.00Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
25.00Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
25.00Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
25.00Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
25.00Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
25.00Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
25.00Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
25.00Single7QA8Peptide7QA8-STE2-Peptide
25.00Single7QA8Peptide7QA8-STE2-Peptide
25.00Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
25.00Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
25.00Single7SINNPS-21437SIN-CaS-NPS-2143
25.00Single7SINNPS-21437SIN-CaS-NPS-2143
25.00Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
25.00Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
25.00Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
25.00Single7WC5Psilocin7WC5-5-HT2A-Psilocin
25.00Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
25.00Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
25.00Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
25.00Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
25.00Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8GNEKW-63568GNE-A2A-KW-6356-Na
25.00Single8IEIA1LYA8IEI-GPR156-A1LYA
25.00Single8IEIA1LYA8IEI-GPR156-A1LYA
25.00Single8IEPA1LYA8IEP-GPR156-A1LYA
25.00Single8IEPA1LYA8IEP-GPR156-A1LYA
25.00Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
25.00Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
25.00Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
25.00Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
25.00Single8QOTNanobody-E8QOT-μ-Nanobody-E
25.00Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
25.00Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
25.00Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
25.00Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
25.00Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
25.00Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
25.00Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
25.00Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
25.00Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
25.00Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
25.00Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
25.00Single9LRCHistamine9LRC-H4-Histamine
25.00Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
25.00Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
25.00Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
25.00Consensusblt_offOrthosteric Ligandblt1_off
25.00Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
25.00Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
25.00Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
25.00Consensusdp_offOrthosteric Liganddp2_off
25.00Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
25.00Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
25.00Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
25.00Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
25.00Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
25.00Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
25.00Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
25.00Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
25.00Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
24.32Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
24.32Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
24.24Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
24.24Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
24.24Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
24.24Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
24.24Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
24.24Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
24.24Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
24.24Consensusglp_onOrthosteric Ligandglp1_on glp2_on
24.24Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
24.24Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
24.14Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
24.14Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
24.14Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
24.14Single8IEBA1LYA8IEB-GPR156-A1LYA
24.14Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
24.14Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
24.14Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
24.14Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
24.14Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
24.14Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
24.00Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
24.00Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
24.00Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
24.00Single7PX4PSB-21137PX4-A2A-PSB-2113
24.00Single7R0CAVP7R0C-V2-AVP-Arrestin2
24.00Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
24.00Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
24.00Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
24.00Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
24.00Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
24.00Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
24.00Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
24.00Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
24.00Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
24.00Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
24.00Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
23.81Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
23.81Single3OE9IT1t3OE9-CXCR4-IT1t
23.81Single6HLLCP999946HLL-NK1-CP99994
23.81Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
23.81Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
23.81Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
23.81Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
23.81Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
23.81Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
23.81Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
23.81Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
23.81Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
23.81Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
23.81Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
23.81Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
23.81Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
23.81Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
23.81Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
23.81Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
23.81Single9AS7Psilocin9AS7-5-HT2A-Psilocin
23.81Single9B9Y7DY9B9Y-CB1-7DY
23.81Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
23.81Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
23.81Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
23.81Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
23.53Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
23.53Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
23.53Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
23.53Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
23.53Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
23.53Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
23.53Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
23.33Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
23.33Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.33Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
23.33Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
23.33Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
23.33Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
23.08Single4N4WSANT-14N4W-SMO-SANT-1
23.08Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
23.08Single5X33BIIL2605X33-BLT1-BIIL260
23.08Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
23.08Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
23.08Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
23.08Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.08Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
23.08Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
23.08Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
23.08Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
23.08Single9BJKNAM9BJK-μ-Naloxone-NAM
23.08Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
23.08Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
23.08Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.08Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
22.86Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
22.73Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
22.73Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
22.73Single3ODUIT1t3ODU-CXCR4-IT1t
22.73Single3PWHZM-2413853PWH-A2A-ZM-241385
22.73Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
22.73Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
22.73Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
22.73Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
22.73Single5ZKQABT-4915ZKQ-PAF-ABT-491
22.73Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
22.73Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
22.73Single6ME9Ramelteon6ME9-MT2-Ramelteon
22.73Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
22.73Single7BR3Elagolix7BR3-GnRH1-Elagolix
22.73Single7F8ULintitript7F8U-CCKA-Lintitript
22.73Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
22.73Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.73Single8GNGIstradefylline8GNG-A2A-Istradefylline
22.73Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
22.73Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
22.73Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
22.73Single8IWESpermidine8IWE-TA9-Spermidine
22.73Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
22.73Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
22.73Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
22.73Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
22.73Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
22.73Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
22.73Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
22.73Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
22.73Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
22.58Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
22.58Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
22.58Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
22.58Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
22.58Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
22.58Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
22.58Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
22.58Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
22.50Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
22.22Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
22.22Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
22.22Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
22.22Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
22.22Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
22.22Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
22.22Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
22.22Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
22.22Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
22.22Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
22.22Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
22.22Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
22.22Consensuschemerin_onOrthosteric Ligandcml1_on
21.88Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
21.88Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
21.88Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
21.88Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
21.88Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
21.88Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
21.88Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
21.88Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
21.88Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
21.88Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
21.74Single3REYXAC3REY-A2A-XAC
21.74Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
21.74Single5IUBQ274563445IUB-A2A-Q27456344-Na
21.74Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
21.74Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
21.74Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
21.74Single5UVIZM-2413855UVI-A2A-ZM-241385
21.74Single6MH8ZM-2413856MH8-A2A-ZM-241385
21.74Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
21.74Single7AROLUF58337ARO-A2A-LUF5833-Na
21.74Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
21.74Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
21.74Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.74Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
21.74Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
21.74Single9BA0A1AKN9BA0-CB1-A1AKN
21.74Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
21.74Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
21.74Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
21.74Consensusgrh_offOrthosteric Ligandgnrh1_off
21.74Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
21.74Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
21.62Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
21.62Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
21.43Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
21.43Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
21.43Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
21.43Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
21.43Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
21.43Single7XN9L-054,5227XN9-SST2-L-054,522
21.43Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
21.43Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
21.43Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
21.43Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
21.21Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
21.21Single6FJ3PTH6FJ3-PTH1-PTH
21.21Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
21.21Single7SK3CXCL127SK3-ACKR3-CXCL12
21.21Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
21.21Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
21.21Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
21.21Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
21.21Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
21.21Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
21.21Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
21.05Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
21.05Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
21.05Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
21.05Single7WC4Serotonin7WC4-5-HT2A-Serotonin
21.05Single8PWNTheophylline8PWN-A2A-Theophylline
21.05Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
21.05Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
20.83Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
20.83Single5UENDU1725UEN-A1-DU172
20.83Single6GPSMK08126GPS-CCR2-MK0812
20.83Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
20.83Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
20.83Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
20.83Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
20.83Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.83Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
20.83Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
20.83Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
20.83Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
20.83Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
20.69Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
20.69Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
20.69Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
20.69Single8KIGSHU91198KIG-MC3-SHU9119-Ca
20.69Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
20.69Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
20.69Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
20.69Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
20.69Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
20.69Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
20.59Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
20.59Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
20.59Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
20.59Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.59Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
20.59Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
20.59Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
20.59Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
20.59Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
20.51Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
20.00Single4NTJAZD12834NTJ-P2Y12-AZD1283
20.00Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
20.00Single5CGCHTL142425CGC-mGlu5-HTL14242
20.00Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
20.00Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
20.00Single6GPXMK08126GPX-CCR2-MK0812
20.00Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
20.00Single6TQ9SB-4081246TQ9-OX1-SB-408124
20.00Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
20.00Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
20.00Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
20.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
20.00Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
20.00Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
20.00Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
20.00Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
20.00Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
20.00Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
20.00Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
20.00Single8A2OTheophylline8A2O-A2A-Theophylline-Na
20.00Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
20.00Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
20.00Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
20.00Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
20.00Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
20.00Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
20.00Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
20.00Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
20.00Single9B9ZA1AKO9B9Z-CB1-A1AKO
20.00Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
20.00Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
20.00Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
20.00Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
20.00Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
20.00Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
20.00Consensusep_offOrthosteric Ligandep4_off
20.00Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
20.00Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
20.00Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
20.00Consensussensory_onOrthosteric Ligandopsins_on
20.00Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
20.00Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
19.51Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
19.44Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
19.35Single3OE0CVX153OE0-CXCR4-CVX15
19.35Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
19.35Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
19.35Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
19.35Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
19.35Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
19.35Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
19.35Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
19.35Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
19.35Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
19.35Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
19.35Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
19.23Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
19.23Single4BV0Neurotensin4BV0-NTS1-Neurotensin
19.23Single5TZRMK86665TZR-FFA1-MK8666
19.23Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
19.23Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
19.23Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
19.23Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
19.23Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
19.23Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
19.23Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
19.23Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
19.23Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
19.23Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
19.23Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
19.23Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
19.23Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
19.23Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
19.23Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
19.23Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
19.23Consensusneurotensin_onOrthosteric Ligandnts1_on
19.23Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
19.23Consensusrelaxin_onOrthosteric Ligandrxfp4_on
19.23Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
19.05Single3UZAGTPL92363UZA-A2A-GTPL9236
19.05Single6ME5Agomelatine6ME5-MT1-Agomelatine
19.05Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.05Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
19.05Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
19.05Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
19.05Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
19.05Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
19.05Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
19.05Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
19.05Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
19.05Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
19.05Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
19.05Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
19.05Consensusgi_sensoryOrthosteric Ligandgi_opsins
19.05Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
19.05Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
18.92Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
18.92Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
18.92Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
18.75Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
18.75Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
18.75Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
18.75Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.75Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
18.75Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
18.75Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
18.75Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
18.75Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
18.60Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
18.52Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
18.52Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
18.52Single4XEENeurotensin4XEE-NTS1-Neurotensin
18.52Single4XESNeurotensin4XES-NTS1-Neurotensin
18.52Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
18.52Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
18.52Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
18.52Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
18.52Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
18.52Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
18.52Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
18.52Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.52Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
18.52Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
18.52Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
18.42Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
18.42Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
18.42Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
18.18Single6LI0C176LI0-GPR52-C17
18.18Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
18.18Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
18.18Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
18.18Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
18.18Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
18.18Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
18.18Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
18.18Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
18.18Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
18.18Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
18.18Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
18.18Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
18.18Consensuspac_onOrthosteric Ligandpac1_on
18.18Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
17.95Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
17.86Single4BUONeurotensin4BUO-NTS1-Neurotensin
17.86Single5CGDHTL142425CGD-mGlu5-HTL14242
17.86Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
17.86Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
17.86Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.86Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
17.86Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
17.86Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
17.86Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
17.86Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
17.86Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
17.86Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
17.86Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
17.86Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
17.86Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
17.78Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
17.65Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
17.65Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
17.65Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
17.65Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
17.65Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
17.65Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
17.65Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
17.65Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
17.65Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
17.65Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
17.50Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
17.39Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
17.39Single5U09Taranabant5U09-CB1-Taranabant
17.39Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
17.39Single7F8YDevazepide7F8Y-CCKA-Devazepide
17.39Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
17.39Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.39Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
17.39Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
17.39Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
17.39Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
17.39Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
17.39Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
17.39Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
17.39Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.39Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
17.39Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
17.39Consensusangiotensin_offOrthosteric Ligandat1_off
17.39Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
17.24Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
17.24Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
17.24Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
17.24Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
17.14Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
17.14Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
17.14Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
17.14Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
17.14Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
17.14Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
16.67Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
16.67Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
16.67Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
16.67Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
16.67Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
16.67Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
16.67Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
16.67Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
16.67Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
16.67Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
16.67Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
16.67Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
16.67Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
16.67Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
16.67Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
16.67Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
16.67Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
16.67Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
16.22Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
16.22Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
16.13Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
16.13Single7XNACYN1548067XNA-SST2-CYN154806
16.13Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
16.13Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
16.13Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
16.00Single4QIMANTA XV4QIM-SMO-ANTA XV
16.00Single5T04Neurotensin5T04-NTS1-Neurotensin
16.00Single6D27CAY104716D27-DP2-CAY10471
16.00Single6IIVDaltroban6IIV-TXA2-Daltroban
16.00Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
16.00Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
16.00Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
16.00Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
16.00Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
16.00Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
16.00Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
16.00Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
16.00Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
16.00Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
16.00Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
16.00Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
16.00Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
15.79Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
15.79Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
15.79Single5MZPCaffeine5MZP-A2A-Caffeine-Na
15.79Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
15.79Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
15.79Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
15.62Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
15.62Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
15.62Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
15.62Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
15.38Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
15.38Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
15.38Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
15.38Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
15.38Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
15.38Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
15.38Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
15.38Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
15.38Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
15.38Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
15.38Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
15.38Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
15.38Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single9HC04YI9HC0-mGlu5-4YI
15.38Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
15.15Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
15.15Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
15.15Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
15.15Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
15.15Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
15.00Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
15.00Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
14.81Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
14.81Single5V56TC1145V56-SMO-TC114
14.81Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
14.81Single6OS1TRV0266OS1-AT1-TRV026
14.81Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
14.81Single7P2L4YI7P2L-mGlu5-4YI
14.81Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.81Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
14.81Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
14.81Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
14.81Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
14.81Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
14.71Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
14.71Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
14.71Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
14.71Consensuscalcitonin_onOrthosteric Ligandctlike_on
14.63Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
14.29Single3RFMCaffeine3RFM-A2A-Caffeine
14.29Single4PY02MeSATP4PY0-P2Y12-2MeSATP
14.29Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
14.29Single6IIURamatroban6IIU-TXA2-Ramatroban
14.29Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
14.29Single6OS2TRV0266OS2-AT1-TRV026
14.29Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
14.29Single6YVRNTS8-136YVR-NTS1-NTS8-13
14.29Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
14.29Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
14.29Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
14.29Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
14.29Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
14.29Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
14.29Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
14.29Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
14.29Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
14.29Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
14.29Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
14.29Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
14.29Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
14.29Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
14.29Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
14.29Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
14.29Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
14.29Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
13.89Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
13.89Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
13.79Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
13.79Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
13.79Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
13.79Single8ZPLHF511168ZPL-CXCR4-HF51116
13.79Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.64Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
13.64Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
13.51Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
13.51Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
13.51Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
13.51Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
13.33Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
13.33Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
13.33Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
13.33Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
13.33Single8XQJJN2418XQJ-Apelin-JN241
13.33Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
13.33Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
13.33Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
13.33Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
13.33Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
13.33Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
13.16Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
13.04Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
13.04Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
13.04Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
13.04Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
13.04Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
13.04Consensusgq_nucleotideOrthosteric Ligandgq_p2y
13.04Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
12.90Single8XWNCXCL88XWN-CXCR2-CXCL8
12.90Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
12.90Consensussomatostatin_offOrthosteric Ligandsst2_off
12.50Single4BWBNeurotensin4BWB-NTS1-Neurotensin
12.50Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
12.50Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
12.50Single7SK5CXCL127SK5-ACKR3-CXCL12
12.50Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
12.50Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
12.50Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
12.50Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
12.50Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
12.50Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
12.50Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
12.20Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
12.20Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
12.00Single6FFIMMPEP6FFI-mGlu5-MMPEP
12.00Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
12.00Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
12.00Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
12.00Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
12.00Single7VV6C48/807VV6-MRGPRX2-C48/80
12.00Single8K2WAMG4878K2W-CXCR3-AMG487
12.00Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
12.00Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single8ZPMAMD0708ZPM-CXCR4-AMD070
12.00Single8ZPNAMD31008ZPN-CXCR4-AMD3100
12.00Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
12.00Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
11.76Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
11.54Single6FFHFenobam6FFH-mGlu5-Fenobam
11.54Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
11.54Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
11.54Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
11.54Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
11.54Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
11.54Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
11.54Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
11.54Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
11.43Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
11.11Single4JKVTaladegib4JKV-SMO-Taladegib
11.11Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
11.11Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
11.11Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
11.11Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
11.11Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
11.11Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
11.11Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
11.11Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
10.71Single5V57TC1145V57-SMO-TC114
10.71Single7F1TMIP-1a7F1T-CCR5-MIP-1a
10.71Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
10.71Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
10.71Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
10.71Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.71Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
10.53Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
10.34Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
10.34Single8XQJJN2418XQJ-Apelin-JN241
10.34Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
10.34Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.00Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
10.00Single8XVUCXCL28XVU-CXCR2-CXCL2
10.00Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
10.00Single9JH5C16:0 Ceramide9JH5-CysLT2-C16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Single6KNMJN241-96KNM-Apelin-JN241-9
9.68Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
9.52Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
9.52Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
9.38Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
9.38Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.38Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
9.38Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
9.09Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
9.09Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
9.09Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
9.09Consensusp2y_offOrthosteric Ligandp2y1_off
8.70Single4XNWMRS25004XNW-P2Y1-MRS2500
8.70Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
8.70Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
8.70Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
8.70Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
8.70Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
8.70Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
8.70Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
8.57Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
8.33Single4O9RCyclopamine4O9R-SMO-Cyclopamine
8.33Single5L7IVismodegib5L7I-SMO-Vismodegib
8.33Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
8.33Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
8.33Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
8.33Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
8.33Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.33Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
8.33Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
8.11Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
8.00Single4QINSAG1.54QIN-SMO-SAG1.5
8.00Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
8.00Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
8.00Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
8.00Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
8.00Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.00Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
8.00Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
8.00Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
8.00Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
8.00Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
7.69Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
7.69Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
7.69Single6ZINSR486926ZIN-NTS1-SR48692
7.69Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
7.69Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single8IYXYL-3658IYX-GPR34-YL-365
7.41Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
7.14Single6Z4SSR486926Z4S-NTS1-SR48692
7.14Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
6.90Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
6.90Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
6.90Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
6.90Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
6.67Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.67Single8XWACXCL18XWA-CXCR2-CXCL1
6.67Single8XWMCXCL68XWM-CXCR2-CXCL6
6.67Single8XWSCXCL58XWS-CXCR2-CXCL5
6.67Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
6.45Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
6.45Single8XWFCXCL38XWF-CXCR2-CXCL3
6.45Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
6.25Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
6.06Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
5.56Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
5.56Single6D35Cholesterol6D35-SMO-Cholesterol
5.56Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
5.56Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
5.56Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
5.56Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
5.56Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042
5.56Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
5.56Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
5.56Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-BHFF
5.56Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
5.56Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626
5.56Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.56Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.56Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.56Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.56Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
5.56Single7DTTCa7DTT-CaS-Ca-Ca
5.56Single7DTTCa7DTT-CaS-Ca-Ca
5.56Single7DTUTryptophan7DTU-CaS-Tryptophan
5.56Single7DTUTryptophan7DTU-CaS-Tryptophan
5.56Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
5.56Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
5.56Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
5.56Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
5.56Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.56Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.56Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.56Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.56Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
5.56Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
5.56Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
5.56Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
5.56Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
5.56Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
5.56Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
5.56Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
5.56Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
5.56Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
5.56Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
5.56Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
5.56Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
5.56Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
5.56Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
5.56Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
5.56Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
5.56Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.56Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.56Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.56Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.56Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
5.56Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
5.56Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
5.56Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
5.56Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
5.56Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
5.56Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.56Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.56Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.56Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.56Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.56Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.56Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.56Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.56Single7T9NM22 Fab7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
5.56Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
5.56Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
5.56Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
5.56Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
5.56Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
5.56Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
5.56Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
5.56Single7XW7K1-707XW7-TSH-K1-70
5.56Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
5.56Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
5.56Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
5.56Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
5.56Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
5.56Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
5.56Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
5.56Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
5.56Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
5.56Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
5.56Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
5.56Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
5.56Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
5.56Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
5.56Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
5.56Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
5.56Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
5.56Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
5.56Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
5.56Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
5.56Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
5.56Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
5.56Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
5.56Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
5.56Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
5.56Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
5.56Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
5.56Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
5.56Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
5.56Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
5.56Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
5.56Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
5.56Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
5.56Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
5.56Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
5.56Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
5.56Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
5.56Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
5.56Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
5.56Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
5.56Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
5.56Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
5.56Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
5.56Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
5.56Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
5.56Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
5.56Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
5.56Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
5.56Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
5.56Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
5.56Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
5.56Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
5.56Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.56Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.56Single8WVXNorrin8WVX-LGR4-Norrin
5.56Single8WVYNorrin8WVY-LGR4-Norrin
5.56Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
5.56Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
5.56Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
5.56Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
5.56Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
5.56Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
5.56Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
5.56Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
5.56Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
5.56Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
5.56Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
5.56Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
5.56Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
5.56Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
5.56Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
5.56Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.56Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.56Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.56Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.56Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.56Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.56Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.56Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.56Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.56Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.56Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.56Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.56Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
5.56Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
5.56Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
5.56Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
5.56Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
5.56Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
5.56Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
5.56Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
5.56Single9KHHNorrin9KHH-LGR4-Norrin
5.56Single9S37NB219S37-LGR4-NB21
5.56Single9UTBSucralose9UTB-TAS1R2; TAS1R3-Sucralose
5.26Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.26Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.26Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.26Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.26Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.26Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.26Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.26Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.26Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
5.26Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
5.26Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.26Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.26Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.26Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.26Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
5.26Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
5.00Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
5.00Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
5.00Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
4.76Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
4.76Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
4.76Single7UTZTR14027UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
4.76Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
4.76Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
4.76Single8JGBConorfamide-Tx28JGB-MRGPRX1-Conorfamide-Tx2-Gi1/β1/γ2
4.55Single5L7DCholesterol5L7D-SMO-Cholesterol
4.55Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
4.55Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
4.55Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
4.55Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
4.55Single8HS2Fab0468HS2-GPR20-Fab046
4.55Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
4.55Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
4.35Single7Y14Beta-Alanine7Y14-MRGPRD-β-Alanine
4.35Single9IVMLSN33188399IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
4.17Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
4.17Single7Y12Beta-Alanine7Y12-MRGPRD-β-Alanine-Gi1/β1/γ2
4.17Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
4.17Single8JPSCCL78JPS-ACKR1-CCL7
4.00Single8HNNSCH5467388HNN-CXCR3-SCH546738
4.00Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
4.00Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
4.00Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
4.00Single8YKDDehydroepiandrosterone8YKD-ADGRG2-Dehydroepiandrosterone-chim(NtGi1-Gs)/β1/γ2
3.85Single4K5YCP-3763954K5Y-CRF1-CP-376395
3.85Single4XNVBPTU4XNV-P2Y1-BPTU
3.85Single7WV9ZCZ0117WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
3.70Single8JD6VU03647708JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
3.57Single4Z9GCP-3763954Z9G-CRF1-CP-376395
3.57Single8GTIBMK-C2058GTI-CRF1-BMK-C205
3.57Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
3.57Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
3.45Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
3.45Single8GTGBMK-I1528GTG-CRF1-BMK-I152
3.45Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
3.45Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
3.45Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
3.45Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
3.33Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
3.23Single8GTMBMK-C2038GTM-CRF1-BMK-C203
2.94Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.94Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.78Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.78Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.70Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.50Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
7EW3 7EW3-S1P3-S1P-Gi1/β1/γ2
7EW4 7EW4-S1P3-CYM5541-Gi1/β1/γ2
7EW2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
Net Summary
Imin 2.28
Number of Linked Nodes 890
Number of Links 1119
Number of Hubs 196
Number of Links mediated by Hubs 715
Number of Communities 23
Number of Nodes involved in Communities 261
Number of Links involved in Communities 399
Path Summary
Number Of Nodes in MetaPath 87
Number Of Links MetaPath 86
Number of Shortest Paths 2416982
Length Of Smallest Path 3
Average Path Length 30.0252
Length of Longest Path 52
Minimum Path Strength 0.486667
Average Path Strength 5.28797
Maximum Path Strength 21.8733
Minimum Path Correlation 0.703333
Average Path Correlation 0.987368
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 3.0303
Average % Of Corr. Nodes 42.1403
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 55.0172
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
s1p_on_gps1p1_on_gp
s1p3_on_gp
s1p5_on_gp



You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

Download s1p3_on_gp.zip



You can click to copy the link of this page to easily come back here later

or use this QR code to link and share this page.



You can also  read or  download a guide explaining the meaning of all files and numerical data.