Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.11 1.30369502
2G.H1.01 4.43653459
3G.S2.03 5.77179419
4G.S2.04 1.90773406
5G.S2.05 5.60814413
6G.S2.08 5.839644105
7G.S3.03 7.08295557
8G.S3.04 8.96878416
9G.S3.05 3.61497457
10G.S3.06 8.20341515
11G.s3h2.03 4.03415419
12G.H2.04 4.16828409
13G.H2.06 4.6101719
14G.H2.07 4.82854619
15G.h2s4.01 6.19392519
16G.S4.04 5.86883449
17G.s4h3.04 5.604796118
18G.H3.01 5.65257509
19G.H3.09 5.16173749
20G.H3.13 4.29089645
21G.H3.17 7.11444615
22G.H3.18 5.37069419
23G.S5.04 3.77325549
24G.S5.05 3.80676679
25G.S5.07 3.6214579
26G.HG.04 5.04844409
27G.HG.14 2.31704405
28G.HG.15 4.44161407
29G.hgh4.02 5.33965187
30G.hgh4.05 7.94217407
31G.hgh4.08 2.78121403
32G.H4.03 4.79133504
33G.H4.10 7.521955186
34G.H4.12 5.94897445
35G.H4.15 5.43967448
36G.h4s6.02 4.62073448
37G.S6.02 4.942578197
38G.S6.05 4.93611404
39G.H5.03 5.06014478
40G.H5.08 5.582984108
41G.H5.13 3.69447508
42G.H5.26 2.936555205
43b.1x4 1.99487408
44b.b1x4 2.99733597
45b.b1x6 6.98261409
46b.l1x3 7.92275669
47b.l1x6 9.67175419
48b.b2x1 6.69702518
49b.b2x5 7.13581507
50b.l3x2 5.22516569
51b.b4x3 4.419534127
52b.b4x6 8.89975669
53b.l4x2 7.89152504
54b.b5x2 5.55019407
55b.b5x3 6.20381669
56b.b5x5 4.856774175
57b.b5x7 5.89626407
58b.l5x1 4.298375128
59b.l5x2 2.91358406
60b.l5x5 6.92041719
61b.b6x5 4.02103606
62b.l6x5 5.887184134
63b.b7x1 5.876855134
64b.l7x2 3.9141419
65b.b8x4 5.597185126
66b.l8x3 2.75661403
67b.l8x5 2.39158403
68b.b9x4 6.04094409
69b.l9x3 6.70676619
70b.l9x6 4.38524818
71b.b10x5 4.34097509
72b.l10x1 3.92796403
73b.b11x4 5.12085419
74b.l11x2 7.76767419
75b.b12x6 8.6659618
76b.b13x7 7.14452537
77b.l13x3 7.57783639
78b.l13x6 4.4231519
79b.l13x7 4.28183439
80b.b14x3 4.65675435
81b.b15x1 6.20607539
82b.b15x2 5.90395416
83b.l15x2 5.81008439
84b.b16x4 10.3525436
85b.b16x5 4.36251405
86b.b16x6 8.47945638
87b.b17x5 6.74528417
88b.b17x7 8.37681418
89b.l17x3 7.37769719
90b.l17x6 5.92714519
91b.b18x3 4.35024418
92b.b18x5 4.97593405
93b.l18x1 5.183667236
94b.l18x3 7.06789405
95b.b19x2 6.41334616
96b.b19x4 5.85159418
97b.l19x2 5.67537519
98b.b20x4 10.0641518
99b.b20x6 6.71308616
100b.b20x7 3.31997409
101b.b21x1 7.48813517
102b.b21x5 5.37007404
103b.b21x7 6.25653505
104b.l21x2 5.17005404
105b.b22x5 4.885746237
106b.l22x5 6.953154219
107b.b23x6 6.347616147
108b.l23x1 7.14878416
109b.b24x4 6.373794146
110b.b24x6 5.797534148
111b.l24x3 3.46565405
112b.l25x3 7.91407589
113b.l25x4 2.25752505
114b.l25x6 11.5173418
115b.l26x1 6.46364227
116b.l27x1 10.0034719
117b.l27x2 7.03777489
118b.b28x2 4.73335404
119b.b28x3 3.84503407
120b.b28x4 6.62176486
121b.b28x6 8.06362589
122g.h1x1 0.732671502
123g.h1x5 1.29397406
124g.l1x4 3.92576408
125g.ctx3 5.184035249
126g.ctx16 3.53963698
127NT 9.36472725
1281x36 1.79382405
1291x50 5.24624409
1301x56 1.94249408
1312x40 3.31059408
1322x41 1.99909404
1332x42 3.28244408
1342x46 4.110594259
1352x50 5.512385259
1362x51 3.02277407
1372x57 3.35371506
1383x25 4.46927429
1393x29 3.93459424
1403x49 4.17302409
1413x50 5.4198409
1423x55 4.614294156
143I2x53 4.04671407
144E2 7.69742825
1455x50 2.89261407
1465x51 2.42726507
1475x58 3.57744609
1485x60 3.685575155
1495x64 3.120764156
1506x30 2.08335507
1516x32 2.302935208
1526x48 5.48264508
1536x59 2.12679403
154E3 4.67458621
1557x53 3.97197509
1568x47 2.43968408
157Lig 5.202571220
158H.HA.19 0.06791674160
159H.HC.03 0.03325160
160H.HC.07 0.05466674160
161H.HD.07 0.0764167400
162H.hdhe.01 0.0609722600
163H.HE.05 0.0583500
164H.HE.06 0.0715417400
165H.HF.06 0.099125400
166E1x52 1.38074400
1674x65 2.76725420
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1b.l2x3 b.l2x5 63.57442.98728NoNo085
2b.b3x1 b.l2x3 63.31245.78442NoNo058
3b.b3x1 b.b6x5 63.05044.28602NoYes056
4b.l2x5 b.l4x2 68.772723.9303NoYes054
5b.l4x2 g.ctx15 72.95787.02665YesNo049
6b.l26x5 g.ctx15 76.10484.08388NoNo059
7b.l26x5 g.ctx4 85.8265.71393NoNo057
8g.ctx3 g.ctx4 86.07484.32644YesNo097
9b.l22x1 g.ctx3 87.5426.41575NoYes2499
10b.b23x1 b.l22x1 88.0613.33179NoNo059
11b.b23x1 b.lhb1x9 44.59333.56217NoNo053
12b.lhb1x11 b.lhb1x9 44.81962.91648NoNo043
13b.b25x7 b.lhb1x11 44.93274.358NoNo074
14b.b25x7 b.b28x6 45.158716.0765NoYes079
15b.b27x3 b.b28x6 45.43067.49024NoYes089
16b.b26x3 b.b27x3 47.79973.64055NoNo068
17b.b22x2 b.b26x3 92.14585.61862NoNo086
18b.b22x1 b.b22x2 92.22992.96NoNo088
19b.b22x1 b.l25x6 87.94554.01087NoYes188
20b.l25x6 b.l27x1 98.598318.5958YesYes189
21b.b2x1 b.l27x1 99.03196.85517YesYes189
22b.b2x1 b.l3x1 99.803912.813YesNo189
23b.l3x1 b.l5x5 1007.07392NoYes199
24b.b23x1 b.b24x5 43.72465.26467NoNo055
25b.b23x3 b.b24x5 43.83314.3683NoNo075
26b.b23x3 b.b27x1 43.94464.18028NoNo076
27b.b26x5 b.b27x1 44.05654.07221NoNo076
28b.b22x4 b.b26x5 44.16853.63138NoNo057
29b.b22x4 b.b26x3 44.28063.22276NoNo056
30G.h2s4.01 b.l5x5 45.247210.8507YesYes199
31G.H2.07 G.h2s4.01 46.76073.61412YesYes199
32G.H2.04 G.H2.07 80.68394.85873YesYes099
33G.H2.04 G.H3.08 80.976.65433YesNo099
34G.H3.08 G.S4.04 80.92315.10494NoYes099
35G.S4.04 G.S5.04 62.82413.40104YesYes499
36G.S5.04 G.S5.06 57.17534.00597YesNo098
37G.S5.06 G.s4h3.01 54.39515.43506NoNo087
38G.HG.04 G.s4h3.01 54.19987.62768YesNo097
39G.HG.04 G.s4h3.04 53.78024.85256YesYes098
40G.HG.07 G.s4h3.04 55.93835.99967NoYes1198
41G.HG.07 G.s4h3.02 56.02512.37879NoNo099
42G.s4h3.02 G.s5hg.01 55.68693.40364NoNo099
43G.S5.07 G.s5hg.01 53.86292.52356YesNo099
44G.S5.07 G.s6h5.01 53.28445.16348YesNo799
45G.S5.05 G.s6h5.01 52.31185.11298YesNo799
46G.S4.03 G.S5.05 42.35323.14261NoYes079
47G.S1.04 G.S4.03 42.22444.79008NoNo077
48G.S1.04 G.S3.03 42.09543.29694NoYes077
49b.l5x5 b.l7x2 54.78984.79355YesYes199
50G.H2.07 b.l7x2 45.23883.19086YesYes199
51G.S3.01 G.S3.03 39.17936.91464NoYes047
52G.S3.01 I2x51 37.46364.359NoNo047
53G.H2.07 b.l9x6 26.46153.4404YesYes198
54G.H2.06 b.l9x6 21.68974.161YesYes198
55G.H2.06 b.l17x6 20.43987.10455YesYes199
56G.H3.09 G.S4.04 12.307812.1216YesYes499
57G.H3.06 G.hgh4.02 22.05544.24166NoYes067
58G.H3.06 G.H4.15 16.46745.96355NoYes068
59G.S5.03 G.S5.05 12.8733.25913NoYes089
60G.H5.10 G.S5.03 12.55665.20517NoNo068
61G.H5.10 G.S6.02 12.39817.11515NoYes067
62G.H4.10 G.hgh4.02 12.57816.3261YesYes1867
63G.H5.15 I2x51 37.32942.66733NoNo077
64G.H5.15 G.H5.19 37.06062.99755NoNo078
65G.H5.19 I2x53 36.9263.92617NoYes087
663x49 I2x53 36.52156.25567YesYes097
67b.b2x4 b.b6x5 44.38383.24059NoYes066
68b.b10x4 b.b2x4 44.105511.3609NoNo066
69b.b10x2 b.b10x4 20.52523.19694NoNo066
70b.b10x2 b.b14x3 20.25235.3706NoYes065
71b.b14x3 b.b15x1 16.30054.30121YesYes359
72b.b15x1 b.b16x6 14.600211.0578YesYes398
73b.b16x4 b.b16x6 11.40678.99736YesYes368
74b.b16x4 b.b17x6 11.15310.5497YesNo067
75b.b17x6 g.l1x1 10.57651.694NoNo071
76g.h1x12 g.l1x1 10.28672.17067NoNo061
77b.l17x5 b.l17x6 20.04463.3529NoYes169
78b.l17x5 b.l19x2 19.83714.18221NoYes169
79b.l17x3 b.l19x2 18.04533.519YesYes199
80b.b20x6 b.l17x3 12.1943.15386YesYes169
81b.l21x7 b.l23x1 15.25554.72151NoYes056
82b.l21x7 b.l23x2 14.91196.97111NoNo058
83b.b23x6 b.l23x2 14.21752.93067YesNo078
84b.b23x6 b.b24x6 12.10346.43083YesYes1478
85b.b21x7 b.b24x6 11.78777.81282YesYes058
86b.b3x3 b.b6x5 16.6214.51824NoYes086
87b.b3x3 b.b4x3 16.33453.12545NoYes087
88b.l11x1 b.l9x6 13.02125.09155NoYes198
89b.b11x6 b.l11x1 12.81812.99643NoNo199
90b.b11x6 b.l9x3 10.841814.5315NoYes199
91b.b10x4 b.b14x5 23.30933.92683NoNo065
92b.b14x5 b.l10x1 23.03584.98359NoYes053
93b.b11x1 b.l10x1 22.20693.89356NoYes053
94b.b11x1 b.b12x5 21.65053.04144NoNo056
95b.b12x5 b.b13x4 21.08012.96507NoNo364
96b.b12x7 b.b13x4 21.15062.66398NoNo094
97b.b12x7 b.l12x3 20.30137.03792NoNo095
98b.b13x2 b.l12x3 20.01793.60992NoNo045
992x42 3x49 30.88794.46965YesYes089
1002x42 3x46 30.47783.71321YesNo089
1013x46 7x53 30.34094.1271NoYes099
1023x43 7x53 29.17123.59637NoYes089
1032x46 3x43 29.02863.19194YesNo098
1042x46 7x49 22.83194.25535YesNo2599
1057x45 7x49 22.92927.37644NoNo099
1066x48 7x45 22.63399.19152YesNo089
1073x36 6x48 20.90313.99965NoYes068
1083x36 Lig 20.75293.96804NoYes060
109H.hdhe.01 b.b13x2 19.72890.0375YesNo004
110H.hdhe.01 H.hdhe.03 18.08480.039YesNo000
111H.HD.07 H.hdhe.03 17.61510.0406667YesNo000
112b.l23x1 b.l25x6 11.230217.1285YesYes168
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
NTNT18.44442YesYes5522
E2NT18.70262YesYes5512
2x572x613.220210YesNo6612
2x573x322.955740YesNo6512
2x577x424.208320YesNo6612
2x57Lig4.121330YesYes6010
2x603x285.403310NoNo4512
2x60Lig5.681380NoYes4010
2x64Lig5.150230NoYes3010
3x22E24.647312NoYes3521
3x253x294.365072YesYes9421
3x25E26.1032YesYes9521
3x26E23.82662NoYes5521
3x29Lig3.162072YesYes4010
3x33Lig7.79370NoYes4010
3x366x483.999650NoYes6812
3x36Lig3.968040NoYes6010
3x375x433.230330NoNo6521
4x60E26.094982NoYes5521
4x605x397.127362NoNo5722
E2E244.35842YesYes5511
5x36E28.670442NoYes4521
5x38E23.085530NoYes4521
6x58E27.165752NoYes3521
7x31E23.407830NoYes2521
E2E33.100672YesYes5112
7x34E24.723392NoYes4511
E2Lig9.932332YesYes5010
5x39E27.528392NoYes7521
5x395x432.989392NoNo7521
5x406x554.759940NoNo5612
5x43Lig7.043820NoYes5010
6x547x343.272980NoNo4421
7x34Lig4.327642NoYes4010
7x38Lig5.677120NoYes5010
3x29E25.277222YesYes4511
2x603x323.345660NoNo4512
3x223x264.122972NoNo3522
E3E35.237432YesYes1122
4x64E29.0130NoYes0521
4x65E24.4662YesYes0521
E2E2x523.8612YesNo5012
E2E2x514.249332YesNo5012
E3NT3.510032YesYes1522
E2x51E2x523.3222NoNo0022
3x294x652.9342YesYes4012
4x65E2x523.172YesNo0022
7x35Lig2.800810NoYes4010
5x40Lig2.772330NoYes5010
5x32E22.750NoYes0521
5x34E22.5150NoYes0521
5x37E22.476852NoYes4521
1x432x572.262970NoYes7621
5x35E21.6350NoYes0521
7x28E21.5430NoYes3521
1x357x351.405620NoNo5421
E1x49E21.1962NoYes0521
4x63E20.7022942NoYes4521
4x66E20.1372NoYes0521

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
100.00Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
83.33Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
73.33Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
71.43Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
71.43Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
69.23Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
69.23Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
68.75Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
66.67Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
64.71Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
64.29Single7V3ZCP559407V3Z-CB1-CP55940
62.50Single9DGIZ85267113509DGI-CB1-Z8526711350
62.50Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
62.50Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
62.50Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
62.50Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
61.11Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
58.82Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
58.82Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
58.82Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
56.25Single5XR8AM8415XR8-CB1-AM841
56.25Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
56.25Single7FEECP559407FEE-CB1-CP55940-ZCZ011
56.25Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
56.25Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
56.25Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
56.25Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
56.25Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
55.56Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
53.33Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
52.94Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
52.94Single6KQICP559406KQI-CB1-CP55940-Org27569
52.94Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
52.63Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
52.63Consensuslpl_onOrthosteric Ligands1p_on lpa_on
52.63Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
50.00Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
50.00Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
50.00Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
50.00Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
50.00Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
50.00Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
50.00Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
50.00Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
50.00Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
50.00Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
50.00Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
50.00Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
47.62Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
47.62Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
47.37Single5ZTYAM102575ZTY-CB2-AM10257
47.37Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
47.37Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
47.37Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
47.37Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
47.06Single5XRAAM115425XRA-CB1-AM11542
47.06Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
47.06Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
47.06Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
47.06Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
47.06Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
47.06Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
47.06Consensuslpa_onOrthosteric Ligandlpa1_on
47.06Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
46.67Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
46.67Single8K5CAcipimox8K5C-HCA2-Acipimox
46.67Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
45.83Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
45.45Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
45.00Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
44.44Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
44.44Single7YITNalfurafine7YIT-κ-Nalfurafine
44.44Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
44.44Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
44.44Consensuslpl_offOrthosteric Ligands1p_off lpa_off
44.44Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
43.75Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
43.75Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
43.75Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
43.75Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
43.75Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
43.75Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
43.75Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
43.75Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
43.75Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
43.75Consensusblt_onOrthosteric Ligandblt1_on
43.75Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
43.75Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
43.75Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
43.75Consensusleukotriene_onOrthosteric Ligandblt_on
43.75Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
42.86Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
42.86Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
42.11Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
42.11Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
42.11Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
42.11Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
41.18Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
41.18Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
41.18Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
41.18Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
41.18Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
41.18Single8JXSPF-61428JXS-D1-PF-6142
41.18Single8TF5Oleic acid8TF5-GPR6-Oleic acid
41.18Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
41.18Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
41.18Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
41.18Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
41.18Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
41.18Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
41.18Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
40.91Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
40.91Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
40.00Single3PWHZM-2413853PWH-A2A-ZM-241385
40.00Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
40.00Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
40.00Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
40.00Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
40.00Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
40.00Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
40.00Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
40.00Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
40.00Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
40.00Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
40.00Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
40.00Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
40.00Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
40.00Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
40.00Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
39.29Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
39.13Single6JODAngiotensin II6JOD-AT2-Angiotensin II
39.13Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
39.13Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
39.13Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
39.13Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
39.13Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
38.89Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
38.89Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
38.89Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
38.89Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
38.89Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
38.89Single8E0GBU728E0G-μ-BU72
38.89Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
38.89Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
38.89Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
38.89Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
38.89Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
38.89Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
38.89Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
38.89Consensusa2_onOrthosteric Liganda2b_on
38.89Consensusa2_on_gpOrthosteric Liganda2b_on_gp
38.89Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
38.89Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
38.89Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
38.89Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
38.89Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
38.89Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
38.10Single7QA8Peptide7QA8-STE2-Peptide
38.10Single7QA8Peptide7QA8-STE2-Peptide
38.10Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
38.10Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
38.10Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
38.10Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
37.50Single7F61PF-036547467F61-H3-PF-03654746
37.50Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
37.50Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
37.50Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
37.50Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
37.50Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
37.50Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
37.50Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
37.50Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
37.50Single8ZRTET-18ZRT-ETB-ET-1
37.50Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
37.50Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
37.50Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
37.50Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
37.50Consensushca_onOrthosteric Ligandhca2_on
37.50Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
37.50Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
37.50Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
36.84Single4RWADIPP-NH24RWA-δ-DIPP-NH2
36.84Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
36.84Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
36.84Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
36.84Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
36.84Single8JWY2-1188JWY-A2A-2-118
36.84Single8JWZAB9288JWZ-A2A-AB928-Na
36.84Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
36.84Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
36.84Single8XYIVUF106618XYI-CXCR3-VUF10661
36.84Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
36.84Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
36.84Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
36.84Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
36.84Consensuslpa_offOrthosteric Ligandlpa1_off
36.84Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
36.84Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
36.36Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
36.36Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
36.36Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
36.36Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
36.36Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
36.36Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
36.00Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
36.00Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
36.00Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
36.00Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
35.71Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
35.71Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
35.71Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
35.71Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
35.29Single5UIGCmpd-15UIG-A2A-Cmpd-1
35.29Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
35.29Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
35.29Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
35.29Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
35.29Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
35.29Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
35.29Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
35.29Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
35.29Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
35.29Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
35.29Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
35.29Consensusa3_onOrthosteric Liganda3a_on
35.29Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
35.29Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
35.29Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
35.29Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
35.29Consensushca_on_gpOrthosteric Ligandhca2_on_gp
35.29Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
35.00Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
35.00Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
35.00Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
35.00Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
35.00Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
35.00Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
35.00Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
35.00Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
35.00Single8ZPLHF511168ZPL-CXCR4-HF51116
35.00Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
35.00Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
34.78Single6W25SHU91196W25-MC4-SHU9119-Ca
34.78Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
34.78Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
34.78Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
34.78Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
34.78Consensusangiotensin_onOrthosteric Ligandat1_on
34.78Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
34.78Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
34.62Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
34.62Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
34.62Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
34.62Single9KDFRES-701-39KDF-ETB-RES-701-3
34.62Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
34.62Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
34.62Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
33.33Single3NY9ICI118-5513NY9-β2-ICI118-551
33.33Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
33.33Single4UG2CGS216804UG2-A2A-CGS21680
33.33Single5C1MBU725C1M-μ-BU72
33.33Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
33.33Single6IGLIRL16206IGL-ETB-IRL1620
33.33Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
33.33Single7C4SS1P7C4S-S1P3-S1P
33.33Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
33.33Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
33.33Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
33.33Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
33.33Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
33.33Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
33.33Single7SK9CCX6627SK9-ACKR3-CCX662
33.33Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
33.33Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
33.33Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
33.33Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
33.33Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
33.33Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
33.33Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
33.33Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
33.33Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
33.33Single8K5BNiacin8K5B-HCA2-Niacin
33.33Single8QJ2pN1628QJ2-MC4-pN162-Gs
33.33Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
33.33Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
33.33Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
33.33Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
33.33Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
33.33Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
33.33Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
33.33Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
33.33Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single9EHSLUF76029EHS-A3A-LUF7602
33.33Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
33.33Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
33.33Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
33.33Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
33.33Consensusa3_on_gpOrthosteric Liganda3a_on_gp
33.33Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
33.33Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
33.33Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
33.33Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
33.33Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
33.33Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
33.33Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
33.33Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
33.33Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
33.33Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
33.33Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
33.33Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
33.33Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
33.33Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
33.33Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
33.33Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
33.33Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
32.00Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
32.00Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
32.00Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
32.00Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
32.00Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
32.00Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
32.00Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
32.00Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
31.82Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
31.82Single4XT1Fractalkine4XT1-US28-Fractalkine
31.82Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
31.82Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
31.82Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
31.82Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
31.82Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
31.82Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
31.82Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
31.82Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
31.82Single8WDTphotoNECA8WDT-A2A-photoNECA
31.82Single8WKYPG-9348WKY-MC4-PG-934
31.82Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
31.82Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
31.82Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
31.82Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
31.82Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
31.82Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
31.82Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
31.82Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
31.82Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
31.58Single3P0GBI1671073P0G-β2-BI167107
31.58Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
31.58Single4DJHJDTic4DJH-κ-JDTic
31.58Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
31.58Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
31.58Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
31.58Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
31.58Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
31.58Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
31.58Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
31.58Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
31.58Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
31.58Single7TUYGSK682753A7TUY-GPR183-GSK682753A
31.58Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
31.58Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
31.58Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
31.58Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
31.58Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
31.58Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
31.58Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
31.58Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
31.58Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
31.58Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
31.58Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
31.58Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
31.58Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
31.58Single9BJKNaloxone9BJK-μ-Naloxone-NAM
31.58Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
31.58Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
31.58Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
31.58Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
31.58Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
31.58Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
31.58Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
31.58Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
31.58Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
31.58Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
31.58Consensusrelaxin_onOrthosteric Ligandrxfp4_on
31.58Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
31.25Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
31.25Single5ZKQABT-4915ZKQ-PAF-ABT-491
31.25Single6AKXA4R6AKX-CCR5-A4R
31.25Single6AKYMaraviroc6AKY-CCR5-Maraviroc
31.25Single6B73MP11046B73-κ-MP1104
31.25Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
31.25Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.25Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
31.25Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
31.25Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
31.25Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
31.25Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
31.25Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
31.25Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
31.25Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
31.25Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
31.25Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
31.25Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
31.25Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
31.25Consensusorexin_offOrthosteric Ligandox2_off ox1_off
31.25Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
31.25Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
31.25Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
31.25Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
30.77Single4XT3Fractalkine4XT3-US28-Fractalkine
30.77Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
30.77Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
30.77Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
30.77Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
30.77Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
30.77Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
30.77Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
30.77Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
30.43Single3QAKUK-4320973QAK-A2A-UK-432097
30.43Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
30.43Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
30.43Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
30.43Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
30.43Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
30.43Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
30.43Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
30.43Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
30.43Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
30.43Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
30.43Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
30.43Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
30.43Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
30.30Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
30.00Single4LDEBI1671074LDE-β2-BI167107
30.00Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
30.00Single4PY02MeSATP4PY0-P2Y12-2MeSATP
30.00Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
30.00Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
30.00Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
30.00Single6A93Risperidone6A93-5-HT2A-Risperidone
30.00Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
30.00Single6MXTSalmeterol6MXT-β2-Salmeterol
30.00Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
30.00Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
30.00Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
30.00Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
30.00Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
30.00Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
30.00Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
30.00Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
30.00Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
30.00Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
30.00Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
30.00Single8JJ8Formoterol8JJ8-β2-Formoterol
30.00Single8JJLOlodaterol8JJL-β2-Olodaterol
30.00Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
30.00Consensusalpha1_offOrthosteric Ligandalpha1a_off
30.00Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
30.00Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
30.00Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
30.00Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
30.00Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
30.00Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
30.00Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Consensusorexin_onOrthosteric Ligandox2_on
30.00Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
29.63Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
29.63Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
29.63Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
29.63Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
29.63Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
29.63Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
29.63Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
29.63Consensusglp_onOrthosteric Ligandglp1_on glp2_on
29.63Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
29.63Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
29.63Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
29.41Single3REYXAC3REY-A2A-XAC
29.41Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
29.41Single4MBSMaraviroc4MBS-CCR5-Maraviroc
29.41Single4ZJCSB-6740424ZJC-OX1-SB-674042
29.41Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
29.41Single5IUBQ274563445IUB-A2A-Q27456344-Na
29.41Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
29.41Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
29.41Single6AQFZM-2413856AQF-A2A-ZM-241385
29.41Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
29.41Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
29.41Single6TPGEMPA6TPG-OX2-EMPA
29.41Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
29.41Single7AROLUF58337ARO-A2A-LUF5833-Na
29.41Single7T32ZM-2413857T32-A2A-ZM-241385
29.41Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
29.41Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
29.41Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
29.41Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
29.41Single8IHKAcifran8IHK-HCA3-Acifran
29.41Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
29.41Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
29.41Single8K2WAMG4878K2W-CXCR3-AMG487
29.41Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
29.41Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.41Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
29.41Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
29.41Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
29.41Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
29.41Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
29.41Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
29.41Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
29.41Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
29.17Single3OE0CVX153OE0-CXCR4-CVX15
29.17Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
29.17Single6PT2KGCHM076PT2-δ-KGCHM07
29.17Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
29.17Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
29.17Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
29.17Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
29.17Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
29.17Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
29.17Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
29.17Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
29.17Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
29.17Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
29.17Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
29.17Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
29.17Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
29.03Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
28.57Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
28.57Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
28.57Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
28.57Single5X93K-87945X93-ETB-K-8794
28.57Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
28.57Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
28.57Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
28.57Single7EZCUKA7EZC-A2A-UKA
28.57Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
28.57Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
28.57Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
28.57Single7UM4AS26747237UM4-5-HT5A-AS2674723
28.57Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
28.57Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
28.57Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
28.57Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
28.57Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
28.57Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
28.57Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
28.57Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
28.57Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
28.57Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
28.57Consensusbradykinin_onOrthosteric Ligandbk2_on
28.57Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
28.57Consensusendothelin_offOrthosteric Ligandetb_off
28.57Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
28.57Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
28.57Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
28.57Consensusprostanoid_offOrthosteric Ligandep_off dp_off
28.57Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
28.12Consensuspth_onOrthosteric Ligandpth1_on pth2_on
28.00Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
28.00Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
28.00Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
28.00Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
28.00Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
28.00Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
28.00Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
28.00Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
28.00Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
28.00Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
28.00Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
28.00Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
28.00Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
28.00Consensusvasop-oxy_onOrthosteric Ligandv2_on
28.00Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
27.78Single2Y04Salbutamol2Y04-β1-Salbutamol
27.78Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
27.78Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
27.78Single4EJ4Naltrindole4EJ4-δ-Naltrindole
27.78Single4QIMANTA XV4QIM-SMO-ANTA XV
27.78Single4YAYZD-71554YAY-AT1-ZD-7155
27.78Single5IU8Q274563475IU8-A2A-Q27456347-Na
27.78Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
27.78Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
27.78Single5UENDU1725UEN-A1-DU172
27.78Single6GPSMK08126GPS-CCR2-MK0812
27.78Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
27.78Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
27.78Single6TOTLemborexant6TOT-OX1-Lemborexant
27.78Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
27.78Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
27.78Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
27.78Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
27.78Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
27.78Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
27.78Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
27.78Single7PYRPSB-21157PYR-A2A-PSB-2115
27.78Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
27.78Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
27.78Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
27.78Single7UL4Alvimopan7UL4-μ-Alvimopan
27.78Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
27.78Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
27.78Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
27.78Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
27.78Single7YXAONO-54306087YXA-S1P5-ONO-5430608
27.78Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
27.78Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.78Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
27.78Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
27.78Single8JXRLSD8JXR-D1-LSD
27.78Single8K5DGSK2560738K5D-HCA2-GSK256073
27.78Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
27.78Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
27.78Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
27.78Single8T1WCVN4248T1W-GPR6-CVN424
27.78Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
27.78Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
27.78Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
27.78Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
27.78Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
27.78Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
27.78Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
27.78Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
27.78Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
27.78Single9CHXS-Carazolol9CHX-β2-S-Carazolol
27.78Single9H37A1IR09H37-A2A-A1IR0-Na
27.78Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
27.78Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
27.78Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
27.78Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
27.78Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
27.78Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
27.78Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
27.78Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
27.78Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
27.78Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
27.59Single5GLHEndothelin-15GLH-ETB-Endothelin-1
27.59Single6IGKEndothelin-36IGK-ETB-Endothelin-3
27.59Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
27.59Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
27.59Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
27.59Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
27.59Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
27.59Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
27.27Single5WF6UK-4320975WF6-A2A-UK-432097
27.27Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
27.27Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
27.27Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
27.27Single6PT3DPI-2876PT3-δ-DPI-287
27.27Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
27.27Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
27.27Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
27.27Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
27.27Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
27.27Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
27.27Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.27Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
27.27Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
27.27Single8X5YAstemizole8X5Y-H1-Astemizole
27.27Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
27.27Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
27.27Single9IPYJR14a9IPY-C3aB-JR14a
27.27Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
27.27Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
26.92Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
26.92Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
26.92Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
26.92Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
26.92Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
26.92Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
26.92Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
26.92Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
26.92Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
26.92Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
26.92Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
26.92Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
26.67Single3OE6IT1t3OE6-CXCR4-IT1t
26.67Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
26.67Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
26.67Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
26.67Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
26.67Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
26.67Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
26.67Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.67Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
26.67Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
26.67Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
26.67Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
26.67Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
26.67Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
26.67Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
26.47Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
26.32Single2Y03Isoprenaline2Y03-β1-Isoprenaline
26.32Single4JKVTaladegib4JKV-SMO-Taladegib
26.32Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
26.32Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
26.32Single5IUAQ274563485IUA-A2A-Q27456348-Na
26.32Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
26.32Single5WQCEMPA5WQC-OX2-EMPA
26.32Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
26.32Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
26.32Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
26.32Single6D26Fevipiprant6D26-DP2-Fevipiprant
26.32Single6E67BI1671076E67-β2-BI167107-Gs(CT)
26.32Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
26.32Single6GPXMK08126GPX-CCR2-MK0812
26.32Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
26.32Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
26.32Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
26.32Single6S0QZM-2413856S0Q-A2A-ZM-241385
26.32Single6TP6Filorexant6TP6-OX1-Filorexant
26.32Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
26.32Single7C61Ergotamine7C61-5-HT1B-Ergotamine
26.32Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
26.32Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
26.32Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
26.32Single7WC6LSD7WC6-5-HT2A-LSD
26.32Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.32Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
26.32Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
26.32Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
26.32Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
26.32Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
26.32Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
26.32Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
26.32Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.32Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
26.32Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
26.32Single8S4DCMF-0198S4D-Apelin-CMF-019
26.32Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
26.32Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.32Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.32Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
26.32Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
26.32Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
26.32Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
26.32Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
26.32Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
26.32Single9HAPTolvaptan9HAP-V2-Tolvaptan
26.32Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
26.32Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
26.32Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
26.32Consensusadenosine_offOrthosteric Liganda1_off a2_off
26.32Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
26.32Consensusblt_offOrthosteric Ligandblt1_off
26.32Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
26.32Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
26.32Consensusdp_offOrthosteric Liganddp2_off
26.32Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
26.32Consensusep_offOrthosteric Ligandep4_off
26.32Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
26.32Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
26.32Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
26.32Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
26.32Consensustrace-amine_onOrthosteric Ligandta1_on
26.09Single4IARErgotamine4IAR-5-HT1B-Ergotamine
26.09Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
26.09Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
26.09Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
26.09Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
26.09Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
26.09Single8KIGSHU91198KIG-MC3-SHU9119-Ca
26.09Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
26.09Single8XWNCXCL88XWN-CXCR2-CXCL8
26.09Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
26.09Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
26.09Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
26.09Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
26.09Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
26.09Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
26.09Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
26.09Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
26.09Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
26.09Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
25.93Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
25.93Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
25.93Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
25.93Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
25.93Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
25.93Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
25.93Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
25.93Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
25.93Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
25.93Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
25.93Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
25.81Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
25.81Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.81Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
25.00Single2YDVNECA2YDV-A2A-NECA
25.00Single3OE9IT1t3OE9-CXCR4-IT1t
25.00Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
25.00Single4UHRCGS216804UHR-A2A-CGS21680
25.00Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
25.00Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
25.00Single5G53NECA5G53-A2A-NECA-Gs
25.00Single5L7IVismodegib5L7I-SMO-Vismodegib
25.00Single5TZRMK86665TZR-FFA1-MK8666
25.00Single5V56TC1145V56-SMO-TC114
25.00Single5V57TC1145V57-SMO-TC114
25.00Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
25.00Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
25.00Single6H7JIsoprenaline6H7J-β1-Isoprenaline
25.00Single6J21Aprepitant6J21-NK1-Aprepitant
25.00Single6LI0C176LI0-GPR52-C17
25.00Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
25.00Single6OS1TRV0266OS1-AT1-TRV026
25.00Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
25.00Single6TQ7SB-3348676TQ7-OX1-SB-334867
25.00Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
25.00Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
25.00Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
25.00Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
25.00Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
25.00Single7PX4PSB-21137PX4-A2A-PSB-2113
25.00Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
25.00Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
25.00Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
25.00Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
25.00Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
25.00Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
25.00Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
25.00Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
25.00Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
25.00Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
25.00Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
25.00Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single7XNACYN1548067XNA-SST2-CYN154806
25.00Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
25.00Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
25.00Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
25.00Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
25.00Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
25.00Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
25.00Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
25.00Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
25.00Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
25.00Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
25.00Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
25.00Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
25.00Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
25.00Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
25.00Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
25.00Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
25.00Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
25.00Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
25.00Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
25.00Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
25.00Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
25.00Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
25.00Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
25.00Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
25.00Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
25.00Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
25.00Single8ZWFJR14a8ZWF-C3aB-JR14a
25.00Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
25.00Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
25.00Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
25.00Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
25.00Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
25.00Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
25.00Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
25.00Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
25.00Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
25.00Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
25.00Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
25.00Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
25.00Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
25.00Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
25.00Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
25.00Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
25.00Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
25.00Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
25.00Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
25.00Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
25.00Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
25.00Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
25.00Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
25.00Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
25.00Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
25.00Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
25.00Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
25.00Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
25.00Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
25.00Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
25.00Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
24.24Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
24.14Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
24.14Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
24.14Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
24.14Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
24.14Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
24.14Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
24.14Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
24.14Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
24.14Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
24.14Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
24.14Consensusendothelin_onOrthosteric Ligandetb_on eta_on
24.14Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
24.00Single5WF5UK-4320975WF5-A2A-UK-432097
24.00Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
24.00Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
24.00Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
24.00Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
24.00Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
24.00Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
24.00Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
24.00Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
24.00Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
24.00Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
24.00Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
23.81Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
23.81Single4N4WSANT-14N4W-SMO-SANT-1
23.81Single5X33BIIL2605X33-BLT1-BIIL260
23.81Single6CM4Risperidone6CM4-D2-Risperidone
23.81Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
23.81Single6OS2TRV0266OS2-AT1-TRV026
23.81Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
23.81Single6ZG4HTL00099366ZG4-M1-HTL0009936
23.81Single7DFPSpiperone7DFP-D2-Spiperone
23.81Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
23.81Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
23.81Single7K15MKD0467K15-BLT1-MKD046-Na
23.81Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
23.81Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
23.81Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
23.81Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
23.81Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
23.81Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
23.81Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.81Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
23.81Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
23.81Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
23.81Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
23.81Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
23.81Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
23.81Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
23.81Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
23.81Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
23.81Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
23.81Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
23.81Single9BJKNAM9BJK-μ-Naloxone-NAM
23.81Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
23.81Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
23.81Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
23.81Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
23.81Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
23.81Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
23.81Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
23.81Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
23.81Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
23.81Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
23.81Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
23.81Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
23.81Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
23.81Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
23.81Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
23.81Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
23.53Single3ODUIT1t3ODU-CXCR4-IT1t
23.53Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
23.53Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
23.53Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
23.53Single5WS3EMPA5WS3-OX2-EMPA
23.53Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
23.53Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
23.53Single6ME2Ramelteon6ME2-MT1-Ramelteon
23.53Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
23.53Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
23.53Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
23.53Single6TODEMPA6TOD-OX1-EMPA-Na
23.53Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
23.53Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
23.53Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
23.53Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
23.53Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
23.53Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
23.53Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
23.53Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
23.53Single7XRRLemborexant7XRR-OX2-Lemborexant
23.53Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
23.53Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
23.53Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.53Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.53Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.53Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
23.53Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
23.53Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
23.53Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
23.53Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
23.53Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
23.53Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
23.53Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
23.53Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
23.53Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
23.53Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
23.53Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.53Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.53Single8Y0HVUF114188Y0H-CXCR3-VUF11418
23.53Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
23.53Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
23.53Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
23.53Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
23.53Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
23.53Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
23.53Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
23.53Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
23.53Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
23.33Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
23.33Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
23.33Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
23.33Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
23.33Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
23.33Consensusbombesin_onOrthosteric Ligandbb2_on
23.33Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
23.33Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
23.33Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
23.33Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
23.08Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
23.08Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
23.08Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
23.08Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
23.08Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
23.08Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
23.08Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.08Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
23.08Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
23.08Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
23.08Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
22.73Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
22.73Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
22.73Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
22.73Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
22.73Single6H7LDobutamine6H7L-β1-Dobutamine
22.73Single6IBLArformoterol6IBL-β1-Arformoterol
22.73Single6K1QIRL25006K1Q-ETB-IRL2500
22.73Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
22.73Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
22.73Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
22.73Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
22.73Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
22.73Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
22.73Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
22.73Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
22.73Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
22.73Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
22.73Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.73Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
22.73Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
22.73Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.73Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
22.73Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
22.73Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
22.73Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
22.73Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
22.73Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
22.73Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
22.73Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
22.73Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
22.73Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
22.73Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
22.73Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
22.73Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
22.73Consensuscck_onOrthosteric Ligandccka_on cckb_on
22.73Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
22.73Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
22.73Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
22.73Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
22.73Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.73Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.73Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
22.58Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
22.58Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
22.58Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
22.58Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
22.58Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
22.22Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
22.22Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
22.22Single5IU7Q274563465IU7-A2A-Q27456346-Na
22.22Single5JTBZM-2413855JTB-A2A-ZM-241385
22.22Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
22.22Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
22.22Single6MH8ZM-2413856MH8-A2A-ZM-241385
22.22Single6PS0S-Carazolol6PS0-β2-S-Carazolol
22.22Single6PS4ICI118-5516PS4-β2-ICI118-551
22.22Single6PS5S-Propranolol6PS5-β2-S-Propranolol
22.22Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
22.22Single6TPNHTL66416TPN-OX2-HTL6641
22.22Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
22.22Single6VI4JDTic6VI4-κ-JDTic
22.22Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
22.22Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
22.22Single6ZG9GSK10347026ZG9-M1-GSK1034702
22.22Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
22.22Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
22.22Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
22.22Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
22.22Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
22.22Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
22.22Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
22.22Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
22.22Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.22Single7UL3Famotidine7UL3-H2-Famotidine
22.22Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
22.22Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
22.22Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
22.22Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
22.22Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
22.22Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
22.22Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
22.22Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
22.22Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
22.22Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
22.22Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
22.22Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
22.22Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
22.22Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.22Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.22Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.22Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
22.22Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
22.22Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
22.22Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
22.22Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
22.22Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
22.22Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
22.22Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
22.22Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
22.22Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
22.22Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
22.22Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
22.22Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
22.22Single8RLNLUF58348RLN-A2A-LUF5834
22.22Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
22.22Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
22.22Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
22.22Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.22Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.22Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.22Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.22Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
22.22Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
22.22Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
22.22Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
22.22Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
22.22Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
22.22Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single8ZPMAMD0708ZPM-CXCR4-AMD070
22.22Single8ZPNAMD31008ZPN-CXCR4-AMD3100
22.22Single9ARXSerotonin9ARX-5-HT2A-Serotonin
22.22Single9BA0A1AKN9BA0-CB1-A1AKN
22.22Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
22.22Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
22.22Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
22.22Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
22.22Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
22.22Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
22.22Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
22.22Consensusa2_offOrthosteric Liganda2a_off
22.22Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
22.22Consensusalpha1_onOrthosteric Ligandalpha1a_on
22.22Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
22.22Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
22.22Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
22.22Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
22.22Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
22.22Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
22.22Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
22.22Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
22.22Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
22.22Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
22.22Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
22.22Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
21.88Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
21.88Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
21.88Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
21.88Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
21.88Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
21.88Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
21.88Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
21.74Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
21.74Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
21.74Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
21.74Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
21.74Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
21.74Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
21.74Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
21.74Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
21.74Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
21.74Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
21.74Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
21.74Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
21.74Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
21.74Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
21.74Consensuskisspeptin_onOrthosteric Ligandkiss1_on
21.74Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single6FJ3PTH6FJ3-PTH1-PTH
21.43Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
21.43Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
21.43Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
21.43Single7SK3CXCL127SK3-ACKR3-CXCL12
21.43Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
21.43Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
21.43Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
21.43Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
21.43Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
21.43Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
21.43Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
21.43Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
21.43Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
21.21Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
21.21Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
21.05Single2Y01Dobutamine2Y01-β1-Dobutamine
21.05Single3EMLZM-2413853EML-A2A-ZM-241385
21.05Single3NY8ICI118-5513NY8-β2-ICI118-551
21.05Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
21.05Single4GBRS-Carazolol4GBR-β2-S-Carazolol
21.05Single4QKX35V4QKX-β2-35V
21.05Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
21.05Single5DHGC-355DHG-NOP-C-35
21.05Single5DHHSB-6121115DHH-NOP-SB-612111
21.05Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
21.05Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
21.05Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
21.05Single5TGZAM65385TGZ-CB1-AM6538
21.05Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
21.05Single6DRXLisuride6DRX-5-HT2B-Lisuride
21.05Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
21.05Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
21.05Single6H7MSalbutamol6H7M-β1-Salbutamol
21.05Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
21.05Single6PS1Timolol6PS1-β2-Timolol
21.05Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
21.05Single6S0LZM-2413856S0L-A2A-ZM-241385
21.05Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
21.05Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
21.05Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
21.05Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
21.05Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
21.05Single7BU7BI1671077BU7-β1-BI167107
21.05Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
21.05Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
21.05Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
21.05Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
21.05Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
21.05Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
21.05Single7WC7Lisuride7WC7-5-HT2A-Lisuride
21.05Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
21.05Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
21.05Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
21.05Single8CU6LJ-45178CU6-A2A-LJ-4517
21.05Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
21.05Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
21.05Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
21.05Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
21.05Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
21.05Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
21.05Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.05Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.05Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.05Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.05Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.05Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.05Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.05Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.05Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.05Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.05Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
21.05Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
21.05Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
21.05Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
21.05Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
21.05Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
21.05Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
21.05Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
21.05Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
21.05Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
21.05Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
21.05Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
21.05Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
21.05Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
21.05Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.05Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.05Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.05Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.05Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
21.05Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
21.05Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
21.05Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
21.05Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
21.05Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
21.05Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
21.05Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
21.05Single9IYAONO-97105319IYA-GPR55-ONO-9710531
21.05Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
21.05Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
21.05Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
21.05Consensus5ht5_onOrthosteric Ligand5ht5a_on
21.05Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
21.05Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
21.05Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
21.05Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
21.05Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
21.05Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
21.05Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
21.05Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
21.05Consensusdopamine_offOrthosteric Ligandd2_off d3_off
21.05Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
21.05Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
21.05Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
21.05Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
21.05Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
20.83Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
20.83Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
20.83Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
20.83Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
20.83Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
20.83Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
20.83Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
20.83Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
20.83Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
20.83Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
20.83Single8IEBA1LYA8IEB-GPR156-A1LYA
20.83Single8IEIA1LYA8IEI-GPR156-A1LYA
20.83Single8IEPA1LYA8IEP-GPR156-A1LYA
20.83Single8IEPA1LYA8IEP-GPR156-A1LYA
20.83Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
20.83Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
20.83Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
20.83Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
20.83Single9M4TSilodosin9M4T-Alpha1A-Silodosin
20.83Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
20.83Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
20.83Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
20.83Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
20.83Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
20.83Consensussomatostatin_offOrthosteric Ligandsst2_off
20.69Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
20.69Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
20.69Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
20.69Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
20.69Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
20.69Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
20.69Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
20.00Single2RH1S-Carazolol2RH1-β2-S-Carazolol
20.00Single2Y00Dobutamine2Y00-β1-Dobutamine
20.00Single2YCWS-Carazolol2YCW-β1-S-Carazolol
20.00Single3OE8IT1t3OE8-CXCR4-IT1t
20.00Single3RFMCaffeine3RFM-A2A-Caffeine
20.00Single4NTJAZD12834NTJ-P2Y12-AZD1283
20.00Single5D6LS-Carazolol5D6L-β2-S-Carazolol
20.00Single5JQHS-Carazolol5JQH-β2-S-Carazolol
20.00Single5N2RPSB-365N2R-A2A-PSB-36-Na
20.00Single5N2SPSB365N2S-A1-PSB36
20.00Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
20.00Single5TVNLSD5TVN-5-HT2B-LSD
20.00Single5WIUNemonapride5WIU-D4-Nemonapride
20.00Single5WIVNemonapride5WIV-D4-Nemonapride-Na
20.00Single5XPRBosentan5XPR-ETB-Bosentan
20.00Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
20.00Single6HLOAprepitant6HLO-NK1-Aprepitant
20.00Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
20.00Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
20.00Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
20.00Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
20.00Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
20.00Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
20.00Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
20.00Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
20.00Single6TQ9SB-4081246TQ9-OX1-SB-408124
20.00Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
20.00Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
20.00Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
20.00Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
20.00Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
20.00Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
20.00Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
20.00Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
20.00Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
20.00Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8A2OTheophylline8A2O-A2A-Theophylline-Na
20.00Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
20.00Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
20.00Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8GNEKW-63568GNE-A2A-KW-6356-Na
20.00Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
20.00Single8IEBA1LYA8IEB-GPR156-A1LYA
20.00Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
20.00Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
20.00Single8IY6Endothelin-18IY6-ETB-Endothelin-1
20.00Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
20.00Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
20.00Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
20.00Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
20.00Single8QOTNanobody-E8QOT-μ-Nanobody-E
20.00Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
20.00Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
20.00Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
20.00Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
20.00Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
20.00Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
20.00Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9B9ZA1AKO9B9Z-CB1-A1AKO
20.00Single9CHUNoradrenaline9CHU-β2-Noradrenaline
20.00Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
20.00Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
20.00Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
20.00Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
20.00Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
20.00Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
20.00Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
20.00Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
20.00Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
20.00Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
20.00Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
20.00Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
20.00Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
20.00Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
20.00Consensusamine_offonOrthosteric Ligandamine_off amine_on
20.00Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
20.00Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
20.00Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
20.00Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
20.00Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
20.00Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
20.00Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
20.00Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
20.00Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
20.00Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
20.00Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
20.00Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
20.00Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
20.00Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
20.00Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
19.44Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
19.35Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
19.23Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
19.23Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
19.23Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
19.23Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
19.23Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
19.23Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
19.23Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
19.23Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
19.05Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
19.05Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
19.05Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
19.05Single4BV0Neurotensin4BV0-NTS1-Neurotensin
19.05Single4U15Tiotropium4U15-M3-Tiotropium
19.05Single5D5AS-Carazolol5D5A-β2-S-Carazolol
19.05Single5D5BS-Carazolol5D5B-β2-S-Carazolol
19.05Single5V54Methiothepin5V54-5-HT1B-Methiothepin
19.05Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
19.05Single6E59L-7607356E59-NK1-L-760735
19.05Single6J20Aprepitant6J20-NK1-Aprepitant
19.05Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
19.05Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
19.05Single6OL9Tiotropium6OL9-M5-Tiotropium
19.05Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
19.05Single6WGTLSD6WGT-5-HT2A-LSD
19.05Single7B6WCyclazosin7B6W-α1b-Cyclazosin
19.05Single7F1TMIP-1a7F1T-CCR5-MIP-1a
19.05Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
19.05Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
19.05Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
19.05Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
19.05Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.05Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
19.05Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
19.05Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
19.05Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
19.05Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
19.05Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
19.05Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
19.05Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
19.05Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
19.05Single8XVLZibotentan8XVL-ETA-Zibotentan
19.05Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
19.05Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
19.05Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
19.05Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
19.05Consensus5ht1_offOrthosteric Ligand5ht1b_off
19.05Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
19.05Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
19.05Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
19.05Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
19.05Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
19.05Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
19.05Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
19.05Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
19.05Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
19.05Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
19.05Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
19.05Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
19.05Consensusneurotensin_onOrthosteric Ligandnts1_on
19.05Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
19.05Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
19.05Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
18.75Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
18.75Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
18.75Single6ME5Agomelatine6ME5-MT1-Agomelatine
18.75Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
18.75Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
18.75Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
18.75Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
18.75Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
18.75Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
18.75Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
18.75Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
18.75Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
18.75Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
18.75Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
18.75Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
18.75Single9LRCHistamine9LRC-H4-Histamine
18.75Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
18.75Consensus5ht2_onOrthosteric Ligand5ht2b_on
18.75Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.75Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
18.75Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
18.75Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
18.75Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
18.52Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
18.52Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
18.52Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
18.52Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
18.52Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
18.52Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
18.52Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
18.52Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
18.18Single3D4STimolol3D4S-β2-Timolol
18.18Single4AMIBucindolol4AMI-β1-Bucindolol
18.18Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
18.18Single4XEENeurotensin4XEE-NTS1-Neurotensin
18.18Single4XESNeurotensin4XES-NTS1-Neurotensin
18.18Single5CXVTiotropium5CXV-M1-Tiotropium
18.18Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
18.18Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
18.18Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
18.18Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
18.18Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
18.18Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
18.18Single6YVRNTS8-136YVR-NTS1-NTS8-13
18.18Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
18.18Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
18.18Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
18.18Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.18Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
18.18Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
18.18Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.18Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
18.18Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
18.18Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
18.18Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
18.18Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.18Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
18.18Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
18.18Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
18.18Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
18.18Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.18Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.18Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
18.18Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
18.18Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
18.18Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
18.18Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
18.18Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
18.18Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
18.18Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
18.18Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
18.18Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
18.18Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
18.18Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.18Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.86Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
17.86Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
17.86Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.86Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
17.86Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
17.86Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
17.86Consensuspac_onOrthosteric Ligandpac1_on
17.86Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
17.65Single6HLLCP999946HLL-NK1-CP99994
17.65Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
17.65Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
17.65Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
17.65Single7SRQLSD7SRQ-5-HT2B-LSD
17.65Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
17.65Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
17.65Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
17.65Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
17.65Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.65Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
17.65Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
17.65Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
17.65Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
17.65Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
17.65Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.65Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
17.65Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
17.65Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
17.65Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
17.65Single9B9Y7DY9B9Y-CB1-7DY
17.65Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
17.65Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
17.65Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
17.65Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
17.65Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
17.65Consensusgq_nucleotideOrthosteric Ligandgq_p2y
17.65Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
17.65Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
17.50Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
17.39Single4BUONeurotensin4BUO-NTS1-Neurotensin
17.39Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
17.39Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
17.39Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
17.39Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
17.39Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
17.39Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
17.39Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
17.39Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.39Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Single8XVJMacitentan8XVJ-ETA-Macitentan
17.39Single8XVUCXCL28XVU-CXCR2-CXCL2
17.39Single8XWFCXCL38XWF-CXCR2-CXCL3
17.39Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
17.39Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
17.39Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
17.39Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.39Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Consensuschemerin_onOrthosteric Ligandcml1_on
17.39Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
17.39Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
17.39Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
17.39Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
17.24Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
17.24Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
17.24Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
17.24Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
17.24Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
17.14Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
16.67Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
16.67Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
16.67Single4BWBNeurotensin4BWB-NTS1-Neurotensin
16.67Single4S0VSuvorexant4S0V-OX2-Suvorexant
16.67Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
16.67Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
16.67Single5U09Taranabant5U09-CB1-Taranabant
16.67Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
16.67Single6DS0Ly2660976DS0-5-HT2B-Ly266097
16.67Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
16.67Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
16.67Single6ME9Ramelteon6ME9-MT2-Ramelteon
16.67Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
16.67Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
16.67Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
16.67Single6TPJSuvorexant6TPJ-OX2-Suvorexant
16.67Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
16.67Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
16.67Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
16.67Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
16.67Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
16.67Single7F8YDevazepide7F8Y-CCKA-Devazepide
16.67Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
16.67Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
16.67Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
16.67Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
16.67Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
16.67Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
16.67Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
16.67Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
16.67Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
16.67Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
16.67Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
16.67Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
16.67Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
16.67Single7XN9L-054,5227XN9-SST2-L-054,522
16.67Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
16.67Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
16.67Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
16.67Single8GNGIstradefylline8GNG-A2A-Istradefylline
16.67Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
16.67Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
16.67Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
16.67Single8IWESpermidine8IWE-TA9-Spermidine
16.67Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
16.67Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
16.67Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
16.67Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
16.67Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
16.67Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
16.67Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
16.67Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
16.67Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
16.67Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
16.67Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
16.67Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
16.67Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
16.67Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
16.67Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
16.67Single9H2XA1IR19H2X-A2A-A1IR1-Na
16.67Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
16.67Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
16.67Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
16.67Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
16.67Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
16.67Consensusalpha2_offOrthosteric Ligandalpha2c_off
16.67Consensusangiotensin_offOrthosteric Ligandat1_off
16.67Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
16.67Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
16.67Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
16.67Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
16.67Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
16.67Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
16.67Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
16.67Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
16.67Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
16.67Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
16.67Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
16.13Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
16.13Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
16.13Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
16.13Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
16.13Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
16.00Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
16.00Single7F8XNN90567F8X-CCKA-NN9056
16.00Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
16.00Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.00Single8IEIA1LYA8IEI-GPR156-A1LYA
16.00Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.00Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
16.00Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
16.00Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
16.00Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
16.00Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
15.79Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
15.79Single2YDOAdenosine2YDO-A2A-Adenosine
15.79Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
15.79Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
15.79Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
15.79Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
15.79Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
15.79Single5UVIZM-2413855UVI-A2A-ZM-241385
15.79Single6A94Zotepine6A94-5-HT2A-Zotepine
15.79Single6IQLL7458706IQL-D4-L745870
15.79Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
15.79Single6KUXRS-799486KUX-α2a-RS-79948
15.79Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
15.79Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
15.79Single6TP3Nemorexant6TP3-OX1-Nemorexant
15.79Single6TPKRetosiban6TPK-OT-Retosiban
15.79Single6V9SGTPL114036V9S-OX1-GTPL11403
15.79Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
15.79Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
15.79Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
15.79Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
15.79Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
15.79Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
15.79Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
15.79Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
15.79Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
15.79Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
15.79Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
15.79Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
15.79Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
15.79Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.79Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
15.79Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
15.79Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
15.79Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
15.79Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
15.79Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
15.79Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
15.79Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.79Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.79Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
15.79Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.79Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
15.79Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
15.79Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
15.79Single9AS5Mescaline9AS5-5-HT2A-Mescaline
15.79Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
15.79Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
15.79Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
15.79Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
15.79Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
15.79Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
15.79Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
15.79Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
15.79Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
15.79Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
15.79Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
15.79Consensusvasop-oxy_offOrthosteric Ligandot_off
15.62Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
15.62Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
15.62Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
15.38Single7SK5CXCL127SK5-ACKR3-CXCL12
15.38Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
15.38Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
15.15Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
15.15Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
15.00Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
15.00Single2Y02Carmoterol2Y02-β1-Carmoterol
15.00Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
15.00Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
15.00Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
15.00Single4DAJTiotropium4DAJ-M3-Tiotropium
15.00Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
15.00Single4MQSIperoxo4MQS-M2-Iperoxo
15.00Single4U14Tiotropium4U14-M3-Tiotropium
15.00Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
15.00Single5DSGTiotropium5DSG-M4-Tiotropium
15.00Single5T04Neurotensin5T04-NTS1-Neurotensin
15.00Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
15.00Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
15.00Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
15.00Single6D27CAY104716D27-DP2-CAY10471
15.00Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
15.00Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
15.00Single6IIVDaltroban6IIV-TXA2-Daltroban
15.00Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
15.00Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
15.00Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.00Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
15.00Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
15.00Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
15.00Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
15.00Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
15.00Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
15.00Single8JJOAlprenolol8JJO-β2-Alprenolol
15.00Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
15.00Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
15.00Single8X63Mepyramine8X63-H1-Mepyramine
15.00Single8X64Desloratadine8X64-H1-Desloratadine
15.00Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
15.00Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
15.00Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
15.00Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
15.00Single9AS1DMT9AS1-5-HT2A-DMT
15.00Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
15.00Single9JEAAtropine9JEA-M1-Atropine
15.00Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
15.00Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
15.00Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
15.00Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
15.00Consensusalpha2_onOrthosteric Ligandalpha2b_on
15.00Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
15.00Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
15.00Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
15.00Consensuscck_offOrthosteric Ligandccka_off
15.00Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
15.00Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
15.00Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
15.00Consensushistamine_offOrthosteric Ligandh1_off
15.00Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
15.00Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
15.00Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
14.81Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
14.81Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
14.81Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
14.81Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
14.81Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
14.29Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
14.29Single6HLPNetupitant6HLP-NK1-Netupitant
14.29Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
14.29Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
14.29Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
14.29Single6PS6Timolol6PS6-β2-Timolol
14.29Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
14.29Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
14.29Single6Z4SSR486926Z4S-NTS1-SR48692
14.29Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
14.29Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
14.29Single7SINNPS-21437SIN-CaS-NPS-2143
14.29Single7SINNPS-21437SIN-CaS-NPS-2143
14.29Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
14.29Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
14.29Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
14.29Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
14.29Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
14.29Single7W41PD1762527W41-BB2-PD176252
14.29Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
14.29Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
14.29Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
14.29Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
14.29Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
14.29Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
14.29Single8ZMFA1L108ZMF-5-HT2C-A1L10
14.29Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
14.29Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
14.29Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
14.29Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
14.29Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
14.29Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
14.29Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
14.29Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
14.29Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
14.29Consensusbombesin_offOrthosteric Ligandbb2_off
14.29Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
14.29Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
14.29Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
14.29Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
14.29Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
14.29Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
13.89Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
13.79Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
13.64Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
13.64Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
13.64Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
13.64Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
13.64Single8EA0Iperoxo8EA0-M3-Iperoxo
13.64Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
13.64Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
13.64Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
13.64Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
13.64Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
13.64Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.64Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
13.64Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
13.64Consensustachykinin_offOrthosteric Ligandnk1_off
13.51Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
13.33Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
13.33Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
13.33Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
13.33Single8PWNTheophylline8PWN-A2A-Theophylline
13.33Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
13.04Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
13.04Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
13.04Single6IIURamatroban6IIU-TXA2-Ramatroban
13.04Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
13.04Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
13.04Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
13.04Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.04Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
13.04Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
13.04Single8XWACXCL18XWA-CXCR2-CXCL1
13.04Single8XWMCXCL68XWM-CXCR2-CXCL6
13.04Single8XWSCXCL58XWS-CXCR2-CXCL5
12.90Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
12.90Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
12.90Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
12.82Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
12.50Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
12.50Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
12.50Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
12.50Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
12.50Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
12.50Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
12.50Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
12.50Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
12.50Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
12.50Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
12.50Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
12.50Consensusp2y_offOrthosteric Ligandp2y1_off
12.00Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
12.00Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
12.00Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
12.00Single9JF4PD1683689JF4-BB1-PD168368
11.76Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
11.76Single3UZAGTPL92363UZA-A2A-GTPL9236
11.76Single4XNWMRS25004XNW-P2Y1-MRS2500
11.76Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
11.76Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
11.76Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
11.76Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
11.76Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
11.76Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
11.76Single7WC5Psilocin7WC5-5-HT2A-Psilocin
11.76Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.76Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
11.76Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
11.76Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
11.76Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
11.54Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
11.54Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
11.54Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
11.54Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
11.11Single3PBLEticlopride3PBL-D3-Eticlopride
11.11Single4O9RCyclopamine4O9R-SMO-Cyclopamine
11.11Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
11.11Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
11.11Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
11.11Single6TP4ACT-4622066TP4-OX1-ACT-462206
11.11Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
11.11Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
11.11Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
11.11Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
11.11Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
11.11Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
11.11Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
11.11Single7UL2SR486927UL2-NTS1-SR48692-Na
11.11Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
11.11Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
11.11Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
11.11Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
11.11Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
11.11Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
11.11Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
11.11Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
11.11Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.11Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single9AS7Psilocin9AS7-5-HT2A-Psilocin
11.11Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
11.11Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
11.11Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
11.11Consensusneurotensin_offOrthosteric Ligandnts1_off
11.11Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
10.53Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
10.53Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
10.53Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
10.53Single4QINSAG1.54QIN-SMO-SAG1.5
10.53Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
10.53Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
10.53Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
10.53Single7BR3Elagolix7BR3-GnRH1-Elagolix
10.53Single7F8ULintitript7F8U-CCKA-Lintitript
10.53Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
10.53Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
10.53Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
10.53Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
10.53Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
10.53Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
10.53Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
10.53Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
10.53Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
10.53Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
10.53Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
10.53Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
10.53Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
10.53Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
10.53Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
10.53Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
10.53Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
10.34Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
10.34Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
10.00Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
10.00Single3RZECidoxepin3RZE-H1-Cidoxepin
10.00Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
10.00Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
10.00Single6ZINSR486926ZIN-NTS1-SR48692
10.00Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
10.00Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
10.00Single7VV6C48/807VV6-MRGPRX2-C48/80
10.00Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
10.00Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
10.00Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
10.00Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
10.00Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
10.00Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single9AS3LSD9AS3-5-HT2A-LSD
10.00Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
10.00Consensuscalcitonin_onOrthosteric Ligandctlike_on
10.00Consensusgrh_offOrthosteric Ligandgnrh1_off
10.00Consensusopsins_offOrthosteric Ligandrhodopsin_off
10.00Consensussensory_offOrthosteric Ligandopsins_off
9.76Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
9.68Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
9.68Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
9.68Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
9.68Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
9.52Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
9.52Single7F83PF-051904577F83-Ghrelin-PF-05190457
9.52Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
9.52Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
9.52Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
9.52Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
9.52Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
9.52Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
9.38Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
9.09Single5CGCHTL142425CGC-mGlu5-HTL14242
9.09Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
9.09Single6LUQHaloperidol6LUQ-D2-Haloperidol
9.09Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
9.09Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
9.09Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
9.09Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
9.09Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
9.09Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
9.09Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
9.09Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
9.09Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
9.09Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
9.09Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
9.09Single9HC04YI9HC0-mGlu5-4YI
9.09Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
8.70Single7P2L4YI7P2L-mGlu5-4YI
8.70Single7R0CAVP7R0C-V2-AVP-Arrestin2
8.70Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
8.70Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
8.70Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
8.70Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
8.70Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
8.70Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
8.70Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
8.70Single9AS9RS130-1809AS9-5-HT2A-RS130-180
8.70Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single8XQJJN2418XQJ-Apelin-JN241
8.00Single5CGDHTL142425CGD-mGlu5-HTL14242
8.00Single9JH5C16:0 Ceramide9JH5-CysLT2-C16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single6KNMJN241-96KNM-Apelin-JN241-9
7.69Single8XQJJN2418XQJ-Apelin-JN241
7.69Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
7.69Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
7.14Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
7.14Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
6.67Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
6.67Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
6.67Single5MZPCaffeine5MZP-A2A-Caffeine-Na
6.67Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
6.25Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
6.25Single7WC4Serotonin7WC4-5-HT2A-Serotonin
6.25Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
6.25Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
6.25Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
5.88Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
5.88Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
5.88Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
5.88Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.88Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
5.88Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
5.88Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
5.88Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
5.88Single9IVMLSN33188399IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
5.88Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
5.88Consensussensory_onOrthosteric Ligandopsins_on
5.56Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
5.56Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
5.56Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
5.56Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
5.56Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
5.56Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
5.56Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
5.56Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
5.56Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
5.56Consensusgi_sensoryOrthosteric Ligandgi_opsins
5.56Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
5.56Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
5.56Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
5.56Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
5.56Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
5.26Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
5.26Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
5.26Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
5.26Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
5.26Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
5.26Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
5.26Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
5.26Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
5.26Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
5.26Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
5.26Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
5.26Single8YKDDehydroepiandrosterone8YKD-ADGRG2-Dehydroepiandrosterone-chim(NtGi1-Gs)/β1/γ2
5.26Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.00Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
5.00Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
5.00Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
5.00Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
5.00Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
5.00Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
5.00Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
5.00Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
4.76Single6FFIMMPEP6FFI-mGlu5-MMPEP
4.76Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
4.76Single7VODCariprazine7VOD-5-HT2A-Cariprazine
4.76Single8IYXYL-3658IYX-GPR34-YL-365
4.76Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
4.55Single6FFHFenobam6FFH-mGlu5-Fenobam
4.35Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
4.35Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
4.17Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
4.17Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB

Consensus Members
Id Members
cannabinoid_on_gp cb2_on_gp
cb1_on_gp
ffa_on_gp ffa2_on_gp
ffa3_on_gp
lpl_on_gp s1p_on_gp
lpa_on_gp
prostanoid_on_gp tp_on_gp
fp-alpha_on_gp
leukotriene_on_gp blt_on_gp
Net Summary
Imin 2.80538
Number of Linked Nodes 1069
Number of Links 1221
Number of Hubs 167
Number of Links mediated by Hubs 674
Number of Communities 25
Number of Nodes involved in Communities 199
Number of Links involved in Communities 276
Path Summary
Number Of Nodes in MetaPath 113
Number Of Links MetaPath 112
Number of Shortest Paths 1997408
Length Of Smallest Path 3
Average Path Length 42.0673
Length of Longest Path 91
Minimum Path Strength 0.257635
Average Path Strength 5.5056
Maximum Path Strength 20.9905
Minimum Path Correlation 0.7005
Average Path Correlation 0.968898
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 1.14943
Average % Of Corr. Nodes 29.6351
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 43.311
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following differences:
Id1st Network2nd Network
lipid_off_on_gplipid_on_gplipid_off
This network is also present in following consensuses:
IdComponents
lipid_offon_gplipid_on_gp
lipid_off
class-a_on_gpsensory_on_gp
alicarboxylic_on_gp
amine_on_gp
lipid_on_gp
nucleotide_on_gp
peptide_on_gp
protein_on_gp



You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

Download lipid_on_gp.zip



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