Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
11x32 2.86562404
21x39 3.22312407
31x43 4.38625427
41x57 2.9795136
52x38 6.08125476
62x42 3.45958677
72x50 5.105509
82x53 3.712527
92x56 5.13875427
102x57 7.40312427
112x60 6.515426
122x64 5.1345525
13E1x50 7.35208628
14E1x52 7.4525406
153x29 8.29938424
163x30 4.47655116
173x33 6.4175504
183x34 3.7385114
193x49 7.9275478
203x50 6.813579
213x51 5.278508
22I2x50 3.52375408
23I2x57 6.683576
244x50 5.573124119
254x56 3.87625404
264x61 7.145404
274x64 7.6425624
284x65 9.86438425
29E2 15.26881323
305x36 9.58424
315x47 5.93055148
325x57 3.69563407
335x58 5.58917679
345x64 5.82375405
356x44 3.9585579
366x48 6.0715529
376x54 4.45424
386x59 8.90187424
39E3 7.20344823
407x27 2.7475423
417x31 5.89375423
427x34 7.12792623
437x38 9.40812425
447x42 6.91625627
457x53 5.2165579
468x50 5.128756138
478x57 2.23125405
48Lig 10.1131620
49G.HN.50 3.71813405
50G.S1.02 5.0975446
51G.S1.06 6.02813448
52G.H1.01 5.61063449
53G.H1.04 3.97875407
54G.S2.03 4.51419
55G.S2.04 3.10625447
56G.S2.06 4.6775449
57G.S2.08 6.32446
58G.S3.03 6.413548
59G.S3.04 8.14313417
60G.S3.06 6.70958617
61G.s3h2.03 4.01562419
62G.H2.03 4.08875619
63G.H2.06 5.84571719
64G.H2.07 5.458509
65G.H2.09 4.63188418
66G.h2s4.01 6.9095519
67G.S4.03 3.23312447
68G.S4.04 4.59125439
69G.S4.06 3.74563437
70G.s4h3.03 5.224168
71G.s4h3.04 6.32875638
72G.H3.01 3.85757169
73G.H3.03 2.29187404
74G.H3.06 3.6195536
75G.H3.09 4.411509
76G.H3.13 6.786254176
77G.H3.17 7.15715
78G.H3.18 5.878134159
79G.S5.03 3.9415549
80G.S5.04 4.29875439
81G.S5.05 4.21542649
82G.S5.06 4.7025438
83G.s5hg.01 4.25375409
84G.HG.01 4.9925436
85G.HG.03 3.585406
86G.HG.04 4.67125438
87G.HG.07 3.90438439
88G.HG.13 3.06062437
89G.hgh4.01 4.66687406
90G.hgh4.02 4.51458638
91G.hgh4.04 3.97563436
92G.hgh4.05 9.6975406
93G.hgh4.08 3.81687406
94G.H4.03 5.31687434
95G.H4.10 8.2025537
96G.H4.12 6.46125434
97G.H4.15 4.974538
98G.h4s6.02 5.643134177
99G.h4s6.12 4.7375402
100G.S6.02 5.64708648
101G.S6.05 6.34188435
102G.s6h5.01 6.03449
103G.s6h5.02 3.47937408
104G.s6h5.05 6.1375449
105G.H5.03 6.06812449
106G.H5.08 5.32893748
107G.H5.23 4.87042674
108G.H5.26 3.7475508
109b.1x2 3.676501
110b.h2x1 5.6175405
111b.h2x5 4.195455
112b.lhb1x6 3.84917653
113b.lhb1x9 2.60187453
114b.lhb1x11 3.596554
115b.l1x3 8.91417699
116b.l1x6 8.3915519
117b.b2x1 6.91958618
118b.b2x3 4.2586
119b.b2x5 7.31958687
120b.b3x4 5.27437499
121b.l3x2 4.875599
122b.b4x2 5.12687408
123b.b4x4 7.0825598
124b.b4x6 10.7317699
125b.l4x2 10.6187484
126b.b5x2 4.98062407
127b.b5x3 5.715799
128b.b5x7 5.85407
129b.l5x1 4.928124198
130b.l5x5 8.34143719
131b.b6x1 3.8805519
132b.b6x5 4.03937406
133b.b7x1 6.07438404
134b.b7x4 3.404384198
135b.l7x2 4.40938419
136b.b8x3 3.82625416
137b.b8x4 5.84625406
138b.l8x3 1.81813403
139b.l9x3 7.0425519
140b.l9x6 4.95718
141b.l9x7 2.973517
142b.b10x5 4.0685519
143b.l10x1 4.38062403
144b.b11x2 4.47125417
145b.b11x4 4.89062419
146b.l11x2 5.5685519
147b.b12x6 10.0805518
148b.l12x3 4.94688405
149b.b13x7 7.09655107
150b.l13x3 8.59955109
151b.l13x7 3.811254109
152b.b14x3 5.38563405
153b.b15x1 6.309374109
154b.b15x2 4.679566
155b.b15x3 4.123134109
156b.l15x1 4.94312417
157b.l15x2 4.59937409
158b.b16x4 12.02564106
159b.b16x6 8.822086108
160b.l16x3 5.889384123
161b.b17x7 8.56063468
162b.l17x3 9.69792669
163b.l17x6 5.704519
164b.b18x3 3.5305568
165b.b18x5 4.567565
166b.l18x1 5.40375816
167b.l18x2 5.21625417
168b.l18x3 9.58875415
169b.b19x2 6.41917666
170b.b19x4 5.731568
171b.l19x1 6.05937419
172b.l19x2 5.2565569
173b.b20x4 8.45917668
174b.b20x6 7.16875666
175b.b21x1 9.14563467
176b.b21x2 2.30083606
177b.b21x5 5.69375414
178b.b21x7 4.92429715
179b.l21x2 7.14563404
180b.b22x5 6.618517
181b.l22x5 6.68659
182b.b23x6 6.21625617
183b.l23x1 7.21375416
184b.b24x4 6.44063416
185b.b24x6 6.80125418
186b.b25x3 6.06188415
187b.b25x6 3.06312413
188b.l25x3 7.9965559
189b.l25x6 7.59143718
190b.b26x3 4.37375406
191b.l27x1 9.17071717
192b.b28x2 4.60375454
193b.b28x3 4.57312497
194b.b28x4 7.72456
195b.b28x6 7.67083659
196g.h1x11 2.29875409
197g.h2x11 8.36813416
198g.ctx3 5.36875609
199g.ctx4 3.21813407
200g.ctx6 2.666556
201g.ctx14 5.61125489
202g.ctx15 6.29938489
203g.ctx16 5.45536788
204I1 4.453550
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
12x56 2x60 14.99624.575YesYes276
22x53 2x56 18.66343.7375YesYes277
32x53 7x46 19.83483.8925YesNo079
42x50 7x46 24.97656.995YesNo099
52x46 2x50 26.74965.4275NoYes099
62x46 3x43 27.00463.8075NoNo098
73x43 7x53 29.26796.1525NoYes089
82x60 Lig 11.97766.7625YesYes260
92x45 4x46 35.848510.42NoNo097
102x42 4x46 39.65662.88YesNo077
112x38 2x42 13.63522.915YesYes767
123x33 4x57 28.03532.67YesNo047
133x34 4x57 28.35883.1025YesNo1147
143x34 4x50 33.20212.5625YesYes1149
152x45 4x50 34.94888.1925NoYes099
164x61 4x64 13.02013.7225YesYes044
173x33 4x61 22.364916.5625YesYes044
182x42 3x49 27.19028.36YesYes778
193x50 7x53 34.56937.2025YesYes799
203x50 G.H5.23 45.13535.915YesYes794
213x49 G.H5.23 13.7445.17YesYes784
223x53 G.H5.23 59.23232.905NoYes784
233x53 G.H5.19 87.23512.345NoNo088
24G.H5.19 I2x50 87.48383.05NoYes088
25G.H5.12 I2x50 87.85645.0175NoYes078
26G.H5.08 G.H5.12 87.95865.13YesNo487
27G.H5.08 G.S3.03 89.30773.215YesYes488
28G.S2.06 G.S3.03 90.18486.43YesYes498
29G.H1.08 G.S2.06 89.83995.6NoYes099
30G.H1.08 G.H5.07 57.75723.01NoNo099
31G.H5.07 G.S5.05 57.16893.82NoYes499
32G.H1.04 G.H1.08 32.23552.9175YesNo079
33G.H1.04 G.S5.07 32.4266.7275YesNo079
34G.S5.07 G.s6h5.01 28.5526.58NoYes099
35G.s6h5.01 G.s6h5.05 58.37463.2525YesYes499
36G.s6h5.02 G.s6h5.05 88.55872.725YesYes089
37G.HG.01 G.s6h5.02 88.67563.6175YesYes068
38G.HG.01 G.S6.05 88.44327.6825YesYes365
39G.S5.06 G.S6.05 88.27284.26YesYes385
40G.S5.04 G.S5.06 88.67054.845YesYes398
41G.S4.04 G.S5.04 92.52442.74YesYes399
42G.H3.08 G.S4.04 99.99725.4325NoYes389
43G.H2.04 G.H3.08 1005.11NoNo098
44G.H2.04 G.H2.07 99.96597.25NoYes099
45G.H2.07 G.h2s4.01 13.28764.26YesYes099
46G.h2s4.01 b.l5x5 11.543111.0275YesYes199
47b.l5x4 b.l5x5 23.7075.56NoYes089
48b.b4x1 b.l5x4 23.50092.785NoNo088
49b.b4x1 b.l5x1 23.29833.42NoYes088
50b.b4x3 b.l5x1 10.19397.2625NoYes1978
51b.b4x3 b.b5x7 10.15743.5675NoYes077
52b.b5x7 b.b5x8 19.42863.39YesNo075
53b.b4x2 b.b5x8 19.0544.185YesNo085
54G.HN.47 b.b4x2 10.20213.8775NoYes058
55G.S5.05 G.s6h5.01 30.18325.5125YesYes499
56G.H5.03 G.S5.05 30.15013.0225YesYes499
57G.H5.03 G.s6h5.05 30.17569.7625YesYes499
58G.H2.07 b.l7x2 58.63522.85YesYes099
59b.l5x5 b.l7x2 12.39846.2625YesYes199
60b.b8x4 b.l5x1 12.07625.86YesYes068
61b.b5x7 b.b8x4 10.0664.535YesYes076
62b.b6x1 b.l7x2 48.15243.8875YesYes199
63b.b2x1 b.b6x1 53.25824.1925YesYes189
64b.b2x1 b.l27x1 30.036211.0925YesYes187
65G.H2.07 G.s3h2.03 28.37694.655YesYes099
66G.s3h2.03 b.l9x6 24.08624.2275YesYes198
67G.H2.06 b.l9x6 20.40684.1775YesYes198
68G.H2.06 b.l19x1 13.60614.1475YesYes199
69G.H2.09 b.b2x1 23.90324.0925YesYes188
70b.l25x6 b.l27x1 15.472513.995YesYes187
71G.H2.09 b.l25x6 15.05472.6275YesYes188
72G.H3.17 b.l23x1 17.59622.7925YesYes156
73b.l23x1 b.l25x6 17.43218.46YesYes168
74b.l17x5 b.l19x1 13.79093.31NoYes069
75b.l17x5 b.l19x2 13.6794.785NoYes069
76b.b20x4 b.l19x2 12.17253.575YesYes689
77b.b20x4 b.b20x6 10.90758.015YesYes686
78b.l21x7 b.l23x1 34.21814.6675NoYes156
79b.b23x6 b.l21x7 30.5553.695YesNo175
80b.b23x6 b.b24x6 23.65667.4775YesYes178
81b.b21x7 b.b24x6 20.90455.545YesYes158
82b.b22x1 b.l25x6 12.85594.53NoYes088
83b.b22x1 b.b22x2 12.65513.6NoNo088
84b.b22x2 b.b26x3 12.46427.1325NoYes086
85b.l13x5 b.l15x1 13.65491.96NoYes057
86b.l13x5 b.l15x2 13.19552.0975NoYes059
87b.b15x5 b.l15x2 12.04554.63NoYes089
88b.b15x5 b.l13x3 11.81535.85NoYes089
89b.b21x7 b.b23x2 11.39294.1025YesNo156
90b.b22x5 b.b23x2 10.605912.785YesNo176
912x38 I2x57 13.877610.35YesYes766
923x53 I2x57 27.87834.145NoYes786
933x49 I2x57 13.727411.315YesYes786
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
2x562x604.5752YesYes7621
2x567x424.372YesYes7722
2x607x387.11252YesYes6512
2x607x427.612YesYes6712
2x60Lig6.76252YesYes6010
2x63E1x503.282NoYes5812
2x63Lig10.2352NoYes5010
2x647x313.26252YesYes5311
2x647x345.1452YesYes5311
2x647x353.0252YesNo5312
2x647x3810.07252YesYes5512
2x64Lig4.16752YesYes5010
3x25E1x504.572NoYes9822
E1x50E23.6052YesYes8321
E1x50E2x5016.652YesNo8922
3x25E24.85252NoYes9321
3x25E2x507.282NoNo9922
3x283x294.70NoYes5421
3x294x6516.552YesYes4511
3x29E2x504.05252YesNo4912
3x29Lig7.8952YesYes4010
4x63E23.482NoYes4321
4x644x655.70752YesYes4521
4x64E222.3552YesYes4321
4x645x364.37252YesYes4422
4x65E2x5212.1652YesNo5411
4x65Lig5.0352YesYes5010
E2E245.822YesYes3311
E2Lig18.2252YesYes3010
E2E2x5124.12252YesNo3411
E2x51Lig8.9152NoYes4010
5x36E2x524.32252YesNo4421
E2x52Lig3.5452NoYes4010
5x35E24.562NoYes2321
5x36E215.9252YesYes4321
5x39E23.95752NoYes5321
5x325x3515.32752NoNo4222
6x516x5512.53752NoNo7622
6x517x343.38752NoYes7321
6x54E34.2852YesYes4321
6x547x345.5252YesYes4321
6x557x343.69752NoYes6321
6x57E35.07750NoYes4321
6x58E34.62752NoYes4311
6x58Lig3.492NoYes4010
E3E34.582YesYes3311
7x30E39.33252NoYes4311
E3Lig22.08252YesYes3010
7x277x305.14752YesNo3421
7x30Lig3.63752NoYes4010
7x317x3510.4652YesNo3312
7x31Lig9.23752YesYes3010
7x347x3816.36252YesYes3512
7x34Lig8.652YesYes3010
7x387x424.0852YesYes5722
5x32E23.83752NoYes4321
7x27E33.06252YesYes3321
4x634x646.5352NoYes4422
E1x49Lig2.5050NoYes5010
3x22E21.9350NoYes3321
7x317x320.612YesNo3112

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
100.00Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
92.86Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
86.67Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
81.25Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
81.25Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
75.00Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
68.75Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
66.67Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
66.67Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
66.67Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
66.67Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
64.29Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
60.00Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
58.82Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
55.56Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
55.56Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
55.56Single6YVRNTS8-136YVR-NTS1-NTS8-13
55.56Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
55.56Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
55.56Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
55.56Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
55.56Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
55.00Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
54.55Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
53.33Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
52.63Single4BUONeurotensin4BUO-NTS1-Neurotensin
52.63Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
50.00Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
50.00Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
50.00Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
50.00Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
50.00Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
50.00Consensusneurotensin_onOrthosteric Ligandnts1_on
50.00Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
47.62Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
47.37Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
47.37Single4XEENeurotensin4XEE-NTS1-Neurotensin
47.37Single4XESNeurotensin4XES-NTS1-Neurotensin
47.37Single6OS2TRV0266OS2-AT1-TRV026
47.37Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
47.37Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
47.37Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
47.37Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
47.37Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
47.06Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
46.67Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
46.67Consensusgq_nucleotideOrthosteric Ligandgq_p2y
46.67Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
45.45Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
45.45Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
45.00Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
45.00Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
45.00Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
44.00Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
44.00Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
44.00Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
43.75Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
43.48Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
43.48Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
43.48Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
43.48Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
43.48Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
42.86Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
42.31Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
42.31Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
42.31Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
42.31Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
42.31Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
42.31Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
42.11Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
42.11Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
42.11Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
42.11Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
42.11Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
42.11Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
41.67Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
41.67Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
41.67Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
41.18Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
41.18Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
41.18Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
41.18Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
40.91Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
40.91Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
40.00Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
40.00Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
40.00Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
40.00Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
40.00Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
40.00Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
40.00Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
40.00Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
39.29Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
39.29Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
39.29Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
39.13Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
39.13Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
39.13Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
39.13Single7XNACYN1548067XNA-SST2-CYN154806
39.13Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
39.13Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
39.13Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
39.13Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
39.13Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
39.13Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
39.13Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
38.89Single5T04Neurotensin5T04-NTS1-Neurotensin
38.89Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
38.89Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
38.89Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
38.89Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
38.89Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
38.46Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
38.46Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
38.46Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
38.46Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
38.46Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
38.10Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
38.10Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
38.10Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
38.10Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
38.10Single8ZPLHF511168ZPL-CXCR4-HF51116
38.10Consensuscck_onOrthosteric Ligandccka_on cckb_on
38.10Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
38.10Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
38.10Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
38.10Consensusprostanoid_offOrthosteric Ligandep_off dp_off
37.93Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
37.50Single3OE9IT1t3OE9-CXCR4-IT1t
37.50Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
37.50Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
37.50Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
37.50Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
37.50Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
37.50Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
37.50Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
37.50Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
37.50Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
37.50Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
37.50Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
37.50Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
37.50Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
37.04Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
37.04Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
36.84Single6D26Fevipiprant6D26-DP2-Fevipiprant
36.84Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
36.84Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
36.84Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
36.84Consensusdp_offOrthosteric Liganddp2_off
36.36Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
36.36Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
36.36Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
36.36Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
36.36Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
36.36Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
36.36Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
36.36Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
36.36Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
36.36Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
36.36Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
36.36Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
36.00Single6JODAngiotensin II6JOD-AT2-Angiotensin II
36.00Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
36.00Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
36.00Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
35.29Single4BWBNeurotensin4BWB-NTS1-Neurotensin
35.29Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
35.29Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
35.29Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
35.29Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
35.29Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
35.00Single4BV0Neurotensin4BV0-NTS1-Neurotensin
35.00Single6OS1TRV0266OS1-AT1-TRV026
35.00Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
35.00Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
35.00Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
35.00Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
35.00Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
35.00Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
35.00Consensusrelaxin_onOrthosteric Ligandrxfp4_on
35.00Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
34.78Single4XT1Fractalkine4XT1-US28-Fractalkine
34.78Single7F8XNN90567F8X-CCKA-NN9056
34.78Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
34.78Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
34.78Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
34.78Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
34.78Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
34.78Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
34.78Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
34.78Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
34.78Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
34.78Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
34.78Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
34.78Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
34.78Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
34.78Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
34.78Consensussomatostatin_offOrthosteric Ligandsst2_off
34.62Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
34.62Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
34.62Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
34.62Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
34.62Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
34.62Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
34.62Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
34.62Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
34.62Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
34.48Single5GLHEndothelin-15GLH-ETB-Endothelin-1
34.48Single6IGKEndothelin-36IGK-ETB-Endothelin-3
34.48Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
34.48Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
34.48Consensusbombesin_onOrthosteric Ligandbb2_on
34.48Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
34.48Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
34.48Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
33.33Single4XT3Fractalkine4XT3-US28-Fractalkine
33.33Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
33.33Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
33.33Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
33.33Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
33.33Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
33.33Single7SK3CXCL127SK3-ACKR3-CXCL12
33.33Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
33.33Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
33.33Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
33.33Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
33.33Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
33.33Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
33.33Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
33.33Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
33.33Single8XWSCXCL58XWS-CXCR2-CXCL5
33.33Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
33.33Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
33.33Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
33.33Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
33.33Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
33.33Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
33.33Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
33.33Consensushca_onOrthosteric Ligandhca2_on
33.33Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
33.33Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
33.33Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
33.33Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
33.33Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
32.26Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
32.14Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
32.14Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
32.14Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
32.14Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
32.00Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
32.00Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
32.00Consensusangiotensin_onOrthosteric Ligandat1_on
32.00Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
32.00Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
32.00Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
32.00Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
32.00Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
31.82Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
31.82Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
31.82Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
31.82Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
31.82Consensuschemerin_onOrthosteric Ligandcml1_on
31.82Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
31.58Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
31.58Single6D27CAY104716D27-DP2-CAY10471
31.58Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
31.58Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
31.58Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
31.58Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
31.58Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
31.58Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
31.58Single8K5DGSK2560738K5D-HCA2-GSK256073
31.58Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
31.58Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
31.58Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
31.58Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
31.58Consensushca_on_gpOrthosteric Ligandhca2_on_gp
31.25Single3OE6IT1t3OE6-CXCR4-IT1t
31.25Single4XNWMRS25004XNW-P2Y1-MRS2500
31.25Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
31.25Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
31.25Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
31.03Single6IGLIRL16206IGL-ETB-IRL1620
31.03Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
31.03Single8IY6Endothelin-18IY6-ETB-Endothelin-1
31.03Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
31.03Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
31.03Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
30.77Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
30.77Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
30.77Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
30.77Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
30.77Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
30.77Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
30.77Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
30.77Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
30.77Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
30.77Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
30.77Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
30.77Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
30.77Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
30.77Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
30.77Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
30.77Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
30.43Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
30.43Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
30.43Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
30.43Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
30.43Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
30.43Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
30.43Single8QJ2pN1628QJ2-MC4-pN162-Gs
30.43Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
30.43Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
30.43Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
30.00Single5N2SPSB365N2S-A1-PSB36
30.00Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
30.00Single6Z4SSR486926Z4S-NTS1-SR48692
30.00Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
30.00Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
30.00Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.00Single8GNEKW-63568GNE-A2A-KW-6356-Na
30.00Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
30.00Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
30.00Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
30.00Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
30.00Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
30.00Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
30.00Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
30.00Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
30.00Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
29.63Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
29.63Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
29.63Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
29.63Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
29.63Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
29.63Single8ZRTET-18ZRT-ETB-ET-1
29.63Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
29.63Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
29.41Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
29.41Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
29.41Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
29.41Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
29.17Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
29.17Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
29.17Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
29.17Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
29.17Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
29.17Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
29.17Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
29.17Single8XWNCXCL88XWN-CXCR2-CXCL8
29.17Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
29.17Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
29.17Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
29.17Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
29.17Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
29.17Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
29.17Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
29.03Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
28.57Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
28.57Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
28.57Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
28.57Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
28.57Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
28.57Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
28.57Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
28.57Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
28.57Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
28.57Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
28.57Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
28.57Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
28.57Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
28.57Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
28.12Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
28.00Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
28.00Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
28.00Single7SK5CXCL127SK5-ACKR3-CXCL12
28.00Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
28.00Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
28.00Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
28.00Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
28.00Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
28.00Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
28.00Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
28.00Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
28.00Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
28.00Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
28.00Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
28.00Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
28.00Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
27.78Single3ODUIT1t3ODU-CXCR4-IT1t
27.78Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
27.78Single7F8YDevazepide7F8Y-CCKA-Devazepide
27.78Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
27.78Single8GNGIstradefylline8GNG-A2A-Istradefylline
27.78Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
27.78Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
27.78Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
27.78Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
27.78Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
27.78Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
27.78Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
27.78Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
27.59Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
27.59Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
27.27Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
27.27Single7K15MKD0467K15-BLT1-MKD046-Na
27.27Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
27.27Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
27.27Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
27.27Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
27.27Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
27.27Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
27.27Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
27.27Single8XWACXCL18XWA-CXCR2-CXCL1
27.27Single8XWMCXCL68XWM-CXCR2-CXCL6
26.92Single3OE0CVX153OE0-CXCR4-CVX15
26.92Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
26.92Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
26.92Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
26.92Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
26.92Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
26.92Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
26.92Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
26.92Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
26.92Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
26.92Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
26.67Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
26.67Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
26.67Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
26.67Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
26.67Consensusbradykinin_onOrthosteric Ligandbk2_on
26.67Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
26.67Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
26.67Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
26.32Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
26.32Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
26.32Single5UVIZM-2413855UVI-A2A-ZM-241385
26.32Single6MH8ZM-2413856MH8-A2A-ZM-241385
26.32Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
26.32Single6ZINSR486926ZIN-NTS1-SR48692
26.32Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
26.32Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
26.32Single8IHKAcifran8IHK-HCA3-Acifran
26.32Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
26.32Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
26.32Single8K5CAcipimox8K5C-HCA2-Acipimox
26.32Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
26.32Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
26.32Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
26.32Single8ZPMAMD0708ZPM-CXCR4-AMD070
26.32Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
26.32Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
26.32Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
26.32Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
26.09Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
26.09Single7EZCUKA7EZC-A2A-UKA
26.09Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
26.09Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
26.09Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
26.09Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
26.09Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
26.09Single8XVUCXCL28XVU-CXCR2-CXCL2
26.09Single8XWFCXCL38XWF-CXCR2-CXCL3
26.09Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
26.09Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
26.09Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
26.09Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
26.09Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
26.09Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
26.09Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
25.93Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
25.93Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
25.93Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
25.93Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
25.93Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
25.93Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
25.81Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
25.71Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
25.71Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
25.00Single3EMLZM-2413853EML-A2A-ZM-241385
25.00Single4YAYZD-71554YAY-AT1-ZD-7155
25.00Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
25.00Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
25.00Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
25.00Single5WF6UK-4320975WF6-A2A-UK-432097
25.00Single6KNMJN241-96KNM-Apelin-JN241-9
25.00Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
25.00Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
25.00Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
25.00Single6S0LZM-2413856S0L-A2A-ZM-241385
25.00Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
25.00Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
25.00Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
25.00Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
25.00Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
25.00Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
25.00Single7V3ZCP559407V3Z-CB1-CP55940
25.00Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
25.00Single7XN9L-054,5227XN9-SST2-L-054,522
25.00Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
25.00Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
25.00Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
25.00Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
25.00Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
25.00Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
25.00Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
25.00Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
25.00Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
25.00Single8XQJJN2418XQJ-Apelin-JN241
25.00Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
25.00Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
25.00Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
25.00Single9H37A1IR09H37-A2A-A1IR0-Na
25.00Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
25.00Single9IPYJR14a9IPY-C3aB-JR14a
25.00Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
25.00Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
25.00Consensuscck_offOrthosteric Ligandccka_off
25.00Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
25.00Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
25.00Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
25.00Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
25.00Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
25.00Consensuskisspeptin_onOrthosteric Ligandkiss1_on
25.00Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
25.00Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
25.00Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
25.00Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
25.00Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
25.00Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
25.00Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
25.00Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
25.00Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensusp2y_offOrthosteric Ligandp2y1_off
25.00Consensuspac_onOrthosteric Ligandpac1_on
24.14Single6FJ3PTH6FJ3-PTH1-PTH
24.14Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
24.14Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
24.14Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
24.14Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
24.14Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
24.00Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
24.00Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
24.00Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
24.00Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
24.00Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
24.00Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
24.00Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
24.00Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
24.00Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
24.00Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
24.00Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
24.00Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
24.00Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
23.81Single5IUAQ274563485IUA-A2A-Q27456348-Na
23.81Single5N2RPSB-365N2R-A2A-PSB-36-Na
23.81Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
23.81Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
23.81Single6S0QZM-2413856S0Q-A2A-ZM-241385
23.81Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
23.81Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
23.81Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
23.81Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
23.81Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
23.81Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
23.81Single8QOTNanobody-E8QOT-μ-Nanobody-E
23.81Single8S4DCMF-0198S4D-Apelin-CMF-019
23.81Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
23.81Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
23.81Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
23.81Single9EHSLUF76029EHS-A3A-LUF7602
23.81Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
23.81Consensusblt_offOrthosteric Ligandblt1_off
23.81Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
23.81Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
23.81Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
23.81Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
23.81Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
23.33Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
23.33Single9KDFRES-701-39KDF-ETB-RES-701-3
23.08Single3QAKUK-4320973QAK-A2A-UK-432097
23.08Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
23.08Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
23.08Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
23.08Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
22.86Consensuspth_onOrthosteric Ligandpth1_on pth2_on
22.73Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
22.73Single7F1TMIP-1a7F1T-CCR5-MIP-1a
22.73Single7FEECP559407FEE-CB1-CP55940-ZCZ011
22.73Single7PX4PSB-21137PX4-A2A-PSB-2113
22.73Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
22.73Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
22.73Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
22.73Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
22.73Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
22.73Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
22.73Single8ZWFJR14a8ZWF-C3aB-JR14a
22.73Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
22.73Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
22.58Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
22.58Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
22.58Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
22.58Consensusendothelin_onOrthosteric Ligandetb_on eta_on
22.22Single5WF5UK-4320975WF5-A2A-UK-432097
22.22Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
22.22Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
22.22Single7UL2SR486927UL2-NTS1-SR48692-Na
22.22Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
22.22Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
22.22Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
22.22Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
22.22Single8K5BNiacin8K5B-HCA2-Niacin
22.22Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
22.22Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
22.22Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
22.22Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
22.22Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
22.22Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
22.22Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
22.22Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
22.22Consensusneurotensin_offOrthosteric Ligandnts1_off
22.22Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
21.95Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
21.88Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
21.88Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
21.88Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
21.74Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
21.74Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
21.74Single6KQICP559406KQI-CB1-CP55940-Org27569
21.74Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
21.74Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
21.74Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
21.74Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
21.74Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.74Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
21.74Single8XQJJN2418XQJ-Apelin-JN241
21.74Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
21.74Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
21.74Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
21.74Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
21.74Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
21.74Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
21.74Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
21.74Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
21.74Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
21.74Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
21.74Consensusorexin_onOrthosteric Ligandox2_on
21.43Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
21.43Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
21.43Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
21.43Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
21.43Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
21.43Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
21.21Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
21.21Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
21.05Single3PWHZM-2413853PWH-A2A-ZM-241385
21.05Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
21.05Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
21.05Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
21.05Single5ZKQABT-4915ZKQ-PAF-ABT-491
21.05Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
21.05Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
21.05Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
21.05Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.05Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
21.05Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
21.05Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
21.05Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
21.05Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
21.05Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
21.05Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
21.05Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
21.05Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
21.05Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
21.05Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
21.05Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
21.05Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
21.05Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
21.05Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
21.05Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
20.83Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
20.83Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
20.83Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
20.83Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.83Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
20.83Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
20.83Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
20.83Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
20.83Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
20.83Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
20.83Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
20.69Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
20.69Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
20.69Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
20.69Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
20.69Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
20.69Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
20.51Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
20.00Single3REYXAC3REY-A2A-XAC
20.00Single4UG2CGS216804UG2-A2A-CGS21680
20.00Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
20.00Single5IU7Q274563465IU7-A2A-Q27456346-Na
20.00Single5IUBQ274563445IUB-A2A-Q27456344-Na
20.00Single5JTBZM-2413855JTB-A2A-ZM-241385
20.00Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
20.00Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
20.00Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
20.00Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
20.00Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
20.00Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
20.00Single7AROLUF58337ARO-A2A-LUF5833-Na
20.00Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
20.00Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
20.00Single7F61PF-036547467F61-H3-PF-03654746
20.00Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
20.00Single7T32ZM-2413857T32-A2A-ZM-241385
20.00Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
20.00Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
20.00Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
20.00Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
20.00Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
20.00Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
20.00Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
20.00Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
20.00Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
20.00Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
20.00Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
20.00Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
20.00Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
20.00Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
20.00Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
20.00Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
20.00Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
20.00Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
20.00Single8ZPNAMD31008ZPN-CXCR4-AMD3100
20.00Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
20.00Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
20.00Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Consensusa2_offOrthosteric Liganda2a_off
20.00Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
20.00Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
20.00Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
20.00Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
20.00Consensusgrh_offOrthosteric Ligandgnrh1_off
19.35Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
19.35Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
19.35Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
19.35Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
19.35Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
19.35Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
19.35Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
19.35Consensusglp_onOrthosteric Ligandglp1_on glp2_on
19.35Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
19.35Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
19.23Single4IARErgotamine4IAR-5-HT1B-Ergotamine
19.23Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
19.23Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
19.23Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
19.23Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
19.23Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
19.23Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
19.23Single8WDTphotoNECA8WDT-A2A-photoNECA
19.23Single8WKYPG-9348WKY-MC4-PG-934
19.23Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.23Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
19.23Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
19.23Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
19.23Consensuslpl_onOrthosteric Ligands1p_on lpa_on
19.23Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
19.23Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
19.23Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
19.05Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
19.05Single5IU8Q274563475IU8-A2A-Q27456347-Na
19.05Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
19.05Single5UIGCmpd-15UIG-A2A-Cmpd-1
19.05Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
19.05Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
19.05Single7PYRPSB-21157PYR-A2A-PSB-2115
19.05Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
19.05Single8CU6LJ-45178CU6-A2A-LJ-4517
19.05Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
19.05Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
19.05Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
19.05Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
19.05Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
19.05Consensusa3_onOrthosteric Liganda3a_on
19.05Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
18.75Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
18.75Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
18.75Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
18.75Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
18.75Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
18.75Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
18.75Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
18.75Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
18.52Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
18.52Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
18.52Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
18.52Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
18.52Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
18.52Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
18.52Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
18.42Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
18.18Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
18.18Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
18.18Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
18.18Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
18.18Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
18.18Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
18.18Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
18.18Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
18.18Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
18.18Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.18Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
18.18Single8JXSPF-61428JXS-D1-PF-6142
18.18Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
18.18Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
18.18Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
18.18Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
18.18Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
18.18Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
18.18Consensusa3_on_gpOrthosteric Liganda3a_on_gp
18.18Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
18.18Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
18.18Consensusadenosine_offOrthosteric Liganda1_off a2_off
17.86Single6PT2KGCHM076PT2-δ-KGCHM07
17.86Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
17.86Single6W25SHU91196W25-MC4-SHU9119-Ca
17.86Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
17.86Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
17.86Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
17.65Single3OE8IT1t3OE8-CXCR4-IT1t
17.65Single8A2OTheophylline8A2O-A2A-Theophylline-Na
17.65Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
17.39Single5TZRMK86665TZR-FFA1-MK8666
17.39Single5XR8AM8415XR8-CB1-AM841
17.39Single5XRAAM115425XRA-CB1-AM11542
17.39Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
17.39Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
17.39Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
17.39Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
17.39Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
17.39Single7B6WCyclazosin7B6W-α1b-Cyclazosin
17.39Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
17.39Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
17.39Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
17.39Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
17.39Single7TUYGSK682753A7TUY-GPR183-GSK682753A
17.39Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
17.39Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
17.39Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
17.39Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
17.39Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
17.39Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
17.39Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
17.39Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
17.39Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
17.39Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
17.39Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
17.39Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
17.39Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
17.39Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
17.39Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
17.39Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
17.39Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
17.39Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
17.39Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Consensusa2_onOrthosteric Liganda2b_on
17.39Consensusa2_on_gpOrthosteric Liganda2b_on_gp
17.39Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
17.39Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
17.39Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
17.39Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
17.39Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
17.39Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
17.39Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
17.24Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
17.24Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
17.24Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
17.24Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
17.24Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
17.24Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
17.24Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
17.24Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
17.24Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
17.24Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
17.24Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
17.24Consensusvasop-oxy_onOrthosteric Ligandv2_on
17.24Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
17.14Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
17.14Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
17.14Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
16.67Single4PY02MeSATP4PY0-P2Y12-2MeSATP
16.67Single4RWADIPP-NH24RWA-δ-DIPP-NH2
16.67Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
16.67Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
16.67Single6ME5Agomelatine6ME5-MT1-Agomelatine
16.67Single6MXTSalmeterol6MXT-β2-Salmeterol
16.67Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
16.67Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
16.67Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
16.67Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
16.67Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
16.67Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
16.67Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
16.67Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
16.67Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
16.67Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
16.67Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
16.67Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
16.67Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
16.67Single8JJLOlodaterol8JJL-β2-Olodaterol
16.67Single8JWY2-1188JWY-A2A-2-118
16.67Single8JWZAB9288JWZ-A2A-AB928-Na
16.67Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
16.67Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
16.67Single8XYIVUF106618XYI-CXCR3-VUF10661
16.67Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
16.67Single9BJKNAM9BJK-μ-Naloxone-NAM
16.67Single9DGIZ85267113509DGI-CB1-Z8526711350
16.67Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
16.67Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
16.67Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
16.67Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
16.67Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
16.67Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
16.67Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
16.67Consensuslpl_offOrthosteric Ligands1p_off lpa_off
16.67Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
16.67Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
16.67Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
16.67Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
16.67Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.22Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
16.13Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
16.13Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
16.13Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
16.13Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
16.13Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
16.13Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
16.13Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
16.13Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
16.00Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
16.00Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
16.00Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
16.00Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
16.00Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
16.00Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
16.00Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
16.00Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
16.00Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
16.00Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
16.00Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
16.00Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
16.00Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
16.00Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
16.00Consensusendothelin_offOrthosteric Ligandetb_off
16.00Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
16.00Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
16.00Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
15.79Single4O9RCyclopamine4O9R-SMO-Cyclopamine
15.79Single5L7IVismodegib5L7I-SMO-Vismodegib
15.79Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
15.79Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
15.79Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
15.62Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
15.62Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
15.62Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
15.62Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
15.62Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
15.62Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
15.38Single5ZTYAM102575ZTY-CB2-AM10257
15.38Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
15.38Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
15.38Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
15.38Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
15.38Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
15.38Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
15.38Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
15.15Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
15.15Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
15.15Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
15.15Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
15.15Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
15.15Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
15.15Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
15.15Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
15.00Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
15.00Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
15.00Single4QINSAG1.54QIN-SMO-SAG1.5
15.00Single6ME9Ramelteon6ME9-MT2-Ramelteon
15.00Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
15.00Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
15.00Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
15.00Single7BR3Elagolix7BR3-GnRH1-Elagolix
15.00Single7F8ULintitript7F8U-CCKA-Lintitript
15.00Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
15.00Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
15.00Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
15.00Single7XRRLemborexant7XRR-OX2-Lemborexant
15.00Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
15.00Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.00Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
15.00Single9H2XA1IR19H2X-A2A-A1IR1-Na
15.00Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
15.00Consensusangiotensin_offOrthosteric Ligandat1_off
15.00Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
14.81Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
14.81Single7QA8Peptide7QA8-STE2-Peptide
14.81Single7QA8Peptide7QA8-STE2-Peptide
14.81Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
14.81Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
14.81Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
14.81Single8KIGSHU91198KIG-MC3-SHU9119-Ca
14.81Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
14.81Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
14.71Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
14.71Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
14.71Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
14.29Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
14.29Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
14.29Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
14.29Single6AQFZM-2413856AQF-A2A-ZM-241385
14.29Single6IQLL7458706IQL-D4-L745870
14.29Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
14.29Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
14.29Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
14.29Single6V9SGTPL114036V9S-OX1-GTPL11403
14.29Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
14.29Single6ZG9GSK10347026ZG9-M1-GSK1034702
14.29Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
14.29Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
14.29Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
14.29Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
14.29Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
14.29Single8IEBA1LYA8IEB-GPR156-A1LYA
14.29Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
14.29Single8K2WAMG4878K2W-CXCR3-AMG487
14.29Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
14.29Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.29Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
14.29Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
14.29Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
14.29Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
14.29Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
14.29Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
14.29Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
14.29Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
14.29Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
14.29Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
13.95Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
13.89Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
13.89Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
13.89Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
13.89Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
13.89Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
13.89Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
13.79Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
13.79Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
13.79Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
13.79Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
13.79Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
13.64Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
13.64Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
13.64Single4QIMANTA XV4QIM-SMO-ANTA XV
13.64Single5DHGC-355DHG-NOP-C-35
13.64Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
13.64Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
13.64Single5UENDU1725UEN-A1-DU172
13.64Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
13.64Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
13.64Single6TOTLemborexant6TOT-OX1-Lemborexant
13.64Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
13.64Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
13.64Single7F83PF-051904577F83-Ghrelin-PF-05190457
13.64Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
13.64Single7UL4Alvimopan7UL4-μ-Alvimopan
13.64Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
13.64Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
13.64Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
13.64Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
13.64Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
13.64Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.64Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
13.64Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
13.64Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
13.64Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
13.64Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
13.64Single9IYAONO-97105319IYA-GPR55-ONO-9710531
13.64Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
13.64Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
13.64Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
13.64Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
13.64Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
13.51Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
13.51Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
13.51Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
13.33Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
13.33Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
13.33Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
13.33Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
13.33Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
13.33Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
13.33Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
13.04Single4JKVTaladegib4JKV-SMO-Taladegib
13.04Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
13.04Single5WIUNemonapride5WIU-D4-Nemonapride
13.04Single5WIVNemonapride5WIV-D4-Nemonapride-Na
13.04Single5WQCEMPA5WQC-OX2-EMPA
13.04Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
13.04Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
13.04Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
13.04Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
13.04Single6LUQHaloperidol6LUQ-D2-Haloperidol
13.04Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
13.04Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
13.04Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
13.04Single7C4SS1P7C4S-S1P3-S1P
13.04Single7C61Ergotamine7C61-5-HT1B-Ergotamine
13.04Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
13.04Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
13.04Single7W41PD1762527W41-BB2-PD176252
13.04Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
13.04Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
13.04Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.04Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
13.04Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
13.04Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
13.04Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
13.04Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
13.04Single8TF5Oleic acid8TF5-GPR6-Oleic acid
13.04Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
13.04Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
13.04Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
13.04Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
13.04Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
13.04Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
13.04Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
13.04Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
13.04Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
13.04Consensusbombesin_offOrthosteric Ligandbb2_off
13.04Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
13.04Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
13.04Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
13.04Consensusep_offOrthosteric Ligandep4_off
13.04Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
13.04Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
13.04Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
12.90Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
12.90Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
12.90Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
12.50Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
12.50Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
12.50Single5V56TC1145V56-SMO-TC114
12.50Single5V57TC1145V57-SMO-TC114
12.50Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
12.50Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
12.50Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
12.50Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
12.50Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
12.50Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
12.50Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
12.50Single7R0CAVP7R0C-V2-AVP-Arrestin2
12.50Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
12.50Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
12.50Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
12.50Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
12.50Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
12.50Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
12.50Single8E0GBU728E0G-μ-BU72
12.50Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
12.50Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
12.50Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
12.50Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
12.50Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
12.50Single8XVLZibotentan8XVL-ETA-Zibotentan
12.50Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
12.50Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
12.50Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
12.50Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
12.50Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
12.50Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
12.50Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
12.50Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
12.50Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
12.50Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
12.50Consensuslpa_onOrthosteric Ligandlpa1_on
12.50Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
12.50Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
12.50Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
12.50Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
12.50Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
12.50Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
12.50Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
12.50Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
12.12Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
12.12Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
12.12Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
12.12Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
12.12Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
12.12Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
12.00Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
12.00Single5X33BIIL2605X33-BLT1-BIIL260
12.00Single6A93Risperidone6A93-5-HT2A-Risperidone
12.00Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
12.00Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
12.00Single6ZG4HTL00099366ZG4-M1-HTL0009936
12.00Single7DFPSpiperone7DFP-D2-Spiperone
12.00Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
12.00Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
12.00Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
12.00Single7YITNalfurafine7YIT-κ-Nalfurafine
12.00Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
12.00Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
12.00Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
12.00Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
12.00Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
12.00Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
12.00Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
12.00Consensusalpha1_offOrthosteric Ligandalpha1a_off
12.00Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
12.00Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
12.00Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
12.00Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
12.00Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
12.00Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
12.00Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
12.00Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
12.00Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
12.00Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
12.00Consensuslpa_offOrthosteric Ligandlpa1_off
12.00Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
12.00Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
12.00Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
12.00Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
12.00Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
11.76Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
11.76Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
11.76Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
11.76Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
11.76Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
11.76Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
11.76Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
11.76Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
11.76Single8PWNTheophylline8PWN-A2A-Theophylline
11.76Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
11.54Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
11.54Single5X93K-87945X93-ETB-K-8794
11.54Single6IBLArformoterol6IBL-β1-Arformoterol
11.54Single6K1QIRL25006K1Q-ETB-IRL2500
11.54Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
11.54Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
11.54Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
11.54Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
11.54Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
11.54Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
11.54Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
11.54Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
11.54Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
11.54Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
11.43Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
11.43Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
11.43Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
11.11Single3NY9ICI118-5513NY9-β2-ICI118-551
11.11Single3RFMCaffeine3RFM-A2A-Caffeine
11.11Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
11.11Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
11.11Single6TQ9SB-4081246TQ9-OX1-SB-408124
11.11Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
11.11Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
11.11Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
11.11Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
11.11Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
11.11Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
11.11Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single9JF4PD1683689JF4-BB1-PD168368
11.11Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
11.11Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
10.81Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
10.71Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
10.71Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
10.71Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
10.71Single8IEBA1LYA8IEB-GPR156-A1LYA
10.71Single8IEIA1LYA8IEI-GPR156-A1LYA
10.71Single8IEIA1LYA8IEI-GPR156-A1LYA
10.71Single8IEPA1LYA8IEP-GPR156-A1LYA
10.71Single8IEPA1LYA8IEP-GPR156-A1LYA
10.71Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
10.71Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
10.71Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
10.71Single9M4TSilodosin9M4T-Alpha1A-Silodosin
10.53Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
10.53Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
10.53Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
10.53Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
10.53Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
10.53Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.53Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
10.53Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
10.53Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
10.53Single8JPSCCL78JPS-ACKR1-CCL7
10.53Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
10.53Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
10.53Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
10.34Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
10.26Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
10.26Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
10.00Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
10.00Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
10.00Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
10.00Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
10.00Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
10.00Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
10.00Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
10.00Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
10.00Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
10.00Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
10.00Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
10.00Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
10.00Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
10.00Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
9.68Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
9.68Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
9.68Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
9.52Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
9.52Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
9.52Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
9.52Single4S0VSuvorexant4S0V-OX2-Suvorexant
9.52Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
9.52Single5WS3EMPA5WS3-OX2-EMPA
9.52Single6B73MP11046B73-κ-MP1104
9.52Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
9.52Single6ME2Ramelteon6ME2-MT1-Ramelteon
9.52Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
9.52Single6TPJSuvorexant6TPJ-OX2-Suvorexant
9.52Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
9.52Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
9.52Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
9.52Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
9.52Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
9.52Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.52Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
9.52Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
9.52Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.52Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
9.52Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.52Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
9.52Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
9.52Single8Y0HVUF114188Y0H-CXCR3-VUF11418
9.52Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
9.52Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
9.52Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
9.52Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
9.52Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
9.52Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
9.52Consensusorexin_offOrthosteric Ligandox2_off ox1_off
9.52Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
9.52Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
9.52Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
9.52Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
9.38Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
9.38Consensuscalcitonin_onOrthosteric Ligandctlike_on
9.38Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
9.30Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
9.09Single2YDOAdenosine2YDO-A2A-Adenosine
9.09Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
9.09Single4ZJCSB-6740424ZJC-OX1-SB-674042
9.09Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
9.09Single6KUXRS-799486KUX-α2a-RS-79948
9.09Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
9.09Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
9.09Single6TP3Nemorexant6TP3-OX1-Nemorexant
9.09Single6TPGEMPA6TPG-OX2-EMPA
9.09Single6TPKRetosiban6TPK-OT-Retosiban
9.09Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
9.09Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
9.09Single7UL3Famotidine7UL3-H2-Famotidine
9.09Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
9.09Single7VV6C48/807VV6-MRGPRX2-C48/80
9.09Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
9.09Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
9.09Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.09Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
9.09Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
9.09Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
9.09Single8RLNLUF58348RLN-A2A-LUF5834
9.09Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
9.09Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.09Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
9.09Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
9.09Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
9.09Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
9.09Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
9.09Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
9.09Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
9.09Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
9.09Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
9.09Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
9.09Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
9.09Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
9.09Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
9.09Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
9.09Consensusvasop-oxy_offOrthosteric Ligandot_off
8.82Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
8.82Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
8.82Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
8.82Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
8.82Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
8.70Single2Y02Carmoterol2Y02-β1-Carmoterol
8.70Single2Y04Salbutamol2Y04-β1-Salbutamol
8.70Single4QKX35V4QKX-β2-35V
8.70Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
8.70Single5DHHSB-6121115DHH-NOP-SB-612111
8.70Single5TGZAM65385TGZ-CB1-AM6538
8.70Single6DRXLisuride6DRX-5-HT2B-Lisuride
8.70Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
8.70Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
8.70Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
8.70Single6GPSMK08126GPS-CCR2-MK0812
8.70Single6PS1Timolol6PS1-β2-Timolol
8.70Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
8.70Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
8.70Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
8.70Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
8.70Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
8.70Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
8.70Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
8.70Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
8.70Single7YXAONO-54306087YXA-S1P5-ONO-5430608
8.70Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
8.70Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
8.70Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
8.70Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
8.70Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
8.70Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
8.70Single8T1WCVN4248T1W-GPR6-CVN424
8.70Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
8.70Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
8.70Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.70Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.70Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.70Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.70Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.70Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
8.70Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
8.70Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
8.70Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
8.70Single9CHXS-Carazolol9CHX-β2-S-Carazolol
8.70Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
8.70Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
8.70Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
8.70Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
8.70Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
8.70Consensusblt_onOrthosteric Ligandblt1_on
8.70Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
8.70Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
8.70Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
8.70Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
8.70Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
8.70Consensusleukotriene_onOrthosteric Ligandblt_on
8.70Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
8.57Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
8.57Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
8.33Single2Y00Dobutamine2Y00-β1-Dobutamine
8.33Single2Y03Isoprenaline2Y03-β1-Isoprenaline
8.33Single4NTJAZD12834NTJ-P2Y12-AZD1283
8.33Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
8.33Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
8.33Single5C1MBU725C1M-μ-BU72
8.33Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
8.33Single6GPXMK08126GPX-CCR2-MK0812
8.33Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
8.33Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
8.33Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
8.33Single6TP6Filorexant6TP6-OX1-Filorexant
8.33Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
8.33Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
8.33Single7SINNPS-21437SIN-CaS-NPS-2143
8.33Single7SINNPS-21437SIN-CaS-NPS-2143
8.33Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
8.33Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
8.33Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
8.33Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
8.33Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
8.33Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
8.33Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
8.33Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
8.33Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.33Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.33Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.33Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
8.33Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
8.33Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
8.33Single9HAPTolvaptan9HAP-V2-Tolvaptan
8.33Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
8.33Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
8.33Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
8.33Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
8.33Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
8.33Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
8.33Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
8.33Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.33Consensustrace-amine_onOrthosteric Ligandta1_on
8.11Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
8.11Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
8.00Single2YDVNECA2YDV-A2A-NECA
8.00Single3P0GBI1671073P0G-β2-BI167107
8.00Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
8.00Single4DJHJDTic4DJH-κ-JDTic
8.00Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
8.00Single4UHRCGS216804UHR-A2A-CGS21680
8.00Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
8.00Single5G53NECA5G53-A2A-NECA-Gs
8.00Single6H7JIsoprenaline6H7J-β1-Isoprenaline
8.00Single6J20Aprepitant6J20-NK1-Aprepitant
8.00Single6J21Aprepitant6J21-NK1-Aprepitant
8.00Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
8.00Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
8.00Single6TQ7SB-3348676TQ7-OX1-SB-334867
8.00Single6WGTLSD6WGT-5-HT2A-LSD
8.00Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
8.00Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
8.00Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
8.00Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
8.00Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
8.00Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
8.00Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
8.00Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
8.00Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
8.00Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
8.00Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
8.00Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
8.00Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
8.00Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
8.00Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
8.00Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
8.00Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
8.00Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.00Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
7.69Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
7.69Single4AMIBucindolol4AMI-β1-Bucindolol
7.69Single4LDEBI1671074LDE-β2-BI167107
7.69Single4N4WSANT-14N4W-SMO-SANT-1
7.69Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
7.69Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
7.69Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
7.69Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
7.69Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
7.69Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
7.69Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
7.69Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
7.69Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
7.69Single8JJ8Formoterol8JJ8-β2-Formoterol
7.69Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.69Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
7.69Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
7.69Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
7.69Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
7.69Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
7.41Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
7.41Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
7.41Single6H7LDobutamine6H7L-β1-Dobutamine
7.41Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
7.41Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
7.41Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
7.41Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
7.41Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
7.41Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
7.41Single7UM4AS26747237UM4-5-HT5A-AS2674723
7.41Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
7.41Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
7.41Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
7.41Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
7.41Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
7.41Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.41Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
7.41Single9JH5C16:0 Ceramide9JH5-CysLT2-C16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
7.41Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
7.41Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
7.14Single6PT3DPI-2876PT3-δ-DPI-287
7.14Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
7.14Single7SK9CCX6627SK9-ACKR3-CCX662
7.14Single8X5YAstemizole8X5Y-H1-Astemizole
7.14Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
7.14Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
7.14Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
6.90Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
6.67Single6HLOAprepitant6HLO-NK1-Aprepitant
6.67Single8W8SAA-148W8S-GPR101-AA-14
6.67Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
6.67Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
6.45Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
6.25Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
6.25Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
6.25Single8W8RAA-148W8R-GPR101-AA-14-chim(NtGi1-Gs)/β1/γ2
6.25Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
6.25Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
6.25Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
6.06Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
5.88Single5MZPCaffeine5MZP-A2A-Caffeine-Na
5.88Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
5.88Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
5.88Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
5.56Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
5.56Single7WC4Serotonin7WC4-5-HT2A-Serotonin
5.56Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
5.56Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
5.56Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
5.26Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
5.26Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
5.26Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
5.26Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
5.26Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
5.26Single9IVMLSN33188399IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
5.26Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
5.26Consensussensory_onOrthosteric Ligandopsins_on
5.00Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
5.00Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
5.00Single3UZAGTPL92363UZA-A2A-GTPL9236
5.00Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
5.00Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
5.00Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
5.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.00Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
5.00Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
5.00Single7WC5Psilocin7WC5-5-HT2A-Psilocin
5.00Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.00Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
5.00Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
5.00Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
5.00Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
5.00Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
5.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
5.00Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
5.00Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
5.00Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
5.00Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
5.00Consensusgi_sensoryOrthosteric Ligandgi_opsins
5.00Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
5.00Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
5.00Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
5.00Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
5.00Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
4.76Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
4.76Single3PBLEticlopride3PBL-D3-Eticlopride
4.76Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
4.76Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
4.76Single6HLLCP999946HLL-NK1-CP99994
4.76Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
4.76Single6LI0C176LI0-GPR52-C17
4.76Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
4.76Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
4.76Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
4.76Single6TP4ACT-4622066TP4-OX1-ACT-462206
4.76Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.76Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.76Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
4.76Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
4.76Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
4.76Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
4.76Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
4.76Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
4.76Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
4.76Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
4.76Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
4.76Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
4.76Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
4.76Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.76Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
4.76Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
4.76Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.76Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
4.76Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
4.76Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9B9Y7DY9B9Y-CB1-7DY
4.76Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.76Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
4.76Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
4.76Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
4.55Single5U09Taranabant5U09-CB1-Taranabant
4.55Single6AKXA4R6AKX-CCR5-A4R
4.55Single6AKYMaraviroc6AKY-CCR5-Maraviroc
4.55Single6DS0Ly2660976DS0-5-HT2B-Ly266097
4.55Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
4.55Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
4.55Single6TODEMPA6TOD-OX1-EMPA-Na
4.55Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
4.55Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
4.55Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
4.55Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.55Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.55Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.55Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.55Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
4.55Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
4.55Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
4.55Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
4.55Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.55Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
4.55Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
4.55Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
4.55Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
4.55Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
4.55Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
4.55Single8IWESpermidine8IWE-TA9-Spermidine
4.55Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
4.55Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
4.55Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.55Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
4.55Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.55Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.55Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.55Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
4.55Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
4.55Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.55Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.55Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
4.55Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
4.55Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
4.55Consensusalpha2_offOrthosteric Ligandalpha2c_off
4.55Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
4.55Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
4.55Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
4.35Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
4.35Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
4.35Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
4.35Single4MBSMaraviroc4MBS-CCR5-Maraviroc
4.35Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
4.35Single6A94Zotepine6A94-5-HT2A-Zotepine
4.35Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
4.35Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
4.35Single6PS0S-Carazolol6PS0-β2-S-Carazolol
4.35Single6PS4ICI118-5516PS4-β2-ICI118-551
4.35Single6PS5S-Propranolol6PS5-β2-S-Propranolol
4.35Single6TPNHTL66416TPN-OX2-HTL6641
4.35Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
4.35Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
4.35Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
4.35Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
4.35Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
4.35Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
4.35Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.35Single7VODCariprazine7VOD-5-HT2A-Cariprazine
4.35Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
4.35Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
4.35Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
4.35Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
4.35Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
4.35Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
4.35Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
4.35Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.35Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.35Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
4.35Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
4.35Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
4.35Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
4.35Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
4.35Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
4.35Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
4.35Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
4.35Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
4.35Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.35Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.35Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.35Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.35Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
4.35Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
4.35Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
4.35Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.35Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.35Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
4.35Single9AS3LSD9AS3-5-HT2A-LSD
4.35Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9AS5Mescaline9AS5-5-HT2A-Mescaline
4.35Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.35Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9BA0A1AKN9BA0-CB1-A1AKN
4.35Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
4.35Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
4.35Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
4.35Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
4.35Consensusopsins_offOrthosteric Ligandrhodopsin_off
4.35Consensussensory_offOrthosteric Ligandopsins_off
4.17Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
4.17Single2Y01Dobutamine2Y01-β1-Dobutamine
4.17Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
4.17Single3NY8ICI118-5513NY8-β2-ICI118-551
4.17Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
4.17Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
4.17Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
4.17Single4EJ4Naltrindole4EJ4-δ-Naltrindole
4.17Single4GBRS-Carazolol4GBR-β2-S-Carazolol
4.17Single6H7MSalbutamol6H7M-β1-Salbutamol
4.17Single6IIVDaltroban6IIV-TXA2-Daltroban
4.17Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
4.17Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
4.17Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
4.17Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
4.17Single7BU7BI1671077BU7-β1-BI167107
4.17Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
4.17Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
4.17Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
4.17Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
4.17Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
4.17Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
4.17Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
4.17Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
4.17Single7WC7Lisuride7WC7-5-HT2A-Lisuride
4.17Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
4.17Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
4.17Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
4.17Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
4.17Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
4.17Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
4.17Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
4.17Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
4.17Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.17Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.17Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.17Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.17Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.17Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.17Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.17Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.17Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.17Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.17Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
4.17Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
4.17Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
4.17Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
4.17Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
4.17Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
4.17Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
4.17Single8JJOAlprenolol8JJO-β2-Alprenolol
4.17Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
4.17Single8JXRLSD8JXR-D1-LSD
4.17Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.17Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.17Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
4.17Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
4.17Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
4.17Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
4.17Single9AS1DMT9AS1-5-HT2A-DMT
4.17Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
4.17Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
4.17Consensus5ht5_onOrthosteric Ligand5ht5a_on
4.17Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
4.17Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
4.17Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
4.17Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
4.17Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
4.17Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
4.17Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
4.17Consensusdopamine_offOrthosteric Ligandd2_off d3_off
4.17Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
4.17Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
4.17Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
4.00Single2RH1S-Carazolol2RH1-β2-S-Carazolol
4.00Single2YCWS-Carazolol2YCW-β1-S-Carazolol
4.00Single5D6LS-Carazolol5D6L-β2-S-Carazolol
4.00Single5JQHS-Carazolol5JQH-β2-S-Carazolol
4.00Single5TVNLSD5TVN-5-HT2B-LSD
4.00Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
4.00Single5XPRBosentan5XPR-ETB-Bosentan
4.00Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
4.00Single6E67BI1671076E67-β2-BI167107-Gs(CT)
4.00Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
4.00Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
4.00Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
4.00Single6PS6Timolol6PS6-β2-Timolol
4.00Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
4.00Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.00Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
4.00Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
4.00Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
4.00Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
4.00Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
4.00Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
4.00Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.00Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.00Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
4.00Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
4.00Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
4.00Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
4.00Single8ZMFA1L108ZMF-5-HT2C-A1L10
4.00Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
4.00Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
4.00Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
4.00Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.00Single9B9ZA1AKO9B9Z-CB1-A1AKO
4.00Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
4.00Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
4.00Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
4.00Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
4.00Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.00Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
4.00Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
4.00Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
4.00Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
4.00Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
4.00Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
4.00Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
4.00Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
4.00Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
4.00Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
4.00Consensusamine_offonOrthosteric Ligandamine_off amine_on
4.00Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
4.00Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
4.00Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
4.00Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
4.00Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
3.85Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
3.85Single5D5AS-Carazolol5D5A-β2-S-Carazolol
3.85Single5D5BS-Carazolol5D5B-β2-S-Carazolol
3.85Single5V54Methiothepin5V54-5-HT1B-Methiothepin
3.85Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
3.85Single6E59L-7607356E59-NK1-L-760735
3.85Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
3.85Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
3.85Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
3.85Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
3.85Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
3.85Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
3.85Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
3.85Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
3.85Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
3.85Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
3.85Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
3.85Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
3.85Single9BJKNaloxone9BJK-μ-Naloxone-NAM
3.85Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.85Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
3.85Consensus5ht1_offOrthosteric Ligand5ht1b_off
3.85Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
3.85Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
3.85Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
3.85Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
3.85Consensustachykinin_offOrthosteric Ligandnk1_off
3.70Single3D4STimolol3D4S-β2-Timolol
3.70Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
3.70Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
3.70Single6CM4Risperidone6CM4-D2-Risperidone
3.70Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
3.70Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
3.70Single6IIURamatroban6IIU-TXA2-Ramatroban
3.70Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
3.70Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
3.70Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
3.70Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
3.70Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
3.70Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
3.57Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
3.57Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
3.57Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
3.57Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
3.57Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
3.57Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
3.57Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
3.57Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
3.57Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
3.57Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
3.45Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
3.45Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
3.45Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
3.45Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
3.33Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
3.03Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2

Consensus Members
Id Members
gal2_on_gp 7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
gal1_on_gp 7WQ3-GAL1-Galanin-Gi1/β1/γ2
Net Summary
Imin 2.5425
Number of Linked Nodes 898
Number of Links 1143
Number of Hubs 204
Number of Links mediated by Hubs 756
Number of Communities 23
Number of Nodes involved in Communities 293
Number of Links involved in Communities 445
Path Summary
Number Of Nodes in MetaPath 94
Number Of Links MetaPath 93
Number of Shortest Paths 3495358
Length Of Smallest Path 3
Average Path Length 35.502
Length of Longest Path 63
Minimum Path Strength 0.7125
Average Path Strength 5.12124
Maximum Path Strength 23.2388
Minimum Path Correlation 0.7
Average Path Correlation 0.985789
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 1.78571
Average % Of Corr. Nodes 32.7315
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 63.7243
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
peptide_on_gpcck_on_gp
angiotensin_on_gp
apelin_on_gp
bombesin_on_gp
bradykinin_on_gp
compl-peptide_on_gp
endothelin_on_gp
formylpeptide_on_gp
galanin_on_gp
ghrelin_on_gp
kisspeptin_on_gp
melanocortin_on_gp
motilin_on_gp
neuromedin-u_on_gp
npy_on_gp
neurotensin_on_gp
opioid_on_gp
orexin_on_gp
relaxin_on_gp
somatostatin_on_gp
tachykinin_on_gp
trh_on_gp
vasop-oxy_on_gp



You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

Download galanin_on_gp.zip



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You can also  read or  download a guide explaining the meaning of all files and numerical data.